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—— (E)-3-(4-bromofuran-2-yl)-2-cyano-N-(3-ethoxypropyl)prop-2-enamide —— C13H15BrN2O3
(E)-3-(4-bromofuran-2-yl)-2-cyano-N-(3-ethoxypropyl)prop-2-enamide
—— (E)-N-[2-[[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl]-3-(4-fluorophenyl)but-2-enamide —— C16H19FN2O4S
(E)-N-[2-[[(3S)-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl]-3-(4-fluorophenyl)but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)but-2-enamide —— C19H21FN2O2
(E)-3-(4-fluorophenyl)-N-(2-methoxyethyl)-N-(pyridin-2-ylmethyl)but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-methyl-N-(2-oxo-2-pyrrolidin-1-ylethyl)but-2-enamide —— C17H21FN2O2
(E)-3-(4-fluorophenyl)-N-methyl-N-(2-oxo-2-pyrrolidin-1-ylethyl)but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[(1S,3S)-3-methylcyclohexyl]but-2-enamide —— C17H22FNO
(E)-3-(4-fluorophenyl)-N-[(1S,3S)-3-methylcyclohexyl]but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[(2R)-1-oxo-1-(propylamino)propan-2-yl]but-2-enamide —— C16H21FN2O2
(E)-3-(4-fluorophenyl)-N-[(2R)-1-oxo-1-(propylamino)propan-2-yl]but-2-enamide
—— (E)-N-[(2S)-1-(ethylamino)-1-oxopropan-2-yl]-3-(4-fluorophenyl)but-2-enamide —— C15H19FN2O2
(E)-N-[(2S)-1-(ethylamino)-1-oxopropan-2-yl]-3-(4-fluorophenyl)but-2-enamide
—— (E)-N-(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)-3-(4-fluorophenyl)but-2-enamide —— C18H22FN3O
(E)-N-(3,5-dimethyl-1-propan-2-ylpyrazol-4-yl)-3-(4-fluorophenyl)but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[[1-(2-methoxyethyl)-3,5-dimethylpyrazol-4-yl]methyl]but-2-enamide —— C19H24FN3O2
(E)-3-(4-fluorophenyl)-N-[[1-(2-methoxyethyl)-3,5-dimethylpyrazol-4-yl]methyl]but-2-enamide
—— (E)-3-(7-methoxy-1,3-benzodioxol-5-yl)-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)prop-2-enenitrile —— C20H16N4O3
(E)-3-(7-methoxy-1,3-benzodioxol-5-yl)-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)prop-2-enenitrile
—— (E)-3-(4-fluorophenyl)-N-[3-[methyl(methylsulfonyl)amino]propyl]but-2-enamide —— C15H21FN2O3S
(E)-3-(4-fluorophenyl)-N-[3-[methyl(methylsulfonyl)amino]propyl]but-2-enamide
—— ethyl (Z)-2-(1-methylimidazol-2-yl)-3-(3-propan-2-yloxyphenyl)prop-2-enoate —— C18H22N2O3
ethyl (Z)-2-(1-methylimidazol-2-yl)-3-(3-propan-2-yloxyphenyl)prop-2-enoate
—— (E)-3-(4-fluorophenyl)-N-[[2-(1,2,4-triazol-1-yl)pyridin-3-yl]methyl]but-2-enamide —— C18H16FN5O
(E)-3-(4-fluorophenyl)-N-[[2-(1,2,4-triazol-1-yl)pyridin-3-yl]methyl]but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[1-[2-(methylamino)-2-oxoethyl]piperidin-4-yl]but-2-enamide —— C18H24FN3O2
(E)-3-(4-fluorophenyl)-N-[1-[2-(methylamino)-2-oxoethyl]piperidin-4-yl]but-2-enamide
—— (E)-3-(4-fluorophenyl)-N-methyl-N-(pyridin-2-ylmethyl)but-2-enamide —— C17H17FN2O
(E)-3-(4-fluorophenyl)-N-methyl-N-(pyridin-2-ylmethyl)but-2-enamide
—— (E)-N-[2-(cyclopropylamino)-2-oxoethyl]-3-(4-fluorophenyl)-N-methylbut-2-enamide —— C16H19FN2O2
(E)-N-[2-(cyclopropylamino)-2-oxoethyl]-3-(4-fluorophenyl)-N-methylbut-2-enamide
—— (E)-3-(4-fluorophenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)but-2-enamide —— C18H23FN2O2
(E)-3-(4-fluorophenyl)-N-(3-oxo-3-piperidin-1-ylpropyl)but-2-enamide
—— (E)-N-[(1S)-1-(1,5-dimethylpyrazol-4-yl)ethyl]-3-(4-fluorophenyl)but-2-enamide —— C17H20FN3O
(E)-N-[(1S)-1-(1,5-dimethylpyrazol-4-yl)ethyl]-3-(4-fluorophenyl)but-2-enamide
—— (E)-4-(1,3-benzothiazol-2-yl)-5-[5-methoxy-2-(pyridin-2-ylmethoxy)phenyl]pent-4-enoic acid —— C25H22N2O4S
(E)-4-(1,3-benzothiazol-2-yl)-5-[5-methoxy-2-(pyridin-2-ylmethoxy)phenyl]pent-4-enoic acid
—— (E)-3-(4-fluorophenyl)-N-propan-2-ylsulfonylbut-2-enamide —— C13H16FNO3S
(E)-3-(4-fluorophenyl)-N-propan-2-ylsulfonylbut-2-enamide
—— (E)-3-(4-fluorophenyl)-N-[6-(1,2,4-triazol-1-yl)pyridin-3-yl]but-2-enamide —— C17H14FN5O
(E)-3-(4-fluorophenyl)-N-[6-(1,2,4-triazol-1-yl)pyridin-3-yl]but-2-enamide
—— (E)-N-[(1R)-1-(1,5-dimethylpyrazol-4-yl)ethyl]-3-(4-fluorophenyl)but-2-enamide —— C17H20FN3O
(E)-N-[(1R)-1-(1,5-dimethylpyrazol-4-yl)ethyl]-3-(4-fluorophenyl)but-2-enamide
—— ethyl (Z)-3-[4-[[3-(4-fluorophenyl)thiophene-2-carbonyl]amino]phenyl]prop-2-enoate —— C22H18FNO3S
ethyl (Z)-3-[4-[[3-(4-fluorophenyl)thiophene-2-carbonyl]amino]phenyl]prop-2-enoate
—— (E)-3-(4-fluorophenyl)-N-[(2S)-1-oxo-1-(propylamino)propan-2-yl]but-2-enamide —— C16H21FN2O2
(E)-3-(4-fluorophenyl)-N-[(2S)-1-oxo-1-(propylamino)propan-2-yl]but-2-enamide
—— (E)-3-(4-fluorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]but-2-en-1-one —— C20H27FN2O2
(E)-3-(4-fluorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]but-2-en-1-one
—— (E)-N-[1-(2-amino-2-oxoethyl)pyrazol-3-yl]-3-(4-fluorophenyl)but-2-enamide —— C15H15FN4O2
(E)-N-[1-(2-amino-2-oxoethyl)pyrazol-3-yl]-3-(4-fluorophenyl)but-2-enamide
—— (E)-N-(dimethylsulfamoyl)-3-(4-fluorophenyl)but-2-enamide —— C12H15FN2O3S
(E)-N-(dimethylsulfamoyl)-3-(4-fluorophenyl)but-2-enamide
—— (E)-N-[(2R)-1-(ethylamino)-1-oxopropan-2-yl]-3-(4-fluorophenyl)but-2-enamide —— C15H19FN2O2
(E)-N-[(2R)-1-(ethylamino)-1-oxopropan-2-yl]-3-(4-fluorophenyl)but-2-enamide
—— (E)-3-cyclopropyl-N-[1-[2-(diethylamino)ethyl]pyrazol-4-yl]but-2-enamide —— C16H26N4O
(E)-3-cyclopropyl-N-[1-[2-(diethylamino)ethyl]pyrazol-4-yl]but-2-enamide
—— (E)-N-[2-(tert-butylamino)-2-oxoethyl]-3-(4-fluorophenyl)-N-methylbut-2-enamide —— C17H23FN2O2
(E)-N-[2-(tert-butylamino)-2-oxoethyl]-3-(4-fluorophenyl)-N-methylbut-2-enamide
—— ethyl (Z)-3-(3,4-diethoxyphenyl)-2-(1-methylimidazol-2-yl)prop-2-enoate —— C19H24N2O4
ethyl (Z)-3-(3,4-diethoxyphenyl)-2-(1-methylimidazol-2-yl)prop-2-enoate
—— (E)-3-(1-adamantyl)-N-[2-(methanesulfonamido)phenyl]but-2-enamide —— C21H28N2O3S
(E)-3-(1-adamantyl)-N-[2-(methanesulfonamido)phenyl]but-2-enamide
—— ethyl (2S)-2-[[(Z)-3-(4-carbamoylphenyl)prop-2-enoyl]amino]-3-methylbutanoate —— C17H22N2O4
ethyl (2S)-2-[[(Z)-3-(4-carbamoylphenyl)prop-2-enoyl]amino]-3-methylbutanoate
—— ethyl (2R)-2-[[(Z)-3-(4-carbamoylphenyl)prop-2-enoyl]amino]-3-methylbutanoate —— C17H22N2O4
ethyl (2R)-2-[[(Z)-3-(4-carbamoylphenyl)prop-2-enoyl]amino]-3-methylbutanoate
—— (E)-3-(4-fluorophenyl)-N-[(1S,3R)-3-methylcyclohexyl]but-2-enamide —— C17H22FNO
(E)-3-(4-fluorophenyl)-N-[(1S,3R)-3-methylcyclohexyl]but-2-enamide
—— (E)-3-(2,3-dihydro-1,4-benzodioxin-5-yl)-2-(4-pyridin-2-yl-1,3-thiazol-2-yl)prop-2-enenitrile —— C19H13N3O2S
(E)-3-(2,3-dihydro-1,4-benzodioxin-5-yl)-2-(4-pyridin-2-yl-1,3-thiazol-2-yl)prop-2-enenitrile
—— (E)-3-(furan-2-yl)-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)prop-2-enenitrile —— C16H12N4O
(E)-3-(furan-2-yl)-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)prop-2-enenitrile
—— (E)-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)-3-(4-prop-2-ynoxyphenyl)prop-2-enenitrile —— C21H16N4O
(E)-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)-3-(4-prop-2-ynoxyphenyl)prop-2-enenitrile
—— (E)-3-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)prop-2-enenitrile —— C21H15FN6
(E)-3-[5-(4-fluorophenyl)-1H-pyrazol-4-yl]-2-(4-methyl-5-phenyl-1,2,4-triazol-3-yl)prop-2-enenitrile
—— (E)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-N-[(2R)-butan-2-yl]-2-cyanoprop-2-enamide —— C17H17BrN4O
(E)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-N-[(2R)-butan-2-yl]-2-cyanoprop-2-enamide
—— (E)-3-(5-chlorothiophen-2-yl)-2-(4-pyridin-4-yl-1,3-thiazol-2-yl)prop-2-enenitrile —— C15H8ClN3S2
(E)-3-(5-chlorothiophen-2-yl)-2-(4-pyridin-4-yl-1,3-thiazol-2-yl)prop-2-enenitrile
—— (E)-3-(5-methylfuran-2-yl)-N-[4-[[(Z)-3-(5-methylfuran-2-yl)prop-2-enoyl]-(pyridin-2-ylmethyl)amino]phenyl]prop-2-enamide —— C28H25N3O4
(E)-3-(5-methylfuran-2-yl)-N-[4-[[(Z)-3-(5-methylfuran-2-yl)prop-2-enoyl]-(pyridin-2-ylmethyl)amino]phenyl]prop-2-enamide
—— (E)-3-(4-fluorophenyl)-N-(1-methylpyrazol-3-yl)but-2-enamide —— C14H14FN3O
(E)-3-(4-fluorophenyl)-N-(1-methylpyrazol-3-yl)but-2-enamide
—— (E)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide —— C18H17BrN4O2
(E)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-[[(2R)-oxolan-2-yl]methyl]prop-2-enamide
—— (E)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide —— C18H17BrN4O2
(E)-3-[5-(4-bromophenyl)-1H-pyrazol-4-yl]-2-cyano-N-[[(2S)-oxolan-2-yl]methyl]prop-2-enamide
—— ethyl 2,5-dimethyl-4-[2-[2-(2-oxo-1,3-thiazolidin-3-yl)acetyl]oxyacetyl]-1H-pyrrole-3-carboxylate —— C16H20N2O6S
ethyl 2,5-dimethyl-4-[2-[2-(2-oxo-1,3-thiazolidin-3-yl)acetyl]oxyacetyl]-1H-pyrrole-3-carboxylate
—— ethyl 4-[[2-[(4S)-4-cyclopropyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-ium-5-yl]acetyl]amino]piperidine-1-carboxylate —— C20H30N3O3S+
ethyl 4-[[2-[(4S)-4-cyclopropyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-ium-5-yl]acetyl]amino]piperidine-1-carboxylate
—— (E)-2-cyano-3-(2,2-dimethyl-3,4-dihydrochromen-6-yl)-N-(2,4-dimethylphenyl)prop-2-enamide —— C23H24N2O2
(E)-2-cyano-3-(2,2-dimethyl-3,4-dihydrochromen-6-yl)-N-(2,4-dimethylphenyl)prop-2-enamide
—— ethyl 4-[[2-[(4R)-4-cyclopropyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-ium-5-yl]acetyl]amino]piperidine-1-carboxylate —— C20H30N3O3S+
ethyl 4-[[2-[(4R)-4-cyclopropyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-ium-5-yl]acetyl]amino]piperidine-1-carboxylate
—— ethyl 6-[[(4S)-4-cyclopropyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-ium-5-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate —— C18H24N3O3S+
ethyl 6-[[(4S)-4-cyclopropyl-4,5,6,7-tetrahydrothieno[3,2-c]pyridin-5-ium-5-yl]methyl]-2-oxo-3,4-dihydro-1H-pyrimidine-5-carboxylate