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—— (E)-1-[4-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(2-methoxy-5-methylphenyl)prop-2-en-1-one —— C23H24N2O2S
(E)-1-[4-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(2-methoxy-5-methylphenyl)prop-2-en-1-one
—— ethyl (4R)-6-[[(Z)-3-(2,4-dimethoxyphenyl)prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H24N2O7
ethyl (4R)-6-[[(Z)-3-(2,4-dimethoxyphenyl)prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(4-methylphenyl)-N-[(2R)-2-pyridin-3-yl-2-thiophen-2-ylsulfonylethyl]prop-2-enamide —— C21H20N2O3S2
(E)-3-(4-methylphenyl)-N-[(2R)-2-pyridin-3-yl-2-thiophen-2-ylsulfonylethyl]prop-2-enamide
—— (E)-1-[4-(2-methylphenyl)piperazin-1-yl]-3-(3-methylthiophen-2-yl)prop-2-en-1-one —— C19H22N2OS
(E)-1-[4-(2-methylphenyl)piperazin-1-yl]-3-(3-methylthiophen-2-yl)prop-2-en-1-one
—— (E)-3-(3-chloro-4-methylphenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one —— C21H23ClN2O
(E)-3-(3-chloro-4-methylphenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one
—— (E)-1-[4-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(3-fluoro-4-methoxyphenyl)prop-2-en-1-one —— C22H21FN2O2S
(E)-1-[4-(1,3-benzothiazol-2-yl)piperidin-1-yl]-3-(3-fluoro-4-methoxyphenyl)prop-2-en-1-one
—— (E)-3-(2-fluorophenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C17H19FN4O2
(E)-3-(2-fluorophenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C19H23ClN4O4
(E)-3-(3-chloro-4,5-dimethoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(3-chloro-4-fluorophenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C17H18ClFN4O2
(E)-3-(3-chloro-4-fluorophenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[(2R)-2-pyridin-3-yl-2-thiophen-2-ylsulfonylethyl]prop-2-enamide —— C20H17FN2O3S2
(E)-3-(4-fluorophenyl)-N-[(2R)-2-pyridin-3-yl-2-thiophen-2-ylsulfonylethyl]prop-2-enamide
—— (E)-3-(3-chloro-1-benzothiophen-2-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C19H19ClN4O2S
(E)-3-(3-chloro-1-benzothiophen-2-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— ethyl N-[3-[[(1R)-1-(2-bromophenyl)ethyl]carbamoyl]phenyl]carbamate —— C18H19BrN2O3
ethyl N-[3-[[(1R)-1-(2-bromophenyl)ethyl]carbamoyl]phenyl]carbamate
—— ethyl 4-[[2-[(Z)-3-(2-nitrophenyl)prop-2-enoyl]oxyacetyl]amino]butanoate —— C17H20N2O7
ethyl 4-[[2-[(Z)-3-(2-nitrophenyl)prop-2-enoyl]oxyacetyl]amino]butanoate
—— ethyl (4S)-6-[[(Z)-3-(3-chlorophenyl)prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H19ClN2O5
ethyl (4S)-6-[[(Z)-3-(3-chlorophenyl)prop-2-enoyl]oxymethyl]-4-methyl-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-3-(2-methylphenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one —— C21H24N2O
(E)-3-(2-methylphenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one
—— ethyl N-[4-[4-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]phenyl]carbamate —— C22H23N3O3S
ethyl N-[4-[4-(1,3-benzothiazol-2-yl)piperidine-1-carbonyl]phenyl]carbamate
—— (E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C20H25ClN4O4
(E)-3-(3-chloro-5-ethoxy-4-methoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— ethyl N-[3-[[(1S)-1-(2-bromophenyl)ethyl]carbamoyl]phenyl]carbamate —— C18H19BrN2O3
ethyl N-[3-[[(1S)-1-(2-bromophenyl)ethyl]carbamoyl]phenyl]carbamate
—— (E)-3-(2,3-dichlorophenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C17H18Cl2N4O2
(E)-3-(2,3-dichlorophenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C19H22N4O4
(E)-3-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one —— C24H29ClN2O3
(E)-3-(3-chloro-5-methoxy-4-propan-2-yloxyphenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one
—— (E)-N-[2-(2,5-dichloroanilino)-2-oxoethyl]-3-(3-fluoro-4-methoxyphenyl)prop-2-enamide —— C18H15Cl2FN2O3
(E)-N-[2-(2,5-dichloroanilino)-2-oxoethyl]-3-(3-fluoro-4-methoxyphenyl)prop-2-enamide
—— (E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one —— C25H27FN4O
(E)-3-[1-(4-fluorophenyl)-3,5-dimethylpyrazol-4-yl]-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one
—— (E)-3-(4-methylphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C18H22N4O2
(E)-3-(4-methylphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(4-methylphenyl)-N-[(2S)-2-pyridin-3-yl-2-thiophen-2-ylsulfonylethyl]prop-2-enamide —— C21H20N2O3S2
(E)-3-(4-methylphenyl)-N-[(2S)-2-pyridin-3-yl-2-thiophen-2-ylsulfonylethyl]prop-2-enamide
—— (E)-1-[4-(2-methylphenyl)piperazin-1-yl]-3-(4-prop-2-enoxyphenyl)prop-2-en-1-one —— C23H26N2O2
(E)-1-[4-(2-methylphenyl)piperazin-1-yl]-3-(4-prop-2-enoxyphenyl)prop-2-en-1-one
—— (E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(2-ethoxyphenyl)prop-2-en-1-one —— C20H25N3O5S
(E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(2-ethoxyphenyl)prop-2-en-1-one
—— (E)-3-(furan-2-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C15H18N4O3
(E)-3-(furan-2-yl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(3,4-dimethoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C19H24N4O4
(E)-3-(3,4-dimethoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— (E)-3-(4-bromophenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one —— C20H21BrN2O
(E)-3-(4-bromophenyl)-1-[4-(2-methylphenyl)piperazin-1-yl]prop-2-en-1-one
—— Ethyl 4-[4-(diethylamino)anilino]-2-methylsulfanylpyrimidine-5-carboxylate —— C18H24N4O2S
Ethyl 4-[4-(diethylamino)anilino]-2-methylsulfanylpyrimidine-5-carboxylate
—— Ethyl 4-(3-imidazol-1-ylpropylamino)-2-methylsulfanylpyrimidine-5-carboxylate —— C14H19N5O2S
Ethyl 4-(3-imidazol-1-ylpropylamino)-2-methylsulfanylpyrimidine-5-carboxylate
—— Ethyl 4-[2-(4-methoxyphenoxy)ethylamino]-2-methylsulfanylpyrimidine-5-carboxylate —— C17H21N3O4S
Ethyl 4-[2-(4-methoxyphenoxy)ethylamino]-2-methylsulfanylpyrimidine-5-carboxylate
—— (E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(4-methylphenyl)prop-2-en-1-one —— C19H23N3O4S
(E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(4-methylphenyl)prop-2-en-1-one
—— ethyl 4,5-difluoro-2-[[(3R)-1-methyl-2-oxopyrrolidin-3-yl]amino]benzoate —— C14H16F2N2O3
ethyl 4,5-difluoro-2-[[(3R)-1-methyl-2-oxopyrrolidin-3-yl]amino]benzoate
—— ethyl 4-methyl-2-[(1S)-1-[(4-methylthiophene-3-carbonyl)amino]ethyl]-1,3-thiazole-5-carboxylate —— C15H18N2O3S2
ethyl 4-methyl-2-[(1S)-1-[(4-methylthiophene-3-carbonyl)amino]ethyl]-1,3-thiazole-5-carboxylate
—— ethyl 4,5-difluoro-2-[[(3S)-1-methyl-2-oxopyrrolidin-3-yl]amino]benzoate —— C14H16F2N2O3
ethyl 4,5-difluoro-2-[[(3S)-1-methyl-2-oxopyrrolidin-3-yl]amino]benzoate
—— (E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(4-ethoxyphenyl)prop-2-en-1-one —— C20H25N3O5S
(E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(4-ethoxyphenyl)prop-2-en-1-one
—— ethyl 4-methyl-2-[(1R)-1-[(4-methylthiophene-3-carbonyl)amino]ethyl]-1,3-thiazole-5-carboxylate —— C15H18N2O3S2
ethyl 4-methyl-2-[(1R)-1-[(4-methylthiophene-3-carbonyl)amino]ethyl]-1,3-thiazole-5-carboxylate
—— (E)-3-(2,4-dimethoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide —— C19H24N4O4
(E)-3-(2,4-dimethoxyphenyl)-N-[2-oxo-2-[(1,3,5-trimethylpyrazol-4-yl)amino]ethyl]prop-2-enamide
—— Ethyl 4-(3-chloro-4-fluoroanilino)-2-methylsulfanylpyrimidine-5-carboxylate —— C14H13ClFN3O2S
Ethyl 4-(3-chloro-4-fluoroanilino)-2-methylsulfanylpyrimidine-5-carboxylate
—— Ethyl 4-(4-carbamoylanilino)-2-methylsulfanylpyrimidine-5-carboxylate —— C15H16N4O3S
Ethyl 4-(4-carbamoylanilino)-2-methylsulfanylpyrimidine-5-carboxylate
—— ethyl 4-[[(3S)-7-chloro-1-oxo-3,4-dihydroisochromene-3-carbonyl]amino]benzoate —— C19H16ClNO5
ethyl 4-[[(3S)-7-chloro-1-oxo-3,4-dihydroisochromene-3-carbonyl]amino]benzoate
—— (E)-3-(6-methoxynaphthalen-2-yl)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]prop-2-enamide —— C26H28N2O3
(E)-3-(6-methoxynaphthalen-2-yl)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]prop-2-enamide
—— (E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(4-fluorophenyl)prop-2-en-1-one —— C18H20FN3O4S
(E)-1-[4-[(3,5-dimethyl-1,2-oxazol-4-yl)sulfonyl]piperazin-1-yl]-3-(4-fluorophenyl)prop-2-en-1-one
—— (E)-3-(1-benzylpyrazol-4-yl)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]prop-2-enamide —— C25H28N4O2
(E)-3-(1-benzylpyrazol-4-yl)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]prop-2-enamide
—— ethyl 5-(dimethylcarbamoyl)-2-[[2-[(2Z,4E)-hexa-2,4-dienoyl]oxyacetyl]amino]-4-methylthiophene-3-carboxylate —— C19H24N2O6S
ethyl 5-(dimethylcarbamoyl)-2-[[2-[(2Z,4E)-hexa-2,4-dienoyl]oxyacetyl]amino]-4-methylthiophene-3-carboxylate
—— (E)-3-(3,5-dimethoxyphenyl)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]prop-2-enamide —— C23H28N2O4
(E)-3-(3,5-dimethoxyphenyl)-N-[(1S)-2-morpholin-4-yl-1-phenylethyl]prop-2-enamide
—— (E)-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methyl-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide —— C19H16FN3O6
(E)-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methyl-3-(6-nitro-1,3-benzodioxol-5-yl)prop-2-enamide
—— (E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methylprop-2-enamide —— C20H24ClFN4O2
(E)-3-[5-chloro-3-methyl-1-(2-methylpropyl)pyrazol-4-yl]-N-[2-(3-fluoroanilino)-2-oxoethyl]-N-methylprop-2-enamide