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—— (7R)-1-(2-aminophenyl)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7,8-dihydro-6H-quinoline-2,5-dione —— C31H24N4O5S
(7R)-1-(2-aminophenyl)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7,8-dihydro-6H-quinoline-2,5-dione
—— (7S)-3-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C26H21ClN2O3S
(7S)-3-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-7-(2,4-dimethoxyphenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C31H33N5O3S
(7S)-7-(2,4-dimethoxyphenyl)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-5-methyl-7-propan-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5OS
(7R)-N-(4-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-5-methyl-7-propan-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-1-(3,5-dimethylphenyl)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7,8-dihydro-6H-quinoline-2,5-dione —— C33H27N3O5S
(7R)-1-(3,5-dimethylphenyl)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7,8-dihydro-6H-quinoline-2,5-dione
—— (7R)-1-(3,4-dimethylphenyl)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7,8-dihydro-6H-quinoline-2,5-dione —— C33H27N3O5S
(7R)-1-(3,4-dimethylphenyl)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-7,8-dihydro-6H-quinoline-2,5-dione
—— (7R)-2-[(2-methoxyphenyl)methylsulfanyl]-5-methyl-N-(4-methylphenyl)-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H27N5O2S
(7R)-2-[(2-methoxyphenyl)methylsulfanyl]-5-methyl-N-(4-methylphenyl)-7-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-[(2-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O5S
(7R)-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-[(2-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H20N2O2S
(7S)-3-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-3-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H19ClN2O2S
(7R)-3-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-2,5-dioxo-7-phenyl-N-[4-(trifluoromethoxy)phenyl]-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C23H17F3N2O4
(7S)-2,5-dioxo-7-phenyl-N-[4-(trifluoromethoxy)phenyl]-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— (7S)-3-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H17FN2O2S
(7S)-3-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-1-phenyl-7,8-dihydro-6H-quinoline-2,5-dione —— C31H23N3O5S
(7R)-7-(4-methoxyphenyl)-3-[4-(3-nitrophenyl)-1,3-thiazol-2-yl]-1-phenyl-7,8-dihydro-6H-quinoline-2,5-dione
—— (7S)-N-(4-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-5-methyl-7-propan-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H23Cl2N5OS
(7S)-N-(4-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-5-methyl-7-propan-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H17ClN2O2S
(7S)-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— 7-methoxy-3-[(S)-(4-methylpiperazin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H29N7O3
7-methoxy-3-[(S)-(4-methylpiperazin-1-yl)-[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (7S)-7-(4-bromo-2-methoxyphenyl)-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21BrN6O2
(7S)-7-(4-bromo-2-methoxyphenyl)-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H17ClN2O2S
(7R)-3-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-7-(2-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23Cl2N5O2S
(7R)-7-(2-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-ethoxy-4-hydroxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C23H25N5O4S
(7S)-7-(3-ethoxy-4-hydroxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-methylsulfanyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H19ClN2O3S
(7R)-3-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-N-(4-chlorophenyl)-7-(4-ethoxyphenyl)-5-methyl-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C22H19ClF3N5O2
(7S)-N-(4-chlorophenyl)-7-(4-ethoxyphenyl)-5-methyl-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H19ClN2O3S
(7S)-3-[4-(3-chlorophenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26FN5O3
(7S)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H17ClN2O2S
(7R)-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-6-N-(4-chlorophenyl)-7-(2,3-dimethoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26ClN5O4
(7S)-6-N-(4-chlorophenyl)-7-(2,3-dimethoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— 7-methoxy-3-[(R)-(4-methylpiperazin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one —— C22H29N7O3
7-methoxy-3-[(R)-(4-methylpiperazin-1-yl)-[1-[[(2R)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl]-1H-quinolin-2-one
—— (7S)-6-N-(4-chlorophenyl)-5-methyl-3-N,7-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C27H22ClN5O2
(7S)-6-N-(4-chlorophenyl)-5-methyl-3-N,7-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5O4S
(7R)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H26F3N5O
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7S)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-bromophenyl)-N-(4-methoxyphenyl)-5-methyl-2-[(2-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C28H26BrN5O2S
(7R)-7-(4-bromophenyl)-N-(4-methoxyphenyl)-5-methyl-2-[(2-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-6-N-(4-chlorophenyl)-7-(2,3-dimethoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26ClN5O4
(7R)-6-N-(4-chlorophenyl)-7-(2,3-dimethoxyphenyl)-5-methyl-3-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-7-(2-chlorophenyl)-5-(4-chlorophenyl)-2-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C24H18Cl2N4
(7R)-7-(2-chlorophenyl)-5-(4-chlorophenyl)-2-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7S)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N,7-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H27N5O2
(7S)-6-N-(2,4-dimethylphenyl)-5-methyl-3-N,7-diphenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-6-N-(4-chlorophenyl)-7-(3,4-dimethoxyphenyl)-3-N-(4-ethoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C31H30ClN5O5
(7S)-6-N-(4-chlorophenyl)-7-(3,4-dimethoxyphenyl)-3-N-(4-ethoxyphenyl)-5-methyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(2-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H23Cl2N5O2S
(7S)-7-(2-chlorophenyl)-2-[(4-chlorophenyl)methylsulfanyl]-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H19ClN2O3S
(7R)-3-[4-(4-chlorophenyl)-1,3-thiazol-2-yl]-7-(4-methoxyphenyl)-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26FN5O3
(7R)-7-(2-ethoxyphenyl)-3-N-(4-fluorophenyl)-5-methyl-6-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7S)-7-(2-chlorophenyl)-5-(4-chlorophenyl)-2-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C24H18Cl2N4
(7S)-7-(2-chlorophenyl)-5-(4-chlorophenyl)-2-(4-methylphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H26F3N5O
(7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(4-propan-2-ylphenyl)-2-(trifluoromethyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-N-(2,4-dimethylphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C31H33N5O4S
(7S)-2-benzylsulfanyl-N-(2,4-dimethylphenyl)-5-methyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H29N5O2S
(7R)-2-benzylsulfanyl-7-(4-ethylphenyl)-N-(2-methoxyphenyl)-5-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-[(2-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C30H31N5O5S
(7S)-7-(4-hydroxy-3,5-dimethoxyphenyl)-N-(4-methoxyphenyl)-5-methyl-2-[(2-methylphenyl)methylsulfanyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-6-N-(4-chlorophenyl)-5-methyl-7-(2-methylphenyl)-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide —— C29H26ClN5O2
(7S)-6-N-(4-chlorophenyl)-5-methyl-7-(2-methylphenyl)-3-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3,6-dicarboxamide
—— (7R)-3-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C25H20N2O2S
(7R)-3-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C29H28FN5O4S
(7S)-2-[(2-fluorophenyl)methylsulfanyl]-5-methyl-N-phenyl-7-(3,4,5-trimethoxyphenyl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-7-(4-methoxyphenyl)-3-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione —— C26H22N2O3S
(7R)-7-(4-methoxyphenyl)-3-[4-(4-methylphenyl)-1,3-thiazol-2-yl]-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7R)-7-(4-bromo-2-methoxyphenyl)-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide —— C21H21BrN6O2
(7R)-7-(4-bromo-2-methoxyphenyl)-N-(2,4-dimethylphenyl)-5-methyl-4,7-dihydrotetrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-2-benzylsulfanyl-7-(3-bromophenyl)-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C25H21BrN6OS
(7S)-2-benzylsulfanyl-7-(3-bromophenyl)-5-methyl-N-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide