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—— (7S)-9-(4-chlorophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21Cl2N5O2
(7S)-9-(4-chlorophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-2-[(1S)-1-[[5-(3-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H23N5O2S3
(7R)-2-[(1S)-1-[[5-(3-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-9-(4-chlorophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21Cl2N5O2
(7R)-9-(4-chlorophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-2-[(1R)-1-[[5-(3-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H23N5O2S3
(7R)-2-[(1R)-1-[[5-(3-methoxyanilino)-1,3,4-thiadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C26H29N5O2
(7S)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-9-benzyl-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C24H23Cl2N5O2
(7R)-9-benzyl-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-[(2S)-3-(1,3-benzothiazol-2-ylsulfanyl)-2-methylpropyl]-3-methyl-8-piperidin-1-ylpurine-2,6-dione —— C22H26N6O2S2
7-[(2S)-3-(1,3-benzothiazol-2-ylsulfanyl)-2-methylpropyl]-3-methyl-8-piperidin-1-ylpurine-2,6-dione
—— (7R)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7R)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-1,7-dimethyl-3-[(3-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7S)-1,7-dimethyl-3-[(3-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-9-benzyl-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C24H23Cl2N5O2
(7S)-9-benzyl-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-9-(4-bromophenyl)-1,7-dimethyl-3-(3-phenylpropyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C25H26BrN5O2
(7R)-9-(4-bromophenyl)-1,7-dimethyl-3-(3-phenylpropyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-1,7-dimethyl-9-(4-phenoxyphenyl)-3-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7R)-1,7-dimethyl-9-(4-phenoxyphenyl)-3-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-methyl-8-[(3R)-3-methylpiperidin-1-yl]purine-2,6-dione —— C20H27N7O2S
7-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-methyl-8-[(3R)-3-methylpiperidin-1-yl]purine-2,6-dione
—— 7-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-methyl-8-[(3S)-3-methylpiperidin-1-yl]purine-2,6-dione —— C20H27N7O2S
7-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-3-methyl-8-[(3S)-3-methylpiperidin-1-yl]purine-2,6-dione
—— (7R)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C26H29N5O2
(7R)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-1,7-dimethyl-3-[(2-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7S)-1,7-dimethyl-3-[(2-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-[2-[(3S)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]-4-propylchromen-2-one —— C25H22N2O5S
7-[2-[(3S)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]-4-propylchromen-2-one
—— (7S)-1,7-dimethyl-9-(4-phenoxyphenyl)-3-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7S)-1,7-dimethyl-9-(4-phenoxyphenyl)-3-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-3-[(2,5-dimethylphenyl)methyl]-1,7-dimethyl-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C31H31N5O3
(7S)-3-[(2,5-dimethylphenyl)methyl]-1,7-dimethyl-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-9-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C25H25Cl2N5O2
(7R)-3-[(2,4-dichlorophenyl)methyl]-1,7-dimethyl-9-(2-phenylethyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-[[4-[(4S)-7-fluoro-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C21H20FN5O3S
7-[[4-[(4S)-7-fluoro-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7R)-9-cyclohexyl-3-[(3,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H27Cl2N5O2
(7R)-9-cyclohexyl-3-[(3,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-9-cyclohexyl-3-[(3,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H27Cl2N5O2
(7S)-9-cyclohexyl-3-[(3,4-dichlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-9-(4-chlorophenyl)-3-[(2-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21Cl2N5O2
(7S)-9-(4-chlorophenyl)-3-[(2-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-9-(4-bromophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21BrClN5O2
(7R)-9-(4-bromophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-[[4-[(4R)-7-fluoro-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C21H20FN5O3S
7-[[4-[(4R)-7-fluoro-2-oxo-3,4-dihydro-1H-quinoline-4-carbonyl]piperazin-1-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[(2S)-3-(1,3-benzothiazol-2-ylsulfanyl)-2-methylpropyl]-3-methyl-8-(4-methylpiperazin-1-yl)purine-2,6-dione —— C22H27N7O2S2
7-[(2S)-3-(1,3-benzothiazol-2-ylsulfanyl)-2-methylpropyl]-3-methyl-8-(4-methylpiperazin-1-yl)purine-2,6-dione
—— 7-[2-(1,3-benzothiazol-2-ylsulfanyl)ethyl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-1,3-dimethylpurine-2,6-dione —— C22H26N6O3S2
7-[2-(1,3-benzothiazol-2-ylsulfanyl)ethyl]-8-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-1,3-dimethylpurine-2,6-dione
—— 7-Bicyclo[4.2.0]octa-1,3,5-trienyl-[4-[1-(2-thiophen-3-ylethyl)imidazol-2-yl]piperidin-1-yl]methanone —— C23H25N3OS
7-Bicyclo[4.2.0]octa-1,3,5-trienyl-[4-[1-(2-thiophen-3-ylethyl)imidazol-2-yl]piperidin-1-yl]methanone
—— (7R)-3-[(2,5-dimethylphenyl)methyl]-1,7-dimethyl-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C31H31N5O3
(7R)-3-[(2,5-dimethylphenyl)methyl]-1,7-dimethyl-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-9-(4-bromophenyl)-1,7-dimethyl-3-(3-phenylpropyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C25H26BrN5O2
(7S)-9-(4-bromophenyl)-1,7-dimethyl-3-(3-phenylpropyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-1,3-dimethyl-8-[(3R)-3-methylpiperidin-1-yl]purine-2,6-dione —— C21H29N7O2S
7-[2-(4,6-dimethylpyrimidin-2-yl)sulfanylethyl]-1,3-dimethyl-8-[(3R)-3-methylpiperidin-1-yl]purine-2,6-dione
—— (7S)-9-(4-bromophenyl)-3-[(2-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21BrClN5O2
(7S)-9-(4-bromophenyl)-3-[(2-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-9-(4-bromophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21BrClN5O2
(7S)-9-(4-bromophenyl)-3-[(4-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7S)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7S)-1,7-dimethyl-3-[(4-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-1,7-dimethyl-3-[(2-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C30H29N5O3
(7R)-1,7-dimethyl-3-[(2-methylphenyl)methyl]-9-(4-phenoxyphenyl)-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— (7R)-9-(4-chlorophenyl)-3-[(2-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione —— C23H21Cl2N5O2
(7R)-9-(4-chlorophenyl)-3-[(2-chlorophenyl)methyl]-1,7-dimethyl-7,8-dihydro-6H-purino[7,8-a]pyrimidine-2,4-dione
—— 7-{(2-Hydroxy-5-methylphenyl)[(4-methylpyridin-2-yl)amino]methyl}quinolin-8-ol —— C23H21N3O2
7-{(2-Hydroxy-5-methylphenyl)[(4-methylpyridin-2-yl)amino]methyl}quinolin-8-ol
—— 7-[2-[(6-Bromo-2-chloroquinolin-3-yl)methylidene]hydrazinyl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylic acid —— C22H15BrClFN4O3
7-[2-[(6-Bromo-2-chloroquinolin-3-yl)methylidene]hydrazinyl]-1-ethyl-6-fluoro-4-oxoquinoline-3-carboxylic acid
—— 7-[2-[(3R)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]-4-propylchromen-2-one —— C25H22N2O5S
7-[2-[(3R)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethoxy]-4-propylchromen-2-one
—— 7-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethoxy]-4-ethylchromen-2-one —— C20H25NO4
7-[2-[(3S,5S)-3,5-dimethylpiperidin-1-yl]-2-oxoethoxy]-4-ethylchromen-2-one
—— [(7S)-2,5-dimethyl-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-morpholin-4-ylmethanone —— C17H20N6O2
[(7S)-2,5-dimethyl-7-pyridin-3-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-morpholin-4-ylmethanone
—— 7-methyl-4,6,6a,8,9,10,10a,11-octahydro-3aH-indolo[4,3-fg]quinoline-9-carboxamide —— C16H21N3O
7-methyl-4,6,6a,8,9,10,10a,11-octahydro-3aH-indolo[4,3-fg]quinoline-9-carboxamide
—— (7S)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C21H19N5O5
(7S)-N-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— 7-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethoxy]-4-ethylchromen-2-one —— C20H25NO4
7-[2-[(3S,5R)-3,5-dimethylpiperidin-1-yl]-2-oxoethoxy]-4-ethylchromen-2-one
—— (7R)-7-(3,4-dimethoxyphenyl)-5-(furan-2-yl)-2-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H18N4O3
(7R)-7-(3,4-dimethoxyphenyl)-5-(furan-2-yl)-2-methyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— [(7S)-2,5-dimethyl-7-pyridin-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-morpholin-4-ylmethanone —— C17H20N6O2
[(7S)-2,5-dimethyl-7-pyridin-2-yl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-morpholin-4-ylmethanone
—— (7R)-N-(2,3-dichlorophenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H15Cl2N5O3
(7R)-N-(2,3-dichlorophenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide
—— [(7R)-7-(furan-2-yl)-2,5-dimethyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-morpholin-4-ylmethanone —— C16H19N5O3
[(7R)-7-(furan-2-yl)-2,5-dimethyl-4,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl]-morpholin-4-ylmethanone
—— (7R)-N-(3-chloro-4-fluorophenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide —— C19H15ClFN5O3
(7R)-N-(3-chloro-4-fluorophenyl)-2-(4-methoxyphenyl)-5-oxo-6,7-dihydro-4H-[1,2,4]triazolo[1,5-a]pyrimidine-7-carboxamide