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中文名称 英文名称 CAS号 化学式 结构式图片
—— (7R)-5-methyl-7-phenyl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H16F3N5O
(7R)-5-methyl-7-phenyl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methoxy-3-[[(4-methoxyphenyl)methyl-[[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one —— C29H30N6O4
7-methoxy-3-[[(4-methoxyphenyl)methyl-[[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl]amino]methyl]-1H-quinolin-2-one
—— 7-Benzyl-8-[2-(2-fluorophenyl)-2-oxoethyl]sulfanyl-1,3-dimethylpurine-2,6-dione —— C22H19FN4O3S
7-Benzyl-8-[2-(2-fluorophenyl)-2-oxoethyl]sulfanyl-1,3-dimethylpurine-2,6-dione
—— (7R)-7-methyl-3-[(4-methylphenyl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C20H21N3O
(7R)-7-methyl-3-[(4-methylphenyl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-3-[(4-chlorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C19H18ClN3O
(7R)-3-[(4-chlorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7S)-3-[(3-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C19H18FN3O
(7S)-3-[(3-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(1-methylpyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H22N6O
(7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(1-methylpyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-methyl-3-[(4-methylphenyl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C20H21N3O
(7S)-7-methyl-3-[(4-methylphenyl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-3-[(3-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C19H18FN3O
(7R)-3-[(3-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C27H27N5OS2
(7R)-N-(2,4-dimethylphenyl)-5-methyl-2-[(3-methylphenyl)methylsulfanyl]-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-(3-bromo-5-ethoxy-4-hydroxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20BrN5O3
(7S)-7-(3-bromo-5-ethoxy-4-hydroxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(1H-pyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H20N6O
(7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(1H-pyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-5-methyl-N-(2-methylphenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5OS
(7R)-5-methyl-N-(2-methylphenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[(2-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C19H18FN3O
(7R)-3-[(2-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-7-(3-bromo-5-ethoxy-4-hydroxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C21H20BrN5O3
(7R)-7-(3-bromo-5-ethoxy-4-hydroxyphenyl)-5-methyl-N-phenyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-methoxyphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5O2S
(7S)-N-(2-methoxyphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-3-[(2-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C19H18FN3O
(7S)-3-[(2-fluorophenyl)methyl]-7-methyl-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-5-methyl-N-(2-methylphenyl)-7-(1H-pyrrol-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C18H18N6O
(7R)-5-methyl-N-(2-methylphenyl)-7-(1H-pyrrol-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-7-methyl-3-[(2-methylphenyl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one —— C20H21N3O
(7S)-7-methyl-3-[(2-methylphenyl)methyl]-6,7,8,9-tetrahydropyrimido[4,5-b]quinolin-4-one
—— (7R)-5-methyl-7-pyridin-2-yl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H15F3N6O
(7R)-5-methyl-7-pyridin-2-yl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— 7-methoxy-3-[[[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl-(3-morpholin-4-ylpropyl)amino]methyl]-1H-quinolin-2-one —— C28H35N7O4
7-methoxy-3-[[[1-[(4-methoxyphenyl)methyl]tetrazol-5-yl]methyl-(3-morpholin-4-ylpropyl)amino]methyl]-1H-quinolin-2-one
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(1-methylpyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H22N6O
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(1-methylpyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2-chlorophenyl)-5-methyl-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H14ClN5OS
(7S)-N-(2-chlorophenyl)-5-methyl-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(1H-pyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H20N6O
(7S)-N-(2,4-dimethylphenyl)-5-methyl-7-(1H-pyrrol-2-yl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2-methoxyphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5O2S
(7R)-N-(2-methoxyphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-N-(2-methylphenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H19N5OS
(7S)-5-methyl-N-(2-methylphenyl)-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-5-methyl-7-pyridin-2-yl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C19H15F3N6O
(7S)-5-methyl-7-pyridin-2-yl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7S)-N-(4-acetylphenyl)-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C24H20N2O4
(7S)-N-(4-acetylphenyl)-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— 7-methyl-3-[[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one —— C24H27N7O2
7-methyl-3-[[[1-[[(2S)-oxolan-2-yl]methyl]tetrazol-5-yl]methyl-(pyridin-3-ylmethyl)amino]methyl]-1H-quinolin-2-one
—— 7-methyl-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-(2-morpholin-4-ylethyl)amino]methyl]-1H-quinolin-2-one —— C24H35N7O2
7-methyl-3-[[[1-(2-methylbutan-2-yl)tetrazol-5-yl]methyl-(2-morpholin-4-ylethyl)amino]methyl]-1H-quinolin-2-one
—— (7R)-N-(2-chlorophenyl)-5-methyl-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C17H14ClN5OS
(7R)-N-(2-chlorophenyl)-5-methyl-7-thiophen-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-3-[4-(3,4-dichlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione —— C24H16Cl2N2O2S
(7R)-3-[4-(3,4-dichlorophenyl)-1,3-thiazol-2-yl]-7-phenyl-1,6,7,8-tetrahydroquinoline-2,5-dione
—— (7S)-5-methyl-7-phenyl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H16F3N5O
(7S)-5-methyl-7-phenyl-N-[3-(trifluoromethyl)phenyl]-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide —— C20H21N5OS
(7R)-N-(2,4-dimethylphenyl)-5-methyl-7-(3-methylthiophen-2-yl)-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
—— (7R)-N-(4-acetylphenyl)-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C24H20N2O4
(7R)-N-(4-acetylphenyl)-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— (7S)-3-ethyl-6-[(4-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24FNS
(7S)-3-ethyl-6-[(4-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-6-benzyl-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H25NS
(7R)-6-benzyl-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7S)-3-ethyl-6-[(3-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24FNS
(7S)-3-ethyl-6-[(3-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-N-(2-chlorophenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C24H25ClN2O2S
(7R)-N-(2-chlorophenyl)-3-ethyl-7-(4-methoxyphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-3-ethyl-6-[(3-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24FNS
(7R)-3-ethyl-6-[(3-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-3-ethyl-6-[(4-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24FNS
(7R)-3-ethyl-6-[(4-fluorophenyl)methyl]-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-N-(2-ethoxyphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C25H28N2O2S
(7R)-N-(2-ethoxyphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7S)-N-(3,5-dimethylphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C25H28N2OS
(7S)-N-(3,5-dimethylphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7S)-3-ethyl-2-methyl-7-phenyl-N-(3,4,5-trimethoxyphenyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C26H30N2O4S
(7S)-3-ethyl-2-methyl-7-phenyl-N-(3,4,5-trimethoxyphenyl)-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-N-(5-chloro-2,4-dimethoxyphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C25H27ClN2O3S
(7R)-N-(5-chloro-2,4-dimethoxyphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7R)-3-ethyl-2-methyl-7-phenyl-N-[2-(trifluoromethyl)phenyl]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C24H23F3N2OS
(7R)-3-ethyl-2-methyl-7-phenyl-N-[2-(trifluoromethyl)phenyl]-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7S)-6-benzyl-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H25NS
(7S)-6-benzyl-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-3-ethyl-7-(4-fluorophenyl)-N-(2-methoxy-5-methylphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C25H27FN2O2S
(7R)-3-ethyl-7-(4-fluorophenyl)-N-(2-methoxy-5-methylphenyl)-2-methyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide
—— (7S)-N-(3-chlorophenyl)-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide —— C22H17ClN2O3
(7S)-N-(3-chlorophenyl)-2,5-dioxo-7-phenyl-1,6,7,8-tetrahydroquinoline-3-carboxamide
—— (7S)-N-(5-chloro-2,4-dimethoxyphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide —— C25H27ClN2O3S
(7S)-N-(5-chloro-2,4-dimethoxyphenyl)-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine-6-carboxamide