| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | 20-0-Val-gimatecan | 870136-98-4 | C30H34N4O6 |
| —— | (E)-7-tert-butoxyiminomethyl-20-O-hemisuccinyl-camptothecin | 630096-28-5 | C29H29N3O8 |
| —— | (3S)-4-[[(2S)-1-[[(19S)-19-ethyl-10-[(E)-(2-methylpropan-2-yl)oxyiminomethyl]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-19-yl]oxy]-3-methyl-1-oxobutan-2-yl]amino]-3-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxobutanoic acid | 870136-99-5 | C39H47N5O11 |
| —— | (9S)-9-ethyl-9-hydroxy-1-(1-methylethyl)-1H,12H-pyrano[3",4":6',7']indolizino-[1',2':6,5]pyrido[4,3,2-de]quinazoline-10,13(9H,15H)-dione | 538374-71-9 | C24H22N4O4 |
| —— | (E)-7-tert-butoxyiminomethyl-20-O-[2-(dimethylamino)ethylamino]succinyl-camptothecin hydrochloride | 630390-98-6 | C33H39N5O7*ClH |
| —— | (E)-7-tert-butoxyiminomethyl-20-O-(tert-butylglycyl)succinyl-camptothecin | 630391-01-4 | C35H40N4O9 |
| —— | (S)-4-Ethyl-4-hydroxy-10-((E)-2-trimethylsilanyl-vinyl)-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione | 189312-00-3 | C25H26N2O4Si |
| —— | (E)-7-tert-butoxyiminomethyl-20-O-(4-trimethylammonium)-butanoyl-camptothecin bromide | 630390-97-5 | Br*C32H39N4O6 |
| —— | (S)-11-((E)-(tert-butoxyimino)methyl)-4-ethyl-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-4-yl (tert-butoxycarbonyl)-L-valinate | 870137-00-1 | C35H42N4O8 |
| —— | Dxd | 1599440-33-1 | C26H24FN3O6 |
| —— | 9-nitrocamptothecin-20-chloroacetate | 623114-14-7 | C22H16ClN3O7 |
| —— | 1185274-92-3 | C2HF3O2*C26H25N3O5 | |
| —— | 10-OTBDMS 20-OTES topotecan | 1004511-36-7 | C35H51N3O5Si2 |
| —— | Butanedioic acid, 1-[(3R,5aS,6R,8aS,9R,10S,12R,12aR)-decahydro-3,6,9-trimethyl-3,12-epoxy-12H-pyrano[4,3-j]-1,2-benzodioxepin-10-yl] 4-[(4S)-4-ethyl-3,4,12,14-tetrahydro-3,14-dioxo-1H-pyrano[3a(2),4a(2):6,7]indolizino[1,2-b]quinolin-4-yl] ester | 1639110-38-5 | C39H42N2O11 |
| —— | 20-OTES topotecan | 1004511-35-6 | C29H37N3O5Si |
| —— | acetic acid (4S)-{[2-(4-ethyl-4-hydroxy-3,13-dioxo-3,4,12,13-tetrahydro-1H-2-oxa-6,12a-diaza-dibenzo[b,h]fluoren-11-yl)-ethyl]-dimethylsilanyl}-methyl ester | 1142936-56-8 | C27H30N2O6Si |
| —— | 882214-67-7 | C31H28FN3O7 | |
| —— | 4-(((S)-1-((2-(((S)-4-ethyl-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-4-yl)oxy)-2-oxoethyl)amino)-1-oxo-3-phenylpropan-2-yl)amino)-4-oxobutanoic acid | 1004317-72-9 | C35H32N4O9 |
| —— | O-{2-[(1,2,3-triazolyl)-4-[4-(N-maleimidomethyl)cyclohexane-1-carboxamidomethyl]]ethyl}-O'-[(N-diglycolyl-2-aminoethyl)-Phe-Lys-PAB-OCO-20-O-SN-38]heptaethyleneglycol trifluoroacetate | 1083198-45-1 | C2HF3O2*C82H106N12O23 |
| —— | (4S)-10-bromo-4-ethyl-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1 ,2-b]quinolin-4-yl N-[6-(2,5-dioxo-2,5-dihydro-1H-pyrrol-1-yl)hexanoyl]-L-phenylalanyl-L-leucylglycinate | 1609075-08-2 | C47H49BrN6O10 |
| —— | 10-(3-bromo-propoxy)-(20S)-camptothecin | 744221-15-6 | C23H21BrN2O5 |
| —— | camptothecin-10-O-tert-butoxycarbonyl-20-O-[(S)-(-)-2-hydroxypropionate] | 1243484-01-6 | C28H28N2O9 |
| —— | 9-<(cyclopropylamino)methyl>-10-hydroxy-(20S)-camptothecin acetate salt | 130064-59-4 | C2H4O2*C24H23N3O5 |
| —— | (19S)-19-ethyl-19-hydroxy-7-[(2-sulfanylidene-1,3,2lambda5-benzodioxaphosphol-2-yl)oxy]-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaene-14,18-dione | 1381808-62-3 | C26H19N2O7PS |
| —— | (2R,3R,4S,5R)-2-(acetoxymethyl)-6-(((((S)-4-ethyl-4-hydroxy-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl)oxy)(hydroxy)phosphoryl)oxy)tetrahydro-2H-pyran-3,4,5-triyl triacetate | 1011298-89-7 | C34H35N2O17P |
| —— | tert-butyl 3-[2-[2-[2-[6-[[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaen-7-yl]oxycarbonylamino]hexylcarbamoyloxy]ethoxy]ethoxy]ethoxy]propanoate | 945867-59-4 | C41H54N4O13 |
| —— | 4-methoxy-benzenesulfonic acid 4-ethyl-4-hydroxy-10-nitro-3,13-dioxo-3,4,12,13-tetrahydro-1H-2-oxa-6,12a-diaza-dibenzo[b,h]fluoren-9-yl ester | 172917-97-4 | C27H21N3O10S |
| —— | O-(2,4-dichlorophenyl) O-ethyl O-((S)-4-ethyl-4-hydroxy-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl) phosphorothioate | 1381809-70-6 | C28H23Cl2N2O7PS |
| —— | 10-hydroxy-9-<(N-methylpiperazinyl)methyl>-(20S)-camptothecin acetate salt | 130064-58-3 | 3C2H4O2*2C26H28N4O5 |
| —— | 10-methoxycamptothecin-20-O-2-(tert-butoxycarbonylamino)acetic acid ester | 1394865-81-6 | C28H29N3O8 |
| —— | (19S)-19-ethyl-19-hydroxy-7-(methoxymethoxy)-8-prop-2-enyl-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione | 1256544-06-5 | C25H24N2O6 |
| —— | N-(6-(2-(((S)-4-ethyl-4-hydroxy-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl)oxy)acetamido)hexyl)-5-((3aS,4S,6aR)-2-oxohexahydro-1H-thieno[3,4-d]imidazol-4-yl)pentanamide | 960230-28-8 | C38H46N6O8S |
| —— | 9-<<<2-(N,N-dimethyloamino)ethyl>thio>methyl>-10-hydroxy-(20S)-camptothecin hydrochloride | 123949-05-3 | C25H27N3O5S*ClH |
| —— | (4S)-4-ethyl-4-hydroxy-9-((5-methyl-2-sulfidobenzo[d][1,3,2]dioxaphosphol-2-yl)oxy)-1,12-dihydro-14H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H)-dione | 1381808-82-7 | C27H21N2O7PS |
| —— | (4S)-9-((5-chloro-2-sulfidobenzo[d][1,3,2]dioxaphosphol-2-yl)oxy)-4-ethyl-4-hydroxy-1,12-dihydro-14H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H)-dione | 1381809-13-7 | C26H18ClN2O7PS |
| —— | 10-hydroxy-9-<(trimethylammonio)methyl>-(20S)-camptothecin methanosulfonate | 123948-98-1 | CH3O3S*C24H26N3O5 |
| —— | (19S)-19-ethyl-7,19-dihydroxy-6-prop-2-enyl-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaene-14,18-dione | 1623024-40-7 | C23H20N2O5 |
| —— | (S)-2,5-dioxopyrrolidin-1-yl (4-ethyl-4-hydroxy-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl) glutarate | 1353778-73-0 | C29H25N3O10 |
| —— | (S)-5-((4-ethyl-4-hydroxy-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl)oxy)-5-oxopentanoic acid | 1353778-70-7 | C25H22N2O8 |
| —— | 9-iodine-10-methoxymethoxycamptothecin | 1256544-05-4 | C22H19IN2O6 |
| —— | camptothecin-10-O-tert-butoxycarbonyl-20-O-[(R)-(+)-2-hydroxypropionate] | 1243484-02-7 | C28H28N2O9 |
| —— | O-ethyl O-((S)-4-ethyl-4-hydroxy-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl) O-(4-nitrophenyl) phosphorothioate | 1381809-60-4 | C28H24N3O9PS |
| —— | 10-methoxycamptothecin-20-O-2-(tert-butoxycarbonylamino)-3-phenylpropanoic acid ester | 1394865-84-9 | C35H35N3O8 |
| —— | 10-hydroxy-9-<<(2-hydroxyethyl)amino>methyl>-(20S)-camptothecin acetate salt | 123948-96-9 | C2H4O2*C23H23N3O6 |
| —— | tert-butyl 3-[2-[2-[2-[2-[6-[[(19S)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaen-7-yl]oxycarbonylamino]hexylcarbamoyloxy]ethoxy]ethoxy]ethoxy]ethoxy]propanoate | 945867-60-7 | C43H58N4O14 |
| —— | Trifluoro-methanesulfonic acid (S)-4-ethyl-4-hydroxy-10-nitro-3,13-dioxo-3,4,12,13-tetrahydro-1H-2-oxa-6,12a-diaza-dibenzo[b,h]fluoren-9-yl ester | 164159-92-6 | C21H14F3N3O9S |
| —— | (20S)-10-acetoxy-20-O-acetyl-7,12-bis(tert-butyldimethylsilyl)camptothecin | 521061-98-3 | C36H48N2O7Si2 |
| —— | 20(S)-OTES-10-OTBDMS-camptothecin | 1004265-04-6 | C32H44N2O5Si2 |
| —— | 10-[4-(2,3,4-tri-O-acetyl-6-O-methyl-β-D-glucuronyloxy)-3-nitrobenzyloxy]camptothecin | 1018932-85-8 | C40H37N3O17 |
| —— | (S)-4-ethyl-4-hydroxy-10-nitro-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-9-yl benzenesulfonate | 172917-94-1 | C26H19N3O9S |