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血液系统用药

造血系统包括血液、骨髓、脾脏、淋巴结以及散布于全身各处的淋巴组织和单核-巨噬细胞组织。血液病,即所谓的造血系统疾病,主要表现为周围血细胞成分及功能的变化,以及出凝血机制障碍。尽管目前临床用于治疗血液病的药物种类较多,但大多数缺乏针对性,其疗效与实际需求仍存在一定差距。

中文名称 英文名称 CAS号 化学式 结构式图片
双香豆乙酯 ethyl biscoumacetate 548-00-5 C22H16O8
双香豆乙酯
卡巴克络 Carbazochrome 69-81-8 C10H12N4O3
卡巴克络
华法林钠 warfarin sodium 129-06-6 C19H16O4*Na
华法林钠
华法林 warfarin 81-81-2 C19H16O4
华法林
千金藤素 cepharanthine 481-49-2 C37H38N2O6
千金藤素
匹卡米隆 N-nicotinoyl-gamma-aminobutyric acid 34562-97-5 C10H12N2O3
匹卡米隆
利可君 leucogen 1950-36-3 C14H17NO4S
利可君
利伐沙班 Rivaroxaban 366789-02-8 C19H18ClN3O5S
利伐沙班
凝血酸 4-aminomethyl-cyclohexanecarboxylic acid 701-54-2 C8H15NO2
凝血酸
依度沙班 edoxaban 480449-70-5 C24H30ClN7O4S
依度沙班
伊波格雷 isbogrel 89667-40-3 C18H19NO2
伊波格雷
二甲基丙烯酸氧化锆 2-Methylprop-2-enoate;oxozirconium(2+) 97171-79-4 C8H10O5Zr
二甲基丙烯酸氧化锆
二(D-谷氨酸基-kappaO1)铁水合物(1:1) Ferrous gluconate hydrate 299-29-6 C12H26FeO15
二(D-谷氨酸基-kappaO1)铁水合物(1:1)
三甲硅基丙炔醇 3-trimethylsilyl-2-propyn-1-ol 5272-36-6 C6H12OSi
三甲硅基丙炔醇
三氯化铁 iron(III) chloride 7705-08-0 Cl3Fe
三氯化铁
丁二酸亚铁 Iron(II)succinate 10030-90-7 C4H6FeO4
丁二酸亚铁
6-氨基己酸 6-aminohexanoic acid 60-32-2 C6H13NO2
6-氨基己酸
4-氨甲基苯甲酸 p-aminomethylbenzoic acid 56-91-7 C8H9NO2
4-氨甲基苯甲酸
4-[(4-甲基哌嗪-1-基)甲基]苯甲酸二盐酸盐 4-[(4-methylpiperazin-1-yl)methyl]benzoic Acid Dihydrochloride 106261-49-8 C13H20Cl2N2O2
4-[(4-甲基哌嗪-1-基)甲基]苯甲酸二盐酸盐
4-[(4-甲基-1-哌嗪基)甲基]-N-[6-甲基-5-[[4-(3-吡啶基)-2-嘧啶基]氨基]-3-吡啶基]-3-(三氟甲基)苯甲酰胺 flumatinib 895519-90-1 C29H29F3N8O
4-[(4-甲基-1-哌嗪基)甲基]-N-[6-甲基-5-[[4-(3-吡啶基)-2-嘧啶基]氨基]-3-吡啶基]-3-(三氟甲基)苯甲酰胺
2-甲氧基-5-(1-丙烯基)苯酚 2-methoxy-5-(1-propenyl)phenol 501-20-2 C10H12O2
2-甲氧基-5-(1-丙烯基)苯酚
2-氧代-4-苯基丁酸乙酯 2-oxo-4-phenylbutanoic acid ethyl ester 64920-29-2 C12H14O3
2-氧代-4-苯基丁酸乙酯
1-环丙基-2-(2-氟苯基)乙酮 1-cyclopropyl-2-(2-fluorophenyl)ethanone 150322-73-9 C11H11FO
1-环丙基-2-(2-氟苯基)乙酮
1-[3-氯-5-[[[4-(4-氯-2-噻吩基)-5-(4-环己基-1-哌嗪基)-2-噻唑基]氨基]羰基]-2-吡啶基]-4-哌啶羧酸 avatrombopag 570406-98-3 C29H34Cl2N6O3S2
1-[3-氯-5-[[[4-(4-氯-2-噻吩基)-5-(4-环己基-1-哌嗪基)-2-噻唑基]氨基]羰基]-2-吡啶基]-4-哌啶羧酸
—— ferroheme b 14875-96-8 C34H32N4O4*Fe
ferroheme b
—— Injectafer 9007-72-1 C24H44FeO25-
Injectafer
—— heme b 927179-10-0 C34H32FeN4O4
heme b
—— (+/-)-2-(dimethylamino)-1-<<o-(m-methoxyphenethyl)phenoxy>methyl>ethyl hydrogen succinate 125926-17-2 C4H6O4*C20H27NO2
(+/-)-2-(dimethylamino)-1-<<o-(m-methoxyphenethyl)phenoxy>methyl>ethyl hydrogen succinate
—— Ferrous Gluconate 6047-12-7 C12H22FeO14
Ferrous Gluconate
—— Iron gluconate 299-29-6 C12H24FeO14
Iron gluconate
—— Zirconium methacrylate 84057-81-8 C16H20O8Zr
Zirconium methacrylate
—— Naftazone 15687-37-3 C11H9N3O2
Naftazone
—— Ferrous lactate 85993-25-5 C6H10FeO6
Ferrous lactate
—— Unii-mul7onl3Z6 1301-70-8 C8H18Fe2O12P2
Unii-mul7onl3Z6
—— Ferroheme 14875-96-8 C34H32FeN4O4
Ferroheme
—— argatroban 121785-71-5 C23H36N6O5S
argatroban
—— ferrous succinate 10030-90-7 C4H4O4*Fe
ferrous succinate
—— 1-Methyl-17β-acetoxy-Δ<sup>1</sup>-5α-androsten 434-05-9 C22H32O3
1-Methyl-17β-acetoxy-Δ<sup>1</sup>-5α-androsten
—— Argatroban, 21R- 1379603-43-6 C23H38N6O6S
Argatroban, 21R-
—— 2-methylprop-2-enoic acid;zirconium 84057-81-8 C16H24O8Zr
2-methylprop-2-enoic acid;zirconium
—— 6132-04-3 C6H10NaO8
—— Iron,7,12,17-tetramethyl-8,13-divinyl-2,18-porphinedipropionato(2-)]- 14875-96-8 C34H32FeN4O4
Iron,7,12,17-tetramethyl-8,13-divinyl-2,18-porphinedipropionato(2-)]-
—— Iron;2,3,4,5,6-pentahydroxyhexanoic acid 299-29-6 C12H24FeO14
Iron;2,3,4,5,6-pentahydroxyhexanoic acid
—— (2R,4R)-1-[5-(diaminomethylideneamino)-2-[(3-methyl-1,2,3,4-tetrahydroquinolin-8-yl)sulfonylamino]pentanoyl]-4-methylpiperidine-2-carboxylic acid 74863-84-6 C23H36N6O5S
(2R,4R)-1-[5-(diaminomethylideneamino)-2-[(3-methyl-1,2,3,4-tetrahydroquinolin-8-yl)sulfonylamino]pentanoyl]-4-methylpiperidine-2-carboxylic acid
—— Berbamine (dihydrochloride) 6078-17-7 C37H42Cl2N2O6
Berbamine (dihydrochloride)
—— ozagrel sodium 82571-53-7 C13H11N2O2*Na
ozagrel sodium
—— 4-((4-methylpiperazin-1-yl)methyl)benzoic acid dihydrochloride 106261-49-8 C13H18N2O2*2ClH
4-((4-methylpiperazin-1-yl)methyl)benzoic acid dihydrochloride
—— Adrenochrom-semicarbazon 69-81-8 C10H12N4O3
Adrenochrom-semicarbazon
—— warfarin 129-06-6 C19H15O4*Na
warfarin
—— iron(II) fumarate 141-01-5 C4H2O4*Fe
iron(II) fumarate