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中文名称 英文名称 CAS号 化学式 结构式图片
—— 7-methoxy-1'-(1,5,7-trimethylindole-2-carbonyl)spiro[3H-chromene-2,4'-piperidine]-4-one —— C26H28N2O4
7-methoxy-1'-(1,5,7-trimethylindole-2-carbonyl)spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-[(2,5-dimethylthiophen-3-yl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H22N4OS
7-[(2,5-dimethylthiophen-3-yl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-cyano-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]prop-2-enoate —— C28H32N2O4
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 2-cyano-3-[2,5-dimethyl-1-(2-methylpropyl)pyrrol-3-yl]prop-2-enoate
—— 7-[1-(2-imidazol-1-ylacetyl)piperidin-4-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H20F3N5O2
7-[1-(2-imidazol-1-ylacetyl)piperidin-4-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-[(2,5-dimethylthiophen-3-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H21N5OS
7-[(2,5-dimethylthiophen-3-yl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,3-dimethoxyphenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H28N4O3
7-[(2,3-dimethoxyphenyl)methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,5-dimethylthiophen-3-yl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C16H21N3OS
7-[(2,5-dimethylthiophen-3-yl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one —— C20H19F3N4O3
7-[(3S)-1-(3,5-dimethyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]-2-methyl-4-(trifluoromethyl)-6H-1,6-naphthyridin-5-one
—— 7-(difluoromethyl)-5-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H23F2N5O2
7-(difluoromethyl)-5-[(3R)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[(2,5-dimethylthiophen-3-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C18H25N3OS
7-[(2,5-dimethylthiophen-3-yl)methyl]-2-propan-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,5-dimethylthiophen-3-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H22N4OS
7-[(2,5-dimethylthiophen-3-yl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,5-Dimethylthiophen-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C19H20N4OS
7-[(2,5-Dimethylthiophen-3-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,3-dimethoxyphenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C22H24N4O3
7-[(2,3-dimethoxyphenyl)methyl]-2-pyridin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,5-dimethylthiophen-3-yl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H26N4O2S
7-[(2,5-dimethylthiophen-3-yl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(4,5-Dimethoxy-2-methylphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H24N4O3
7-[(4,5-Dimethoxy-2-methylphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-Methoxy-2,5-dimethylphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H25N5O2
7-[(4-Methoxy-2,5-dimethylphenyl)methyl]-2-(5-methylpyrazin-2-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[(2,5-Dimethyl-1-pyridin-2-ylpyrrol-3-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[2-(difluoromethoxy)-3-methoxyphenyl]methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H26F2N4O3
7-[[2-(difluoromethoxy)-3-methoxyphenyl]methyl]-2-pyrrolidin-1-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[[1-(Furan-2-ylmethyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H25N5O2
7-[[1-(Furan-2-ylmethyl)-2,5-dimethylpyrrol-3-yl]methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-(difluoromethyl)-5-[(3S)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine —— C20H23F2N5O2
7-(difluoromethyl)-5-[(3S)-1-[(2,3-dimethoxyphenyl)methyl]piperidin-3-yl]-[1,2,4]triazolo[1,5-a]pyrimidine
—— 7-[(2-fluoro-3-methoxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C20H25FN4O3
7-[(2-fluoro-3-methoxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,6-dimethoxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H28N4O4
7-[(2,6-dimethoxyphenyl)methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2-Hydroxy-3-methoxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H20N4O3
7-[(2-Hydroxy-3-methoxyphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2,5-Dimethyl-1-pyridin-3-ylpyrrol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[(2,5-Dimethyl-1-pyridin-3-ylpyrrol-3-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4,5-Dimethoxy-2-methylphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H24N4O3
7-[(4,5-Dimethoxy-2-methylphenyl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C19H25N3O2
7-[(4-methoxy-2,5-dimethylphenyl)methyl]-2-methyl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2,6-dimethoxyphenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H23N5O3
7-[(2,6-dimethoxyphenyl)methyl]-2-pyrazin-2-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(2-fluoro-3-methoxyphenyl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H21FN4O2
7-[(2-fluoro-3-methoxyphenyl)methyl]-2-pyridin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-[(3,5-Dimethyl-2-pyrazol-1-ylphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H24N6O
7-[(3,5-Dimethyl-2-pyrazol-1-ylphenyl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-[(4,5-Dimethoxy-2-methylphenyl)methyl]piperidin-4-yl]-1,6-naphthyridine —— C23H27N3O2
7-[1-[(4,5-Dimethoxy-2-methylphenyl)methyl]piperidin-4-yl]-1,6-naphthyridine
—— (7-Methoxy-2-oxochromen-4-yl)methyl 3-bromobenzoate —— C18H13BrO5
(7-Methoxy-2-oxochromen-4-yl)methyl 3-bromobenzoate
—— 7-[[1-(3-Methoxyphenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C24H23N5O2
7-[[1-(3-Methoxyphenyl)pyrrol-2-yl]methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[1-(5,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one —— C21H22N4O3
7-[1-(5,6-dimethyl-2-oxo-1H-pyridine-3-carbonyl)piperidin-4-yl]-6H-1,6-naphthyridin-5-one
—— (7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)methyl 3-chloroadamantane-1-carboxylate —— C23H27ClN2O3S
(7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)methyl 3-chloroadamantane-1-carboxylate
—— 7-chloro-2-(3-ethoxyphenyl)-2,3-dihydro-1H-indole —— C16H16ClNO
7-chloro-2-(3-ethoxyphenyl)-2,3-dihydro-1H-indole
—— 7-acetyl-2-[(2R)-1-[(2-hydroxy-3,5-dimethylphenyl)methyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H28N4O3
7-acetyl-2-[(2R)-1-[(2-hydroxy-3,5-dimethylphenyl)methyl]pyrrolidin-2-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[[2-(difluoromethoxy)-3-methoxyphenyl]methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one —— C21H26F2N4O4
7-[[2-(difluoromethoxy)-3-methoxyphenyl]methyl]-2-morpholin-4-yl-5,6,8,9-tetrahydro-3H-pyrimido[4,5-d]azepin-4-one
—— 7-(4-chlorophenyl)-8-(3-ethoxypropyl)-1,3-dimethyl-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione —— C20H22ClN5O3
7-(4-chlorophenyl)-8-(3-ethoxypropyl)-1,3-dimethyl-1H-imidazo[2,1-f]purine-2,4(3H,8H)-dione
—— 7-[(3-methyl-1H-indol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H21N5O
7-[(3-methyl-1H-indol-2-yl)methyl]-2-pyridin-2-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3-methyl-1H-indol-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H21N5O
7-[(3-methyl-1H-indol-2-yl)methyl]-2-pyridin-3-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-acetyl-2-[(3S)-1-(3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H24N4O4
7-acetyl-2-[(3S)-1-(3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-N-(3-methoxyphenyl)imidazo[5,1-b][1,3]thiazol-5-amine —— C21H24N6OS
7-[(3R)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-N-(3-methoxyphenyl)imidazo[5,1-b][1,3]thiazol-5-amine
—— 7'-chloro-2'-(4-fluorophenyl)-1'-(thiophen-2-ylcarbonyl)-1',2'-dihydro-3a'H-spiro[indene-2,3'-pyrrolo[1,2-a]quinoline]-1,3-dione —— C31H19ClFNO3S
7'-chloro-2'-(4-fluorophenyl)-1'-(thiophen-2-ylcarbonyl)-1',2'-dihydro-3a'H-spiro[indene-2,3'-pyrrolo[1,2-a]quinoline]-1,3-dione
—— 7-[(3S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-N-(3-methoxyphenyl)imidazo[5,1-b][1,3]thiazol-5-amine —— C23H28N4O2S
7-[(3S)-1-(3,6-dihydro-2H-pyran-5-ylmethyl)piperidin-3-yl]-N-(3-methoxyphenyl)imidazo[5,1-b][1,3]thiazol-5-amine
—— 7-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-N-(3-methoxyphenyl)imidazo[5,1-b][1,3]thiazol-5-amine —— C21H24N6OS
7-[(3S)-1-(1H-imidazol-2-ylmethyl)piperidin-3-yl]-N-(3-methoxyphenyl)imidazo[5,1-b][1,3]thiazol-5-amine
—— (7-methoxy-3-methyl-1H-indol-2-yl)-[4-[(2-methyl-5-pyridin-3-ylpyrazol-3-yl)methyl]piperazin-1-yl]methanone —— C25H28N6O2
(7-methoxy-3-methyl-1H-indol-2-yl)-[4-[(2-methyl-5-pyridin-3-ylpyrazol-3-yl)methyl]piperazin-1-yl]methanone
—— 7-[(3-methyl-1H-indol-2-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C22H21N5O
7-[(3-methyl-1H-indol-2-yl)methyl]-2-pyridin-4-yl-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-fluoro-N-[(1R)-1-(4-fluorophenyl)-2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]-3-methyl-1-benzofuran-2-carboxamide —— C23H19F2N3O3
7-fluoro-N-[(1R)-1-(4-fluorophenyl)-2-(2-methyl-6-oxo-1H-pyrimidin-4-yl)ethyl]-3-methyl-1-benzofuran-2-carboxamide
—— 7-acetyl-2-[(3R)-1-(3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C23H24N4O4
7-acetyl-2-[(3R)-1-(3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-fluoro-3-methyl-1-benzofuran-2-yl)-[(3S)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone —— C25H24FN5O2
(7-fluoro-3-methyl-1-benzofuran-2-yl)-[(3S)-3-[6-(methylamino)-2-pyridin-4-ylpyrimidin-4-yl]piperidin-1-yl]methanone