| 中文名称 | 英文名称 | CAS号 | 化学式 |
|---|---|---|---|
| —— | (10S,23S)-10-ethyl-18-fluoro-10-hydroxy-19,23-dimethyl-8-oxa-4,15-diazahexacyclo[14.7.1.02,14.04,13.06,11.020,24]tetracosa-1,6(11),12,14,16,18,20(24)-heptaene-5,9-dione | —— | C50H46F2N4O8 |
| —— | [(19S)-19-ethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaen-19-yl] (2S)-2-[(E)-(4-methyl-2,5,7-trinitrofluoren-9-ylidene)amino]oxypropanoate;[(19S)-19-ethyl-7-[(2-methylpropan-2-yl)oxycarbonyloxy]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaen-19-yl] 2-[(E)-(4-methyl-2,5,7-trinitrofluoren-9-ylidene)amino]oxyacetate | —— | C78H58N12O28 |
| —— | (4-methylphenyl)methyl N-[(10S,23S)-10-ethyl-18-fluoro-10-hydroxy-19-methyl-5,9-dioxo-8-oxa-4,15-diazahexacyclo[14.7.1.02,14.04,13.06,11.020,24]tetracosa-1,6(11),12,14,16,18,20(24)-heptaen-23-yl]carbamate | —— | C33H30FN3O6 |
| —— | ethane;[(19S)-19-ethyl-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-19-yl] 5-methyliminopentanoate | —— | C28H31N3O5 |
| —— | [(19S)-19-ethyl-19-hydroxy-8-[[methyl(methylamino)amino]methyl]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-[[4-(docosa-4,7,10,13,16,19-hexaenoylamino)phenyl]methyl]piperazine-1-carboxylate | —— | C57H69N7O7 |
| —— | (10S)-10-ethyl-10-hydroxy-23-(3-phenylpropyl)-8-oxa-4,15,21-triazahexacyclo[14.7.1.02,14.04,13.06,11.020,24]tetracosa-1(24),2(14),6(11),12,16,18,20,22-octaene-5,9-dione | —— | C31H27N3O4 |
| —— | 4-[[1-[[(19S)-19-ethyl-10-[(2-methylpropan-2-yl)oxyiminomethyl]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-19-yl]oxy]-3-methyl-1-oxobutan-2-yl]amino]-4-oxobutanoic acid | —— | C34H38N4O9 |
| —— | (19S)-10-(butylamino)-19-ethyl-19-hydroxy-8-nitro-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione | —— | C24H24N4O6 |
| —— | (19S)-10-(4-chlorophenyl)-19-ethyl-19-hydroxy-7-methanimidoyl-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione | —— | C27H20ClN3O4 |
| —— | (19S)-8-[(dimethylamino)methyl]-19-ethyl-7,19-dihydroxy-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione;(19S)-19-ethyl-7,19-dihydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-8-carbaldehyde | —— | C45H41N5O10 |
| —— | (19S)-8,10-diamino-19-ethyl-19-hydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaene-14,18-dione | —— | C20H18N4O4 |
| —— | dimethylphosphinic acid;(19S)-19-(dimethylphosphoryloxymethoxy)-19-ethyl-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaene-14,18-dione | —— | C25H30N2O8P2 |
| —— | [(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 6-[[4-[[3-[bis(phosphanyl)methylsulfanyl]-2,5-dihydroxypyrrol-1-yl]methyl]cyclohexanecarbonyl]amino]hexanoate | —— | C41H50N4O9P2S |
| —— | N-[[1-[2-[2-[2-[2-[2-[2-[2-[2-[2-[[2-[2-[[(2S)-1-[[(2S)-6-amino-1-(4-ethylanilino)-1-oxohexan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-2-oxoethoxy]acetyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethyl]triazol-4-yl]methyl]-4-[(3-methyl-2,5-dioxopyrrolidin-1-yl)methyl]cyclohexane-1-carboxamide;[(19S)-10,19-diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] methyl carbonate | —— | C85H116N12O23 |
| —— | (R)-Topotecan | —— | C23H23N3O5 |
| —— | (2R)-2-hydroxy-2-[8-(hydroxymethyl)-9-oxo-11H-indolizino[1,2-b]quinolin-7-yl]butanoic acid | —— | C20H18N2O5 |
| —— | 2-amino-N-[(19R)-19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-8-yl]acetamide | —— | C22H20N4O5 |
| —— | (19S)-10-[2-(2,4-difluorophenyl)ethoxyiminomethyl]-19-ethyl-19-hydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaene-14,18-dione | —— | C29H23F2N3O5 |
| —— | (10,19-Diethyl-19-methoxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl) 5-piperidin-1-ylcyclononane-1-carboxylate | —— | C38H47N3O6 |
| —— | [(19S)-8-[(dimethylamino)methyl]-19-ethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] (2S)-2-[(E)-(4-methyl-2,5,7-trinitrofluoren-9-ylidene)amino]oxypropanoate | —— | C40H33N7O13 |
| —— | (10,19-diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl) [4-[2-[3-(3-methyl-2,5-dioxopyrrolidin-1-yl)propanoylamino]ethylperoxyperoxyperoxyperoxyperoxyperoxymethyl]phenyl]methyl carbonate;ethene | —— | C65H90N4O22 |
| —— | (10,19-Diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl) [2-[[2-[2-[[4-[1-[4-[[[4-[(3-ethyl-2,5-dihydroxypyrrol-1-yl)methyl]cyclohexanecarbonyl]amino]methyl]triazol-1-yl]pentan-3-yloxy]-2-methylbutan-2-yl]amino]-2-oxoethoxy]acetyl]amino]-3-methylbutyl] carbonate | —— | C59H79N9O14 |
| —— | [(19S)-19-ethyl-7-[(2-methylpropan-2-yl)oxycarbonyloxy]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaen-19-yl] (2S)-2-[(E)-(4-methyl-2,5,7-trinitrofluoren-9-ylidene)amino]oxypropanoate | —— | C42H34N6O15 |
| —— | (19S)-10,19-diethyl-19-hydroxy-7-methyl-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione;2-[(2-methylpropan-2-yl)oxycarbonylamino]acetic acid | —— | C30H35N3O8 |
| —— | 3-[(19S)-19-ethyl-7,19-dihydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-10-yl]prop-2-enal | —— | C23H18N2O6 |
| —— | [(19S)-19-ethyl-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-19-yl] 3-[2,5-dihydroxy-3-[[phosphanyl(phosphanylidene)-lambda4-sulfanyl]methyl]pyrrol-1-yl]propanoate | —— | C28H27N3O7P2S |
| —— | disodium;(19S)-19-ethyl-19-hydroxy-10-(2-trimethylsilylethyl)-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaene-14,18-dione;2-(2-sulfonatoethyldisulfanyl)ethanesulfonate | —— | C29H36N2Na2O10S4Si |
| —— | [(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-[6-(2,5-dioxopyrrol-1-yl)hexanoylamino]benzoate | —— | C39H36N4O9 |
| —— | [(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-[[[4-[(2,5-dioxopyrrol-1-yl)methyl]cyclohexanecarbonyl]amino]methyl]cyclohexane-1-carboxylate | —— | C42H46N4O9 |
| —— | (10,19-Diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl) 4-[3-[2-[2-[2-[2-[[4-[(2,5-dioxopyrrol-1-yl)methyl]cyclohexanecarbonyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carboxylate | —— | C50H62N6O14 |
| —— | [(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-[3-[2-[2-[2-[2-[[4-[(2,5-dioxopyrrol-1-yl)methyl]cyclohexanecarbonyl]amino]ethoxy]ethoxy]ethoxy]ethoxy]propanoyl]piperazine-1-carboxylate | —— | C50H62N6O14 |
| —— | [(19S)-10,19-diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] 2-[[4-[[(2S)-6-amino-2-[[(2S)-2-[[2-[2-[2-[2-[2-[4-[[[4-[(2,5-dioxopyrrol-1-yl)methyl]cyclohexanecarbonyl]amino]methyl]triazol-1-yl]ethoxy]ethoxy]ethylamino]-2-oxoethoxy]acetyl]amino]-3-phenylpropanoyl]amino]hexanoyl]amino]phenyl]methoxycarbonylamino]acetate | —— | C72H85N13O18 |
| —— | [(19S)-10,19-diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] 2-(butanoylamino)acetate | —— | C28H29N3O7 |
| —— | [(19S)-10,19-diethyl-7-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] 2-[[4-[[(2S)-6-amino-2-[[(2S)-2-[[2-[2-[2-[2-(2-azidoethoxy)ethoxy]ethylamino]-2-oxoethoxy]acetyl]amino]-3-phenylpropanoyl]amino]hexanoyl]amino]phenyl]methoxycarbonylamino]acetate | —— | C57H67N11O15 |
| —— | (2R)-2-[[4-[[(19S)-19-[4-[[(1R)-1-carboxy-2-phenylethyl]amino]-4-oxobutanoyl]oxy-10,19-diethyl-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl]oxy]-4-oxobutanoyl]amino]-3-phenylpropanoic acid | —— | C48H46N4O13 |
| —— | [(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] N-ethyl-N-methylcarbamate | —— | C26H27N3O6 |
| —— | 6,7-dichloro-3,5-dihydro-1H-imidazo[2,1-b]quinazolin-2-one;[(19S)-10,19-diethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-piperidin-1-ylpiperidine-1-carboxylate;4-[(2S)-2-(3,5-dioxopiperazin-1-yl)propyl]piperazine-2,6-dione | —— | C54H61Cl2N11O11 |
| —— | (19S)-19-ethyl-19-hydroxy-8-nitroso-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione | —— | C20H15N3O5 |
| —— | [(19S)-10,19-diethyl-19-[2-(2-formamidoethoxy)ethoxycarbonyloxy]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl] 4-piperidin-1-ylpiperidine-1-carboxylate | —— | C39H47N5O10 |
| —— | [(2R,3S,4R,5R)-5-(2,6-diaminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methyl [(19S)-19-ethyl-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4,6,8,10,15(20)-heptaen-19-yl] hydrogen phosphate | —— | C30H29N8O10P |
| —— | (19S)-19-aminooxy-8-bromo-19-ethyl-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione | —— | C20H16BrN3O4 |
| —— | L-valyl-N-[4-({[(4-{[(4S)-10-bromo-4-ethyl-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-4-yl]oxy}-2,2-dimethyl-4-oxobutyl)carbamoyl]oxy}methyl)phenyl]-N<sup>5</sup>-carbamoyl-L-onithinamide | 1609075-25-3 | C45H53BrN8O10 |
| —— | L-valyl-N-(4-{[({[1-(2-{[(4S)-10-bromo-4-ethyl-3,14-dioxo-3,4,12,14-tetrahydro-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinolin-4-yl]oxy}2-oxoethyl)cyclohexyl]methyl}carbamoyl)oxy]methyl}phenyl)-N<sup>5</sup>-carbamoyl-L-ornithinamide | 1609075-26-4 | C48H57BrN8O10 |
| —— | [(19S)-8-bromo-19-ethyl-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl] 4-[[4-[[(2S)-5-(carbamoylamino)-2-[[(2S)-3-methyl-2-[(2-methylpropan-2-yl)oxycarbonylamino]butanoyl]amino]pentanoyl]amino]phenyl]methoxycarbonylamino]-3,3-dimethylbutanoate | —— | C50H61BrN8O12 |
| —— | (19S)-8-[(dimethylamino)methyl]-19-ethyl-7,19-dihydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaene-14,18-dione;hydroxyurea | —— | C24H27N5O7 |
| —— | tert-butyl 2-[[6-amino-2-[[4-[[(19S)-10,19-diethyl-7-[(2-methylpropan-2-yl)oxycarbonyloxy]-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl]oxy]-4-oxobutanoyl]amino]hexanoyl]amino]octadecanoate | —— | C59H87N5O12 |
| —— | tert-butyl (2S)-5-[[2-[[(19S)-10,19-diethyl-7-methyl-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-19-yl]oxy]-2-oxoethyl]amino]-2-(hexadecanoylamino)-5-oxopentanoate | —— | C50H70N4O9 |
| —— | tert-butyl 2-[[4-[[(19S)-10,19-diethyl-19-[4-[[1-[(2-methylpropan-2-yl)oxy]-1-oxohexan-2-yl]amino]-4-oxobutanoyl]oxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-7-yl]oxy]-4-oxobutanoyl]amino]hexanoate | —— | C50H66N4O13 |
| —— | Camptothecin phosphate | —— | C20H17N2O7P |
| —— | 2-amino-N-(19-ethyl-19-hydroxy-14,18-dioxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2,4(9),5,7,10,15(20)-heptaen-8-yl)acetamide;chloride | —— | C22H20ClN4O5- |