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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-[(1-ethyl-5-methylpyrazol-4-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H27N5O
7-[(1-ethyl-5-methylpyrazol-4-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(1-Ethylbenzimidazol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H22N6O
7-[(1-Ethylbenzimidazol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Hydroxy-4-methyl-8-diaethylaminomethyl-3-benzyl-cumarin —— C22H25NO3
7-Hydroxy-4-methyl-8-diaethylaminomethyl-3-benzyl-cumarin
—— (7-Methyl-2-oxochromen-4-yl)methyl 5-bromo-2-hydroxybenzoate —— C18H13BrO5
(7-Methyl-2-oxochromen-4-yl)methyl 5-bromo-2-hydroxybenzoate
—— 7-[(3S)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole —— C18H25N5O2S2
7-[(3S)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole
—— 7-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H30N6O2
7-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3R)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole —— C18H25N5O2S2
7-[(3R)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-3,5-dimethylimidazo[5,1-b][1,3]thiazole
—— 7-acetyl-2-[(2R)-1-(2-ethyl-4,5,6,7-tetrahydroindazole-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-acetyl-2-[(2R)-1-(2-ethyl-4,5,6,7-tetrahydroindazole-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-ethyl-5-methylpyrazol-4-yl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H24N6O
7-[(1-ethyl-5-methylpyrazol-4-yl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3S)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-5-methylimidazo[5,1-b][1,3]thiazole —— C17H23N5O2S2
7-[(3S)-1-(1-ethyl-5-methylpyrazol-4-yl)sulfonylpiperidin-3-yl]-5-methylimidazo[5,1-b][1,3]thiazole
—— 7-[(1-ethyl-5-methylpyrazol-4-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H23N7O
7-[(1-ethyl-5-methylpyrazol-4-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(3-bromophenyl)-5-(4-bromophenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine —— C17H15Br2N5
7-(3-bromophenyl)-5-(4-bromophenyl)-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidin-2-amine
—— 7-acetyl-2-[(2S)-1-(2-ethyl-4,5,6,7-tetrahydroindazole-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-acetyl-2-[(2S)-1-(2-ethyl-4,5,6,7-tetrahydroindazole-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H29N5O
7-[(1-ethyl-3,5-dimethylpyrazol-4-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-bromo-1-(4-chlorophenyl)-2-(4,5-dimethyl-1,3-thiazol-2-yl)-1H-chromeno[2,3-c]pyrrole-3,9-dione —— C22H14BrClN2O3S
7-bromo-1-(4-chlorophenyl)-2-(4,5-dimethyl-1,3-thiazol-2-yl)-1H-chromeno[2,3-c]pyrrole-3,9-dione
—— 7-Ethoxy-1-(4-ethylphenyl)-6-methoxy-1,2,3,4-tetrahydroisoquinoline —— C20H25NO2
7-Ethoxy-1-(4-ethylphenyl)-6-methoxy-1,2,3,4-tetrahydroisoquinoline
—— 7-Bromo-2-[[5-(2-methylfuran-3-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one —— C19H16BrN5O2S
7-Bromo-2-[[5-(2-methylfuran-3-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanylmethyl]pyrido[1,2-a]pyrimidin-4-one
—— 7-[(5-ethylfuran-2-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H26N4O2
7-[(5-ethylfuran-2-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-Chloro-1-(2,5-dimethoxyphenyl)-2-(4-methyl-1,3-thiazol-2-yl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione —— C23H17ClN2O5S
7-Chloro-1-(2,5-dimethoxyphenyl)-2-(4-methyl-1,3-thiazol-2-yl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione
—— 7-[(3R)-1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[(3R)-1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-(2-methoxy-4-methylphenoxy)acetate —— C24H26O6
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-(2-methoxy-4-methylphenoxy)acetate
—— 7-[(7-ethyl-1H-indol-3-yl)methyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H22N4O
7-[(7-ethyl-1H-indol-3-yl)methyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[4-Cyclohexyl-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C26H25N5OS2
7-[[4-Cyclohexyl-5-(naphthalen-1-ylmethyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Methyl-1-[(2-propan-2-yloxyphenyl)methyl]-3,4-dihydro-1,4-benzodiazepine-2,5-dione —— C20H22N2O3
7-Methyl-1-[(2-propan-2-yloxyphenyl)methyl]-3,4-dihydro-1,4-benzodiazepine-2,5-dione
—— 7-[(3S)-1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[(3S)-1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(5-ethyl-2-methylpyrazole-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H23N5O2
7-[1-(5-ethyl-2-methylpyrazole-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-phenylsulfanyl-14H-naphtho[3,2-a]phenothiazine-8,13-dione —— C26H15NO2S2
7-phenylsulfanyl-14H-naphtho[3,2-a]phenothiazine-8,13-dione
—— 7-acetyl-2-[(2R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4
7-acetyl-2-[(2R)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-(3,5-diethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C21H24N4O3
7-[1-(3,5-diethyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(5-ethylthiophene-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H21N3O2S
7-[1-(5-ethylthiophene-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— (7-methyl-2-oxochromen-4-yl)methyl 3-(1H-indol-3-yl)propanoate —— C22H19NO4
(7-methyl-2-oxochromen-4-yl)methyl 3-(1H-indol-3-yl)propanoate
—— 7-[(3R)-1-(3,5-diethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H22N4O3
7-[(3R)-1-(3,5-diethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[(3S)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-acetyl-2-[(2S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4
7-acetyl-2-[(2S)-1-(5-ethyl-3-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C19H20N4O3
7-[(3R)-1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[[5-(4-Chlorophenyl)-4-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C22H16ClN5OS2
7-[[5-(4-Chlorophenyl)-4-(3-methylphenyl)-1,2,4-triazol-3-yl]sulfanylmethyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-Bromo-2-(furan-2-ylmethyl)-1-(4-hydroxyphenyl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione —— C22H14BrNO5
7-Bromo-2-(furan-2-ylmethyl)-1-(4-hydroxyphenyl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione
—— 7-chloro-2-(4-fluorophenyl)-2,3-dihydro-1H-indole —— C14H11ClFN
7-chloro-2-(4-fluorophenyl)-2,3-dihydro-1H-indole
—— 7-cyclopentyl-2-[(2R)-1-(5-ethyl-4-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclopentyl-2-[(2R)-1-(5-ethyl-4-methyl-1H-pyrazole-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4S
7-ethylsulfonyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H28N4O5S
7-ethylsulfonyl-2-[(2R)-1-(3-methoxypropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4S
7-ethylsulfonyl-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H25FN4O4S
7-ethylsulfonyl-2-[(2R)-1-(2-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H28N4O5S
7-ethylsulfonyl-2-[(2S)-1-[(2S)-oxolane-2-carbonyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4S
7-ethylsulfonyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H28N4O4S
7-ethylsulfonyl-2-[(2S)-1-[(1R,2S)-2-methylcyclopropanecarbonyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4S
7-ethylsulfonyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25N5O4S
7-ethylsulfonyl-2-[(2S)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-ethylsulfonyl-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4S
7-ethylsulfonyl-2-[(2R)-1-(3-methylbenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one