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—— 7-[(3S)-1-(cyclopropylmethyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine —— C22H25N5
7-[(3S)-1-(cyclopropylmethyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C18H21F3N4O4
7-[(2R)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-benzyl-2-[(3R)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-benzyl-2-[(3R)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C17H19F3N4O4
7-[(2R)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-(benzenesulfonyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine —— C24H23N5O2S
7-[(3S)-1-(benzenesulfonyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C21H25F3N4O3
7-[(3S)-1-(cyclopentanecarbonyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C19H19F3N6
7-[(3R)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(2R)-1-(cyclopropylmethyl)piperidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C19H23F3N4O2
7-[(2R)-1-(cyclopropylmethyl)piperidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(benzenesulfonyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine —— C24H23N5O2S
7-[(3R)-1-(benzenesulfonyl)piperidin-3-yl]-2-phenylpyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3R)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H23FN4O3
7-[(3R)-1-[2-(4-fluorophenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-(1-Benzoylpiperidin-4-yl)-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H26N4O4
7-(1-Benzoylpiperidin-4-yl)-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H19ClF3N5
7-[(3R)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O3
7-[(3-fluorophenyl)methyl]-2-[(3S)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H27ClN4O3
7-[(3S)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H26F3N5
7-[(3R)-1-(cyclohexylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H19F4N5
7-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3R)-1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H25FN4O3
7-[(3R)-1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H27FN4O3
7-[(3S)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(quinolin-6-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C23H21F3N6
7-[(3R)-1-(quinolin-6-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3R)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H27ClN4O3
7-[(3R)-1-[(4-chlorophenyl)methyl]piperidin-3-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[1-[(4-Methoxyphenyl)methyl]piperidin-4-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-diamine —— C21H23F3N6O
7-[1-[(4-Methoxyphenyl)methyl]piperidin-4-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-diamine
—— 7-[(3R)-1-(3-phenylpropyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C22H24F3N5
7-[(3R)-1-(3-phenylpropyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3R)-1-benzylpiperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H20F3N5
7-[(3R)-1-benzylpiperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3R)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H25N5O2
7-[(3R)-1-(1H-indol-5-ylmethyl)piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H25FN4O3
7-[(3S)-1-[3-(4-fluorophenyl)propanoyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-ethenyl-8-[5-(hydroxymethyl)furan-2-yl]-3,8a-diphenyl-5,8-dihydro-4aH-naphthalene-1,4-dione —— C29H24O4
7-ethenyl-8-[5-(hydroxymethyl)furan-2-yl]-3,8a-diphenyl-5,8-dihydro-4aH-naphthalene-1,4-dione
—— 7-[(3R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H26N4O4
7-[(3R)-1-[2-(4-methoxyphenyl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-(3-methylphenyl)-5-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C19H18N4
7-(3-methylphenyl)-5-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-(1-Acetylpiperidin-4-yl)-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C18H24N4O4
7-(1-Acetylpiperidin-4-yl)-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H19F4N5
7-[(3R)-1-[(4-fluorophenyl)methyl]piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[1-(Cyclopentanecarbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H30N4O4
7-[1-(Cyclopentanecarbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-ethenyl-8-[2-(2-hydroxyethoxy)phenyl]-2,8a-dimethyl-5,8-dihydro-4aH-naphthalene-1,4-dione —— C22H24O4
7-ethenyl-8-[2-(2-hydroxyethoxy)phenyl]-2,8a-dimethyl-5,8-dihydro-4aH-naphthalene-1,4-dione
—— 7-fluoro-3-methyl-6-(4-methylpiperazin-1-yl)-4H-1,4-benzothiazine 1,1-dioxide —— C14H18FN3O2S
7-fluoro-3-methyl-6-(4-methylpiperazin-1-yl)-4H-1,4-benzothiazine 1,1-dioxide
—— 7,9-Dibromo-3a,4,5,6-tetrahydro-[1,3]thiazolo[3,2-a][1,5]benzodiazepine —— C11H10Br2N2S
7,9-Dibromo-3a,4,5,6-tetrahydro-[1,3]thiazolo[3,2-a][1,5]benzodiazepine
—— 7-(3-Chloro-4-methylphenyl)-N-(1-methoxypropan-2-YL)-5-phenyl-7H-pyrrolo[2,3-D]pyrimidin-4-amine —— C23H23ClN4O
7-(3-Chloro-4-methylphenyl)-N-(1-methoxypropan-2-YL)-5-phenyl-7H-pyrrolo[2,3-D]pyrimidin-4-amine
—— 7,9-dibromo-4,5,6,11-tetrahydro-3aH-[1,3]thiazolo[3,2-a][1,5]benzodiazepin-11-ium —— C11H11Br2N2S+
7,9-dibromo-4,5,6,11-tetrahydro-3aH-[1,3]thiazolo[3,2-a][1,5]benzodiazepin-11-ium
—— 7-bromo-4-(cyclohexylcarbonyl)-5-phenyl-1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-one —— C22H23BrN2O2
7-bromo-4-(cyclohexylcarbonyl)-5-phenyl-1,3,4,5-tetrahydro-2H-1,4-benzodiazepin-2-one
—— 7-ethenyl-8-(2-hydroxy-4-methoxyphenyl)-3,8a-diphenyl-5,8-dihydro-4aH-naphthalene-1,4-dione —— C31H26O4
7-ethenyl-8-(2-hydroxy-4-methoxyphenyl)-3,8a-diphenyl-5,8-dihydro-4aH-naphthalene-1,4-dione
—— 7-methyl-5-phenyl-4-(4-(piperidin-1-ylsulfonyl)benzoyl)-4,5-dihydro-1H-benzo[e][1,4]diazepin-2(3H)-one —— C28H29N3O4S
7-methyl-5-phenyl-4-(4-(piperidin-1-ylsulfonyl)benzoyl)-4,5-dihydro-1H-benzo[e][1,4]diazepin-2(3H)-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(5-methyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O2
7-(cyclohexylmethyl)-4-methyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclopropylmethyl)-2-[(2R)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C26H32N4O3
7-(cyclopropylmethyl)-2-[(2R)-1-[3-(4-methoxyphenyl)propanoyl]piperidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-(2-methylpropanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(3-methylbutanoyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H27FN4O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpropanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(2S)-1-(2-morpholin-4-ylacetyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H31N5O3
7-benzyl-4-methyl-2-[(2S)-1-(2-morpholin-4-ylacetyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C20H23FN4O3S
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H36N4O2
7-(cyclohexylmethyl)-4-methyl-2-[(2R)-1-(3-methylbutanoyl)piperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C20H23FN4O3S
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-methylsulfonylpiperidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one