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—— 7-[(3R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-N-(3-fluorophenyl)imidazo[5,1-b][1,3]thiazol-5-amine —— C22H25FN4OS
7-[(3R)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-N-(3-fluorophenyl)imidazo[5,1-b][1,3]thiazol-5-amine
—— 7-Chloro-2-[2-(3,4-dimethoxyphenyl)ethyl]-1-(4-methylphenyl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione —— C28H24ClNO5
7-Chloro-2-[2-(3,4-dimethoxyphenyl)ethyl]-1-(4-methylphenyl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione
—— 7-[1-[(3-fluorophenyl)methyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C20H20FN3O
7-[1-[(3-fluorophenyl)methyl]piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(3-Fluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H16FN5O
7-[(3-Fluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-N-(3-fluorophenyl)imidazo[5,1-b][1,3]thiazol-5-amine —— C22H25FN4OS
7-[(3S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-N-(3-fluorophenyl)imidazo[5,1-b][1,3]thiazol-5-amine
—— 7-[(3-fluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H23FN4O
7-[(3-fluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-Chloro-2-[2-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]-2-oxoethyl]sulfanyl-3-(2-methylpropyl)quinazolin-4-one —— C27H28ClN3O2S
7-Chloro-2-[2-[2,5-dimethyl-1-(4-methylphenyl)pyrrol-3-yl]-2-oxoethyl]sulfanyl-3-(2-methylpropyl)quinazolin-4-one
—— 7-cyclohexyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-cyclohexyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-chloro-4,5-difluorobenzoate —— C18H11ClF2O5
(7-Methoxy-2-oxochromen-4-yl)methyl 2-chloro-4,5-difluorobenzoate
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H29FN4O2
7-cyclopentyl-2-[(2R)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H23FN4O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H25FN4O3
7-(cyclopropanecarbonyl)-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-cyclohexyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H29FN4O2
7-cyclopentyl-2-[(2S)-1-(3-fluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-tert-butyl-2-{4-[3-(3,5-dimethylphenoxy)propoxy]-3-methoxyphenyl}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one —— C32H38N2O4S
7-tert-butyl-2-{4-[3-(3,5-dimethylphenoxy)propoxy]-3-methoxyphenyl}-5,6,7,8-tetrahydro[1]benzothieno[2,3-d]pyrimidin-4(3H)-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H23FN4O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-(3-fluorobenzoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H22F2N4O
7-[(3,4-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(5-Chloro-2-hydroxyphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H17ClN4O2
7-[(5-Chloro-2-hydroxyphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-difluorophenyl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H18F2N4O
7-[(3,4-difluorophenyl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,5-difluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H17F2N5O
7-[(2,5-difluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[[4-Hydroxy-3-(piperidin-1-ylmethyl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H29N5O2
7-[[4-Hydroxy-3-(piperidin-1-ylmethyl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Chloro-2-(5-chlorothien-2-yl)-8-methylquinoline-4-carboxylic acid —— C15H9Cl2NO2S
7-Chloro-2-(5-chlorothien-2-yl)-8-methylquinoline-4-carboxylic acid
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[(3,4-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H26F2N4O2
7-(cyclobutanecarbonyl)-2-[(3S)-1-[(3,4-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-Difluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H15F2N5O
7-[(3,4-Difluorophenyl)methyl]-2-pyrazin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3,4-difluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H17F2N5O
7-[(3,4-difluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-cyclopentyl-2-[(2R)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28F2N4O2
7-cyclopentyl-2-[(2R)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H22F2N4O
7-[(2,5-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,3-difluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H17F2N5O
7-[(2,3-difluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[[4-Hydroxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H27N5O3
7-[[4-Hydroxy-3-(morpholin-4-ylmethyl)phenyl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(2,4-difluorobenzoyl)-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H16F2N4O2
7-(2,4-difluorobenzoyl)-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[(3,4-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H26F2N4O2
7-(cyclobutanecarbonyl)-2-[(3R)-1-[(3,4-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Ethoxy-6-methoxy-1-(2,4,5-trimethoxyphenyl)-1,2,3,4-tetrahydroisoquinoline —— C21H27NO5
7-Ethoxy-6-methoxy-1-(2,4,5-trimethoxyphenyl)-1,2,3,4-tetrahydroisoquinoline
—— 7-cyclopentyl-2-[(2S)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28F2N4O2
7-cyclopentyl-2-[(2S)-1-(3,4-difluorobenzoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,3-difluorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H18F2N4O
7-[(2,3-difluorophenyl)methyl]-2-pyridin-3-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,3-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H22F2N4O
7-[(2,3-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,4-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H22F2N4O
7-[(2,4-difluorophenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2-chloro-6-fluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H17ClFN5O
7-[(2-chloro-6-fluorophenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,3-difluorophenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H22F2N4O2
7-[(2,3-difluorophenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3,4-Dichlorophenyl)methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H22Cl2N4O
7-[(3,4-Dichlorophenyl)methyl]-2-piperidin-1-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[(2,3-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H26F2N4O2
7-(cyclobutanecarbonyl)-2-[(3S)-1-[(2,3-difluorophenyl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-nitrophenyl)methylsulfanyl]-5,6-dihydroimidazo[4,5-d]pyridazine-4-thione —— C12H9N5O2S2
7-[(4-nitrophenyl)methylsulfanyl]-5,6-dihydroimidazo[4,5-d]pyridazine-4-thione
—— 7-Methyl-4-[2-oxo-2-[4-(3-phenylprop-2-enyl)piperazin-1-yl]ethyl]-1,4-benzoxazin-3-one —— C24H27N3O3
7-Methyl-4-[2-oxo-2-[4-(3-phenylprop-2-enyl)piperazin-1-yl]ethyl]-1,4-benzoxazin-3-one
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-chloro-5-piperidin-1-ylsulfonylbenzoate —— C23H22ClNO7S
(7-Methoxy-2-oxochromen-4-yl)methyl 2-chloro-5-piperidin-1-ylsulfonylbenzoate
—— 7-(2-chlorophenyl)-5-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C18H15ClN4
7-(2-chlorophenyl)-5-(4-methylphenyl)-1,7-dihydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[(3S)-1-(1-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C17H17N5O2
7-[(3S)-1-(1-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-(4-formylphenoxy)acetate —— C20H16O7
(7-Methoxy-2-oxochromen-4-yl)methyl 2-(4-formylphenoxy)acetate
—— 7-[(3R)-1-(1-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C17H17N5O2
7-[(3R)-1-(1-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(4-fluorophenyl)methylsulfanyl]-5,6-dihydroimidazo[4,5-d]pyridazine-4-thione —— C12H9FN4S2
7-[(4-fluorophenyl)methylsulfanyl]-5,6-dihydroimidazo[4,5-d]pyridazine-4-thione
—— 7-[(4-methoxyphenyl)methyl]-2-[(3R)-1-(1-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H28N6O3
7-[(4-methoxyphenyl)methyl]-2-[(3R)-1-(1-methylpyrazole-3-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one