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—— (7R)-3-ethyl-2-methyl-6-[(3-methylphenyl)methyl]-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C24H27NS
(7R)-3-ethyl-2-methyl-6-[(3-methylphenyl)methyl]-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7S)-7-(4-methylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-7-(4-methylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-6-[(2-chloro-4-fluorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H23ClFNS
(7R)-6-[(2-chloro-4-fluorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-6-[(2-chloro-6-fluorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H23ClFNS
(7S)-6-[(2-chloro-6-fluorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7S)-N-(2,5-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-N-(2,5-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS2
(7R)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-7-(4-methylphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS2
(7S)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-6-[(3-chlorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24ClNS
(7R)-6-[(3-chlorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7S)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS2
(7S)-7-(4-methylsulfanylphenyl)-N-(2-phenylethyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7S)-7-(4-ethoxyphenyl)-N-[(4-methylphenyl)methyl]-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,4-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(2,4-dimethylphenyl)-7-(3-fluorophenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS2
(7R)-N-[(4-fluorophenyl)methyl]-7-(4-methylsulfanylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-3-ethyl-2-methyl-6-[(3-methylphenyl)methyl]-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C24H27NS
(7S)-3-ethyl-2-methyl-6-[(3-methylphenyl)methyl]-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-N-(2,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-N-(2,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7R)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-6-[(4-chlorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24ClNS
(7R)-6-[(4-chlorophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— 7-methoxy-3-[(3R)-3-methylpiperidin-1-yl]sulfonylchromen-2-one —— C16H19NO5S
7-methoxy-3-[(3R)-3-methylpiperidin-1-yl]sulfonylchromen-2-one
—— (7S)-N-benzyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-N-benzyl-7-(4-ethylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— 7-(4-Methylpiperazin-1-yl)-5-(morpholin-4-yl)-4-nitro-2,1,3-benzoxadiazole —— C15H20N6O4
7-(4-Methylpiperazin-1-yl)-5-(morpholin-4-yl)-4-nitro-2,1,3-benzoxadiazole
—— (7R)-6-[(3-bromophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine —— C23H24BrNS
(7R)-6-[(3-bromophenyl)methyl]-3-ethyl-2-methyl-7-phenyl-5,7-dihydro-4H-thieno[2,3-c]pyridine
—— (7R)-N-(2,5-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7R)-N-(2,5-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C30H31N3OS
(7S)-N-(2,3-dimethylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7R)-N-(3-fluoro-4-methylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C29H28FN3OS
(7R)-N-(3-fluoro-4-methylphenyl)-7-(4-methylphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— (7S)-N-(3,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide —— C31H33N3O2S
(7S)-N-(3,4-dimethylphenyl)-7-(4-ethoxyphenyl)-17-thia-2,8-diazatetracyclo[8.7.0.02,6.011,16]heptadeca-1(10),3,5,11(16)-tetraene-8-carboxamide
—— 7-methoxy-3-[(3S)-3-methylpiperidin-1-yl]sulfonylchromen-2-one —— C16H19NO5S
7-methoxy-3-[(3S)-3-methylpiperidin-1-yl]sulfonylchromen-2-one
—— (7R)-7-tert-butyl-2-[3-[4-(2,4-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C29H38N4O2S
(7R)-7-tert-butyl-2-[3-[4-(2,4-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[3-[4-(4-acetylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H30N4O3S
(7R)-2-[3-[4-(4-acetylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-ethyl-2-methyl-3-phenyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide —— C22H21N5O
7-ethyl-2-methyl-3-phenyl-N-(pyridin-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 3-methylbenzoate —— C22H22O4
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 3-methylbenzoate
—— 7-[(2-Chloro-6-fluorophenyl)methyl]-8-[2-(3,4-dimethoxyphenyl)ethylamino]-1,3-dimethylpurine-2,6-dione —— C24H25ClFN5O4
7-[(2-Chloro-6-fluorophenyl)methyl]-8-[2-(3,4-dimethoxyphenyl)ethylamino]-1,3-dimethylpurine-2,6-dione
—— (7S)-2-[3-[4-(4-acetylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C26H30N4O3S
(7S)-2-[3-[4-(4-acetylphenyl)piperazin-1-yl]-3-oxopropyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-5-(4-chlorophenyl)-7-(4-methylphenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H21ClN4O
(7R)-5-(4-chlorophenyl)-7-(4-methylphenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-7-tert-butyl-2-[3-[4-(2,4-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C29H38N4O2S
(7S)-7-tert-butyl-2-[3-[4-(2,4-dimethylphenyl)piperazin-1-yl]-3-oxopropyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-[[2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-7-oxoheptanoic acid —— C41H53N3O6
7-[[3-[3-[4-[4-(Hydroxymethyl)phenyl]-6-[[2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]methyl]-1,3-dioxan-2-yl]phenyl]phenyl]methylamino]-7-oxoheptanoic acid
—— (7R)-5-(4-bromophenyl)-N-(4-fluorophenyl)-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C25H18BrFN4O
(7R)-5-(4-bromophenyl)-N-(4-fluorophenyl)-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-5-(4-bromophenyl)-7-(4-fluorophenyl)-N-(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20BrFN4O
(7R)-5-(4-bromophenyl)-7-(4-fluorophenyl)-N-(3-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-N-(4-ethoxyphenyl)-7-(2-fluorophenyl)-5-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C28H25FN4O2
(7R)-N-(4-ethoxyphenyl)-7-(2-fluorophenyl)-5-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-5-(4-bromophenyl)-N-(3-methylphenyl)-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H21BrN4O
(7R)-5-(4-bromophenyl)-N-(3-methylphenyl)-7-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-5-(4-chlorophenyl)-N-(4-ethoxyphenyl)-7-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C28H25ClN4O3
(7R)-5-(4-chlorophenyl)-N-(4-ethoxyphenyl)-7-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— 7-(4-chlorophenyl)-8-(2-hydroxyethyl)-1,3-dimethyl-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione —— C17H16ClN5O3
7-(4-chlorophenyl)-8-(2-hydroxyethyl)-1,3-dimethyl-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione
—— (7S)-5-(3-methoxyphenyl)-N-phenyl-7-(2,3,4-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C29H28N4O5
(7S)-5-(3-methoxyphenyl)-N-phenyl-7-(2,3,4-trimethoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-5-(4-bromophenyl)-7-(2-fluorophenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20BrFN4O
(7S)-5-(4-bromophenyl)-7-(2-fluorophenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-N-(4-chlorophenyl)-7-(2-fluorophenyl)-5-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C26H20ClFN4O
(7R)-N-(4-chlorophenyl)-7-(2-fluorophenyl)-5-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-N-(4-chlorophenyl)-5-(4-ethylphenyl)-7-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C28H25ClN4O2
(7R)-N-(4-chlorophenyl)-5-(4-ethylphenyl)-7-(3-methoxyphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(4-bromophenyl)-5-(4-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23BrN4O2
(7R)-7-(4-bromophenyl)-5-(4-methoxyphenyl)-N-(4-methylphenyl)-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7S)-7-(4-chlorophenyl)-5-(4-ethylphenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23ClN4O
(7S)-7-(4-chlorophenyl)-5-(4-ethylphenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (7R)-7-(4-chlorophenyl)-5-(4-ethylphenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C27H23ClN4O
(7R)-7-(4-chlorophenyl)-5-(4-ethylphenyl)-N-phenyl-1,7-dihydropyrazolo[1,5-a]pyrimidine-3-carboxamide