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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-Chloro-4'-(3-oxopiperazine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C19H22ClN3O4
7-Chloro-4'-(3-oxopiperazine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-chloro-N-cyclopropyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C18H21ClN2O3
7-chloro-N-cyclopropyl-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-[1-[(3S)-1,1-dioxothiolane-3-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O4S
7-[1-[(3S)-1,1-dioxothiolane-3-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3R)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O3
7-[(3R)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(cyclopropanecarbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C17H19N3O2
7-[1-(cyclopropanecarbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-(trifluoromethyl)-2-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1H-indole —— C16H11F6N
7-(trifluoromethyl)-2-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1H-indole
—— 7-[1-(3,4-difluorophenyl)sulfonylpiperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C19H17F2N3O3S
7-[1-(3,4-difluorophenyl)sulfonylpiperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C21H19F2N3O2
7-[1-[2-(2,5-difluorophenyl)acetyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-[(3R)-1,1-dioxothiolane-3-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O4S
7-[1-[(3R)-1,1-dioxothiolane-3-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-(4-Piperidyl)-1,6-naphthyridin-5-one —— C13H15N3O
7-(4-Piperidyl)-1,6-naphthyridin-5-one
—— 7-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O3
7-[1-[(2S)-oxolane-2-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H17F2N3O2
7-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(pyridine-4-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C19H18N4O2
7-[1-(pyridine-4-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C12H13N3O
7-[(3S)-pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-[2-(difluoromethyl)pyrazole-3-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C18H17F2N5O2
7-[1-[2-(difluoromethyl)pyrazole-3-carbonyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(2,4-Dichlorophenyl)methyl]-8-[2-methoxy-4-[(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]phenoxy]-1,3-dimethylpurine-2,6-dione —— C26H21Cl2N5O5S2
7-[(2,4-Dichlorophenyl)methyl]-8-[2-methoxy-4-[(3-methyl-4-oxo-2-sulfanylidene-1,3-thiazolidin-5-ylidene)methyl]phenoxy]-1,3-dimethylpurine-2,6-dione
—— 7-[1-(2-cyclopentylacetyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H25N3O2
7-[1-(2-cyclopentylacetyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3S)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C18H21N3O3
7-[(3S)-1-(oxane-4-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[1-(oxane-4-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C19H23N3O3
7-[1-(oxane-4-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-(pyridine-4-carbonyl)-2-[(2S)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H23N5O2S
7-(pyridine-4-carbonyl)-2-[(2S)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-4-carbonyl)-2-[(2S)-1-(thiophen-2-ylmethyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridine-4-carbonyl)-2-[(2S)-1-(thiophen-2-ylmethyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-5-oxo-N-(2-thiophen-2-ylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C21H23ClN2O3S
7-chloro-5-oxo-N-(2-thiophen-2-ylethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-cyclopentyl-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O2S
7-cyclopentyl-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H24N4O3S
7-(cyclopropanecarbonyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclopentyl-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-4-carbonyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23N5O3S
7-(pyridine-4-carbonyl)-2-[(2R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N4O3S
7-(cyclobutanecarbonyl)-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-5-oxo-N-(thiophen-2-ylmethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C20H21ClN2O3S
7-chloro-5-oxo-N-(thiophen-2-ylmethyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-[[1-(thiophen-2-ylmethyl)tetrazol-5-yl]methyl]-2-(trifluoromethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine —— C14H14F3N7S
7-[[1-(thiophen-2-ylmethyl)tetrazol-5-yl]methyl]-2-(trifluoromethyl)-6,8-dihydro-5H-imidazo[1,2-a]pyrazine
—— 7-Tert-butyl-5-methyl-1,2,3,4-tetrahydropyrimido[1,6-a]indole —— C16H22N2
7-Tert-butyl-5-methyl-1,2,3,4-tetrahydropyrimido[1,6-a]indole
—— 7-Ethoxy-1-(2-iodophenyl)-6-methoxy-1,2,3,4-tetrahydroisoquinoline —— C18H20INO2
7-Ethoxy-1-(2-iodophenyl)-6-methoxy-1,2,3,4-tetrahydroisoquinoline
—— 7-cyclohexyl-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H32N4O2S
7-cyclohexyl-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-4-carbonyl)-2-[(2R)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H23N5O2S
7-(pyridine-4-carbonyl)-2-[(2R)-1-(thiophen-2-ylmethyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-[(2S)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H22F3N3O3
7-[(3S)-1-[(2S)-oxane-2-carbonyl]piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H24N4O3S
7-(cyclopropanecarbonyl)-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O2S
7-cyclopentyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclopentyl-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(thiophene-2-carbonyl)-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H20N4O3S2
7-(thiophene-2-carbonyl)-2-[(2R)-1-(thiophene-2-carbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridin-4-ylmethyl)-2-[(2R)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25N5O2S
7-(pyridin-4-ylmethyl)-2-[(2R)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N4O3S
7-(cyclopropanecarbonyl)-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclohexyl-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclohexyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H24N4O3S
7-(cyclopropanecarbonyl)-2-[(2R)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C14H14F3N3O
7-[(3R)-piperidin-3-yl]-2-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-chloro-2-(furan-2-ylmethyl)-1-(4-hydroxyphenyl)-1H-chromeno[2,3-c]pyrrole-3,9-dione —— C22H14ClNO5
7-chloro-2-(furan-2-ylmethyl)-1-(4-hydroxyphenyl)-1H-chromeno[2,3-c]pyrrole-3,9-dione
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H26N4O2S
7-(cyclobutanecarbonyl)-2-[(3S)-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(pyridine-4-carbonyl)-2-[(2S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H23N5O3S
7-(pyridine-4-carbonyl)-2-[(2S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N4O3S
7-(cyclobutanecarbonyl)-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H24N4O3S
7-(cyclopropanecarbonyl)-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N4O2S
7-cyclohexyl-2-[(3R)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one