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—— (5Z)-5-[(3-methylphenyl)methylidene]-2-[(2E)-2-[(1R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one —— C21H25N3OS
(5Z)-5-[(3-methylphenyl)methylidene]-2-[(2E)-2-[(1R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one
—— (5S,7S)-3-bromo-N-[2-[cyclohexyl(methyl)amino]ethyl]-N-methyladamantane-1-carboxamide —— C21H35BrN2O
(5S,7S)-3-bromo-N-[2-[cyclohexyl(methyl)amino]ethyl]-N-methyladamantane-1-carboxamide
—— (5Z)-3-benzyl-5-[(2,5-diphenyl-1,2,4-triazol-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C25H18N4OS2
(5Z)-3-benzyl-5-[(2,5-diphenyl-1,2,4-triazol-3-yl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S,7S)-3-bromo-N-[(2S)-2-cyanopropyl]-N-methyladamantane-1-carboxamide —— C16H23BrN2O
(5S,7S)-3-bromo-N-[(2S)-2-cyanopropyl]-N-methyladamantane-1-carboxamide
—— (5S,7S)-3-bromo-N-(2-tert-butylpyrimidin-5-yl)adamantane-1-carboxamide —— C19H26BrN3O
(5S,7S)-3-bromo-N-(2-tert-butylpyrimidin-5-yl)adamantane-1-carboxamide
—— (5S,7S)-3-bromo-N-[(2R)-2-cyanopropyl]-N-methyladamantane-1-carboxamide —— C16H23BrN2O
(5S,7S)-3-bromo-N-[(2R)-2-cyanopropyl]-N-methyladamantane-1-carboxamide
—— (5E)-5-[[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one —— C22H23FN2O3S
(5E)-5-[[3-ethoxy-4-[(2-fluorophenyl)methoxy]phenyl]methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one
—— (5E)-5-[(2,7-dimethoxynaphthalen-1-yl)methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one —— C19H20N2O3S
(5E)-5-[(2,7-dimethoxynaphthalen-1-yl)methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one
—— (5Z)-3-methyl-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H16N4OS2
(5Z)-3-methyl-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5S)-3-[(E)-benzylideneamino]-5-phenyl-1-prop-2-enyl-2-sulfanylideneimidazolidin-4-one —— C19H17N3OS
(5S)-3-[(E)-benzylideneamino]-5-phenyl-1-prop-2-enyl-2-sulfanylideneimidazolidin-4-one
—— (5E)-3-cyclohexyl-5-[(2,7-diethoxynaphthalen-1-yl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C24H28N2O3S
(5E)-3-cyclohexyl-5-[(2,7-diethoxynaphthalen-1-yl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5S,6R,7aS)-N-(3,5-dimethylphenyl)-1'-methyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide —— C23H25N3O2S
(5S,6R,7aS)-N-(3,5-dimethylphenyl)-1'-methyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(2-tert-butylphenoxy)acetate —— C19H20N2O5
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 2-(2-tert-butylphenoxy)acetate
—— 5-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-3-[(3S)-piperidin-3-yl]-1,2,4-oxadiazole —— C15H23N3O
5-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-3-[(3S)-piperidin-3-yl]-1,2,4-oxadiazole
—— (5Z)-3-benzyl-5-[[5-(3-fluorophenyl)furan-2-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C21H14FNO2S2
(5Z)-3-benzyl-5-[[5-(3-fluorophenyl)furan-2-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R)-3-[(E)-benzylideneamino]-5-phenyl-1-prop-2-enyl-2-sulfanylideneimidazolidin-4-one —— C19H17N3OS
(5R)-3-[(E)-benzylideneamino]-5-phenyl-1-prop-2-enyl-2-sulfanylideneimidazolidin-4-one
—— (5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H20N4OS2
(5Z)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-propan-2-yl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R,10bS)-2-(4-methoxyphenyl)-5-(5-methylfuran-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C22H20N2O3
(5R,10bS)-2-(4-methoxyphenyl)-5-(5-methylfuran-2-yl)-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5Z)-3-(2-methoxyethyl)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C22H20N4O2S2
(5Z)-3-(2-methoxyethyl)-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5R,5'E,10bS)-5'-benzylidene-9-bromo-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazolidine]-2'-one —— C25H18BrN3O2S
(5R,5'E,10bS)-5'-benzylidene-9-bromo-2-phenylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,4'-1,3-thiazolidine]-2'-one
—— (5E)-5-[(1-benzylindol-3-yl)methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one —— C22H21N3OS
(5E)-5-[(1-benzylindol-3-yl)methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one
—— (5Z)-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C20H23N3O3S2
(5Z)-5-[[(1S,9S)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-11-yl]methylidene]-3-[[(2R)-oxolan-2-yl]methyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5Z)-5-[(5-methylfuran-2-yl)methylidene]-2-[(Z)-2-(4-methylphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C19H15N3O2S
(5Z)-5-[(5-methylfuran-2-yl)methylidene]-2-[(Z)-2-(4-methylphenyl)ethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (5S)-3-[(E)-benzylideneamino]-1-methyl-5-phenyl-2-sulfanylideneimidazolidin-4-one —— C17H15N3OS
(5S)-3-[(E)-benzylideneamino]-1-methyl-5-phenyl-2-sulfanylideneimidazolidin-4-one
—— (5Z)-5-[(3-methylphenyl)methylidene]-2-[(2Z)-2-[(1R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one —— C21H25N3OS
(5Z)-5-[(3-methylphenyl)methylidene]-2-[(2Z)-2-[(1R,4S)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one
—— (5Z)-5-[[5-(4-chlorophenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one —— C19H13ClN4OS2
(5Z)-5-[[5-(4-chlorophenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-3-methyl-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[5-(3,4-dichlorophenyl)furan-2-yl]methylidene]-2-[(Z)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one —— C23H13Cl2N3O2S
(5E)-5-[[5-(3,4-dichlorophenyl)furan-2-yl]methylidene]-2-[(Z)-2-phenylethenyl]-[1,3]thiazolo[3,2-b][1,2,4]triazol-6-one
—— (5Z)-3-(4-chlorophenyl)-2-hydrazinyl-5-[(4-methoxyphenyl)methylidene]imidazol-4-one —— C17H15ClN4O2
(5Z)-3-(4-chlorophenyl)-2-hydrazinyl-5-[(4-methoxyphenyl)methylidene]imidazol-4-one
—— (5E)-5-[[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one —— C22H24N2O3S
(5E)-5-[[3-methoxy-4-[(4-methylphenyl)methoxy]phenyl]methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one
—— (5R,10bS)-5-(furan-2-yl)-7-methoxy-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine —— C19H16N2O3S
(5R,10bS)-5-(furan-2-yl)-7-methoxy-2-thiophen-2-yl-5,10b-dihydro-1H-pyrazolo[1,5-c][1,3]benzoxazine
—— (5Z)-3-[(2R)-butan-2-yl]-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C23H22N4OS2
(5Z)-3-[(2R)-butan-2-yl]-5-[[5-(4-methylphenyl)-2-phenyl-1,2,4-triazol-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one —— C15H17BrN2O3S
(5E)-5-[(3-bromo-5-ethoxy-4-hydroxyphenyl)methylidene]-3-propyl-2-sulfanylideneimidazolidin-4-one
—— (5Z)-5-[(3-nitro-4-piperidin-1-ylphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one —— C15H16N4O3S
(5Z)-5-[(3-nitro-4-piperidin-1-ylphenyl)methylidene]-2-sulfanylideneimidazolidin-4-one
—— (5S,6S,7aS)-N-(3,5-dimethylphenyl)-1'-methyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide —— C23H25N3O2S
(5S,6S,7aS)-N-(3,5-dimethylphenyl)-1'-methyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide
—— 5-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-3-[(3R)-piperidin-3-yl]-1,2,4-oxadiazole —— C15H23N3O
5-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]methyl]-3-[(3R)-piperidin-3-yl]-1,2,4-oxadiazole
—— (5R,6R,7aR)-N-(2-ethoxyphenyl)-1'-ethyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide —— C24H27N3O3S
(5R,6R,7aR)-N-(2-ethoxyphenyl)-1'-ethyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide
—— (5R,6S,7aR)-N-(2-ethoxyphenyl)-1'-ethyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide —— C24H27N3O3S
(5R,6S,7aR)-N-(2-ethoxyphenyl)-1'-ethyl-2'-oxospiro[3,6,7,7a-tetrahydro-1H-pyrrolo[1,2-c][1,3]thiazole-5,3'-indole]-6-carboxamide
—— 5-[[1-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
—— (5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-[3-[4-[(5E)-5-[(4-methoxyphenyl)methylidene]-4-oxo-1,3-thiazol-2-yl]piperazin-1-yl]-3-oxopropyl]-2-sulfanylidene-1,3-thiazolidin-4-one —— C29H26N4O6S3
(5Z)-5-(1,3-benzodioxol-5-ylmethylidene)-3-[3-[4-[(5E)-5-[(4-methoxyphenyl)methylidene]-4-oxo-1,3-thiazol-2-yl]piperazin-1-yl]-3-oxopropyl]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[[1-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
—— (5E)-3-(2-methoxyethyl)-5-[[2-[4-(2-methoxyphenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C26H27N5O4S2
(5E)-3-(2-methoxyethyl)-5-[[2-[4-(2-methoxyphenyl)piperazin-1-yl]-4-oxopyrido[1,2-a]pyrimidin-3-yl]methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— (5E)-5-[[4-methoxy-3-[(2,4,6-trichlorophenoxy)methyl]phenyl]methylidene]-2-[(2E)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one —— C28H28Cl3N3O3S
(5E)-5-[[4-methoxy-3-[(2,4,6-trichlorophenoxy)methyl]phenyl]methylidene]-2-[(2E)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one
—— (5E)-4-(4-methoxyanilino)-5-[(E)-3-phenylprop-2-enylidene]-1,3-thiazol-2-one —— C19H16N2O2S
(5E)-4-(4-methoxyanilino)-5-[(E)-3-phenylprop-2-enylidene]-1,3-thiazol-2-one
—— 5-[[1-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole
—— (5E)-5-[[4-methoxy-3-[(2,4,6-trichlorophenoxy)methyl]phenyl]methylidene]-2-[(2Z)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one —— C28H28Cl3N3O3S
(5E)-5-[[4-methoxy-3-[(2,4,6-trichlorophenoxy)methyl]phenyl]methylidene]-2-[(2Z)-2-[(1S,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]hydrazinyl]-1,3-thiazol-4-one
—— (5,6-Dichloropyridin-3-yl)-[2-(2-methylphenyl)imino-1,3-thiazolidin-3-yl]methanone —— C16H13Cl2N3OS
(5,6-Dichloropyridin-3-yl)-[2-(2-methylphenyl)imino-1,3-thiazolidin-3-yl]methanone
—— [5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 1-(thiophene-2-carbonyl)piperidine-4-carboxylate —— C18H17N3O5S
[5-(Furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl 1-(thiophene-2-carbonyl)piperidine-4-carboxylate
—— [5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 1-ethyl-3-methyl-2-oxoquinoxaline-6-carboxylate —— C21H20N4O5
[5-(2,5-Dimethylfuran-3-yl)-1,3,4-oxadiazol-2-yl]methyl 1-ethyl-3-methyl-2-oxoquinoxaline-6-carboxylate
—— (5-Phenyl-1,3-oxazol-2-yl)methyl 1-(thiophene-2-carbonyl)piperidine-4-carboxylate —— C21H20N2O4S
(5-Phenyl-1,3-oxazol-2-yl)methyl 1-(thiophene-2-carbonyl)piperidine-4-carboxylate
—— 5-[[1-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole —— C24H30N4O4S
5-[[1-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-4,5-dimethylimidazol-2-yl]sulfonylmethyl]-3-(4-methoxyphenyl)-1,2,4-oxadiazole