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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— 4-[[2-[(18S,25R,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]amino]-4-oxobut-2-enoic acid —— C51H47N13O10S6
4-[[2-[(18S,25R,35S)-35-[(S)-hydroxy(phenyl)methyl]-28-(methoxymethyl)-21-methyl-18-[2-(methylamino)-2-oxoethyl]-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,6(11),7,9,12(42),14,19(41),21,26(40),28,36(39)-tridecaen-8-yl]-1,3-thiazol-4-yl]amino]-4-oxobut-2-enoic acid
—— [(8R,10R,13S,14R,15S)-14,21,23-trihydroxy-8,15,20-trimethoxy-4,11,13,17-tetramethyl-3-oxo-2-azabicyclo[17.3.1]tricosa-1(22),4,6,11,17,19(23),20-heptaen-10-yl] carbamate —— C30H42N2O9
[(8R,10R,13S,14R,15S)-14,21,23-trihydroxy-8,15,20-trimethoxy-4,11,13,17-tetramethyl-3-oxo-2-azabicyclo[17.3.1]tricosa-1(22),4,6,11,17,19(23),20-heptaen-10-yl] carbamate
—— N-(aminomethyl)-3-(1,3-dioxobenzo[de]isoquinolin-2-yl)-N-methylbenzamide;ethane;N-ethyl-N-methylacetamide —— C28H34N4O4
N-(aminomethyl)-3-(1,3-dioxobenzo[de]isoquinolin-2-yl)-N-methylbenzamide;ethane;N-ethyl-N-methylacetamide
—— (3S,7S,10R,11R,12S)-10-but-3-enyl-3-(1-chloro-2-pyridin-2-ylethenyl)-7,11-dihydroxy-8,8,12,16-tetramethyl-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C30H43ClN2O5
(3S,7S,10R,11R,12S)-10-but-3-enyl-3-(1-chloro-2-pyridin-2-ylethenyl)-7,11-dihydroxy-8,8,12,16-tetramethyl-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— (1S,4R,6S,18S)-18 [6-(4-Methylthiazol-2-yl)-2-(4-trifluoromethylthiazol-2-yl)-pyrimidin-4-yloxy]-13-N-methyl-2,14-dioxo-3,13,15-triazatricyclo[13.4.0.0*4,6*]nonadec-7-ene-4-carboxylic acid —— C30H32F3N7O5S2
(1S,4R,6S,18S)-18 [6-(4-Methylthiazol-2-yl)-2-(4-trifluoromethylthiazol-2-yl)-pyrimidin-4-yloxy]-13-N-methyl-2,14-dioxo-3,13,15-triazatricyclo[13.4.0.0*4,6*]nonadec-7-ene-4-carboxylic acid
—— (1S,4S,6S,14R,18S)-14-[(2-methylpropan-2-yl)oxycarbonylamino]-2,15-dioxo-18-[5-[(4-phenylphenyl)methyl]tetrazol-2-yl]-16-azatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid —— C38H46N6O6
(1S,4S,6S,14R,18S)-14-[(2-methylpropan-2-yl)oxycarbonylamino]-2,15-dioxo-18-[5-[(4-phenylphenyl)methyl]tetrazol-2-yl]-16-azatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid
—— (1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-[7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid —— C41H47N5O7S
(1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-[7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid
—— Ethane;8,16,24,32-tetramethoxy-2,10,18,26-tetrazapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(28),4(9),5,7,12(17),13,15,20(25),21,23,29,31-dodecaene-3,11,19,27-tetrone —— C40H52N4O8
Ethane;8,16,24,32-tetramethoxy-2,10,18,26-tetrazapentacyclo[26.4.0.04,9.012,17.020,25]dotriaconta-1(28),4(9),5,7,12(17),13,15,20(25),21,23,29,31-dodecaene-3,11,19,27-tetrone
—— [(1S,7Z)-4-[2-(3,4-dimethylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate;[(1S,7Z)-4-[2-(4-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate —— C87H110F2N6O14
[(1S,7Z)-4-[2-(3,4-dimethylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate;[(1S,7Z)-4-[2-(4-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate
—— 4,5-Dimethyl-6,9-dithia-3-azatetracyclo[8.8.0.03,7.012,17]octadeca-1(18),10,12,14,16-pentaene-2,8-dione;ethane —— C19H21NO2S2
4,5-Dimethyl-6,9-dithia-3-azatetracyclo[8.8.0.03,7.012,17]octadeca-1(18),10,12,14,16-pentaene-2,8-dione;ethane
—— (21-Bromo-20,22-dihydroxy-8,13,14,17-tetramethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,6,10,16,18,20-heptaen-9-yl) carbamate —— C30H41BrN2O9
(21-Bromo-20,22-dihydroxy-8,13,14,17-tetramethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,6,10,16,18,20-heptaen-9-yl) carbamate
—— 1-[[3-(7-tert-butyl-2-methoxy-12,12-dimethyl-6,9-dioxo-10-oxa-5,8-diazatetracyclo[21.2.2.12,5.017,22]octacosa-1(26),17,19,21,23(27),24-hexaen-4-yl)oxiran-2-yl]amino]-2-cyclopropyl-N-cyclopropylsulfonylcyclopropane-1-carboxamide —— C44H60N4O8S
1-[[3-(7-tert-butyl-2-methoxy-12,12-dimethyl-6,9-dioxo-10-oxa-5,8-diazatetracyclo[21.2.2.12,5.017,22]octacosa-1(26),17,19,21,23(27),24-hexaen-4-yl)oxiran-2-yl]amino]-2-cyclopropyl-N-cyclopropylsulfonylcyclopropane-1-carboxamide
—— 7-Methoxy-17-methyl-14-propan-2-yl-9-oxa-3,14,17,19,21,23-hexazatetracyclo[16.6.1.14,8.022,25]hexacosa-2,5,7,18,20,22(25)-hexaene-13,24-dione —— C24H32N6O4
7-Methoxy-17-methyl-14-propan-2-yl-9-oxa-3,14,17,19,21,23-hexazatetracyclo[16.6.1.14,8.022,25]hexacosa-2,5,7,18,20,22(25)-hexaene-13,24-dione
—— 6-Chloro-18-fluoro-9,11,13,23,37-pentazapentacyclo[25.5.3.14,8.110,14.115,19]octatriaconta-4(38),5,7,10,12,14(37),15(36),16,18,27(35)-decaen-24-one —— C33H39ClFN5O
6-Chloro-18-fluoro-9,11,13,23,37-pentazapentacyclo[25.5.3.14,8.110,14.115,19]octatriaconta-4(38),5,7,10,12,14(37),15(36),16,18,27(35)-decaen-24-one
—— [(9E,19E,21Z,26Z)-26-[[[(2E)-3,7-dimethylocta-2,6-dienoxy]amino]methylidene]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23,27-trioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25(29)-heptaen-13-yl] acetate —— C48H64N2O13
[(9E,19E,21Z,26Z)-26-[[[(2E)-3,7-dimethylocta-2,6-dienoxy]amino]methylidene]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23,27-trioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25(29)-heptaen-13-yl] acetate
—— (1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-(2-methoxy-6-phenylpyrimidin-4-yl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid —— C36H41N5O7
(1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-(2-methoxy-6-phenylpyrimidin-4-yl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid
—— [(16Z,18Z)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] 2-[acetyl(methyl)amino]propanoate —— C34H46ClN3O10
[(16Z,18Z)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] 2-[acetyl(methyl)amino]propanoate
—— (1S,4R,6S,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-2-(1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C34H39N5O7S2
(1S,4R,6S,18R)-N-cyclopropylsulfonyl-18-[7-methoxy-2-(1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (1R,4R,6S,15R,17R)-17-(6-methoxy-2-phenylpyrimidin-4-yl)oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C33H41N5O7S
(1R,4R,6S,15R,17R)-17-(6-methoxy-2-phenylpyrimidin-4-yl)oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— [(1S,4R,6S,14S)-2,15-dioxo-4-(2-phenylethylsulfonylcarbamoyl)-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C31H44N4O7S
[(1S,4R,6S,14S)-2,15-dioxo-4-(2-phenylethylsulfonylcarbamoyl)-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— [(1R,4R,6S,15R,17R)-4-(cyclopropylsulfonylcarbamoyl)-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-(3-methylphenyl)carbamate —— C29H38N4O7S
[(1R,4R,6S,15R,17R)-4-(cyclopropylsulfonylcarbamoyl)-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-(3-methylphenyl)carbamate
—— 2-[(1E,4E)-hepta-1,4-dienyl]-1,5,9-triazacyclotridecan-4-one —— C17H31N3O
2-[(1E,4E)-hepta-1,4-dienyl]-1,5,9-triazacyclotridecan-4-one
—— [(8S,9S,12S,13R,14S)-19-amino-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C28H39N3O8
[(8S,9S,12S,13R,14S)-19-amino-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— (7R,8S,9S,16S)-8-hydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-2,6-dioxo-1-azacyclohexadec-13-ene-4-carbonitrile —— C28H41N3O3S
(7R,8S,9S,16S)-8-hydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-2,6-dioxo-1-azacyclohexadec-13-ene-4-carbonitrile
—— 39-[6-(2,5-Dihydroxypyrrol-1-yl)oxy-6-oxohexyl]-15,39-dimethyl-21,26-dioxo-8-(3-sulfopropyl)-22,25,32-triaza-8-azoniapentacyclo[30.7.0.07,15.09,14.033,38]nonatriaconta-1,3,5,7,9(14),10,12,33(38),34,36-decaene-12,36-disulfonic acid —— C50H66N5O15S3+
39-[6-(2,5-Dihydroxypyrrol-1-yl)oxy-6-oxohexyl]-15,39-dimethyl-21,26-dioxo-8-(3-sulfopropyl)-22,25,32-triaza-8-azoniapentacyclo[30.7.0.07,15.09,14.033,38]nonatriaconta-1,3,5,7,9(14),10,12,33(38),34,36-decaene-12,36-disulfonic acid
—— [(8S,9S,12S,13R,14S,16R)-20-chloro-13,19,21-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate —— C28H41ClN2O8
[(8S,9S,12S,13R,14S,16R)-20-chloro-13,19,21-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate
—— [(8S,9S,12S,13R,14S,16R)-13,21-dihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C28H40N2O7
[(8S,9S,12S,13R,14S,16R)-13,21-dihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— 2-[[5-[Benzyl-[[[6-(hydroxycarbamoyl)-7-(2-methylpropyl)-8-oxo-2-oxa-9-azabicyclo[10.2.2]hexadeca-1(14),12,15-triene-10-carbonyl]amino]methyl]carbamoyl]pyridin-2-yl]-diazenylmethyl]benzenesulfonic acid —— C41H47N7O9S
2-[[5-[Benzyl-[[[6-(hydroxycarbamoyl)-7-(2-methylpropyl)-8-oxo-2-oxa-9-azabicyclo[10.2.2]hexadeca-1(14),12,15-triene-10-carbonyl]amino]methyl]carbamoyl]pyridin-2-yl]-diazenylmethyl]benzenesulfonic acid
—— (3S,7S,10R,11R,12S)-3-(1-chloro-2-pyridin-2-ylethenyl)-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(oxiran-2-ylmethyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C29H41ClN2O6
(3S,7S,10R,11R,12S)-3-(1-chloro-2-pyridin-2-ylethenyl)-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(oxiran-2-ylmethyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— [(8S,9S,12S,13R,14S,16R)-19-(2,3-dihydroxypropylamino)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C31H47N3O10
[(8S,9S,12S,13R,14S,16R)-19-(2,3-dihydroxypropylamino)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— ethyl N-[(8S,9S,12S,13R,14S)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-19-yl]carbamate —— C31H43N3O10
ethyl N-[(8S,9S,12S,13R,14S)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-19-yl]carbamate
—— (9S,10S,11R)-10-hydroxy-9-methoxy-11,13-dimethyl-1-azacyclotetradeca-7,12-dien-2-one —— C16H27NO3
(9S,10S,11R)-10-hydroxy-9-methoxy-11,13-dimethyl-1-azacyclotetradeca-7,12-dien-2-one
—— (1R,4R,6S,15R,17R)-17-[2-methoxy-6-(3-methoxyphenyl)pyrimidin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C34H43N5O8S
(1R,4R,6S,15R,17R)-17-[2-methoxy-6-(3-methoxyphenyl)pyrimidin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— 1-[2-[(22Z)-2,15-dihydroxy-11-methoxy-3,7,12,13,14,16,23,34-octamethyl-1'-(2-methylpropyl)-6,24,33-trioxospiro[8,18,35-trioxa-25,28,30-triazahexacyclo[24.6.1.14,7.117,19.05,32.027,31]pentatriaconta-1(32),2,4,9,20,22,26,30-octaene-29,4'-piperidine]-19-yl]-2-oxoethyl]-3-[4-(2-ethyl-3-oxobutyl)phenyl]urea —— C61H80N6O12
1-[2-[(22Z)-2,15-dihydroxy-11-methoxy-3,7,12,13,14,16,23,34-octamethyl-1'-(2-methylpropyl)-6,24,33-trioxospiro[8,18,35-trioxa-25,28,30-triazahexacyclo[24.6.1.14,7.117,19.05,32.027,31]pentatriaconta-1(32),2,4,9,20,22,26,30-octaene-29,4'-piperidine]-19-yl]-2-oxoethyl]-3-[4-(2-ethyl-3-oxobutyl)phenyl]urea
—— (1R,4R,6S,7Z,15R,17R)-17-(8-bromo-2-ethoxy-7-methoxyquinolin-4-yl)oxy-13-methyl-2,14-dioxo-13-azatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C31H37BrN2O7
(1R,4R,6S,7Z,15R,17R)-17-(8-bromo-2-ethoxy-7-methoxyquinolin-4-yl)oxy-13-methyl-2,14-dioxo-13-azatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— (10S,13S)-13-[(1S)-2-chloro-1-hydroxyethyl]-9,10-dimethyl-2-oxa-9,12-diazabicyclo[13.3.1]nonadeca-1(18),4,15(19),16-tetraene-8,11-dione —— C20H27ClN2O4
(10S,13S)-13-[(1S)-2-chloro-1-hydroxyethyl]-9,10-dimethyl-2-oxa-9,12-diazabicyclo[13.3.1]nonadeca-1(18),4,15(19),16-tetraene-8,11-dione
—— ethane;(1R,7R,9S)-5-methyl-2,5-diazatricyclo[7.5.0.02,7]tetradecan-3-one —— C15H28N2O
ethane;(1R,7R,9S)-5-methyl-2,5-diazatricyclo[7.5.0.02,7]tetradecan-3-one
—— (1R,7S,11S,15S,17R)-11-hydroxy-7-[(1S)-1-hydroxy-3-[(2S)-4-methyl-3,6-dihydro-2H-pyran-2-yl]prop-2-enyl]-15-methyl-13-methylidene-21-oxa-6-azabicyclo[15.3.1]henicosa-3,9,19-trien-5-one —— C30H43NO5
(1R,7S,11S,15S,17R)-11-hydroxy-7-[(1S)-1-hydroxy-3-[(2S)-4-methyl-3,6-dihydro-2H-pyran-2-yl]prop-2-enyl]-15-methyl-13-methylidene-21-oxa-6-azabicyclo[15.3.1]henicosa-3,9,19-trien-5-one
—— (1S,4R,6S,17R)-17-(7-methoxy-6-methyl-2-phenyl-quinazolin-4-yloxy)-13-methyl-2,14-dioxo-3,13,15-triaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carboxylic acid —— C33H37N5O6
(1S,4R,6S,17R)-17-(7-methoxy-6-methyl-2-phenyl-quinazolin-4-yloxy)-13-methyl-2,14-dioxo-3,13,15-triaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carboxylic acid
—— (1R,4R,6S,15R,17R)-17-(6-methoxy-3-pyrazol-1-ylisoquinolin-1-yl)oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C31H35N5O6
(1R,4R,6S,15R,17R)-17-(6-methoxy-3-pyrazol-1-ylisoquinolin-1-yl)oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— (4R,6S,7Z,15S,17S)-17-[8-chloro-2-(4-ethenyl-1,3-thiazol-2-yl)-7-methoxyquinolin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-1,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C37H42ClN5O7S2
(4R,6S,7Z,15S,17S)-17-[8-chloro-2-(4-ethenyl-1,3-thiazol-2-yl)-7-methoxyquinolin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-1,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— 1-Oxa-6-azacyclopentadecan-5-one —— C13H25NO2
1-Oxa-6-azacyclopentadecan-5-one
—— (1S,4R,6S,14R,18R)-18-(8-chloro-7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-N-cyclopropylsulfonyl-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C44H50ClF3N6O8S
(1S,4R,6S,14R,18R)-18-(8-chloro-7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-N-cyclopropylsulfonyl-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— 24-Tert-butyl-27-[4-cyclopropyl-2-(2-ethenylcyclopropyl)-4-hydroxybutanoyl]-7-methoxy-18-methyl-2,21-dioxa-4,11,23,26-tetrazapentacyclo[24.2.1.03,12.05,10.018,20]nonacosa-3,5(10),6,8,11-pentaene-22,25-dione —— C41H56N4O7
24-Tert-butyl-27-[4-cyclopropyl-2-(2-ethenylcyclopropyl)-4-hydroxybutanoyl]-7-methoxy-18-methyl-2,21-dioxa-4,11,23,26-tetrazapentacyclo[24.2.1.03,12.05,10.018,20]nonacosa-3,5(10),6,8,11-pentaene-22,25-dione
—— 1,3-dimethyl-3,3a-dihydro-1H-[1,3]thiazolo[4,3-c][1,4]benzothiazepine-4,10-dione;ethane —— C15H19NO2S2
1,3-dimethyl-3,3a-dihydro-1H-[1,3]thiazolo[4,3-c][1,4]benzothiazepine-4,10-dione;ethane
—— [(9S,12S,13R,14S,16R)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C31H43N3O8
[(9S,12S,13R,14S,16R)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— (1S,4R,6S,18R)-18-(6-methoxy-3-pyrazol-1-ylisoquinolin-1-yl)oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid —— C31H35N5O6
(1S,4R,6S,18R)-18-(6-methoxy-3-pyrazol-1-ylisoquinolin-1-yl)oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid
—— 2,6-Bis[4-(dimethylamino)phenyl]-14-(trifluoromethylperoxysulfanyl)-17-(trifluoromethylsulfonyl)-11,20-dioxa-14,17-diazatricyclo[19.2.2.27,10]heptacosa-1(24),2,5,7,9,21(25),22,26-octaene-15,16-dione —— C41H40F6N4O8S2
2,6-Bis[4-(dimethylamino)phenyl]-14-(trifluoromethylperoxysulfanyl)-17-(trifluoromethylsulfonyl)-11,20-dioxa-14,17-diazatricyclo[19.2.2.27,10]heptacosa-1(24),2,5,7,9,21(25),22,26-octaene-15,16-dione
—— 22-[(2-Acetamidoacetyl)amino]-1-ethyl-5-[(2-fluorophenyl)methyl]-9-hydroxy-3,6,12,19,23-pentaoxo-1,4,7,10,13,18-hexazacyclotricosane-14-carboxamide —— C31H46FN9O9
22-[(2-Acetamidoacetyl)amino]-1-ethyl-5-[(2-fluorophenyl)methyl]-9-hydroxy-3,6,12,19,23-pentaoxo-1,4,7,10,13,18-hexazacyclotricosane-14-carboxamide
—— (4S,7R,8S,9S,16S)-4,8-dihydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-oxazol-4-yl)prop-1-en-2-yl]-1-azacyclohexadeca-11,13-diene-2,6-dione —— C27H40N2O5
(4S,7R,8S,9S,16S)-4,8-dihydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-oxazol-4-yl)prop-1-en-2-yl]-1-azacyclohexadeca-11,13-diene-2,6-dione