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—— 7-methyl-4-[[5-morpholin-4-yl-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one —— C22H26N4O4S
7-methyl-4-[[5-morpholin-4-yl-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanylmethyl]chromen-2-one
—— 7-[(4-cyclopropyl-5-morpholin-4-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one —— C17H20N6O2S2
7-[(4-cyclopropyl-5-morpholin-4-yl-1,2,4-triazol-3-yl)sulfanylmethyl]-3-methyl-[1,3]thiazolo[3,2-a]pyrimidin-5-one
—— (7S)-3-[[5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H18ClN3O2S
(7S)-3-[[5-(4-chlorophenyl)-1,3-oxazol-2-yl]methyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-3-[2-[(3S)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H22N4O3S2
(7S)-3-[2-[(3S)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-3-[2-[(3R)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H22N4O3S2
(7S)-3-[2-[(3R)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-3-[2-[(3S)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C24H22N4O3S2
(7R)-3-[2-[(3S)-3-(furan-2-yl)-5-thiophen-2-yl-3,4-dihydropyrazol-2-yl]-2-oxoethyl]-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methylsulfanyl]-3-(2-fluorophenyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24FN7OS2
(7R)-2-[[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methylsulfanyl]-3-(2-fluorophenyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-2-[[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methylsulfanyl]-3-(2-fluorophenyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H24FN7OS2
(7S)-2-[[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methylsulfanyl]-3-(2-fluorophenyl)-7-methyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-N-[4-[(2,6-dichlorophenyl)sulfonylamino]phenyl]-1,3-benzodioxole-5-carboxamide —— C20H13Cl3N2O5S
7-chloro-N-[4-[(2,6-dichlorophenyl)sulfonylamino]phenyl]-1,3-benzodioxole-5-carboxamide
—— 7-methyl-N-(oxolan-2-ylmethyl)-2-pyridin-3-ylimidazo[1,2-a]pyridin-3-amine —— C18H20N4O
7-methyl-N-(oxolan-2-ylmethyl)-2-pyridin-3-ylimidazo[1,2-a]pyridin-3-amine
—— (7-Methoxy-1-benzofuran-2-yl)-[2-[(1-methylbenzimidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-8-yl]methanone —— C27H30N4O3
(7-Methoxy-1-benzofuran-2-yl)-[2-[(1-methylbenzimidazol-2-yl)methyl]-2,8-diazaspiro[4.5]decan-8-yl]methanone
—— (7-Methoxy-1-benzofuran-2-yl)-[2-[(6-nitro-1,3-benzodioxol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-8-yl]methanone —— C26H27N3O7
(7-Methoxy-1-benzofuran-2-yl)-[2-[(6-nitro-1,3-benzodioxol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-8-yl]methanone
—— (7S)-2-[(1R)-1-[[5-[(4-fluorophenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H21FN4O3S2
(7S)-2-[(1R)-1-[[5-[(4-fluorophenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-2-[(1R)-1-[[5-[(4-fluorophenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H21FN4O3S2
(7R)-2-[(1R)-1-[[5-[(4-fluorophenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2R)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoate —— C22H22N4O4S2
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2R)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoate
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2S)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoate —— C22H22N4O4S2
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl (2S)-2-[(5,6-dimethyl-4-oxo-3H-thieno[2,3-d]pyrimidin-2-yl)methylsulfanyl]propanoate
—— 7-(((5-Methylisoxazol-3-yl)amino)(3-nitrophenyl)methyl)quinolin-8-ol —— C20H16N4O4
7-(((5-Methylisoxazol-3-yl)amino)(3-nitrophenyl)methyl)quinolin-8-ol
—— 7-amino-5-(4-chlorophenyl)-2-methyl-4-oxo-3,5-dihydro-4H-pyrano[2,3-d]pyrimidine-6-carbonitrile —— C15H11ClN4O2
7-amino-5-(4-chlorophenyl)-2-methyl-4-oxo-3,5-dihydro-4H-pyrano[2,3-d]pyrimidine-6-carbonitrile
—— (7S)-2-[(1S)-1-[[5-[(4-fluorophenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H21FN4O3S2
(7S)-2-[(1S)-1-[[5-[(4-fluorophenoxy)methyl]-1,3,4-oxadiazol-2-yl]sulfanyl]ethyl]-7-methyl-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-fluoro-2-methyl-N-[2-(1-phenylpyrazol-4-yl)ethyl]quinoline-3-carboxamide —— C22H19FN4O
7-fluoro-2-methyl-N-[2-(1-phenylpyrazol-4-yl)ethyl]quinoline-3-carboxamide
—— 7-chloro-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one —— C22H20ClN3O3S2
7-chloro-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one
—— 7-chloro-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]-3-[[(2R)-oxolan-2-yl]methyl]quinazolin-4-one —— C22H20ClN3O3S2
7-chloro-2-[(5-methyl-2-thiophen-2-yl-1,3-oxazol-4-yl)methylsulfanyl]-3-[[(2R)-oxolan-2-yl]methyl]quinazolin-4-one
—— 7-Methyl-4-quinolin-8-yloxy-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine —— C20H17N3OS
7-Methyl-4-quinolin-8-yloxy-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidine
—— 7-chloro-3-[[(2R)-oxolan-2-yl]methyl]-2-[(2,3,4,5,6-pentafluorophenyl)methylsulfanyl]quinazolin-4-one —— C20H14ClF5N2O2S
7-chloro-3-[[(2R)-oxolan-2-yl]methyl]-2-[(2,3,4,5,6-pentafluorophenyl)methylsulfanyl]quinazolin-4-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(3,4-dimethylphenyl)sulfonylcyclopentane-1-carboxylate —— C24H26N2O5S
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 1-(3,4-dimethylphenyl)sulfonylcyclopentane-1-carboxylate
—— 7-chloro-3-[[(2S)-oxolan-2-yl]methyl]-2-[(2,3,4,5,6-pentafluorophenyl)methylsulfanyl]quinazolin-4-one —— C20H14ClF5N2O2S
7-chloro-3-[[(2S)-oxolan-2-yl]methyl]-2-[(2,3,4,5,6-pentafluorophenyl)methylsulfanyl]quinazolin-4-one
—— 7-chloro-2-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one —— C21H26ClN3O4S
7-chloro-2-[2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one
—— 7-chloro-2-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one —— C21H26ClN3O4S
7-chloro-2-[2-[(2S,6R)-2,6-dimethylmorpholin-4-yl]-2-oxoethyl]sulfanyl-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2S)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C20H16ClN3O4S
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2S)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— (7-ethyl-2-oxochromen-4-yl)methyl 2-[(2R)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C22H18ClNO5S
(7-ethyl-2-oxochromen-4-yl)methyl 2-[(2R)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— 7-chloro-3-methyl-N-(4-phenoxybutyl)-1-benzofuran-2-carboxamide —— C20H20ClNO3
7-chloro-3-methyl-N-(4-phenoxybutyl)-1-benzofuran-2-carboxamide
—— 7-methyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide —— C15H14N4O
7-methyl-N-(pyridin-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
—— (7-ethyl-2-oxochromen-4-yl)methyl 2-[(2S)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C22H18ClNO5S
(7-ethyl-2-oxochromen-4-yl)methyl 2-[(2S)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— (7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2R)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate —— C20H16ClN3O4S
(7-methyl-4-oxopyrido[1,2-a]pyrimidin-2-yl)methyl 2-[(2R)-6-chloro-3-oxo-4H-1,4-benzothiazin-2-yl]acetate
—— 7-Chloro-3-(oxolan-2-ylmethyl)-2-sulfanyl-3,4-dihydroquinazolin-4-one —— C13H13ClN2O2S
7-Chloro-3-(oxolan-2-ylmethyl)-2-sulfanyl-3,4-dihydroquinazolin-4-one
—— (7S)-7-methyl-2-[(2R)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H29N3O2S2
(7S)-7-methyl-2-[(2R)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(2R)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H29N3O2S2
(7R)-7-methyl-2-[(2R)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-ethyl-2-oxochromen-4-yl)methyl (3S)-1-(phenylcarbamoyl)piperidine-3-carboxylate —— C25H26N2O5
(7-ethyl-2-oxochromen-4-yl)methyl (3S)-1-(phenylcarbamoyl)piperidine-3-carboxylate
—— (7S)-7-methyl-2-[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H29N3O2S2
(7S)-7-methyl-2-[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-2-[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H29N3O2S2
(7R)-7-methyl-2-[(2S)-1-oxo-1-piperidin-1-ylpropan-2-yl]sulfanyl-3-prop-2-enyl-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7-ethyl-2-oxochromen-4-yl)methyl (3R)-1-(phenylcarbamoyl)piperidine-3-carboxylate —— C25H26N2O5
(7-ethyl-2-oxochromen-4-yl)methyl (3R)-1-(phenylcarbamoyl)piperidine-3-carboxylate
—— (7-chloro-3-methyl-1-benzofuran-2-yl)-[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]methanone —— C22H23ClN2O4S
(7-chloro-3-methyl-1-benzofuran-2-yl)-[4-(4-methylphenyl)sulfonyl-1,4-diazepan-1-yl]methanone
—— 7-[(3,4-Dichlorophenyl)methyl]-8-[(2,2-dimethyl-1,3-dioxolan-4-yl)methoxy]-1,3-dimethylpurine-2,6-dione —— C20H22Cl2N4O5
7-[(3,4-Dichlorophenyl)methyl]-8-[(2,2-dimethyl-1,3-dioxolan-4-yl)methoxy]-1,3-dimethylpurine-2,6-dione
—— (7-methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl (3S)-1,1-dioxothiolane-3-carboxylate —— C19H22O6S
(7-methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl (3S)-1,1-dioxothiolane-3-carboxylate
—— 7-fluoro-2-methyl-N-[4-(2,2,2-trifluoroethoxy)phenyl]quinoline-3-carboxamide —— C19H14F4N2O2
7-fluoro-2-methyl-N-[4-(2,2,2-trifluoroethoxy)phenyl]quinoline-3-carboxamide
—— 7-[2-[(2-Acetyl-4-chlorophenoxy)methyl]morpholine-4-carbonyl]-3-methyl-2-methylsulfanylquinazolin-4-one —— C24H24ClN3O5S
7-[2-[(2-Acetyl-4-chlorophenoxy)methyl]morpholine-4-carbonyl]-3-methyl-2-methylsulfanylquinazolin-4-one
—— 7-chloro-2-[[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methylsulfanyl]-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one —— C24H22ClN3O4S
7-chloro-2-[[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methylsulfanyl]-3-[[(2S)-oxolan-2-yl]methyl]quinazolin-4-one
—— (7R)-7-methyl-2-[(1S)-1-[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22N6OS3
(7R)-7-methyl-2-[(1S)-1-[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-2-[(1S)-1-[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C20H22N6OS3
(7S)-7-methyl-2-[(1S)-1-[1-(2-thiophen-2-ylethyl)tetrazol-5-yl]sulfanylethyl]-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— [7-methyl-2-(3-nitrophenyl)-1,3-dioxo-1,2,3,3a,7,7a-hexahydro-4H-4,7-epoxyisoindol-4-yl]methanediyl diacetate —— C20H18N2O9
[7-methyl-2-(3-nitrophenyl)-1,3-dioxo-1,2,3,3a,7,7a-hexahydro-4H-4,7-epoxyisoindol-4-yl]methanediyl diacetate