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—— 7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[2-(2-fluorophenyl)ethyl]-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3R)-1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C24H25N5O3
7-[(3R)-1-[2-(1H-indol-3-yl)acetyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(3-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3S)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-benzyl-4-methyl-2-[(3S)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(2-methoxyphenyl)methyl]-2-[(3R)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(3S)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O3
7-benzyl-2-[(3S)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3S)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H29N5O3
7-benzyl-4-methyl-2-[(3S)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(4-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(3R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H27N5O3
7-benzyl-2-[(3R)-1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H23FN6O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2S)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2S)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C21H25F3N4O3
7-[(2S)-1-(2-cyclopentylacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H30N4O4
7-[(2-methoxyphenyl)methyl]-2-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-pyrazol-1-ylacetyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(4-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-2-[(3S)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H27N5O3
7-benzyl-2-[(3S)-1-(2,4-dimethyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[2-(4-fluorophenyl)ethyl]-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O3
7-[2-(4-fluorophenyl)ethyl]-2-[(2R)-1-(2-methoxy-2-methylpropanoyl)pyrrolidin-2-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2S)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-benzyl-4-methyl-2-[(3R)-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O2
7-benzyl-4-methyl-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H26N4O3
7-[(3S)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C19H23F3N4O4
7-[(3S)-1-(3-methoxypropanoyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C18H21F3N4O4
7-[(3R)-1-(2-methoxyacetyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-benzyl-4-methyl-2-[(3S)-1-(4-methylthiadiazole-5-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H24N6O2S
7-benzyl-4-methyl-2-[(3S)-1-(4-methylthiadiazole-5-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-2-[(3R)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O3
7-[(3-fluorophenyl)methyl]-2-[(3R)-1-(2-methoxy-2-methylpropanoyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-benzylpiperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C22H23F3N4O2
7-[(3S)-1-benzylpiperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione —— C22H26N4O3
7-[(3R)-1-[(4-methoxyphenyl)methyl]piperidin-3-yl]-1,3-dimethylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-(1-Benzylpiperidin-4-yl)-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H28N4O3
7-(1-Benzylpiperidin-4-yl)-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-benzyl-4-methyl-2-[(3S)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H24N6O3
7-benzyl-4-methyl-2-[(3S)-1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H29FN4O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C17H19F3N4O4
7-[(2S)-1-(2-methoxyacetyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H26N6O3
7-[(3-methoxyphenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-benzyl-4-methyl-2-[(3R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H29N5O3
7-benzyl-4-methyl-2-[(3R)-1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3S)-1-(2-pyrazol-1-ylacetyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[1-[(4-Chlorophenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H27ClN4O3
7-[1-[(4-Chlorophenyl)methyl]piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-(3-phenylpropyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C22H24F3N5
7-[(3S)-1-(3-phenylpropyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-benzyl-2-[(3S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H27N5O3
7-benzyl-2-[(3S)-1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[1-(Cyclohexanecarbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H32N4O4
7-[1-(Cyclohexanecarbonyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C18H21F3N4O4
7-[(3S)-1-(2-methoxyacetyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(3S)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C24H25FN6O2
7-[(3-fluorophenyl)methyl]-4-methyl-2-[(3R)-1-(1-methylpyrazole-4-carbonyl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H32N4O3
7-[(2-methoxyphenyl)methyl]-4-methyl-2-[(3R)-1-(oxan-4-yl)piperidin-3-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C20H26F3N5
7-[(3S)-1-(cyclohexylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[1-(Cyclohexylmethyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione —— C23H34N4O3
7-[1-(Cyclohexylmethyl)piperidin-4-yl]-1-(2-methoxyethyl)-3-methylpyrido[2,3-d]pyrimidine-2,4-dione
—— 7-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C19H19F3N6
7-[(3S)-1-(pyridin-3-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3S)-1-(quinolin-6-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine —— C23H21F3N6
7-[(3S)-1-(quinolin-6-ylmethyl)piperidin-3-yl]-5-(trifluoromethyl)pyrido[2,3-d]pyrimidin-4-amine
—— 7-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C21H25F3N4O3
7-[(3R)-1-(cyclopentanecarbonyl)piperidin-3-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione
—— 7-benzyl-2-[(3R)-1-(1-ethylpyrazole-3-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C25H28N6O2
7-benzyl-2-[(3R)-1-(1-ethylpyrazole-3-carbonyl)piperidin-3-yl]-4-methyl-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one —— C23H23FN6O2
7-[(4-fluorophenyl)methyl]-4-methyl-2-[(2R)-1-(2-methylpyrazole-3-carbonyl)pyrrolidin-2-yl]-5H-pyrrolo[2,3-d]pyrimidin-6-one
—— 7-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione —— C18H21F3N4O4
7-[(2S)-1-(3-methoxypropanoyl)pyrrolidin-2-yl]-1,3-dimethyl-5-(trifluoromethyl)pyrido[2,3-d]pyrimidine-2,4-dione