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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S,4R,6S,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-2-(1,3-thiazol-4-yl)quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C34H39N5O7S2
(1S,4R,6S,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-2-(1,3-thiazol-4-yl)quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— 1-Azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one;ethane —— C13H17NO
1-Azatricyclo[6.3.1.04,12]dodeca-4,6,8(12)-trien-2-one;ethane
—— N-cyclopropylsulfonyl-17-[[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxymethyl]-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C39H49N5O7S2
N-cyclopropylsulfonyl-17-[[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxymethyl]-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— cyclopropanesulfonic acid [(1R,4R,6S,15R,17R)-17-(2-isopropylamino-quinazolin-4-yloxy)-13-methyl-2,14-dioxo-3,13-diaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carbonyl]-amide —— C32H42N6O6S
cyclopropanesulfonic acid [(1R,4R,6S,15R,17R)-17-(2-isopropylamino-quinazolin-4-yloxy)-13-methyl-2,14-dioxo-3,13-diaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carbonyl]-amide
—— [(9R,12S,13R,14S,16S,17R)-20-hydroxy-13,14,17-trimethoxy-4,8,10,12,16-pentamethyl-3,22-dioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,19-pentaen-9-yl] carbamate —— C30H44N2O8
[(9R,12S,13R,14S,16S,17R)-20-hydroxy-13,14,17-trimethoxy-4,8,10,12,16-pentamethyl-3,22-dioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,19-pentaen-9-yl] carbamate
—— [(4E)-19-(cyclopropylmethylideneamino)-13,20,22-trihydroxy-4,8,10,12,16-pentamethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C31H43N3O6
[(4E)-19-(cyclopropylmethylideneamino)-13,20,22-trihydroxy-4,8,10,12,16-pentamethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— Azacyclohexadecane-2,8,11,14-tetrone —— C15H23NO4
Azacyclohexadecane-2,8,11,14-tetrone
—— tert-butyl 4-[[4-[[(8S,9S,12S,13R,14S)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-19-yl]carbamoyl]phenyl]methyl]piperazine-1-carboxylate —— C45H61N5O11
tert-butyl 4-[[4-[[(8S,9S,12S,13R,14S)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-19-yl]carbamoyl]phenyl]methyl]piperazine-1-carboxylate
—— 2,2-Dimethyl-1-azatricyclo[6.4.1.04,13]trideca-4(13),5,7-triene-9,12-dione;ethane —— C16H21NO2
2,2-Dimethyl-1-azatricyclo[6.4.1.04,13]trideca-4(13),5,7-triene-9,12-dione;ethane
—— benzyl (1R,7S,9S)-3-oxo-2,5-diazatricyclo[7.5.0.02,7]tetradecane-5-carboxylate;ethane —— C22H32N2O3
benzyl (1R,7S,9S)-3-oxo-2,5-diazatricyclo[7.5.0.02,7]tetradecane-5-carboxylate;ethane
—— cyclopropanesulfonic acid [(1S,4R,6S,18R)-18-[2-(4-fluoro-phenyl)-7-methoxy-8-methyl-quinazolin-4-yloxy]-14-(4-methoxy-benzyl)-2,15-dioxo-3,14,16-triaza-tricyclo[14.3.0.0(4,6)]nonadec-7-ene-4-carboyl]-amide —— C44H49FN6O8S
cyclopropanesulfonic acid [(1S,4R,6S,18R)-18-[2-(4-fluoro-phenyl)-7-methoxy-8-methyl-quinazolin-4-yloxy]-14-(4-methoxy-benzyl)-2,15-dioxo-3,14,16-triaza-tricyclo[14.3.0.0(4,6)]nonadec-7-ene-4-carboyl]-amide
—— methyl (2S)-2-[[(E,2R,3R)-3-(3-hydroxypropyl)-6-methyl-2-(2-methylpropyl)hept-4-enoyl]amino]heptanoate;methyl (8S,11R,12R)-12-[(E)-3-methylbut-1-enyl]-11-(2-methylpropyl)-2,10-dioxo-1-oxa-3,9-diazacyclopentadecane-8-carboxylate —— C46H83N3O9
methyl (2S)-2-[[(E,2R,3R)-3-(3-hydroxypropyl)-6-methyl-2-(2-methylpropyl)hept-4-enoyl]amino]heptanoate;methyl (8S,11R,12R)-12-[(E)-3-methylbut-1-enyl]-11-(2-methylpropyl)-2,10-dioxo-1-oxa-3,9-diazacyclopentadecane-8-carboxylate
—— ethyl (1R,4R,6S,15R,17R)-17-(6-methoxy-2-phenylpyrimidin-4-yl)oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C31H38N4O6
ethyl (1R,4R,6S,15R,17R)-17-(6-methoxy-2-phenylpyrimidin-4-yl)oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— [19-[[(2-tert-butyl-5-methyl-1H-pyrazol-3-ylidene)-hydroxymethyl]amino]-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18-hexaen-9-yl] carbamate —— C37H51N5O9
[19-[[(2-tert-butyl-5-methyl-1H-pyrazol-3-ylidene)-hydroxymethyl]amino]-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18-hexaen-9-yl] carbamate
—— (1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C46H57F3N6O8S2
(1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (1R,4R,6S,7Z,15R,17R)-17-[(2-ethoxy-8,9-dihydrofuro[2,3-h]quinolin-4-yl)oxy]-13-methyl-2,14-dioxo-13-azatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C32H38N2O7
(1R,4R,6S,7Z,15R,17R)-17-[(2-ethoxy-8,9-dihydrofuro[2,3-h]quinolin-4-yl)oxy]-13-methyl-2,14-dioxo-13-azatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— Ethane;5-methyl-3,10-diazapentacyclo[10.7.1.02,10.04,9.016,20]icosa-1(19),2,4,6,8,12,14,16(20),17-nonaen-11-one —— C23H24N2O
Ethane;5-methyl-3,10-diazapentacyclo[10.7.1.02,10.04,9.016,20]icosa-1(19),2,4,6,8,12,14,16(20),17-nonaen-11-one
—— (2R)-7-[cyclopropylsulfonyl(hydroxy)methyl]-4,17-dimethyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione —— C33H34N4O7S
(2R)-7-[cyclopropylsulfonyl(hydroxy)methyl]-4,17-dimethyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione
—— [(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] 4-(4-fluorophenyl)piperazine-1-carboxylate —— C50H61FN4O13
[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] 4-(4-fluorophenyl)piperazine-1-carboxylate
—— [(1S,4R,6S,14S)-4-(cyclopropylsulfamoylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C26H41N5O7S
[(1S,4R,6S,14S)-4-(cyclopropylsulfamoylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— Amino 19-[3-[4-[3-[(9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl)imino]propyl]piperazin-1-yl]propylideneamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaene-9-carboxylate —— C66H96N8O16
Amino 19-[3-[4-[3-[(9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl)imino]propyl]piperazin-1-yl]propylideneamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaene-9-carboxylate
—— 5-Acetyl-6-(2,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one;ethane —— C27H34Cl2N2O2
5-Acetyl-6-(2,4-dichlorophenyl)-9,9-dimethyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one;ethane
—— 4-[(5S)-5-[(5R,6S,7S)-6-amino-7-methoxy-3,5-dimethyl-14-oxo-1-azacyclotetradeca-3,8,12-trien-2-yl]-4-oxohexyl]piperidine-2,6-dione —— C27H41N3O5
4-[(5S)-5-[(5R,6S,7S)-6-amino-7-methoxy-3,5-dimethyl-14-oxo-1-azacyclotetradeca-3,8,12-trien-2-yl]-4-oxohexyl]piperidine-2,6-dione
—— (2R)-5-hydroxy-N-[2-[(18S,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]-2-methylpentanamide —— C53H55N13O9S6
(2R)-5-hydroxy-N-[2-[(18S,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]-2-methylpentanamide
—— Ethane;2-oxaspiro[4.5]decan-1-one —— C11H20O2
Ethane;2-oxaspiro[4.5]decan-1-one
—— ethane;(17S)-17-propyl-15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaene —— C19H25N3O
ethane;(17S)-17-propyl-15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaene
—— [(1S,4R,6S,14S)-4-[(4-cyanophenyl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C30H39N5O7S
[(1S,4R,6S,14S)-4-[(4-cyanophenyl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— 14-Methoxy-7-methyl-12-oxa-3,7,18,20,22,24-hexazapentacyclo[17.6.1.13,5.113,17.023,26]octacosa-14,17,19(26),21-tetraen-25-one —— C23H34N6O3
14-Methoxy-7-methyl-12-oxa-3,7,18,20,22,24-hexazapentacyclo[17.6.1.13,5.113,17.023,26]octacosa-14,17,19(26),21-tetraen-25-one
—— 10-Hydroxy-11,19-dimethyl-1-azacycloicosa-3,5,7,13,15,17-hexaen-2-one —— C21H29NO2
10-Hydroxy-11,19-dimethyl-1-azacycloicosa-3,5,7,13,15,17-hexaen-2-one
—— Ethane;1-methoxy-2,6-dimethyl-1,5-dihydro-[1,2,4]triazino[4,3-a][1,4]benzodiazepin-7-one —— C18H28N4O2
Ethane;1-methoxy-2,6-dimethyl-1,5-dihydro-[1,2,4]triazino[4,3-a][1,4]benzodiazepin-7-one
—— (13R)-13-benzyl-7-methoxy-15-methyl-9-oxa-3,12,15,18,20,22,24-heptazatetracyclo[17.6.1.14,8.023,26]heptacosa-1,4(27),5,7,19(26),20,22-heptaene-11,25-dione 1093797-17-1 C28H31N7O4
(13R)-13-benzyl-7-methoxy-15-methyl-9-oxa-3,12,15,18,20,22,24-heptazatetracyclo[17.6.1.14,8.023,26]heptacosa-1,4(27),5,7,19(26),20,22-heptaene-11,25-dione
—— 14-methyl-9-oxa-3,14,17,19,21,23-hexazatetracyclo[16.6.1.14,8.022,25]hexacosa-1,4(26),5,7,18(25),19,21-heptaene-13,24-dione 1093795-88-0 C20H22N6O3
14-methyl-9-oxa-3,14,17,19,21,23-hexazatetracyclo[16.6.1.14,8.022,25]hexacosa-1,4(26),5,7,18(25),19,21-heptaene-13,24-dione
—— [(8S,9S,12S,13R,14S,16R)-19-[2-[2-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]ethyl-methylamino]ethylideneamino]-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C61H87N7O18
[(8S,9S,12S,13R,14S,16R)-19-[2-[2-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]ethyl-methylamino]ethylideneamino]-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— (1S,4R,6S,14R,18R)-18-(8-chloro-7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-N-cyclopropylsulfonyl-14-[2-(3,3-difluoropiperidin-1-yl)-2-oxoethyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C43H49ClF2N6O8S
(1S,4R,6S,14R,18R)-18-(8-chloro-7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-N-cyclopropylsulfonyl-14-[2-(3,3-difluoropiperidin-1-yl)-2-oxoethyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (1R,4R,6S,7Z,15R,17R)-17-(8-chloro-2-ethoxyquinolin-4-yl)oxy-13-methyl-2,14-dioxo-13-azatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C30H35ClN2O6
(1R,4R,6S,7Z,15R,17R)-17-(8-chloro-2-ethoxyquinolin-4-yl)oxy-13-methyl-2,14-dioxo-13-azatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— 3-[[(6aS)-2-methyl-11-oxo-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxy]-N-methylpropanamide;ethane —— C19H27N3O3
3-[[(6aS)-2-methyl-11-oxo-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxy]-N-methylpropanamide;ethane
—— (11S,12S)-8-[tert-butyl(dimethyl)silyl]oxy-1,11-dimethyl-12-penta-2,4-dien-2-yl-1-azacyclododec-9-en-2-one —— C24H43NO2Si
(11S,12S)-8-[tert-butyl(dimethyl)silyl]oxy-1,11-dimethyl-12-penta-2,4-dien-2-yl-1-azacyclododec-9-en-2-one
—— [(1R,4R,6S,15R,17S)-13-methyl-4-[(1-methylcyclopropyl)sulfonylcarbamoyl]-2,14-dioxo-3-azatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-[3-(methylcarbamoyl)phenyl]carbamate —— C32H42N4O8S
[(1R,4R,6S,15R,17S)-13-methyl-4-[(1-methylcyclopropyl)sulfonylcarbamoyl]-2,14-dioxo-3-azatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-[3-(methylcarbamoyl)phenyl]carbamate
—— (8S)-10,15-dimethyl-7-morpholin-4-yl-3,10,15,19,21,23,25-heptazatetracyclo[18.6.1.14,8.024,27]octacosa-1,3,6,19,21,24(27)-hexaene-14,26-dione —— C27H38N8O3
(8S)-10,15-dimethyl-7-morpholin-4-yl-3,10,15,19,21,23,25-heptazatetracyclo[18.6.1.14,8.024,27]octacosa-1,3,6,19,21,24(27)-hexaene-14,26-dione
—— Ethane;8,16,24,32-tetramethyl-2,10,18-trioxa-26-azapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(32),4,6,8,12,14,16,20,22,24,28,30-dodecaene-3,11,19,27-tetrone —— C40H49NO7
Ethane;8,16,24,32-tetramethyl-2,10,18-trioxa-26-azapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(32),4,6,8,12,14,16,20,22,24,28,30-dodecaene-3,11,19,27-tetrone
—— (1S,4R,6S,18R)-N-cyclopropylsulfonyl-18-(2-methoxy-6-phenylpyrimidin-4-yl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C31H38N6O7S
(1S,4R,6S,18R)-N-cyclopropylsulfonyl-18-(2-methoxy-6-phenylpyrimidin-4-yl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[7-methoxy-8-methyl-2-(6-methylpyridin-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C38H45N5O7S
(1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[7-methoxy-8-methyl-2-(6-methylpyridin-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— Ethane;8,16,24,32-tetramethyl-2-oxa-10,18,26-triazapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(32),4,6,8,12,14,16,20,22,24,28,30-dodecaene-3,11,19,27-tetrone —— C40H51N3O5
Ethane;8,16,24,32-tetramethyl-2-oxa-10,18,26-triazapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(32),4,6,8,12,14,16,20,22,24,28,30-dodecaene-3,11,19,27-tetrone
—— (2R,17S)-7-(difluoromethoxy)-2-[(6-fluoro-3-hydroxy-2H-isoindol-5-yl)amino]-4,17,19-trimethyl-4,11-diazatricyclo[16.2.2.16,10]tricosa-1(20),6,8,10(23),18,21-hexaene-3,12-dione —— C33H35F3N4O4
(2R,17S)-7-(difluoromethoxy)-2-[(6-fluoro-3-hydroxy-2H-isoindol-5-yl)amino]-4,17,19-trimethyl-4,11-diazatricyclo[16.2.2.16,10]tricosa-1(20),6,8,10(23),18,21-hexaene-3,12-dione
—— (2S)-N-[(3R,6R,7S,10S)-7-[(3,5-difluorophenyl)methyl]-6-hydroxy-9-oxo-3-phenyl-1-oxa-4,8-diazacyclotetradec-12-en-10-yl]-N,2-dimethylhexanamide —— C32H43F2N3O4
(2S)-N-[(3R,6R,7S,10S)-7-[(3,5-difluorophenyl)methyl]-6-hydroxy-9-oxo-3-phenyl-1-oxa-4,8-diazacyclotetradec-12-en-10-yl]-N,2-dimethylhexanamide
—— ethyl (4R,6S,15S,17S)-17-[8-chloro-7-methoxy-2-(4-methyl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-1,3,13-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C33H38ClN5O6S
ethyl (4R,6S,15S,17S)-17-[8-chloro-7-methoxy-2-(4-methyl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-1,3,13-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— 22-Chloro-28-[4-[(22-chloro-27-cyclohexyl-10-methyl-7,9,9,16-tetraoxo-9lambda6-thia-1,8,10,15-tetrazapentacyclo[15.8.1.12,6.13,25.019,24]octacosa-2,4,6(28),17,19(24),20,22,25(27)-octaen-15-yl)methyl]cyclohexyl]-10,16-dimethyl-9,9-dioxo-13-oxa-9lambda6-thia-1,8,10,16-tetrazapentacyclo[16.8.1.12,6.13,26.020,25]nonacosa-2,4,6(29),18,21,23,26(28)-heptaene-7,17-dione —— C62H70Cl2N8O9S2
22-Chloro-28-[4-[(22-chloro-27-cyclohexyl-10-methyl-7,9,9,16-tetraoxo-9lambda6-thia-1,8,10,15-tetrazapentacyclo[15.8.1.12,6.13,25.019,24]octacosa-2,4,6(28),17,19(24),20,22,25(27)-octaen-15-yl)methyl]cyclohexyl]-10,16-dimethyl-9,9-dioxo-13-oxa-9lambda6-thia-1,8,10,16-tetrazapentacyclo[16.8.1.12,6.13,26.020,25]nonacosa-2,4,6(29),18,21,23,26(28)-heptaene-7,17-dione
—— (4S,7R,8S,9S,13R,14R,16S)-4,8,13,14-tetrahydroxy-5,5,7,9,13-pentamethyl-16-[2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-azacyclohexadecane-2,6-dione —— C26H42N2O6S
(4S,7R,8S,9S,13R,14R,16S)-4,8,13,14-tetrahydroxy-5,5,7,9,13-pentamethyl-16-[2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-azacyclohexadecane-2,6-dione
—— (1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-[2-(propan-2-ylamino)-1,3-thiazol-4-yl]quinolin-4-yl]oxy-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C46H58F3N7O8S2
(1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-[2-(propan-2-ylamino)-1,3-thiazol-4-yl]quinolin-4-yl]oxy-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— cyclopropanesulfonic acid [(1S,4R,6S,18R)-14-(4-methoxy-benzyl)-18-(7-methoxy-8-methyl-2-phenyl-quinazolin-4-yloxy)-2,15-dioxo-3,14,16-triaza-tricyclo[14.3.0.0(4,6)]nonadec-7-ene-4-carbonyl]-amide —— C44H50N6O8S
cyclopropanesulfonic acid [(1S,4R,6S,18R)-14-(4-methoxy-benzyl)-18-(7-methoxy-8-methyl-2-phenyl-quinazolin-4-yloxy)-2,15-dioxo-3,14,16-triaza-tricyclo[14.3.0.0(4,6)]nonadec-7-ene-4-carbonyl]-amide