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—— ethyl 2-[5-[(1S)-1-[1,3-benzodioxol-5-ylmethyl-[(5,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]amino]butyl]tetrazol-1-yl]acetate —— C29H34N6O5
ethyl 2-[5-[(1S)-1-[1,3-benzodioxol-5-ylmethyl-[(5,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]amino]butyl]tetrazol-1-yl]acetate
—— (E)-3-(2,5-dimethoxyphenyl)-N-(6-ethoxy-1,3-benzothiazol-2-yl)prop-2-enamide —— C20H20N2O4S
(E)-3-(2,5-dimethoxyphenyl)-N-(6-ethoxy-1,3-benzothiazol-2-yl)prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[3-[(4-methoxyphenyl)sulfamoyl]-4-pyrrolidin-1-ylphenyl]prop-2-enamide —— C26H26FN3O4S
(E)-3-(4-fluorophenyl)-N-[3-[(4-methoxyphenyl)sulfamoyl]-4-pyrrolidin-1-ylphenyl]prop-2-enamide
—— (E)-N-benzyl-3-(furan-2-yl)-N-[4-(4-methoxynaphthalen-1-yl)-1,3-thiazol-2-yl]prop-2-enamide —— C28H22N2O3S
(E)-N-benzyl-3-(furan-2-yl)-N-[4-(4-methoxynaphthalen-1-yl)-1,3-thiazol-2-yl]prop-2-enamide
—— (E)-N'-[2-(2-benzylphenoxy)acetyl]-3-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)prop-2-enehydrazide —— C29H31N3O7S
(E)-N'-[2-(2-benzylphenoxy)acetyl]-3-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)prop-2-enehydrazide
—— (E)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]-1-(2-methyl-2,3-dihydroindol-1-yl)prop-2-en-1-one —— C29H23N3O2
(E)-3-[3-(1-benzofuran-2-yl)-1-phenylpyrazol-4-yl]-1-(2-methyl-2,3-dihydroindol-1-yl)prop-2-en-1-one
—— ethyl 2-[5-[(1R)-1-[1,3-benzodioxol-5-ylmethyl-[(5,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]amino]butyl]tetrazol-1-yl]acetate —— C29H34N6O5
ethyl 2-[5-[(1R)-1-[1,3-benzodioxol-5-ylmethyl-[(5,7-dimethyl-2-oxo-1H-quinolin-3-yl)methyl]amino]butyl]tetrazol-1-yl]acetate
—— ethyl 4-[2,5-dimethyl-3-[(Z)-(pyridin-2-ylhydrazinylidene)methyl]pyrrol-1-yl]benzoate —— C21H22N4O2
ethyl 4-[2,5-dimethyl-3-[(Z)-(pyridin-2-ylhydrazinylidene)methyl]pyrrol-1-yl]benzoate
—— (E,4E)-4-[(benzylamino)methylidene]-2,3-dimethylpent-2-enedioic acid —— C15H17NO4
(E,4E)-4-[(benzylamino)methylidene]-2,3-dimethylpent-2-enedioic acid
—— ethyl 4-[(3R)-5-acetyl-4-benzyl-3-[2-[(4-chlorophenyl)methoxy]phenyl]-3H-1,2,4-triazol-2-yl]benzoate —— C33H30ClN3O4
ethyl 4-[(3R)-5-acetyl-4-benzyl-3-[2-[(4-chlorophenyl)methoxy]phenyl]-3H-1,2,4-triazol-2-yl]benzoate
—— ethyl 4-[(4Z)-1,3-dioxo-4-[[2-(trifluoromethyl)phenyl]methylidene]isoquinolin-2-yl]benzoate —— C26H18F3NO4
ethyl 4-[(4Z)-1,3-dioxo-4-[[2-(trifluoromethyl)phenyl]methylidene]isoquinolin-2-yl]benzoate
—— ethyl 2-[3-[(Z)-[[(1S,6R,7R)-1-methylbicyclo[4.1.0]heptane-7-carbonyl]hydrazinylidene]methyl]indol-1-yl]acetate —— C22H27N3O3
ethyl 2-[3-[(Z)-[[(1S,6R,7R)-1-methylbicyclo[4.1.0]heptane-7-carbonyl]hydrazinylidene]methyl]indol-1-yl]acetate
—— (E)-1-(3,4-difluorophenyl)-3-(4-ethylphenyl)prop-2-en-1-one —— C17H14F2O
(E)-1-(3,4-difluorophenyl)-3-(4-ethylphenyl)prop-2-en-1-one
—— (E)-3-[3-ethoxy-4-[(6-nitro-4H-1,3-benzodioxin-8-yl)methoxy]phenyl]-1-(4-methoxyphenyl)prop-2-en-1-one —— C27H25NO8
(E)-3-[3-ethoxy-4-[(6-nitro-4H-1,3-benzodioxin-8-yl)methoxy]phenyl]-1-(4-methoxyphenyl)prop-2-en-1-one
—— ethyl ({(2Z)-2-[(2-methyl-2H-chromen-3-yl)methylidene]-3-oxo-2,3-dihydro-1-benzofuran-6-yl}oxy)acetate —— C23H20O6
ethyl ({(2Z)-2-[(2-methyl-2H-chromen-3-yl)methylidene]-3-oxo-2,3-dihydro-1-benzofuran-6-yl}oxy)acetate
—— (E)-N-[3-(dimethylsulfamoyl)phenyl]-3-[4-[(2-methoxyphenyl)sulfamoyl]phenyl]prop-2-enamide —— C24H25N3O6S2
(E)-N-[3-(dimethylsulfamoyl)phenyl]-3-[4-[(2-methoxyphenyl)sulfamoyl]phenyl]prop-2-enamide
—— ethyl 2-[5-[(1R)-2-methyl-1-[2-(2-methylphenyl)ethyl-[(6-oxo-5H-[1,3]dioxolo[4,5-g]quinolin-7-yl)methyl]amino]propyl]tetrazol-1-yl]acetate —— C29H34N6O5
ethyl 2-[5-[(1R)-2-methyl-1-[2-(2-methylphenyl)ethyl-[(6-oxo-5H-[1,3]dioxolo[4,5-g]quinolin-7-yl)methyl]amino]propyl]tetrazol-1-yl]acetate
—— (E)-N-[2,5-bis(trifluoromethyl)phenyl]-2-cyano-3-hydroxybut-2-enamide —— C13H8F6N2O2
(E)-N-[2,5-bis(trifluoromethyl)phenyl]-2-cyano-3-hydroxybut-2-enamide
—— ethyl 4-[(3S)-5-acetyl-4-benzyl-3-[2-[(4-chlorophenyl)methoxy]phenyl]-3H-1,2,4-triazol-2-yl]benzoate —— C33H30ClN3O4
ethyl 4-[(3S)-5-acetyl-4-benzyl-3-[2-[(4-chlorophenyl)methoxy]phenyl]-3H-1,2,4-triazol-2-yl]benzoate
—— ethyl 2-[3-[(Z)-[[(1S,6R,7S)-1-methylbicyclo[4.1.0]heptane-7-carbonyl]hydrazinylidene]methyl]indol-1-yl]acetate —— C22H27N3O3
ethyl 2-[3-[(Z)-[[(1S,6R,7S)-1-methylbicyclo[4.1.0]heptane-7-carbonyl]hydrazinylidene]methyl]indol-1-yl]acetate
—— ethyl (2Z)-2-[(5Z)-5-[(4-cyanophenyl)methylidene]-3-[2-[(2-methylcyclohexyl)amino]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate —— C24H27N3O4S
ethyl (2Z)-2-[(5Z)-5-[(4-cyanophenyl)methylidene]-3-[2-[(2-methylcyclohexyl)amino]-2-oxoethyl]-4-oxo-1,3-thiazolidin-2-ylidene]acetate
—— (E)-2-cyano-3-[(3-fluorophenyl)methylamino]-N-(2-phenylethyl)but-2-enamide —— C20H20FN3O
(E)-2-cyano-3-[(3-fluorophenyl)methylamino]-N-(2-phenylethyl)but-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 3-oxo-4H-1,4-benzothiazine-6-carboxylate —— C15H13N3O4S
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 3-oxo-4H-1,4-benzothiazine-6-carboxylate
—— (E)-3-(2,4-dimethoxyphenyl)-2-[4-(9H-fluoren-2-yl)-1,3-thiazol-2-yl]prop-2-enenitrile —— C27H20N2O2S
(E)-3-(2,4-dimethoxyphenyl)-2-[4-(9H-fluoren-2-yl)-1,3-thiazol-2-yl]prop-2-enenitrile
—— ethyl 4-(2-chlorophenyl)-2-[[(E)-[2-(3,4-dimethoxyphenyl)-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]thiophene-3-carboxylate —— C31H25ClN2O6S
ethyl 4-(2-chlorophenyl)-2-[[(E)-[2-(3,4-dimethoxyphenyl)-1,3-dioxoisoquinolin-4-ylidene]methyl]amino]thiophene-3-carboxylate
—— (E)-1-(4-benzhydrylpiperazin-1-yl)-3-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]prop-2-en-1-one —— C36H34N4O
(E)-1-(4-benzhydrylpiperazin-1-yl)-3-[3-(4-methylphenyl)-1-phenylpyrazol-4-yl]prop-2-en-1-one
—— (E,2S,3R)-5-amino-3-(2-chlorophenyl)-2,4-dicyano-5-methylsulfanyl-N-phenylpent-4-enamide —— C20H17ClN4OS
(E,2S,3R)-5-amino-3-(2-chlorophenyl)-2,4-dicyano-5-methylsulfanyl-N-phenylpent-4-enamide
—— (E)-1-[4-(difluoromethoxy)phenyl]-3-(4-hydroxy-3,5-dimethylphenyl)prop-2-en-1-one —— C18H16F2O3
(E)-1-[4-(difluoromethoxy)phenyl]-3-(4-hydroxy-3,5-dimethylphenyl)prop-2-en-1-one
—— ethyl 4-[(4Z)-1,3-dioxo-4-[[4-(pyrimidin-2-ylsulfamoyl)anilino]methylidene]isoquinolin-2-yl]benzoate —— C29H23N5O6S
ethyl 4-[(4Z)-1,3-dioxo-4-[[4-(pyrimidin-2-ylsulfamoyl)anilino]methylidene]isoquinolin-2-yl]benzoate
—— (E)-3-(1,3-benzothiazol-2-yl)-4-(3-bromo-5-ethoxy-4-methoxyphenyl)but-3-enoic acid —— C20H18BrNO4S
(E)-3-(1,3-benzothiazol-2-yl)-4-(3-bromo-5-ethoxy-4-methoxyphenyl)but-3-enoic acid
—— (E)-3-[4-(methylamino)-3-nitrophenyl]-1-(4-methyl-3-nitrophenyl)prop-2-en-1-one —— C17H15N3O5
(E)-3-[4-(methylamino)-3-nitrophenyl]-1-(4-methyl-3-nitrophenyl)prop-2-en-1-one
—— ethyl 2-[5-[(1R)-2-methyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl-(thiophen-2-ylmethyl)amino]propyl]tetrazol-1-yl]acetate —— C26H30N6O5S
ethyl 2-[5-[(1R)-2-methyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl-(thiophen-2-ylmethyl)amino]propyl]tetrazol-1-yl]acetate
—— (E)-3-(2-chlorophenyl)-1-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]prop-2-en-1-one —— C19H18ClFN2O3S
(E)-3-(2-chlorophenyl)-1-[4-(3-fluorophenyl)sulfonylpiperazin-1-yl]prop-2-en-1-one
—— (E,2R,3R)-5-amino-3-(2-chlorophenyl)-2,4-dicyano-5-methylsulfanyl-N-phenylpent-4-enamide —— C20H17ClN4OS
(E,2R,3R)-5-amino-3-(2-chlorophenyl)-2,4-dicyano-5-methylsulfanyl-N-phenylpent-4-enamide
—— ethyl 4-[(4Z)-4-[[5-[(2-chlorophenyl)sulfamoyl]-2-piperidin-1-ylanilino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate —— C36H33ClN4O6S
ethyl 4-[(4Z)-4-[[5-[(2-chlorophenyl)sulfamoyl]-2-piperidin-1-ylanilino]methylidene]-1,3-dioxoisoquinolin-2-yl]benzoate
—— (E,2R,3S)-5-amino-3-(2-chlorophenyl)-2,4-dicyano-5-methylsulfanyl-N-phenylpent-4-enamide —— C20H17ClN4OS
(E,2R,3S)-5-amino-3-(2-chlorophenyl)-2,4-dicyano-5-methylsulfanyl-N-phenylpent-4-enamide
—— (E)-1-(6-methoxynaphthalen-2-yl)-3-(4-piperidin-1-ylphenyl)prop-2-en-1-one —— C25H25NO2
(E)-1-(6-methoxynaphthalen-2-yl)-3-(4-piperidin-1-ylphenyl)prop-2-en-1-one
—— (E)-3-(5-bromo-2-fluorophenyl)-1-[4-(2-oxo-2-pyrrolidin-1-ylethoxy)phenyl]prop-2-en-1-one —— C21H19BrFNO3
(E)-3-(5-bromo-2-fluorophenyl)-1-[4-(2-oxo-2-pyrrolidin-1-ylethoxy)phenyl]prop-2-en-1-one
—— (E)-3-(3,4-dichlorophenyl)-N-[3-[(2-methoxyphenyl)sulfamoyl]-4-methylphenyl]prop-2-enamide —— C23H20Cl2N2O4S
(E)-3-(3,4-dichlorophenyl)-N-[3-[(2-methoxyphenyl)sulfamoyl]-4-methylphenyl]prop-2-enamide
—— (E)-3-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)-1-[2-[(E)-3-phenylprop-2-enyl]sulfanylbenzimidazol-1-yl]prop-2-en-1-one —— C30H29N3O5S2
(E)-3-(4-methoxy-3-morpholin-4-ylsulfonylphenyl)-1-[2-[(E)-3-phenylprop-2-enyl]sulfanylbenzimidazol-1-yl]prop-2-en-1-one
—— (E)-3-(furan-2-yl)-N-[5-pyrrolidin-1-ylsulfonyl-2-(2,2,2-trifluoroethoxy)phenyl]prop-2-enamide —— C19H19F3N2O5S
(E)-3-(furan-2-yl)-N-[5-pyrrolidin-1-ylsulfonyl-2-(2,2,2-trifluoroethoxy)phenyl]prop-2-enamide
—— [(E)-4-amino-3-cyano-2-oxopent-3-enyl] 3-(carbamoylamino)-3-(4-chlorophenyl)propanoate —— C16H17ClN4O4
[(E)-4-amino-3-cyano-2-oxopent-3-enyl] 3-(carbamoylamino)-3-(4-chlorophenyl)propanoate
—— ethyl 2-[5-[(1S)-2-methyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl-(thiophen-2-ylmethyl)amino]propyl]tetrazol-1-yl]acetate —— C26H30N6O5S
ethyl 2-[5-[(1S)-2-methyl-1-[(7-oxo-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinolin-8-yl)methyl-(thiophen-2-ylmethyl)amino]propyl]tetrazol-1-yl]acetate
—— (E)-2-(4-bromophenyl)sulfonyl-3-[3-ethoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]prop-2-enenitrile —— C23H23BrN2O6S
(E)-2-(4-bromophenyl)sulfonyl-3-[3-ethoxy-4-(2-morpholin-4-yl-2-oxoethoxy)phenyl]prop-2-enenitrile
—— (E)-N-[5-(diethylsulfamoyl)-2-propan-2-yloxyphenyl]-3-thiophen-2-ylprop-2-enamide —— C20H26N2O4S2
(E)-N-[5-(diethylsulfamoyl)-2-propan-2-yloxyphenyl]-3-thiophen-2-ylprop-2-enamide
—— (E)-N-(2-chloro-4-methylphenyl)-3-(furan-2-yl)prop-2-enamide —— C14H12ClNO2
(E)-N-(2-chloro-4-methylphenyl)-3-(furan-2-yl)prop-2-enamide
—— (E)-1-[4-(2-fluorophenyl)sulfonylpiperazin-1-yl]-3-(furan-2-yl)prop-2-en-1-one —— C17H17FN2O4S
(E)-1-[4-(2-fluorophenyl)sulfonylpiperazin-1-yl]-3-(furan-2-yl)prop-2-en-1-one
—— (E)-1-(1,3-benzodioxol-5-yl)-3-[4-methoxy-3-(2-methylpropoxy)phenyl]prop-2-en-1-one —— C21H22O5
(E)-1-(1,3-benzodioxol-5-yl)-3-[4-methoxy-3-(2-methylpropoxy)phenyl]prop-2-en-1-one
—— (E)-3-(4-bromothiophen-2-yl)-1-(3-methoxyphenyl)prop-2-en-1-one —— C14H11BrO2S
(E)-3-(4-bromothiophen-2-yl)-1-(3-methoxyphenyl)prop-2-en-1-one
—— (E)-N-(2-chloro-4-methylphenyl)-3-thiophen-2-ylprop-2-enamide —— C14H12ClNOS
(E)-N-(2-chloro-4-methylphenyl)-3-thiophen-2-ylprop-2-enamide