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—— 7-[(3S)-1-[(2R)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one —— C21H24ClN5O2
7-[(3S)-1-[(2R)-3-(4-chloro-3,5-dimethylpyrazol-1-yl)-2-methylpropanoyl]pyrrolidin-3-yl]-6H-1,6-naphthyridin-5-one
—— 7-[(4-Hydroxy-3-methoxyphenyl)methyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C16H19N3O3
7-[(4-Hydroxy-3-methoxyphenyl)methyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2S)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H23N3O3
7-[(2S)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2R)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H23N3O3
7-[(2R)-3-(1,3-benzodioxol-5-yl)-2-methylpropyl]-2-methyl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7,9-Dibromo-2-(2-naphthyl)-5-(3,4,5-trimethoxyphenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine —— C29H24Br2N2O4
7,9-Dibromo-2-(2-naphthyl)-5-(3,4,5-trimethoxyphenyl)-1,10b-dihydropyrazolo[1,5-c][1,3]benzoxazine
—— 7-[(4-Fluorophenyl)methyl]-8-[[4-(4-methoxyphenyl)piperazin-1-yl]methyl]-1,3-dimethylpurine-2,6-dione —— C26H29FN6O3
7-[(4-Fluorophenyl)methyl]-8-[[4-(4-methoxyphenyl)piperazin-1-yl]methyl]-1,3-dimethylpurine-2,6-dione
—— 7-[(4-Methylpiperazine-1,4-diium-1-yl)-pyridin-2-ylmethyl]quinolin-8-ol —— C20H24N4O+2
7-[(4-Methylpiperazine-1,4-diium-1-yl)-pyridin-2-ylmethyl]quinolin-8-ol
—— 7-{Pyrrolidin-1-yl[4-(trifluoromethyl)phenyl]methyl}quinolin-8-ol —— C21H19F3N2O
7-{Pyrrolidin-1-yl[4-(trifluoromethyl)phenyl]methyl}quinolin-8-ol
—— 7-[(4-Methylpiperazin-1-yl)(pyridin-2-yl)methyl]quinolin-8-ol —— C20H22N4O
7-[(4-Methylpiperazin-1-yl)(pyridin-2-yl)methyl]quinolin-8-ol
—— 7-[(4-Methylpiperazine-1,4-diium-1-yl)-pyridin-1-ium-2-ylmethyl]quinolin-1-ium-8-ol —— C20H26N4O+4
7-[(4-Methylpiperazine-1,4-diium-1-yl)-pyridin-1-ium-2-ylmethyl]quinolin-1-ium-8-ol
—— 7-[[4-(2-Hydroxyethyl)piperazine-1,4-diium-1-yl]-thiophen-2-ylmethyl]quinolin-8-ol —— C20H25N3O2S+2
7-[[4-(2-Hydroxyethyl)piperazine-1,4-diium-1-yl]-thiophen-2-ylmethyl]quinolin-8-ol
—— 7-[Pyrrolidin-1-ium-1-yl-[4-(trifluoromethyl)phenyl]methyl]quinolin-8-ol —— C21H20F3N2O+
7-[Pyrrolidin-1-ium-1-yl-[4-(trifluoromethyl)phenyl]methyl]quinolin-8-ol
—— 7-[Morpholin-4-ium-4-yl(pyridin-3-yl)methyl]quinolin-8-ol —— C19H20N3O2+
7-[Morpholin-4-ium-4-yl(pyridin-3-yl)methyl]quinolin-8-ol
—— 7-(thieno[2,3-d]pyrimidin-4-yloxy)-2H-chromen-2-one —— C15H8N2O3S
7-(thieno[2,3-d]pyrimidin-4-yloxy)-2H-chromen-2-one
—— 7-methylsulfonyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O4S2
7-methylsulfonyl-2-[(3S)-1-(2-thiophen-2-ylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O4S
7-methylsulfonyl-2-[(2R)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(2-pyridin-2-ylsulfanylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H23N5O4S2
7-methylsulfonyl-2-[(2S)-1-(2-pyridin-2-ylsulfanylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O4S2
7-methylsulfonyl-2-[(2S)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclopropanecarbonyl)-2-[(2S)-1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H23N5O4S
7-methylsulfonyl-2-[(2R)-1-(pyridine-3-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N4O4S
7-methylsulfonyl-2-[(2R)-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H26N4O4S
7-methylsulfonyl-2-[(3S)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(3-phenylpropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4S
7-methylsulfonyl-2-[(2R)-1-(3-phenylpropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H24N4O4S2
7-methylsulfonyl-2-[(2R)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(3R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H24N4O5S
7-methylsulfonyl-2-[(3R)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O4S2
7-methylsulfonyl-2-[(2R)-1-(2-thiophen-3-ylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H26N4O4S
7-methylsulfonyl-2-[(3R)-1-(3-phenylpropanoyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(3S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C17H24N4O5S
7-methylsulfonyl-2-[(3S)-1-[(2S)-oxolane-2-carbonyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O4S
7-methylsulfonyl-2-[(2S)-1-(2-phenylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(3S)-1-(2-phenylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H24N4O4S
7-methylsulfonyl-2-[(3S)-1-(2-phenylacetyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H24N4O4S2
7-methylsulfonyl-2-[(2S)-1-(2-thiophen-2-ylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H23N5O4S
7-methylsulfonyl-2-[(2R)-1-(pyridine-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H30N6O3
7-(cyclopropanecarbonyl)-2-[(2R)-1-[2-(3,5-dimethylpyrazol-1-yl)acetyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(2-pyridin-2-ylsulfanylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H23N5O4S2
7-methylsulfonyl-2-[(2R)-1-(2-pyridin-2-ylsulfanylacetyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Chlorophenyl)methyl]-8-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]-1,3-dimethylpurine-2,6-dione —— C25H26Cl2N6O2
7-[(4-Chlorophenyl)methyl]-8-[[4-(3-chlorophenyl)piperazin-1-yl]methyl]-1,3-dimethylpurine-2,6-dione
—— 7-methylsulfonyl-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H22N4O4S2
7-methylsulfonyl-2-[(2S)-1-(thiophene-2-carbonyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H26N4O4S
7-methylsulfonyl-2-[(2S)-1-(1-phenylcyclopropanecarbonyl)pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H26N4O4S
7-methylsulfonyl-2-[(2R)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H26N4O4S
7-methylsulfonyl-2-[(2S)-1-(2-phenylacetyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-(3-phenylpropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O4S
7-methylsulfonyl-2-[(2S)-1-(3-phenylpropanoyl)piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H30N4O5S
7-methylsulfonyl-2-[(2S)-1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H30N4O5S
7-methylsulfonyl-2-[(2R)-1-[3-[(2S)-oxolan-2-yl]propanoyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3R)-1-[(3S)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N6O3
7-acetyl-2-[(3R)-1-[(3S)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-methylsulfonyl-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C18H26N4O5S
7-methylsulfonyl-2-[(2R)-1-[(2S)-oxolane-2-carbonyl]piperidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(5-methylthiophen-3-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H24N4OS
7-[(5-methylthiophen-3-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-acetyl-2-[(3S)-1-[(3R)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N6O3
7-acetyl-2-[(3S)-1-[(3R)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Methoxy-3-methylphenyl)-[(4-methylpyridin-2-yl)amino]methyl]-2-methylquinolin-8-ol —— C25H25N3O2
7-[(4-Methoxy-3-methylphenyl)-[(4-methylpyridin-2-yl)amino]methyl]-2-methylquinolin-8-ol
—— 7-[(2-methoxypyrimidin-5-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H24N6O2
7-[(2-methoxypyrimidin-5-yl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-acetyl-2-[(3S)-1-[(3S)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N6O3
7-acetyl-2-[(3S)-1-[(3S)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3R)-1-[(3R)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H30N6O3
7-acetyl-2-[(3R)-1-[(3R)-3-(3,5-dimethylpyrazol-1-yl)butanoyl]pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one