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—— (7-chloro-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2S)-2-(2,4-dichlorophenoxy)propanoate —— C18H13Cl3N2O4
(7-chloro-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2S)-2-(2,4-dichlorophenoxy)propanoate
—— 7-[(2-fluorophenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H19FN4O
7-[(2-fluorophenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H27FN4O2
7-(cyclobutanecarbonyl)-2-[(3S)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(3,4-Dimethoxy-phenyl)-9-furan-2-ylmethyl-7,9-dihydro-12-oxa-9,11-diaza-benzo[a]anthracen-8-ylideneamine —— C28H23N3O4
7-(3,4-Dimethoxy-phenyl)-9-furan-2-ylmethyl-7,9-dihydro-12-oxa-9,11-diaza-benzo[a]anthracen-8-ylideneamine
—— 7-[(3S)-1-[2-(2-fluorophenoxy)acetyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H18FN3O3
7-[(3S)-1-[2-(2-fluorophenoxy)acetyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl 5-methyl-3-phenyl-1,2-oxazole-4-carboxylate —— C23H19NO5
(7,8-Dimethyl-2-oxochromen-4-yl)methyl 5-methyl-3-phenyl-1,2-oxazole-4-carboxylate
—— 7-[(4-Fluorobenzyl)sulfanyl]-12-methyl-10,11,12,13-tetrahydro[1]benzothieno[3,2-e]bis[1,2,4]triazolo[4,3-a:1',5'-c]pyrimidine —— C20H17FN6S2
7-[(4-Fluorobenzyl)sulfanyl]-12-methyl-10,11,12,13-tetrahydro[1]benzothieno[3,2-e]bis[1,2,4]triazolo[4,3-a:1',5'-c]pyrimidine
—— 7-(4-methylphenyl)-2-[(tetrahydrofuran-2-ylmethyl)amino]-7,8-dihydroquinazolin-5(6H)-one —— C20H23N3O2
7-(4-methylphenyl)-2-[(tetrahydrofuran-2-ylmethyl)amino]-7,8-dihydroquinazolin-5(6H)-one
—— 7-(4-methylpiperidin-1-yl)-4-(propan-2-yl)-2,3-dihydro-1H-cyclopenta[4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidine —— C21H26N4S
7-(4-methylpiperidin-1-yl)-4-(propan-2-yl)-2,3-dihydro-1H-cyclopenta[4',5']pyrido[3',2':4,5]thieno[3,2-d]pyrimidine
—— 7-[(3R)-1-[2-(2-fluorophenoxy)acetyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H18FN3O3
7-[(3R)-1-[2-(2-fluorophenoxy)acetyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[[2-[(3-Fluorophenyl)methoxy]phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C26H23FN4O2
7-[[2-[(3-Fluorophenyl)methoxy]phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Bromo-2-methylbicyclo[2.2.1]heptan-2-ol —— C8H13BrO
7-Bromo-2-methylbicyclo[2.2.1]heptan-2-ol
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H27FN4O2
7-(cyclobutanecarbonyl)-2-[(3R)-1-[(2-fluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-fluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H23FN4O
7-[(2-fluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(difluoromethyl)-5-[(3S)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H18F3N5
7-(difluoromethyl)-5-[(3S)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-(difluoromethyl)-5-[(3R)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H18F3N5
7-(difluoromethyl)-5-[(3R)-1-[(2-fluorophenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-Methyl-4-[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]chromen-2-one —— C20H17N3O2S
7-Methyl-4-[(5-methyl-4-phenyl-1,2,4-triazol-3-yl)sulfanylmethyl]chromen-2-one
—— 7-cyclohexyl-2-[(3S)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-cyclohexyl-2-[(3S)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-cyclohexyl-2-[(3R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(2-fluorophenyl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27FN4O3
7-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(2-fluorophenyl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27FN4O3
7-(cyclobutanecarbonyl)-2-[(3R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(2-fluorophenyl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27FN4O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(2-fluorophenyl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C23H22FN3O2
7-[1-[1-(2-fluorophenyl)cyclopropanecarbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24FN5O2
7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27FN4O3
7-(cyclobutanecarbonyl)-2-[(3S)-1-[2-(2-fluorophenyl)acetyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24FN5O2
7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O4
7-(2-fluorobenzoyl)-2-[(3S)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O4
7-(2-fluorobenzoyl)-2-[(3R)-1-[(2R)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-[(3,5-Difluorophenyl)methyl]piperidin-4-yl]-1,6-naphthyridine —— C20H19F2N3
7-[1-[(3,5-Difluorophenyl)methyl]piperidin-4-yl]-1,6-naphthyridine
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H22FN5O3
7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H22FN5O3
7-(2-fluorobenzoyl)-2-[(3R)-1-(pyridine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-(2-fluorobenzoyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H18FN3O2
7-[1-(2-fluorobenzoyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O4
7-(2-fluorobenzoyl)-2-[(3S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24FN5O2
7-(2-fluorobenzoyl)-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23FN4O2S
7-(2-fluorobenzoyl)-2-[(3S)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-cyclohexyl-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23FN4O2S
7-(2-fluorobenzoyl)-2-[(3R)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O4
7-(2-fluorobenzoyl)-2-[(3R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)pyrrolidin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H17N5O4S
7-[(2S)-1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)pyrrolidin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-Chloro-3-[[4-hydroxy-1-(2-morpholin-4-ylacetyl)piperidin-4-yl]methyl]quinazolin-4-one —— C20H25ClN4O4
7-Chloro-3-[[4-hydroxy-1-(2-morpholin-4-ylacetyl)piperidin-4-yl]methyl]quinazolin-4-one
—— 7-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O3
7-[1-[(2R)-oxolane-2-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(2R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)pyrrolidin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C17H17N5O4S
7-[(2R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylsulfonyl)pyrrolidin-2-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-chloro-4-(2-oxo-2-pyrrolidin-1-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C19H23ClN2O4
7-chloro-4-(2-oxo-2-pyrrolidin-1-ylethyl)spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-[(2-chloro-6-fluorobenzyl)oxy]-3-[2-(4a-hydroxyoctahydroisoquinolin-2(1H)-yl)-2-oxoethyl]-4-methyl-2H-chromen-2-one —— C28H29ClFNO5
7-[(2-chloro-6-fluorobenzyl)oxy]-3-[2-(4a-hydroxyoctahydroisoquinolin-2(1H)-yl)-2-oxoethyl]-4-methyl-2H-chromen-2-one
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl 2-(2,4-dichlorophenoxy)acetate —— C20H16Cl2O5
(7,8-Dimethyl-2-oxochromen-4-yl)methyl 2-(2,4-dichlorophenoxy)acetate
—— (7-Methyl-2-oxochromen-4-yl)methyl 2-[(4-methoxybenzoyl)amino]-3-methylbutanoate —— C24H25NO6
(7-Methyl-2-oxochromen-4-yl)methyl 2-[(4-methoxybenzoyl)amino]-3-methylbutanoate
—— 7-(3,4-dihydro-2H-chromen-6-ylmethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine —— C15H18N4O
7-(3,4-dihydro-2H-chromen-6-ylmethyl)-6,8-dihydro-5H-[1,2,4]triazolo[4,3-a]pyrazine
—— 7-[(3R)-pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C12H13N3O
7-[(3R)-pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one