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—— (E)-1-[4-[(1S,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C17H21N3O2
(E)-1-[4-[(1S,2S)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2-hydroxy-4-methylphenyl)prop-2-enamide —— C18H20ClN3O4S
(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2-hydroxy-4-methylphenyl)prop-2-enamide
—— (E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2,3-dihydro-1H-inden-5-yl)prop-2-enamide —— C20H22ClN3O3S
(E)-3-[5-chloro-1-[(3R)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2,3-dihydro-1H-inden-5-yl)prop-2-enamide
—— (E)-3-(5-nitrofuran-2-yl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]prop-2-enamide —— C17H21N3O4
(E)-3-(5-nitrofuran-2-yl)-N-[(E)-[(1R,4R)-1,7,7-trimethyl-2-bicyclo[2.2.1]heptanylidene]amino]prop-2-enamide
—— (E)-1-[4-[(1S,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C17H21N3O2
(E)-1-[4-[(1S,2R)-2-methylcyclopropanecarbonyl]piperazin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (E)-3-(3-benzyl-1,2-dihydrotriazol-5-yl)-N-(4-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)prop-2-enamide —— C19H18N4O2
(E)-3-(3-benzyl-1,2-dihydrotriazol-5-yl)-N-(4-methyl-6-oxocyclohexa-2,4-dien-1-ylidene)prop-2-enamide
—— (E)-1-[4-(benzenesulfonyl)piperazin-1-yl]-3-phenylsulfanylprop-2-en-1-one —— C19H20N2O3S2
(E)-1-[4-(benzenesulfonyl)piperazin-1-yl]-3-phenylsulfanylprop-2-en-1-one
—— (E)-N-(2-hydroxy-4-methylphenyl)-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide —— C18H16N2O6
(E)-N-(2-hydroxy-4-methylphenyl)-3-(6-nitro-4H-1,3-benzodioxin-8-yl)prop-2-enamide
—— (E)-3-(3,5-dimethoxyphenyl)-N-(2-hydroxy-4-methylphenyl)prop-2-enamide —— C18H19NO4
(E)-3-(3,5-dimethoxyphenyl)-N-(2-hydroxy-4-methylphenyl)prop-2-enamide
—— ethyl (6R)-3-cyclopropyl-6-[3-(difluoromethoxy)-4-methoxyphenyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H22F2N2O4S
ethyl (6R)-3-cyclopropyl-6-[3-(difluoromethoxy)-4-methoxyphenyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-N-(2-hydroxy-4-methylphenyl)prop-2-enamide —— C21H20ClN3O2
(E)-3-(1-benzyl-5-chloro-3-methylpyrazol-4-yl)-N-(2-hydroxy-4-methylphenyl)prop-2-enamide
—— (E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2-hydroxy-4-methylphenyl)prop-2-enamide —— C18H20ClN3O4S
(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2-hydroxy-4-methylphenyl)prop-2-enamide
—— ethyl (6S)-6-(4-bromothiophen-2-yl)-3-cyclopropyl-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C15H17BrN2O2S2
ethyl (6S)-6-(4-bromothiophen-2-yl)-3-cyclopropyl-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-cyclopropyl-6-(2,4-difluorophenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C17H18F2N2O2S
ethyl (6S)-3-cyclopropyl-6-(2,4-difluorophenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-cyclopropyl-6-(4-methoxycarbonylphenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C19H22N2O4S
ethyl (6S)-3-cyclopropyl-6-(4-methoxycarbonylphenyl)-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-N'-[2-(2,6-dimethylphenoxy)acetyl]-3-(1-phenylpyrazol-4-yl)prop-2-enehydrazide —— C22H22N4O3
(E)-N'-[2-(2,6-dimethylphenoxy)acetyl]-3-(1-phenylpyrazol-4-yl)prop-2-enehydrazide
—— ethyl (6S)-3-cyclopropyl-6-[2-(difluoromethoxy)phenyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C18H20F2N2O3S
ethyl (6S)-3-cyclopropyl-6-[2-(difluoromethoxy)phenyl]-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— (E)-1-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]-3-(5-nitrofuran-2-yl)prop-2-en-1-one —— C19H21N3O6S
(E)-1-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]-3-(5-nitrofuran-2-yl)prop-2-en-1-one
—— (E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-(2-hydroxy-4-methylphenyl)prop-2-enamide —— C22H22ClN3O2
(E)-3-[1-[(2-chlorophenyl)methyl]-3,5-dimethylpyrazol-4-yl]-N-(2-hydroxy-4-methylphenyl)prop-2-enamide
—— (E)-3-phenylsulfanyl-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide —— C22H22N4OS
(E)-3-phenylsulfanyl-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide
—— (E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2,3-dihydro-1H-inden-5-yl)prop-2-enamide —— C20H22ClN3O3S
(E)-3-[5-chloro-1-[(3S)-1,1-dioxothiolan-3-yl]-3-methylpyrazol-4-yl]-N-(2,3-dihydro-1H-inden-5-yl)prop-2-enamide
—— (E)-3-(5-nitrofuran-2-yl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide —— C20H19N5O4
(E)-3-(5-nitrofuran-2-yl)-N-[3-(6,7,8,9-tetrahydro-5H-[1,2,4]triazolo[4,3-a]azepin-3-yl)phenyl]prop-2-enamide
—— ethyl (6S)-6-(4-chlorophenyl)-3-cyclopropyl-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C17H19ClN2O2S
ethyl (6S)-6-(4-chlorophenyl)-3-cyclopropyl-4-methyl-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 4-[2-(3-ethyl-4-oxophthalazine-1-carbonyl)hydrazinyl]-4-oxobutanoate —— C17H20N4O5
Ethyl 4-[2-(3-ethyl-4-oxophthalazine-1-carbonyl)hydrazinyl]-4-oxobutanoate
—— ethyl (6R)-3-cyclopropyl-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate —— C20H24N2O3S
ethyl (6R)-3-cyclopropyl-4-methyl-6-(3-prop-2-enoxyphenyl)-2-sulfanylidene-1,6-dihydropyrimidine-5-carboxylate
—— Ethyl 4-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]-4-oxobutanoate —— C18H26N2O5S
Ethyl 4-[4-(2,5-dimethylphenyl)sulfonylpiperazin-1-yl]-4-oxobutanoate
—— (E)-N-(2,3-dihydro-1H-inden-5-yl)-3-(3,5-dimethoxyphenyl)prop-2-enamide —— C20H21NO3
(E)-N-(2,3-dihydro-1H-inden-5-yl)-3-(3,5-dimethoxyphenyl)prop-2-enamide
—— (E)-1-[(3S)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C20H22N2O2
(E)-1-[(3S)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— (E)-3-(1-benzyltriazol-4-yl)-N-[(5-chlorothiophen-2-yl)methyl]-N-prop-2-enylprop-2-enamide —— C20H19ClN4OS
(E)-3-(1-benzyltriazol-4-yl)-N-[(5-chlorothiophen-2-yl)methyl]-N-prop-2-enylprop-2-enamide
—— (E)-1-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]-3-phenylsulfanylprop-2-en-1-one —— C20H22N2O3S2
(E)-1-[4-(4-methylphenyl)sulfonylpiperazin-1-yl]-3-phenylsulfanylprop-2-en-1-one
—— ethyl 4-oxo-4-[3-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)anilino]butanoate —— C18H25N3O5S
ethyl 4-oxo-4-[3-(3,4,5,6-tetrahydro-2H-azepin-7-ylsulfamoyl)anilino]butanoate
—— (E)-N-[4-(dimethylsulfamoyl)phenyl]-3-phenylsulfanylprop-2-enamide —— C17H18N2O3S2
(E)-N-[4-(dimethylsulfamoyl)phenyl]-3-phenylsulfanylprop-2-enamide
—— (E)-N-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]-3-(5-nitrofuran-2-yl)prop-2-enamide —— C19H21N3O6S
(E)-N-[4-(4-methylpiperidin-1-yl)sulfonylphenyl]-3-(5-nitrofuran-2-yl)prop-2-enamide
—— Ethyl 4-[4-(3,4-dimethylphenyl)sulfonylpiperazin-1-yl]-4-oxobutanoate —— C18H26N2O5S
Ethyl 4-[4-(3,4-dimethylphenyl)sulfonylpiperazin-1-yl]-4-oxobutanoate
—— (E)-N'-[2-(4-cyanophenoxy)acetyl]-3-(3,5-dimethoxyphenyl)prop-2-enehydrazide —— C20H19N3O5
(E)-N'-[2-(4-cyanophenoxy)acetyl]-3-(3,5-dimethoxyphenyl)prop-2-enehydrazide
—— Ethyl 4-oxo-4-[2-(4-pyrrolidin-1-ylsulfonylbenzoyl)hydrazinyl]butanoate —— C17H23N3O6S
Ethyl 4-oxo-4-[2-(4-pyrrolidin-1-ylsulfonylbenzoyl)hydrazinyl]butanoate
—— (E)-1-[(3R)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one —— C20H22N2O2
(E)-1-[(3R)-3-(phenylmethoxymethyl)pyrrolidin-1-yl]-3-pyridin-3-ylprop-2-en-1-one
—— Ethyl 4-[2-(4-tert-butylbenzoyl)hydrazinyl]-4-oxobutanoate —— C17H24N2O4
Ethyl 4-[2-(4-tert-butylbenzoyl)hydrazinyl]-4-oxobutanoate
—— (E)-N'-[2-(1-adamantyl)acetyl]-3-(1-benzylpyrazol-4-yl)prop-2-enehydrazide —— C25H30N4O2
(E)-N'-[2-(1-adamantyl)acetyl]-3-(1-benzylpyrazol-4-yl)prop-2-enehydrazide
—— (E)-N'-[2-(2-methylphenoxy)acetyl]-3-(1-phenylpyrazol-4-yl)prop-2-enehydrazide —— C21H20N4O3
(E)-N'-[2-(2-methylphenoxy)acetyl]-3-(1-phenylpyrazol-4-yl)prop-2-enehydrazide
—— ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C19H21N3O4
ethyl (6S)-6-[4-(cyanomethoxy)phenyl]-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-3-cyclopropyl-6-[4-(difluoromethoxy)-3,5-dimethylphenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C20H24F2N2O4
ethyl (6S)-3-cyclopropyl-6-[4-(difluoromethoxy)-3,5-dimethylphenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— ethyl (6S)-6-(5-bromothiophen-2-yl)-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C15H17BrN2O3S
ethyl (6S)-6-(5-bromothiophen-2-yl)-3-cyclopropyl-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate
—— (E)-N-[(1S)-1-(3-fluoro-4-methylsulfonylphenyl)ethyl]-3-(furan-2-yl)prop-2-enamide —— C16H16FNO4S
(E)-N-[(1S)-1-(3-fluoro-4-methylsulfonylphenyl)ethyl]-3-(furan-2-yl)prop-2-enamide
—— (E)-3-(furan-2-yl)-N-[(2R)-4-(1-methylpyrrol-2-yl)butan-2-yl]prop-2-enamide —— C16H20N2O2
(E)-3-(furan-2-yl)-N-[(2R)-4-(1-methylpyrrol-2-yl)butan-2-yl]prop-2-enamide
—— (E)-3-(3,5-dimethoxyphenyl)-N'-[2-(2-fluorophenoxy)acetyl]prop-2-enehydrazide —— C19H19FN2O5
(E)-3-(3,5-dimethoxyphenyl)-N'-[2-(2-fluorophenoxy)acetyl]prop-2-enehydrazide
—— (E)-N'-[2-(4-ethylphenoxy)acetyl]-3-phenylsulfanylprop-2-enehydrazide —— C19H20N2O3S
(E)-N'-[2-(4-ethylphenoxy)acetyl]-3-phenylsulfanylprop-2-enehydrazide
—— Ethyl 4-[2-(3,5-dimethoxybenzoyl)hydrazinyl]-4-oxobutanoate —— C15H20N2O6
Ethyl 4-[2-(3,5-dimethoxybenzoyl)hydrazinyl]-4-oxobutanoate
—— (E)-N'-[2-(2-chlorophenoxy)acetyl]-3-(2-ethyl-1-benzofuran-3-yl)prop-2-enehydrazide —— C21H19ClN2O4
(E)-N'-[2-(2-chlorophenoxy)acetyl]-3-(2-ethyl-1-benzofuran-3-yl)prop-2-enehydrazide
—— ethyl (6R)-3-cyclopropyl-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate —— C20H24F2N2O5
ethyl (6R)-3-cyclopropyl-6-[4-(difluoromethoxy)-3-ethoxyphenyl]-4-methyl-2-oxo-1,6-dihydropyrimidine-5-carboxylate