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—— ethyl (6S)-3-[2-(diethylamino)ethyl]-4-methyl-6-(3-nitrophenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C20H28N4O4S
ethyl (6S)-3-[2-(diethylamino)ethyl]-4-methyl-6-(3-nitrophenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(2-ethoxyphenyl)prop-2-enamide —— C17H13ClN4O2S
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(2-ethoxyphenyl)prop-2-enamide
—— (E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C22H23ClN6
(E)-3-[5-chloro-3-methyl-1-[(4-methylphenyl)methyl]pyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— ethyl (6S)-6-(2,4-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H25F2N3O2S
ethyl (6S)-6-(2,4-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C18H21ClN6O2S
(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— ethyl 2-[[2-[4-(dimethylamino)pyridin-1-ium-1-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate —— C19H24N3O3S+
ethyl 2-[[2-[4-(dimethylamino)pyridin-1-ium-1-yl]acetyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxylate
—— ethyl (6S)-3,4-dimethyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22N2O3S
ethyl (6S)-3,4-dimethyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N2O4S
ethyl (6S)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 2-[[(2S)-2-[4-(dimethylamino)pyridin-1-ium-1-yl]propanoyl]amino]-5-phenylthiophene-3-carboxylate —— C23H26N3O3S+
ethyl 2-[[(2S)-2-[4-(dimethylamino)pyridin-1-ium-1-yl]propanoyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-N-(4-fluoro-2-methylphenyl)-3-(4-prop-2-enoxyphenyl)prop-2-enamide —— C19H18FNO2
(E)-N-(4-fluoro-2-methylphenyl)-3-(4-prop-2-enoxyphenyl)prop-2-enamide
—— ethyl (6R)-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O4S
ethyl (6R)-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-3,4-dimethyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 4-[2-[4-(dimethylamino)pyridin-1-ium-1-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate —— C18H24N3O3+
ethyl 4-[2-[4-(dimethylamino)pyridin-1-ium-1-yl]acetyl]-2,5-dimethyl-1H-pyrrole-3-carboxylate
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-(3-ethoxypropyl)prop-2-enamide —— C15H16F2N2O2
(E)-2-cyano-3-(3,4-difluorophenyl)-N-(3-ethoxypropyl)prop-2-enamide
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-(2,4,6-trimethylphenyl)prop-2-enamide —— C19H16F2N2O
(E)-2-cyano-3-(3,4-difluorophenyl)-N-(2,4,6-trimethylphenyl)prop-2-enamide
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-(2-ethoxyphenyl)prop-2-enamide —— C18H14F2N2O2
(E)-2-cyano-3-(3,4-difluorophenyl)-N-(2-ethoxyphenyl)prop-2-enamide
—— ethyl (4S)-4-ethyl-2-oxo-6-[[[(R)-phenyl(thiophen-2-yl)methyl]amino]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C21H25N3O3S
ethyl (4S)-4-ethyl-2-oxo-6-[[[(R)-phenyl(thiophen-2-yl)methyl]amino]methyl]-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl (6R)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N2O4S
ethyl (6R)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-N-(4-bromo-2-chlorophenyl)-3-(2-methoxyphenyl)prop-2-enamide —— C16H13BrClNO2
(E)-N-(4-bromo-2-chlorophenyl)-3-(2-methoxyphenyl)prop-2-enamide
—— ethyl (6R)-6-(3,4-difluorophenyl)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O3S
ethyl (6R)-6-(3,4-difluorophenyl)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(3,4-difluorophenyl)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O3S
ethyl (6S)-6-(3,4-difluorophenyl)-3-[(2R)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-2-cyano-3-[3-(4-fluorobenzoyl)-2-methylindolizin-1-yl]-N-prop-2-enylprop-2-enamide —— C23H18FN3O2
(E)-2-cyano-3-[3-(4-fluorobenzoyl)-2-methylindolizin-1-yl]-N-prop-2-enylprop-2-enamide
—— (E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide —— C19H17N5O
(E)-2-cyano-3-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide
—— (E)-N-(4-bromo-2-chlorophenyl)-3-(4-nitrophenyl)prop-2-enamide —— C15H10BrClN2O3
(E)-N-(4-bromo-2-chlorophenyl)-3-(4-nitrophenyl)prop-2-enamide
—— ethyl (6S)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N2O4S
ethyl (6S)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-[2,4-bis(difluoromethoxy)phenyl]-2-cyano-N-prop-2-enylprop-2-enamide —— C15H12F4N2O3
(E)-3-[2,4-bis(difluoromethoxy)phenyl]-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-3-[5-chloro-1-[(4-chlorophenyl)methyl]-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C18H16Cl2N4O
(E)-3-[5-chloro-1-[(4-chlorophenyl)methyl]-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— ethyl (6R)-6-(3,4-difluorophenyl)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H22F2N2O3S
ethyl (6R)-6-(3,4-difluorophenyl)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(2,6-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H25F2N3O2S
ethyl (6S)-6-(2,6-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile —— C20H18ClFN6
(E)-3-[5-chloro-1-(4-fluorophenyl)-3-methylpyrazol-4-yl]-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)prop-2-enenitrile
—— (E)-N-(4-bromo-2-chlorophenyl)-3-thiophen-2-ylprop-2-enamide —— C13H9BrClNOS
(E)-N-(4-bromo-2-chlorophenyl)-3-thiophen-2-ylprop-2-enamide
—— Ethyl 2-[[2-[4-(dimethylamino)pyridin-1-ium-1-yl]acetyl]amino]-5-phenylthiophene-3-carboxylate —— C22H24N3O3S+
Ethyl 2-[[2-[4-(dimethylamino)pyridin-1-ium-1-yl]acetyl]amino]-5-phenylthiophene-3-carboxylate
—— (E)-2-cyano-N-naphthalen-1-yl-3-(2,3,4-trimethoxyphenyl)prop-2-enamide —— C23H20N2O4
(E)-2-cyano-N-naphthalen-1-yl-3-(2,3,4-trimethoxyphenyl)prop-2-enamide
—— Ethyl 2-[[2-(5-ethyl-2-methylpyridin-1-ium-1-yl)acetyl]amino]benzoate —— C19H23N2O3+
Ethyl 2-[[2-(5-ethyl-2-methylpyridin-1-ium-1-yl)acetyl]amino]benzoate
—— ethyl (6S)-3-[3-(dimethylamino)propyl]-6-(3-fluorophenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H26FN3O2S
ethyl (6S)-3-[3-(dimethylamino)propyl]-6-(3-fluorophenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-6-(2,6-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H25F2N3O2S
ethyl (6R)-6-(2,6-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6R)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N2O4S
ethyl (6R)-3-[(2S)-1-methoxypropan-2-yl]-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl 5-amino-4-cyano-3-[[[(R)-phenyl(thiophen-2-yl)methyl]amino]methyl]thiophene-2-carboxylate —— C20H19N3O2S2
ethyl 5-amino-4-cyano-3-[[[(R)-phenyl(thiophen-2-yl)methyl]amino]methyl]thiophene-2-carboxylate
—— ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C23H23N3O5
ethyl (6R)-6-[4-(cyanomethoxy)phenyl]-3-(4-methoxyphenyl)-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(4-ethylphenyl)prop-2-enamide —— C17H13ClN4OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-2-cyano-N-(4-ethylphenyl)prop-2-enamide
—— ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C21H28N4O3S
ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide —— C15H17ClN4O3S
(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-prop-2-enylprop-2-enamide —— C18H17ClN4O
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-2-cyano-N-prop-2-enylprop-2-enamide
—— (E)-2-cyano-3-(3,4-difluorophenyl)-N-(4-ethylphenyl)prop-2-enamide —— C18H14F2N2O
(E)-2-cyano-3-(3,4-difluorophenyl)-N-(4-ethylphenyl)prop-2-enamide
—— (E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-(3-ethoxypropyl)prop-2-enamide —— C17H23ClN4O4S
(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-2-cyano-N-(3-ethoxypropyl)prop-2-enamide
—— ethyl (6S)-6-(3,4-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H25F2N3O2S
ethyl (6S)-6-(3,4-difluorophenyl)-3-[3-(dimethylamino)propyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide —— C20H14Cl2N4O
(E)-3-(5-chloro-3-methyl-1-phenylpyrazol-4-yl)-N-(2-chlorophenyl)-2-cyanoprop-2-enamide
—— (E)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)-3-(2,4,6-trimethylphenyl)prop-2-enenitrile —— C19H22N4
(E)-2-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)-3-(2,4,6-trimethylphenyl)prop-2-enenitrile
—— (E)-2-cyano-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide —— C24H22N4O3
(E)-2-cyano-3-[3-(3,4-dimethoxyphenyl)-1-phenylpyrazol-4-yl]-N-prop-2-enylprop-2-enamide
—— (E)-N-(4-bromo-2-chlorophenyl)-3-(2-fluorophenyl)prop-2-enamide —— C15H10BrClFNO
(E)-N-(4-bromo-2-chlorophenyl)-3-(2-fluorophenyl)prop-2-enamide
—— (E)-2-cyano-N-(4-ethylphenyl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide —— C21H22N2O4
(E)-2-cyano-N-(4-ethylphenyl)-3-(2,4,5-trimethoxyphenyl)prop-2-enamide