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—— ethyl 1-phenyl-4-[(Z)-[(4-phenyl-1,3-thiazol-2-yl)hydrazinylidene]methyl]pyrazole-3-carboxylate —— C22H19N5O2S
ethyl 1-phenyl-4-[(Z)-[(4-phenyl-1,3-thiazol-2-yl)hydrazinylidene]methyl]pyrazole-3-carboxylate
—— ethyl (4R)-4-(3-ethoxycarbonyl-1-phenylpyrazol-4-yl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H22N4O4S
ethyl (4R)-4-(3-ethoxycarbonyl-1-phenylpyrazol-4-yl)-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[(6S,7R)-6-cyano-2-oxo-3,5,6,7-tetrahydrothiopyrano[2,3-d][1,3]thiazol-7-yl]-1-(4-fluorophenyl)pyrazole-3-carboxylate —— C19H15FN4O3S2
ethyl 4-[(6S,7R)-6-cyano-2-oxo-3,5,6,7-tetrahydrothiopyrano[2,3-d][1,3]thiazol-7-yl]-1-(4-fluorophenyl)pyrazole-3-carboxylate
—— ethyl 4-[(Z)-[(Z)-[(5Z)-5-[(4-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]hydrazinylidene]methyl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(Z)-[(Z)-[(5Z)-5-[(4-methoxyphenyl)methylidene]-4-oxo-1,3-thiazolidin-2-ylidene]hydrazinylidene]methyl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2S,5R)-5-cyano-1-(2,5-dimethylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C25H23N5O3S
ethyl 4-[(2S,5R)-5-cyano-1-(2,5-dimethylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2S,5R)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2S,5R)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2S,5S)-5-cyano-1-(4-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O3S
ethyl 4-[(2S,5S)-5-cyano-1-(4-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2R,5S)-5-cyano-1-(4-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2R,5S)-5-cyano-1-(4-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2S,5S)-5-cyano-1-(3-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O3S
ethyl 4-[(2S,5S)-5-cyano-1-(3-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— (E)-3-[1-(cyanomethyl)-2,5-dimethylpyrrol-3-yl]-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile —— C20H17N5O
(E)-3-[1-(cyanomethyl)-2,5-dimethylpyrrol-3-yl]-2-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]prop-2-enenitrile
—— ethyl 4-[(2R,5R)-5-cyano-1-(3-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O3S
ethyl 4-[(2R,5R)-5-cyano-1-(3-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2S,5S)-5-cyano-1-(2,5-dimethylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C25H23N5O3S
ethyl 4-[(2S,5S)-5-cyano-1-(2,5-dimethylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2R,5R)-5-cyano-1-(2,5-dimethylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C25H23N5O3S
ethyl 4-[(2R,5R)-5-cyano-1-(2,5-dimethylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2R,5S)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2R,5S)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl (4S)-4-[1-(4-chlorophenyl)-3-ethoxycarbonylpyrazol-4-yl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H21ClN4O4S
ethyl (4S)-4-[1-(4-chlorophenyl)-3-ethoxycarbonylpyrazol-4-yl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— ethyl 4-[(2R,5S)-5-cyano-1-(4-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O3S
ethyl 4-[(2R,5S)-5-cyano-1-(4-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(2S,5S)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2S,5S)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl (4R)-4-[1-(4-chlorophenyl)-3-ethoxycarbonylpyrazol-4-yl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C20H21ClN4O4S
ethyl (4R)-4-[1-(4-chlorophenyl)-3-ethoxycarbonylpyrazol-4-yl]-6-methyl-2-sulfanylidene-3,4-dihydro-1H-pyrimidine-5-carboxylate
—— (E)-2-methyl-N-[1-[2-(methylamino)-2-oxoethyl]piperidin-4-yl]pent-2-enamide —— C14H25N3O2
(E)-2-methyl-N-[1-[2-(methylamino)-2-oxoethyl]piperidin-4-yl]pent-2-enamide
—— ethyl 4-[(2R,5R)-5-cyano-1-(4-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O3S
ethyl 4-[(2R,5R)-5-cyano-1-(4-methylphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 1-[(2R)-2-hydroxy-3-(2-methylbut-3-yn-2-yloxy)propyl]piperidine-4-carboxylate —— C16H27NO4
ethyl 1-[(2R)-2-hydroxy-3-(2-methylbut-3-yn-2-yloxy)propyl]piperidine-4-carboxylate
—— (E)-N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-2-methylpent-2-enamide —— C16H21NO2
(E)-N-[[(3R)-3,4-dihydro-2H-chromen-3-yl]methyl]-2-methylpent-2-enamide
—— (E)-N-[(2,5-dimethoxyphenyl)methyl]-2-methylpent-2-enamide —— C15H21NO3
(E)-N-[(2,5-dimethoxyphenyl)methyl]-2-methylpent-2-enamide
—— (E)-2-methyl-N-(2-quinolin-8-ylethyl)pent-2-enamide —— C17H20N2O
(E)-2-methyl-N-(2-quinolin-8-ylethyl)pent-2-enamide
—— (E)-N-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]-2-methylpent-2-enamide —— C16H21NO2
(E)-N-[[(3S)-3,4-dihydro-2H-chromen-3-yl]methyl]-2-methylpent-2-enamide
—— (E)-N-[[6-(dimethylamino)pyridin-3-yl]methyl]-2-methylpent-2-enamide —— C14H21N3O
(E)-N-[[6-(dimethylamino)pyridin-3-yl]methyl]-2-methylpent-2-enamide
—— ethyl 4-[(2S,5S)-5-cyano-4-oxo-1-(4-propan-2-ylphenyl)-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C26H25N5O3S
ethyl 4-[(2S,5S)-5-cyano-4-oxo-1-(4-propan-2-ylphenyl)-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 2-[[2-[[(2S)-5,6-dimethyl-4-oxo-3-prop-2-enyl-1,2-dihydrothieno[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H29N3O4S3
ethyl 2-[[2-[[(2S)-5,6-dimethyl-4-oxo-3-prop-2-enyl-1,2-dihydrothieno[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-N-[(5-bromothiophen-2-yl)methyl]-2-methylpent-2-enamide —— C11H14BrNOS
(E)-N-[(5-bromothiophen-2-yl)methyl]-2-methylpent-2-enamide
—— ethyl 4-[(2S,5R)-5-cyano-1-(4-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2S,5R)-5-cyano-1-(4-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— (E)-2-methyl-N-[[(2S)-oxolan-2-yl]methyl]pent-2-enamide —— C11H19NO2
(E)-2-methyl-N-[[(2S)-oxolan-2-yl]methyl]pent-2-enamide
—— ethyl (3R)-1-[(Z)-2-methylpent-2-enoyl]piperidine-3-carboxylate —— C14H23NO3
ethyl (3R)-1-[(Z)-2-methylpent-2-enoyl]piperidine-3-carboxylate
—— ethyl 4-[(2R,5R)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2R,5R)-5-cyano-1-(3-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— ethyl 4-[(Z)-2-methylpent-2-enoyl]piperazine-1-carboxylate —— C13H22N2O3
ethyl 4-[(Z)-2-methylpent-2-enoyl]piperazine-1-carboxylate
—— (E)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(4-thiophen-2-ylthiophen-2-yl)prop-2-enamide —— C22H20N2O3S2
(E)-2-cyano-N-[2-(3,4-dimethoxyphenyl)ethyl]-3-(4-thiophen-2-ylthiophen-2-yl)prop-2-enamide
—— (E)-2-methylsulfonyl-3-(4-thiophen-2-ylthiophen-2-yl)prop-2-enenitrile —— C12H9NO2S3
(E)-2-methylsulfonyl-3-(4-thiophen-2-ylthiophen-2-yl)prop-2-enenitrile
—— ethyl 4-[(2S,5S)-5-cyano-1-(4-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate —— C24H21N5O4S
ethyl 4-[(2S,5S)-5-cyano-1-(4-methoxyphenyl)-4-oxo-6-sulfanylidene-1,3-diazinan-2-yl]-1-phenylpyrazole-3-carboxylate
—— (E)-N-[(2-methoxypyridin-3-yl)methyl]-2-methylpent-2-enamide —— C13H18N2O2
(E)-N-[(2-methoxypyridin-3-yl)methyl]-2-methylpent-2-enamide
—— (E)-2-cyano-N-phenyl-3-(4-thiophen-2-ylthiophen-2-yl)prop-2-enamide —— C18H12N2OS2
(E)-2-cyano-N-phenyl-3-(4-thiophen-2-ylthiophen-2-yl)prop-2-enamide
—— ethyl 1-[(2S)-2-hydroxy-3-(2-methylbut-3-yn-2-yloxy)propyl]piperidine-4-carboxylate —— C16H27NO4
ethyl 1-[(2S)-2-hydroxy-3-(2-methylbut-3-yn-2-yloxy)propyl]piperidine-4-carboxylate
—— ethyl 2-[[2-[[(2R)-5,6-dimethyl-4-oxo-3-prop-2-enyl-1,2-dihydrothieno[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate —— C24H29N3O4S3
ethyl 2-[[2-[[(2R)-5,6-dimethyl-4-oxo-3-prop-2-enyl-1,2-dihydrothieno[2,3-d]pyrimidin-2-yl]sulfanyl]acetyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylate
—— (E)-2-methyl-N-[(2-morpholin-4-ylpyridin-4-yl)methyl]pent-2-enamide —— C16H23N3O2
(E)-2-methyl-N-[(2-morpholin-4-ylpyridin-4-yl)methyl]pent-2-enamide
—— (E)-1-[4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-1-yl]-3-(4-methoxyphenyl)-2-thiophen-2-ylprop-2-en-1-one —— C28H27NO5S
(E)-1-[4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-1-yl]-3-(4-methoxyphenyl)-2-thiophen-2-ylprop-2-en-1-one
—— ethyl (3S)-1-[(Z)-2-methylpent-2-enoyl]piperidine-3-carboxylate —— C14H23NO3
ethyl (3S)-1-[(Z)-2-methylpent-2-enoyl]piperidine-3-carboxylate
—— (E)-2-methyl-N-[3-(propanoylamino)phenyl]pent-2-enamide —— C15H20N2O2
(E)-2-methyl-N-[3-(propanoylamino)phenyl]pent-2-enamide
—— (E)-3-(3-fluorophenyl)-N-methyl-N-[2-(methylamino)-2-oxoethyl]-2-(5-methyltetrazol-1-yl)prop-2-enamide —— C15H17FN6O2
(E)-3-(3-fluorophenyl)-N-methyl-N-[2-(methylamino)-2-oxoethyl]-2-(5-methyltetrazol-1-yl)prop-2-enamide
—— (E)-N-[3-(difluoromethoxy)-4-methoxyphenyl]-2-methylpent-2-enamide —— C14H17F2NO3
(E)-N-[3-(difluoromethoxy)-4-methoxyphenyl]-2-methylpent-2-enamide
—— ethyl 6-[4-[(Z)-3-(furan-2-yl)prop-2-enoyl]piperazin-1-yl]pyridine-3-carboxylate —— C19H21N3O4
ethyl 6-[4-[(Z)-3-(furan-2-yl)prop-2-enoyl]piperazin-1-yl]pyridine-3-carboxylate
—— (E)-N-(5-acetamido-2-fluorophenyl)-2-methylpent-2-enamide —— C14H17FN2O2
(E)-N-(5-acetamido-2-fluorophenyl)-2-methylpent-2-enamide
—— (E)-2-(6-bromo-4-oxo-3H-quinazolin-2-yl)-3-(2-ethyl-1-benzofuran-3-yl)prop-2-enenitrile —— C21H14BrN3O2
(E)-2-(6-bromo-4-oxo-3H-quinazolin-2-yl)-3-(2-ethyl-1-benzofuran-3-yl)prop-2-enenitrile