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—— 5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-4-methyl-1-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H33N5O7S
5-[2-(tert-butylsulfamoyl)-4-nitrophenoxy]-4-methyl-1-(4-methylphenyl)-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— (5R,10bS)-5',5'-dimethyl-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-cyclohexene]-1'-ol —— C21H22N2O2S
(5R,10bS)-5',5'-dimethyl-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-cyclohexene]-1'-ol
—— 5,6-dimethyl-3-[2-oxo-2-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)ethyl]thieno[2,3-d]pyrimidin-4-one —— C19H17N3O3S
5,6-dimethyl-3-[2-oxo-2-(2-oxo-3,4-dihydro-1H-quinolin-6-yl)ethyl]thieno[2,3-d]pyrimidin-4-one
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,5-dimethylphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,5-dimethylphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— (5S,7S)-3-acetamido-N-[(2R)-2-[1-(difluoromethyl)benzimidazol-2-yl]propyl]adamantane-1-carboxamide —— C24H30F2N4O2
(5S,7S)-3-acetamido-N-[(2R)-2-[1-(difluoromethyl)benzimidazol-2-yl]propyl]adamantane-1-carboxamide
—— 5-[[3-(3-bromophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-methyl-1,3,4-thiadiazol-2-amine —— C12H10BrN5OS2
5-[[3-(3-bromophenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-N-methyl-1,3,4-thiadiazol-2-amine
—— 5,6-dimethyl-3-{2-[1-(methylsulfonyl)-2,3-dihydro-1H-indol-5-yl]-2-oxoethyl}thieno[2,3-d]pyrimidin-4(3H)-one —— C19H19N3O4S2
5,6-dimethyl-3-{2-[1-(methylsulfonyl)-2,3-dihydro-1H-indol-5-yl]-2-oxoethyl}thieno[2,3-d]pyrimidin-4(3H)-one
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-4-methyl-1-propan-2-ylpyrazole-3-carboxylic acid —— C27H31F3N4O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-4-methyl-1-propan-2-ylpyrazole-3-carboxylic acid
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C18H11ClN2O4S
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— [5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,3-dihydro-1H-inden-5-ylsulfanyl)acetate —— C21H20N2O3S
[5-(3-methylphenyl)-1,3,4-oxadiazol-2-yl]methyl 2-(2,3-dihydro-1H-inden-5-ylsulfanyl)acetate
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid —— C25H27ClN4O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 5-[4-[(4-fluorobenzoyl)amino]-2-(3-methoxypropylsulfamoyl)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid —— C28H26F2N4O7S
5-[4-[(4-fluorobenzoyl)amino]-2-(3-methoxypropylsulfamoyl)phenoxy]-1-(3-fluorophenyl)-4-methylpyrazole-3-carboxylic acid
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate —— C20H13ClN2O3S
(5-Phenyl-1,2-oxazol-3-yl)methyl 2-(3-chlorophenyl)-1,3-thiazole-4-carboxylate
—— 5,6-Dimethyl-3-[2-oxo-2-(4-propan-2-ylphenyl)ethyl]thieno[2,3-d]pyrimidin-4-one —— C19H20N2O2S
5,6-Dimethyl-3-[2-oxo-2-(4-propan-2-ylphenyl)ethyl]thieno[2,3-d]pyrimidin-4-one
—— 5-[[5-(5-bromothiophen-2-yl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-N-methyl-1,3,4-thiadiazol-2-amine —— C10H8BrN5OS3
5-[[5-(5-bromothiophen-2-yl)-1,3,4-oxadiazol-2-yl]methylsulfanyl]-N-methyl-1,3,4-thiadiazol-2-amine
—— (5-acetyl-2-methoxyphenyl)methyl (2R)-3-phenyl-2-(tetrazol-1-yl)propanoate —— C20H20N4O4
(5-acetyl-2-methoxyphenyl)methyl (2R)-3-phenyl-2-(tetrazol-1-yl)propanoate
—— 5-[2-(1,3-benzodioxol-5-ylmethylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-1-tert-butyl-4-methylpyrazole-3-carboxylic acid —— C28H34N4O8S
5-[2-(1,3-benzodioxol-5-ylmethylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-1-tert-butyl-4-methylpyrazole-3-carboxylic acid
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,5-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,5-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3,3-dimethylbutanoylamino)phenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxylic acid —— C27H33FN4O6S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-(3,3-dimethylbutanoylamino)phenoxy]-1-(4-fluorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 5-[2-(cyclopropylsulfamoyl)-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-1,4-dimethylpyrazole-3-carboxylic acid —— C24H23F3N4O7S
5-[2-(cyclopropylsulfamoyl)-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-1,4-dimethylpyrazole-3-carboxylic acid
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2S)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-tert-butyl-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide —— C24H31N5O7S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-nitrophenoxy]-1-tert-butyl-N-(furan-2-ylmethyl)-4-methylpyrazole-3-carboxamide
—— 5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid —— C25H27ClN4O6S
5-[2-[[(2S)-butan-2-yl]sulfamoyl]-4-(cyclopropanecarbonylamino)phenoxy]-1-(4-chlorophenyl)-4-methylpyrazole-3-carboxylic acid
—— 5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-4-methyl-1-propan-2-ylpyrazole-3-carboxylic acid —— C27H31F3N4O7S
5-[2-[[(2R)-butan-2-yl]sulfamoyl]-4-[[4-methoxy-3-(trifluoromethyl)benzoyl]amino]phenoxy]-4-methyl-1-propan-2-ylpyrazole-3-carboxylic acid
—— (5R,7R)-3-(4-methoxyphenyl)-N-[(2S)-pentan-2-yl]adamantane-1-carboxamide —— C23H33NO2
(5R,7R)-3-(4-methoxyphenyl)-N-[(2S)-pentan-2-yl]adamantane-1-carboxamide
—— 5-[2-(1,3-benzodioxol-5-ylmethylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-1-tert-butyl-4-methylpyrazole-3-carboxylic acid —— C28H34N4O8S
5-[2-(1,3-benzodioxol-5-ylmethylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-1-tert-butyl-4-methylpyrazole-3-carboxylic acid
—— (5S,10bS)-5',5'-dimethyl-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-cyclohexene]-1'-ol —— C21H22N2O2S
(5S,10bS)-5',5'-dimethyl-2-thiophen-2-ylspiro[1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine-5,3'-cyclohexene]-1'-ol
—— 5-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C24H30FN5O2S
5-[[4-[(1R)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— (5R,7R)-3-(4-methoxyphenyl)-N-[(2R)-pentan-2-yl]adamantane-1-carboxamide —— C23H33NO2
(5R,7R)-3-(4-methoxyphenyl)-N-[(2R)-pentan-2-yl]adamantane-1-carboxamide
—— 5-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C24H30FN5O2S
5-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-ethyl-1,2,4-oxadiazole —— C23H28FN5O2S
5-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-ethyl-1,2,4-oxadiazole
—— 5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide —— C27H31N5O7S
5-[2-(cyclopropylsulfamoyl)-4-nitrophenoxy]-1-(2,3-dimethylphenyl)-4-methyl-N-[[(2R)-oxolan-2-yl]methyl]pyrazole-3-carboxamide
—— 5-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-ethyl-1,2,4-oxadiazole —— C23H28FN5O2S
5-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-ethyl-1,2,4-oxadiazole
—— 5-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-ethyl-1,2,4-oxadiazole —— C23H28FN5O2S
5-[[4-[(1S)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-ethyl-1,2,4-oxadiazole
—— 5-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C24H30FN5O2S
5-[[4-[(1S)-1-[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole —— C24H30FN5O2S
5-[[4-[(1R)-1-[(1R,2S,4R)-2-bicyclo[2.2.1]heptanyl]ethyl]-5-[(2-fluorophenoxy)methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]-3-propan-2-yl-1,2,4-oxadiazole
—— 5-[(2,5-Dimethoxyphenyl)methylsulfanyl]-1-(2,6-dimethylphenyl)tetrazole —— C18H20N4O2S
5-[(2,5-Dimethoxyphenyl)methylsulfanyl]-1-(2,6-dimethylphenyl)tetrazole
—— (5E)-5-[(3-bromo-4-phenylmethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C17H12BrNO2S2
(5E)-5-[(3-bromo-4-phenylmethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— 5-[2-(tert-butylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C27H34N4O7S
5-[2-(tert-butylsulfamoyl)-4-[[(2S)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— [5-(diethylamino)-2-[[ethylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate —— C25H33Cl2N3O5S
[5-(diethylamino)-2-[[ethylcarbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate
—— 5-[4-(cyclopentanecarbonylamino)-2-(propylsulfamoyl)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C27H32N4O7S
5-[4-(cyclopentanecarbonylamino)-2-(propylsulfamoyl)phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— 5-[4-(cyclobutanecarbonylamino)-2-morpholin-4-ylsulfonylphenoxy]-1-(2,3-dimethylphenyl)-4-methylpyrazole-3-carboxylic acid —— C28H32N4O7S
5-[4-(cyclobutanecarbonylamino)-2-morpholin-4-ylsulfonylphenoxy]-1-(2,3-dimethylphenyl)-4-methylpyrazole-3-carboxylic acid
—— (5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 5-chloro-1-benzofuran-2-carboxylate —— C16H9ClN2O4S
(5-Oxo-[1,3]thiazolo[3,2-a]pyrimidin-7-yl)methyl 5-chloro-1-benzofuran-2-carboxylate
—— [5-(diethylamino)-2-[[(2-methoxyacetyl)-[[(2R)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate —— C25H32Cl2N2O6S
[5-(diethylamino)-2-[[(2-methoxyacetyl)-[[(2R)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate
—— (5E)-5-[(3-bromo-5-methoxy-4-phenylmethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one —— C18H14BrNO3S2
(5E)-5-[(3-bromo-5-methoxy-4-phenylmethoxyphenyl)methylidene]-2-sulfanylidene-1,3-thiazolidin-4-one
—— [5-(diethylamino)-2-[[(2-methoxyacetyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate —— C25H32Cl2N2O6S
[5-(diethylamino)-2-[[(2-methoxyacetyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate
—— [5-(diethylamino)-2-[[ethylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate —— C25H33Cl2N3O5S
[5-(diethylamino)-2-[[ethylcarbamoyl-[[(2S)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3,4-dichlorobenzenesulfonate
—— 5-[2-(tert-butylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid —— C27H34N4O7S
5-[2-(tert-butylsulfamoyl)-4-[[(2R)-2-methylbutanoyl]amino]phenoxy]-1-(4-methoxyphenyl)-4-methylpyrazole-3-carboxylic acid
—— [5-(diethylamino)-2-[[(2-methoxyphenyl)carbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3-(trifluoromethyl)benzenesulfonate —— C31H36F3N3O6S
[5-(diethylamino)-2-[[(2-methoxyphenyl)carbamoyl-[[(2R)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3-(trifluoromethyl)benzenesulfonate
—— [5-(diethylamino)-2-[[(2-methoxyacetyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3-(trifluoromethyl)benzenesulfonate —— C26H33F3N2O6S
[5-(diethylamino)-2-[[(2-methoxyacetyl)-[[(2S)-oxolan-2-yl]methyl]amino]methyl]phenyl] 3-(trifluoromethyl)benzenesulfonate