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—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N6O3
7-(cyclopropanecarbonyl)-2-[(2S)-1-(5-methylpyrazine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-methylthiophen-2-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H24N4OS
7-[(3-methylthiophen-2-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N6O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Methoxy-4-[(1-methyltetrazol-5-yl)sulfanylmethyl]chromen-2-one —— C13H12N4O3S
7-Methoxy-4-[(1-methyltetrazol-5-yl)sulfanylmethyl]chromen-2-one
—— 7-[(3-methylthiophen-2-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H20N4OS
7-[(3-methylthiophen-2-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-acetyl-2-[(2S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N6O3
7-acetyl-2-[(2S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O2
7-cyclohexyl-2-[(3S)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-methylthiophen-2-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H19N5OS
7-[(3-methylthiophen-2-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-cyclohexyl-2-[(3R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O2
7-cyclohexyl-2-[(3R)-1-(5-methylpyrazine-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7,8-Dimethyl-2-oxochromen-4-yl)methyl 2-phenoxyacetate —— C20H18O5
(7,8-Dimethyl-2-oxochromen-4-yl)methyl 2-phenoxyacetate
—— 7-acetyl-2-[(2R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N6O3
7-acetyl-2-[(2R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7S)-7-methyl-3-[1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H29N5O2S
(7S)-7-methyl-3-[1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-cyclopentyl-2-[(2S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclopentyl-2-[(2S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7R)-7-methyl-3-[1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H29N5O2S
(7R)-7-methyl-3-[1-[3-(5-methylpyrazol-1-yl)propanoyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-cyclohexyl-2-[(3R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclohexyl-2-[(3R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N6O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclobutanecarbonyl)-2-[(3R)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclobutanecarbonyl)-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-Methyl-2-oxochromen-4-yl)methyl 4-amino-3,5,6-trichloropyridine-2-carboxylate —— C17H11Cl3N2O4
(7-Methyl-2-oxochromen-4-yl)methyl 4-amino-3,5,6-trichloropyridine-2-carboxylate
—— 7-cyclohexyl-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclohexyl-2-[(3S)-1-[3-(5-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[4-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]piperazin-1-yl]methanone —— C24H26N6O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[4-[(S)-(1-methylimidazol-2-yl)-phenylmethyl]piperazin-1-yl]methanone
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone —— C23H23N5OS
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3S)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone
—— 7-methyl-N-[[3-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]imidazo[1,2-a]pyridine-2-carboxamide —— C21H23N3O3
7-methyl-N-[[3-[[(2R)-oxolan-2-yl]methoxy]phenyl]methyl]imidazo[1,2-a]pyridine-2-carboxamide
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone —— C22H20F3N5O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-[5-(trifluoromethyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]piperidin-1-yl]methanone
—— 7-cyclohexyl-2-[(3S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H34N6O2
7-cyclohexyl-2-[(3S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[4-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]piperazin-1-yl]methanone —— C24H26N6O
(7-methylimidazo[1,2-a]pyridin-2-yl)-[4-[(R)-(1-methylimidazol-2-yl)-phenylmethyl]piperazin-1-yl]methanone
—— 7-methoxy-1'-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C22H27N3O4
7-methoxy-1'-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-[3-(3-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-[3-(3-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclobutanecarbonyl)-2-[(3R)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3R)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N6O3
7-(cyclopropanecarbonyl)-2-[(3R)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-[(2S)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H23N5O2
7-[(3S)-1-[(2S)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[[(4-methyl-2-oxo-1H-pyridin-3-yl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one —— C17H15N3O4
7-[[(4-methyl-2-oxo-1H-pyridin-3-yl)amino]methyl]-5H-[1,3]dioxolo[4,5-g]quinolin-6-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclopropanecarbonyl)-2-[(2S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(3S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N6O3
7-(cyclopropanecarbonyl)-2-[(3S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H23N5O2
7-[(3R)-1-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-{[(4-bromo-3-methyl-1H-pyrazol-1-yl)acetyl]amino}-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C16H17BrN8O4S2
7-{[(4-bromo-3-methyl-1H-pyrazol-1-yl)acetyl]amino}-3-{[(1-methyl-1H-tetrazol-5-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 7-(cyclobutanecarbonyl)-2-[(3S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclobutanecarbonyl)-2-[(3S)-1-[3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3S)-1-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C20H23N5O2
7-[(3S)-1-[(2R)-2-methyl-3-(3-methylpyrazol-1-yl)propanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— (7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone —— C23H23N5OS
(7-methylimidazo[1,2-a]pyridin-2-yl)-[(3R)-3-(4-methyl-6-thiophen-2-ylpyrimidin-2-yl)piperidin-1-yl]methanone
—— 7,8-Dimethyl-4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]chromen-2-one —— C15H14N2O2S2
7,8-Dimethyl-4-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanylmethyl]chromen-2-one
—— 7-[[2-(3,3-Dimethyl-2-oxobutylidene)-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-3-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C21H19N3O3S3
7-[[2-(3,3-Dimethyl-2-oxobutylidene)-4-oxo-5-(thiophen-3-ylmethylidene)-1,3-thiazolidin-3-yl]methyl]-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— 7-[3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one —— C20H19FN4O3
7-[3-ethoxy-4-[(4-fluorophenyl)methoxy]phenyl]-6,7-dihydro-1H-[1,2,4]triazolo[1,5-a]pyrimidin-5-one
—— [7-(2-Methylpropanoyloxy)naphthalen-2-yl] 2-methylpropanoate —— C18H20O4
[7-(2-Methylpropanoyloxy)naphthalen-2-yl] 2-methylpropanoate
—— 7-[[3,5-Dimethyl-1-(2-methylphenyl)pyrazol-4-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H26N6O
7-[[3,5-Dimethyl-1-(2-methylphenyl)pyrazol-4-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-fluoro-1-(3-methoxyphenyl)-2-[2-(4-methoxyphenyl)ethyl]-1H,2H,3H,9H-chromeno[2,3-c]pyrrole-3,9-dione —— C27H22FNO5
7-fluoro-1-(3-methoxyphenyl)-2-[2-(4-methoxyphenyl)ethyl]-1H,2H,3H,9H-chromeno[2,3-c]pyrrole-3,9-dione
—— 7-cyclohexyl-2-[(2R)-1-[2-(2-methylphenyl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C27H36N4O2
7-cyclohexyl-2-[(2R)-1-[2-(2-methylphenyl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-{[3-(4-chloro-1H-pyrazol-1-yl)-2-methylpropanoyl]amino}-3-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid —— C18H19ClN6O4S3
7-{[3-(4-chloro-1H-pyrazol-1-yl)-2-methylpropanoyl]amino}-3-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-8-oxo-5-thia-1-azabicyclo[4.2.0]oct-2-ene-2-carboxylic acid
—— 7-bromo-1-(4-bromophenyl)-2-(4,5-dimethyl-1,3-thiazol-2-yl)-1H-chromeno[2,3-c]pyrrole-3,9-dione —— C22H14Br2N2O3S
7-bromo-1-(4-bromophenyl)-2-(4,5-dimethyl-1,3-thiazol-2-yl)-1H-chromeno[2,3-c]pyrrole-3,9-dione
—— 7-Chloro-1-(4-methoxyphenyl)-2-(thiazol-2-yl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione —— C21H13ClN2O4S
7-Chloro-1-(4-methoxyphenyl)-2-(thiazol-2-yl)-1,2-dihydrochromeno[2,3-c]pyrrole-3,9-dione
—— 7-(cyclobutanecarbonyl)-2-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H29N5O2
7-(cyclobutanecarbonyl)-2-[(3R)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one