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—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N4O3S
7-(cyclopropanecarbonyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-(5-methylfuran-2-yl)quinoline-4-carboxylate —— C29H25NO5
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-(5-methylfuran-2-yl)quinoline-4-carboxylate
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl adamantane-1-carboxylate —— C23H26O4
(7,8-Dimethyl-2-oxochromen-4-yl)methyl adamantane-1-carboxylate
—— 7-[(3R)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C19H16F3N5O2
7-[(3R)-1-(pyrazine-2-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7,8-Dimethyl-4-[(2-oxochromen-7-yl)oxymethyl]chromen-2-one —— C21H16O5
7,8-Dimethyl-4-[(2-oxochromen-7-yl)oxymethyl]chromen-2-one
—— 7-[(3R)-1-[(2S)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H22F3N3O3
7-[(3R)-1-[(2S)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-chloro-N-[3-(furan-2-yl)propyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H25ClN2O4
7-chloro-N-[3-(furan-2-yl)propyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-[(3S)-1-(1,2-oxazole-5-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C18H15F3N4O3
7-[(3S)-1-(1,2-oxazole-5-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C14H14F3N3O
7-[(3S)-piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-(1,2-oxazole-5-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C18H15F3N4O3
7-[(3R)-1-(1,2-oxazole-5-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-1-[2-[(2R)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C21H24F3N3O3
7-[(3S)-1-[2-[(2R)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H17F3N4O2
7-[(3R)-1-(pyridine-4-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-[2-[(2S)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C21H24F3N3O3
7-[(3R)-1-[2-[(2S)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3,4-difluorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H18F2N4O
7-[(3,4-difluorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3R)-1-[(2R)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H22F3N3O3
7-[(3R)-1-[(2R)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-[2-[(2R)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C21H24F3N3O3
7-[(3R)-1-[2-[(2R)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-1-[(2R)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H22F3N3O3
7-[(3S)-1-[(2R)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-1-[2-[(2S)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C21H24F3N3O3
7-[(3S)-1-[2-[(2S)-oxan-2-yl]acetyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(6-Fluoroquinolin-2-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H18FN5O
7-[(6-Fluoroquinolin-2-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-fluorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H19FN4O
7-[(4-fluorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-hydroxy-3-methylbenzoate —— C19H16O6
(7-Methoxy-2-oxochromen-4-yl)methyl 2-hydroxy-3-methylbenzoate
—— 7-[(4-Hydroxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H18N4O2
7-[(4-Hydroxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[1-(4-Fluorophenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H20FN5O
7-[[1-(4-Fluorophenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-fluorophenyl)methyl]-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine —— C23H24FN5O
7-[(4-fluorophenyl)methyl]-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine
—— 7-[(6-Bromo-1,3-benzodioxol-5-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H17BrN4O3
7-[(6-Bromo-1,3-benzodioxol-5-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-3-ylmethyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridin-3-ylmethyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2,3-Dihydro-1,4-dioxin-5-ylmethyl)-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H18N4O3
7-(2,3-Dihydro-1,4-dioxin-5-ylmethyl)-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[(3R)-oxolan-3-yl]methyl]-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine —— C21H27N5O2
7-[[(3R)-oxolan-3-yl]methyl]-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine
—— 7-[(5-Chloro-2-hydroxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H17ClN4O2
7-[(5-Chloro-2-hydroxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-3-ylmethyl)-2-[(3S)-1-(2-thiophen-3-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridin-3-ylmethyl)-2-[(3S)-1-(2-thiophen-3-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(6-Chloro-1,3-benzodioxol-5-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H17ClN4O3
7-[(6-Chloro-1,3-benzodioxol-5-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-3-ylmethyl)-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridin-3-ylmethyl)-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H19ClN6O
7-[[5-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-3-ylmethyl)-2-[(3R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridin-3-ylmethyl)-2-[(3R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-3-ylmethyl)-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H23N5O
7-(pyridin-3-ylmethyl)-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-(1-adamantyl)acetate —— C26H32O4
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-(1-adamantyl)acetate
—— (7-Acetyloxy-11-ethyl-13-methyl-6-methylidene-4-oxo-11-azoniahexacyclo[7.7.2.15,8.01,10.02,8.013,17]nonadecan-16-yl) acetate —— C26H36NO5+
(7-Acetyloxy-11-ethyl-13-methyl-6-methylidene-4-oxo-11-azoniahexacyclo[7.7.2.15,8.01,10.02,8.013,17]nonadecan-16-yl) acetate
—— 7-(1,3-benzodioxol-5-yl)-5-(3,4-dimethoxyphenyl)-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C21H17F3N4O4
7-(1,3-benzodioxol-5-yl)-5-(3,4-dimethoxyphenyl)-2-(trifluoromethyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl 2-(2-chlorophenyl)quinoline-4-carboxylate —— C28H20ClNO4
(7,8-Dimethyl-2-oxochromen-4-yl)methyl 2-(2-chlorophenyl)quinoline-4-carboxylate
—— 7-[2-bromo-4-[(4-chlorophenyl)methoxy]-5-methoxyphenyl]-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one —— C19H16BrClN4O3
7-[2-bromo-4-[(4-chlorophenyl)methoxy]-5-methoxyphenyl]-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one
—— 7-(pyridin-4-ylmethyl)-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine —— C22H24N6O
7-(pyridin-4-ylmethyl)-4-pyridin-3-yloxy-2-pyrrolidin-1-yl-6,8-dihydro-5H-pyrido[3,4-d]pyrimidine
—— 7-[[(1S)-cyclohex-3-en-1-yl]methyl]-2-pyridin-3-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H22N4O
7-[[(1S)-cyclohex-3-en-1-yl]methyl]-2-pyridin-3-yl-1,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H27N5O2
7-(cyclobutanecarbonyl)-2-[(3S)-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-3-carbonyl)-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O3
7-(pyridine-3-carbonyl)-2-[(2S)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclohexylmethyl)-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H31N5O2
7-(cyclohexylmethyl)-2-[(2S)-1-(pyridine-3-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H29N5O2
7-cyclopentyl-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-3-carbonyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O3
7-(pyridine-3-carbonyl)-2-[(2R)-1-(pyridine-4-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-(pyridine-3-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H17F3N4O2
7-[(3R)-1-(pyridine-3-carbonyl)piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-(pyridine-4-carbonyl)-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O3
7-(pyridine-4-carbonyl)-2-[(2S)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H29N5O2
7-cyclopentyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one