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中文名称 英文名称 CAS号 化学式 结构式图片
—— ethyl (2R)-2-methyl-5-oxo-4-(4-phenyldiazenylanilino)-1-(4-phenyldiazenylphenyl)pyrrole-2-carboxylate —— C32H28N6O3
ethyl (2R)-2-methyl-5-oxo-4-(4-phenyldiazenylanilino)-1-(4-phenyldiazenylphenyl)pyrrole-2-carboxylate
—— ethyl 4-[[(3R)-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]carbamoylamino]benzoate —— C34H30N4O5
ethyl 4-[[(3R)-1-[2-(2-methylphenyl)-2-oxoethyl]-2-oxo-5-phenyl-3H-1,4-benzodiazepin-3-yl]carbamoylamino]benzoate
—— ethyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27N3O4S
ethyl (5S)-3-[2-(cyclopropylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-(cyclopropylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H27N3O4S
ethyl (5R)-3-[2-(cyclopropylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H28FN3O4S
ethyl (5S)-3-[2-[(4-fluorophenyl)methylamino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
ethyl (5S)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
ethyl (5R)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N3O4S
ethyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (2Z,5R)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H23Cl2N3O3S2
ethyl (2Z,5R)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
ethyl (5S)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-methoxyphenyl)-3-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
ethyl (5S)-5-(2-methoxyphenyl)-3-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-fluorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
ethyl (5S)-5-(2-fluorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C31H29N3O4S
ethyl (5R)-3-[2-(benzylamino)-2-oxoethyl]-5-(4-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(3-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N3O4S
ethyl (5R)-5-(3-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E)-3-[3-bromo-4-[(4-bromophenyl)methoxy]phenyl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C22H20Br2N2O3
(E)-3-[3-bromo-4-[(4-bromophenyl)methoxy]phenyl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl (5S)-5-(4-chlorophenyl)-3-[2-(2-methoxyethylamino)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H26ClN3O4S
ethyl (5S)-5-(4-chlorophenyl)-3-[2-(2-methoxyethylamino)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-methoxyphenyl)-3-[2-(2-methylpropylamino)-2-oxoethyl]-7-(trifluoromethyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C23H26F3N3O4S
ethyl (5S)-5-(2-methoxyphenyl)-3-[2-(2-methylpropylamino)-2-oxoethyl]-7-(trifluoromethyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
ethyl (5R)-3-[2-(2-fluoroanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2-methoxyphenyl)-3-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
ethyl (5R)-5-(2-methoxyphenyl)-3-[2-(2-methylpropylamino)-2-oxoethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2,4-dimethylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H33N3O4S
ethyl (5S)-5-(2,4-dimethylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
ethyl (5R)-3-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H29N3O4S
ethyl (5R)-3-[2-(3,4-dimethylanilino)-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H31N3O4S
ethyl (5S)-5-(2-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(4-methylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N3O4S
ethyl (5R)-5-(4-methylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (1S,4S,5S)-5-cyano-2-(4-methylphenyl)sulfonyl-2-azabicyclo[2.2.1]heptane-5-carboxylate —— C17H20N2O4S
ethyl (1S,4S,5S)-5-cyano-2-(4-methylphenyl)sulfonyl-2-azabicyclo[2.2.1]heptane-5-carboxylate
—— ethyl (2Z,5S)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H23Cl2N3O3S2
ethyl (2Z,5S)-2-[[1-[(2,4-dichlorophenyl)methyl]indol-3-yl]methylidene]-7-methyl-3-oxo-5-thiophen-2-yl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2-fluorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C25H24FN3O4S
ethyl (5R)-5-(2-fluorophenyl)-3-[2-(4-methoxyanilino)-2-oxoethyl]-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (1S,4S,5R)-5-cyano-2-(4-methylphenyl)sulfonyl-2-azabicyclo[2.2.1]heptane-5-carboxylate —— C17H20N2O4S
ethyl (1S,4S,5R)-5-cyano-2-(4-methylphenyl)sulfonyl-2-azabicyclo[2.2.1]heptane-5-carboxylate
—— ethyl (5R)-5-(2-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C32H31N3O4S
ethyl (5R)-5-(2-methoxyphenyl)-3-[2-oxo-2-[[(1R)-1-phenylethyl]amino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H28F3N3O4S
ethyl (5R)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-7-methyl-5-(2-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C24H29N3O4S
ethyl (5S)-7-methyl-5-(2-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-chlorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28ClN3O4S
ethyl (5S)-5-(2-chlorophenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(2-chlorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H28ClN3O4S
ethyl (5S)-5-(2-chlorophenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N3O4S
ethyl (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[(1R)-1,2,3,4-tetrahydronaphthalen-1-yl]amino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(4-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H31N3O4S
ethyl (5R)-5-(4-methylphenyl)-3-[2-oxo-2-[[(2R)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
ethyl (5S)-3-[2-[[(2R)-butan-2-yl]amino]-2-oxoethyl]-5-(4-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(2,4-dimethylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H33N3O4S
ethyl (5R)-5-(2,4-dimethylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C28H31N3O4S
ethyl (5R)-3-[2-[[(2S)-butan-2-yl]amino]-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methylanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
ethyl (5R)-5-(3-methoxyphenyl)-7-methyl-3-[2-(4-methylanilino)-2-oxoethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-(ethylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
ethyl (5S)-3-[2-(ethylamino)-2-oxoethyl]-5-(2-methoxyphenyl)-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C29H28F3N3O4S
ethyl (5S)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3aS,6aS)-5-(2-nitrophenyl)-4,6-dioxo-1-phenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C20H16N4O6
ethyl (3aS,6aS)-5-(2-nitrophenyl)-4,6-dioxo-1-phenyl-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— ethyl (5S)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H27N3O4S
ethyl (5S)-3-[2-(3-methoxyanilino)-2-oxoethyl]-7-methyl-5-(2-methylphenyl)-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (3aR,6aR)-5-(2-chlorophenyl)-1-(4-nitrophenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate —— C20H15ClN4O6
ethyl (3aR,6aR)-5-(2-chlorophenyl)-1-(4-nitrophenyl)-4,6-dioxo-3a,6a-dihydropyrrolo[3,4-c]pyrazole-3-carboxylate
—— (E)-3-[3-bromo-4-[(4-bromophenyl)methoxy]phenyl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C22H20Br2N2O3
(E)-3-[3-bromo-4-[(4-bromophenyl)methoxy]phenyl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl (5S)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C26H31N3O4S
ethyl (5S)-3-[2-[[(1R,2R,4R)-2-bicyclo[2.2.1]heptanyl]amino]-2-oxoethyl]-5-(3-methoxyphenyl)-7-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— (E,2R)-2-[2-oxo-2-(4-phenoxyanilino)ethyl]tetradec-4-enoic acid —— C28H37NO4
(E,2R)-2-[2-oxo-2-(4-phenoxyanilino)ethyl]tetradec-4-enoic acid
—— ethyl (5S)-5-(2,4-dimethylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C30H33N3O4S
ethyl (5S)-5-(2,4-dimethylphenyl)-3-[2-oxo-2-[[(2S)-oxolan-2-yl]methylamino]ethyl]-7-phenyl-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5R)-3-[2-(2-methoxyethylamino)-2-oxoethyl]-7-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H26F3N3O4S
ethyl (5R)-3-[2-(2-methoxyethylamino)-2-oxoethyl]-7-phenyl-5-[4-(trifluoromethyl)phenyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate
—— ethyl (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[3-(trifluoromethyl)phenyl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate —— C27H26F3N3O4S
ethyl (5S)-5-(3-methoxyphenyl)-7-methyl-3-[2-oxo-2-[[3-(trifluoromethyl)phenyl]methylamino]ethyl]-5H-[1,3]thiazolo[3,2-a]pyrimidine-6-carboxylate