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—— (7R)-7-methyl-3-[1-(1-propan-2-ylpyrazole-4-carbonyl)piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H29N5O2S
(7R)-7-methyl-3-[1-(1-propan-2-ylpyrazole-4-carbonyl)piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[(5-chloro-2-hydroxyphenyl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25ClN4O3
7-[(5-chloro-2-hydroxyphenyl)methyl]-2-[(2R,6R)-2,6-dimethylmorpholin-4-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7R)-7-methyl-3-[1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S
(7R)-7-methyl-3-[1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[(3-Hydroxy-4-methoxyphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O3
7-[(3-Hydroxy-4-methoxyphenyl)methyl]-2-(4-methylpiperidin-1-yl)-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7S)-7-methyl-3-[1-[2-(2-oxoimidazolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H27N5O3S
(7S)-7-methyl-3-[1-[2-(2-oxoimidazolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-[(1,3-dimethyl-1H-benzimidazol-3-ium-2-yl)methyl]-6-nitro-7H-[1,2,4]triazolo[1,5-a]pyrimidin-4-ide —— C15H15N7O2
7-[(1,3-dimethyl-1H-benzimidazol-3-ium-2-yl)methyl]-6-nitro-7H-[1,2,4]triazolo[1,5-a]pyrimidin-4-ide
—— (7S)-7-methyl-3-[1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S
(7S)-7-methyl-3-[1-[2-(2-oxopyrrolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-3-[1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C23H30N4O3S
(7R)-7-methyl-3-[1-[3-(2-oxopyrrolidin-1-yl)propanoyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-chloro-4'-[(2S,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2S,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— (7R)-7-methyl-3-[1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S
(7R)-7-methyl-3-[1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7R)-7-methyl-3-[1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S
(7R)-7-methyl-3-[1-[(3S)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-(furan-2-yl)-5-thiophen-2-yl-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine —— C13H12N4OS
7-(furan-2-yl)-5-thiophen-2-yl-1,5,6,7-tetrahydro-[1,2,4]triazolo[1,5-a]pyrimidine
—— (7R)-7-methyl-3-[1-[2-(2-oxoimidazolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C21H27N5O3S
(7R)-7-methyl-3-[1-[2-(2-oxoimidazolidin-1-yl)acetyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— (7S)-7-methyl-3-[1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one —— C22H28N4O3S
(7S)-7-methyl-3-[1-[(3R)-1-methyl-5-oxopyrrolidine-3-carbonyl]piperidin-4-yl]-5,6,7,8-tetrahydro-[1]benzothiolo[2,3-d]pyrimidin-4-one
—— 7-methoxy-1'-[(6R)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one —— C24H27NO4S
7-methoxy-1'-[(6R)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl]spiro[3H-chromene-2,4'-piperidine]-4-one
—— 7-[2-(4-Methylpiperidin-1-yl)-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one —— C22H26N6O2
7-[2-(4-Methylpiperidin-1-yl)-2-oxoethyl]-5-phenyl-4,5,7,9,13-pentazatricyclo[7.4.0.02,6]trideca-1(13),2(6),3-trien-8-one
—— 7-chloro-4'-[(2R,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2R,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-[(2-chlorophenyl)methyl]-6-imino-11-methyl-2-oxo-N-(1-phenylethyl)-1,7,9-triazatricyclo[8.4.0.0^{3,8}]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide —— C28H24ClN5O2
7-[(2-chlorophenyl)methyl]-6-imino-11-methyl-2-oxo-N-(1-phenylethyl)-1,7,9-triazatricyclo[8.4.0.0^{3,8}]tetradeca-3(8),4,9,11,13-pentaene-5-carboxamide
—— 7-[(2-hydroxyphenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H26N4O2
7-[(2-hydroxyphenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-fluorophenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25FN4O
7-[(2-fluorophenyl)methyl]-2-[(2R)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H27ClN2O4
7-chloro-4-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-[(2-fluorophenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25FN4O
7-[(2-fluorophenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-Chloro-4'-(4-methylpiperidine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-Chloro-4'-(4-methylpiperidine-1-carbonyl)spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— (7-methyl-2-oxochromen-4-yl)methyl 3-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)benzoate —— C27H23NO6S
(7-methyl-2-oxochromen-4-yl)methyl 3-(3,4-dihydro-1H-isoquinolin-2-ylsulfonyl)benzoate
—— 7-[(2-fluorophenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25FN4O
7-[(2-fluorophenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-4'-[(2S,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2S,3R)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-chloro-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one —— C21H27ClN2O4
7-chloro-4-[2-[(3S)-3-methylpiperidin-1-yl]-2-oxoethyl]spiro[3H-1,4-benzoxazepine-2,4'-oxane]-5-one
—— 7-[(2-methoxyphenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O2
7-[(2-methoxyphenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-hydroxyphenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H26N4O2
7-[(2-hydroxyphenyl)methyl]-2-[(3S)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— (7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 5-chloro-2-hydroxybenzoate —— C21H19ClO5
(7-Methyl-2-oxo-6-propan-2-ylchromen-4-yl)methyl 5-chloro-2-hydroxybenzoate
—— (7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)methyl 4-formylbenzoate —— C20H18N2O4S
(7-methyl-4-oxo-5,6,7,8-tetrahydro-3H-[1]benzothiolo[2,3-d]pyrimidin-2-yl)methyl 4-formylbenzoate
—— 7-[(2-hydroxyphenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H26N4O2
7-[(2-hydroxyphenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(2-fluorophenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H25FN4O
7-[(2-fluorophenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-N-[(1R,2R)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H29ClN2O3
7-chloro-N-[(1R,2R)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-[(2-hydroxyphenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C20H26N4O2
7-[(2-hydroxyphenyl)methyl]-2-[(3R)-3-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-4'-[(2R,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C22H29ClN2O3
7-chloro-4'-[(2R,3S)-2,3-dimethylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-8-oxo-9-propan-2-yl-2-thiophen-2-ylpurine-6-carboxamide —— C21H26N6O3S
7-[2-[(3R)-3-methylpiperidin-1-yl]-2-oxoethyl]-8-oxo-9-propan-2-yl-2-thiophen-2-ylpurine-6-carboxamide
—— 7-[(1R,2R)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one —— C16H23N3O2
7-[(1R,2R)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one
—— 7-chloro-4'-[(2S)-2-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one —— C21H27ClN2O3
7-chloro-4'-[(2S)-2-methylpiperidine-1-carbonyl]spiro[3,4-dihydro-1,4-benzoxazepine-2,1'-cyclohexane]-5-one
—— 7-[(2-methoxyphenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C21H28N4O2
7-[(2-methoxyphenyl)methyl]-2-[(2S)-2-methylpiperidin-1-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-N-(4-methylcyclohexyl)-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H29ClN2O3
7-chloro-N-(4-methylcyclohexyl)-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-(2-fluorobenzoyl)-2-[(3S)-1-(4-methylcyclohexyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-(2-fluorobenzoyl)-2-[(3S)-1-(4-methylcyclohexyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-chloro-N-[(1S,2R)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide —— C22H29ClN2O3
7-chloro-N-[(1S,2R)-2-methylcyclohexyl]-5-oxospiro[3,4-dihydro-1,4-benzoxazepine-2,4'-cyclohexane]-1'-carboxamide
—— 7-[(1R,2S)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one —— C16H23N3O2
7-[(1R,2S)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one
—— 7-[(1S,2S)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one —— C16H23N3O2
7-[(1S,2S)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one
—— 7-(2-fluorobenzoyl)-2-[(3R)-1-(4-methylcyclohexyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one —— C25H31FN4O2
7-(2-fluorobenzoyl)-2-[(3R)-1-(4-methylcyclohexyl)pyrrolidin-3-yl]-3,5,6,8-tetrahydropyrido[3,4-d]pyrimidin-4-one
—— 7-[(1S,2R)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one —— C16H23N3O2
7-[(1S,2R)-2-methylcyclopropanecarbonyl]-2-propan-2-yl-5,6,8,9-tetrahydro-1H-pyrimido[4,5-d]azepin-4-one
—— 7,9-Dichloro-5-methyl-1,2,3,4-tetrahydropyrimido[1,6-a]indole —— C12H12Cl2N2
7,9-Dichloro-5-methyl-1,2,3,4-tetrahydropyrimido[1,6-a]indole
—— (7-Methyl-2-oxochromen-4-yl)methyl 2-(1,3-dioxoisoindol-2-yl)-3-methylbutanoate —— C24H21NO6
(7-Methyl-2-oxochromen-4-yl)methyl 2-(1,3-dioxoisoindol-2-yl)-3-methylbutanoate
—— (7-Methoxy-2-oxochromen-4-yl)methyl 2-ethyl-3-methylquinoline-4-carboxylate —— C24H21NO5
(7-Methoxy-2-oxochromen-4-yl)methyl 2-ethyl-3-methylquinoline-4-carboxylate