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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(8S,9S,12S,13R,14S,16R)-13-hydroxy-8,14,20-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate —— C29H44N2O7
[(8S,9S,12S,13R,14S,16R)-13-hydroxy-8,14,20-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate
—— (5S)-20-methoxy-18-(methoxymethoxy)-7,7,13-trimethyl-6,8-dioxa-15-azatricyclo[15.4.0.05,9]henicosa-1(17),2,12,18,20-pentaene-10,16-dione —— C24H31NO7
(5S)-20-methoxy-18-(methoxymethoxy)-7,7,13-trimethyl-6,8-dioxa-15-azatricyclo[15.4.0.05,9]henicosa-1(17),2,12,18,20-pentaene-10,16-dione
—— [(1S,4R,6S,14S)-4-[(4-methylphenyl)sulfamoylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C30H43N5O7S
[(1S,4R,6S,14S)-4-[(4-methylphenyl)sulfamoylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— [(1S,3S,5S,6S,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-(methylamino)propanoate —— C32H44ClN3O9
[(1S,3S,5S,6S,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-(methylamino)propanoate
—— 1,4-Dioxaspiro[4.5]decan-8-one;ethane —— C10H18O3
1,4-Dioxaspiro[4.5]decan-8-one;ethane
—— [(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13-hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-20-yl] N-methyl-N-[3-(methylamino)propyl]carbamate —— C35H56N4O9
[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13-hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-20-yl] N-methyl-N-[3-(methylamino)propyl]carbamate
—— (10S,14S,18S)-14-hydroxy-18-[(1S)-1-hydroxy-3-[(2S)-4-methyl-3,6-dihydro-2H-pyran-2-yl]prop-2-enyl]-10-methyl-12-methylidene-1-oxa-7-azacyclooctadec-15-ene-2,8-dione —— C27H41NO6
(10S,14S,18S)-14-hydroxy-18-[(1S)-1-hydroxy-3-[(2S)-4-methyl-3,6-dihydro-2H-pyran-2-yl]prop-2-enyl]-10-methyl-12-methylidene-1-oxa-7-azacyclooctadec-15-ene-2,8-dione
—— 2,15,30-trihydroxy-11,13-dimethoxy-27-[[[4-(2-methoxyethyl)piperazin-1-yl]amino]methylidene]-3,7,12,14,16,19,23,31-octamethyl-8,18,32-trioxa-25-azapentacyclo[24.3.1.14,7.117,19.05,29]dotriaconta-1(29),2,4,9,20,22,26(30)-heptaene-6,24,28-trione —— C46H64N4O12
2,15,30-trihydroxy-11,13-dimethoxy-27-[[[4-(2-methoxyethyl)piperazin-1-yl]amino]methylidene]-3,7,12,14,16,19,23,31-octamethyl-8,18,32-trioxa-25-azapentacyclo[24.3.1.14,7.117,19.05,29]dotriaconta-1(29),2,4,9,20,22,26(30)-heptaene-6,24,28-trione
—— (5S,9R,13R,14S)-10-hydroxy-20-methoxy-18-(methoxymethoxy)-7,7,13,14-tetramethyl-6,8,15-trioxa-2-azatricyclo[15.4.0.05,9]henicosa-1(17),11,18,20-tetraene-3,16-dione —— C24H33NO9
(5S,9R,13R,14S)-10-hydroxy-20-methoxy-18-(methoxymethoxy)-7,7,13,14-tetramethyl-6,8,15-trioxa-2-azatricyclo[15.4.0.05,9]henicosa-1(17),11,18,20-tetraene-3,16-dione
—— [4-[(4-Acetyl-5-oxohexanoyl)amino]phenyl] 2,15,17-trihydroxy-11-methoxy-3,7,12,13,14,16,18,22-octamethyl-1'-(2-methylpropyl)-6,23,32-trioxospiro[8,33-dioxa-24,27,29-triazapentacyclo[23.6.1.14,7.05,31.026,30]tritriaconta-1(31),2,4,9,19,21,25,29-octaene-28,4'-piperidine]-27-carboxylate —— C60H77N5O14
[4-[(4-Acetyl-5-oxohexanoyl)amino]phenyl] 2,15,17-trihydroxy-11-methoxy-3,7,12,13,14,16,18,22-octamethyl-1'-(2-methylpropyl)-6,23,32-trioxospiro[8,33-dioxa-24,27,29-triazapentacyclo[23.6.1.14,7.05,31.026,30]tritriaconta-1(31),2,4,9,19,21,25,29-octaene-28,4'-piperidine]-27-carboxylate
—— (1S,5S,6S,7R,10S,14S,16S)-1-chloro-14-[1-fluoro-2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-6,10-dihydroxy-5,7,9,9-tetramethyl-3,17-dioxa-13-azabicyclo[14.1.0]heptadecane-8,12-dione —— C24H34ClFN2O6S
(1S,5S,6S,7R,10S,14S,16S)-1-chloro-14-[1-fluoro-2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-6,10-dihydroxy-5,7,9,9-tetramethyl-3,17-dioxa-13-azabicyclo[14.1.0]heptadecane-8,12-dione
—— [(1S,4R,6S,14S)-2,15-dioxo-4-(propan-2-ylsulfonylcarbamoyl)-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C26H42N4O7S
[(1S,4R,6S,14S)-2,15-dioxo-4-(propan-2-ylsulfonylcarbamoyl)-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— (1R,13R,15S,16R,17S)-16,17-dimethoxy-15-phenylsulfanyl-2,14-dioxa-11-azabicyclo[11.4.0]heptadec-6-en-10-one —— C22H31NO5S
(1R,13R,15S,16R,17S)-16,17-dimethoxy-15-phenylsulfanyl-2,14-dioxa-11-azabicyclo[11.4.0]heptadec-6-en-10-one
—— N-[(4R,5S,8S)-5-benzyl-4-hydroxy-18-methoxy-7-oxo-2,6,13-triazatricyclo[12.6.1.015,20]henicosa-1,16,18-trien-8-yl]-N-methylpentane-1-sulfonamide —— C32H48N4O5S
N-[(4R,5S,8S)-5-benzyl-4-hydroxy-18-methoxy-7-oxo-2,6,13-triazatricyclo[12.6.1.015,20]henicosa-1,16,18-trien-8-yl]-N-methylpentane-1-sulfonamide
—— [(8R,10R,13S,14R,15S,17R)-20-(2,3-dihydroxypropylamino)-14,21,23-trihydroxy-8,15-dimethoxy-4,11,13,17-tetramethyl-3-oxo-2-azabicyclo[17.3.1]tricosa-1(22),4,6,11,19(23),20-hexaen-10-yl] carbamate —— C32H49N3O10
[(8R,10R,13S,14R,15S,17R)-20-(2,3-dihydroxypropylamino)-14,21,23-trihydroxy-8,15-dimethoxy-4,11,13,17-tetramethyl-3-oxo-2-azabicyclo[17.3.1]tricosa-1(22),4,6,11,19(23),20-hexaen-10-yl] carbamate
—— Ethane;4-methyl-1,2,3a,4-tetrahydro-[1,3]thiazolo[2,3-c][1,4]benzothiazepin-10-one —— C14H19NOS2
Ethane;4-methyl-1,2,3a,4-tetrahydro-[1,3]thiazolo[2,3-c][1,4]benzothiazepin-10-one
—— (1R,4R,6S,17R)-N-cyclopropylsulfonyl-17-[2-(4-fluorophenyl)-7-methoxy-8-methylquinazolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C37H42FN5O7S
(1R,4R,6S,17R)-N-cyclopropylsulfonyl-17-[2-(4-fluorophenyl)-7-methoxy-8-methylquinazolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— (2S)-N-[(4R,5S,8S,14R)-5-benzyl-4-hydroxy-18-methyl-7-oxo-13-oxa-2,6-diazatricyclo[12.6.1.015,20]henicosa-10,15(20),16,18-tetraen-8-yl]-N,2-dimethylhexanamide —— C34H47N3O4
(2S)-N-[(4R,5S,8S,14R)-5-benzyl-4-hydroxy-18-methyl-7-oxo-13-oxa-2,6-diazatricyclo[12.6.1.015,20]henicosa-10,15(20),16,18-tetraen-8-yl]-N,2-dimethylhexanamide
—— [(9S,10S,13S,14R,15S,17R)-22,24-dihydroxy-9,14,15-trimethoxy-5,11,13,17-tetramethyl-4-oxo-21-(2-pyrrolidin-1-ylethylideneamino)-3-azabicyclo[18.3.1]tetracosa-1(23),5,7,11,20(24),21-hexaen-10-yl] carbamate —— C37H56N4O8
[(9S,10S,13S,14R,15S,17R)-22,24-dihydroxy-9,14,15-trimethoxy-5,11,13,17-tetramethyl-4-oxo-21-(2-pyrrolidin-1-ylethylideneamino)-3-azabicyclo[18.3.1]tetracosa-1(23),5,7,11,20(24),21-hexaen-10-yl] carbamate
—— 6-(6-Aminohexanoylamino)hexanoic acid;1,8-diazacyclotetradecane-2,9-dione;heptane —— C31H62N4O5
6-(6-Aminohexanoylamino)hexanoic acid;1,8-diazacyclotetradecane-2,9-dione;heptane
—— 14-methyl-7-(4-methylpiperazin-1-yl)-9-oxa-3,14,17,19,21,23-hexazatetracyclo[16.6.1.14,8.022,25]hexacosa-1,4(26),5,7,18(25),19,21-heptaene-13,24-dione 1093796-85-0 C25H32N8O3
14-methyl-7-(4-methylpiperazin-1-yl)-9-oxa-3,14,17,19,21,23-hexazatetracyclo[16.6.1.14,8.022,25]hexacosa-1,4(26),5,7,18(25),19,21-heptaene-13,24-dione
—— [(1S,2R,3R,5S,6S,20R,21R)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9-azatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[methyl-[3-(methyldisulfanyl)propanoyl]amino]propanoate —— C37H51ClN2O10S2
[(1S,2R,3R,5S,6S,20R,21R)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9-azatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[methyl-[3-(methyldisulfanyl)propanoyl]amino]propanoate
—— 12-Oxa-5,9,18,20,24,25-hexazatetracyclo[19.3.1.02,19.03,23]pentacosa-1,3,5,7,9,15,18,20,23-nonaen-17-one —— C18H16N6O2
12-Oxa-5,9,18,20,24,25-hexazatetracyclo[19.3.1.02,19.03,23]pentacosa-1,3,5,7,9,15,18,20,23-nonaen-17-one
—— 2-[2-[3-[2-(1,3-Dioxobenzo[de]isoquinolin-2-yl)ethylsulfanyl]propoxy]ethyl]benzo[de]isoquinoline-1,3-dione;ethane —— C39H50N2O5S
2-[2-[3-[2-(1,3-Dioxobenzo[de]isoquinolin-2-yl)ethylsulfanyl]propoxy]ethyl]benzo[de]isoquinoline-1,3-dione;ethane
—— (4R)-4-[[(3S,7R)-3-[(2S,3S)-2-amino-3-hydroxybutanoyl]-1-[(2S,4S)-4-amino-1-(methylamino)-1,3-dioxo-5-phenylpentan-2-yl]-2,6,9-trioxo-1,4,8-triazacyclotetradec-12-en-7-yl]amino]-5-oxopentanoic acid —— C32H45N7O10
(4R)-4-[[(3S,7R)-3-[(2S,3S)-2-amino-3-hydroxybutanoyl]-1-[(2S,4S)-4-amino-1-(methylamino)-1,3-dioxo-5-phenylpentan-2-yl]-2,6,9-trioxo-1,4,8-triazacyclotetradec-12-en-7-yl]amino]-5-oxopentanoic acid
—— [(1R,4R,6S,15R,17R)-4-(cyclopropylsulfonylcarbamoyl)-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-[4-fluoro-2-(1,3-thiazol-2-yl)phenyl]carbamate —— C31H36FN5O7S2
[(1R,4R,6S,15R,17R)-4-(cyclopropylsulfonylcarbamoyl)-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-[4-fluoro-2-(1,3-thiazol-2-yl)phenyl]carbamate
—— [(1S,4R,6S,14S)-4-[(4-chlorophenyl)methylsulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C30H41ClN4O7S
[(1S,4R,6S,14S)-4-[(4-chlorophenyl)methylsulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— (3R,6S,9R,11S,12Z,19R,24R,27E)-N-cyclopropylsulfonyl-30-methoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,35-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29,31,33,36-heptaene-9-carboxamide —— C41H51N3O9S
(3R,6S,9R,11S,12Z,19R,24R,27E)-N-cyclopropylsulfonyl-30-methoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,35-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29,31,33,36-heptaene-9-carboxamide
—— [(9S,12S,13R,14S,16R)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(propylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C31H45N3O8
[(9S,12S,13R,14S,16R)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(propylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— [(1R,4R,6S,15R,17R)-4-(cyclopropylsulfonylcarbamoyl)-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-[5-methoxy-2-(5-methylpyridin-2-yl)phenyl]carbamate —— C35H43N5O8S
[(1R,4R,6S,15R,17R)-4-(cyclopropylsulfonylcarbamoyl)-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-en-17-yl] N-[5-methoxy-2-(5-methylpyridin-2-yl)phenyl]carbamate
—— N-[(1S,7S,10S,11R,14R)-10-benzyl-11-hydroxy-17-methoxy-8-oxo-2-oxa-9,13-diazatricyclo[12.7.0.015,20]henicosa-16,18,20-trien-7-yl]-N-methylpentane-1-sulfonamide —— C32H47N3O6S
N-[(1S,7S,10S,11R,14R)-10-benzyl-11-hydroxy-17-methoxy-8-oxo-2-oxa-9,13-diazatricyclo[12.7.0.015,20]henicosa-16,18,20-trien-7-yl]-N-methylpentane-1-sulfonamide
—— [(9S,12S,13R,14S)-13,20,22-trihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C29H40N2O9
[(9S,12S,13R,14S)-13,20,22-trihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— (20,22-Dihydroxy-8,13,14,17-tetramethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),6,10,16,18(22),19-hexaen-9-yl) carbamate —— C30H44N2O9
(20,22-Dihydroxy-8,13,14,17-tetramethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),6,10,16,18(22),19-hexaen-9-yl) carbamate
—— 1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-7-[3-[[1-[[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl]oxycarbonyl]piperidin-4-yl]amino]pyrrolidin-1-yl]quinoline-3-carboxylic acid —— C63H77FN6O17
1-cyclopropyl-6-fluoro-8-methoxy-4-oxo-7-[3-[[1-[[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl]oxycarbonyl]piperidin-4-yl]amino]pyrrolidin-1-yl]quinoline-3-carboxylic acid
—— 8-chloro-1-cyclopropyl-6-fluoro-4-oxo-7-[3-[[2-[[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl]oxycarbonylamino]acetyl]amino]pyrrolidin-1-yl]quinoline-3-carboxylic acid —— C59H68ClFN6O17
8-chloro-1-cyclopropyl-6-fluoro-4-oxo-7-[3-[[2-[[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl]oxycarbonylamino]acetyl]amino]pyrrolidin-1-yl]quinoline-3-carboxylic acid
—— [(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] N-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]carbamate —— C49H57N5O14
[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] N-[(3-pyridin-2-yl-1,2-oxazol-5-yl)methyl]carbamate
—— [(8S,9S,12S,13R,14S,16R)-13-hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-20-phosphonooxy-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-9-yl] carbamate —— C29H45N2O11P
[(8S,9S,12S,13R,14S,16R)-13-hydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-20-phosphonooxy-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-9-yl] carbamate
—— [(8S,9S,12S,13R,14S)-19-(azetidin-1-yl)-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C31H43N3O9
[(8S,9S,12S,13R,14S)-19-(azetidin-1-yl)-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— (6S,9S,12R)-6-cyclohexyl-12-[(4-hydroxyphenyl)methyl]-9-(2-hydroxypropan-2-yl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione —— C34H46N4O6
(6S,9S,12R)-6-cyclohexyl-12-[(4-hydroxyphenyl)methyl]-9-(2-hydroxypropan-2-yl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione
—— 19-Methyl-11-oxa-3,16,18-triazatricyclo[15.3.1.16,10]docosa-1(21),6(22),7,9,13,17,19-heptaen-2-one —— C19H21N3O2
19-Methyl-11-oxa-3,16,18-triazatricyclo[15.3.1.16,10]docosa-1(21),6(22),7,9,13,17,19-heptaen-2-one
—— (1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[2-(3,5-dimethylpyrazol-1-yl)-7-methoxy-8-methylquinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C37H46N6O7S
(1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[2-(3,5-dimethylpyrazol-1-yl)-7-methoxy-8-methylquinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— 2,5-dimethyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-1,6-dione;ethane —— C16H24N4O2
2,5-dimethyl-4H-[1,2,4]triazolo[4,3-a][1,4]benzodiazepine-1,6-dione;ethane
—— ethane;2-[2-methyl-6-[(E)-2-(4,4,10,10-tetramethyl-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13)-trien-7-yl)ethenyl]pyran-4-ylidene]indene-1,3-dione —— C35H39NO3
ethane;2-[2-methyl-6-[(E)-2-(4,4,10,10-tetramethyl-1-azatricyclo[7.3.1.05,13]trideca-5,7,9(13)-trien-7-yl)ethenyl]pyran-4-ylidene]indene-1,3-dione
—— 2-[(1S,4R,6S,14R,18R)-18-(8-chloro-7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-4-(cyclopropylsulfonylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl]acetic acid —— C38H42ClN5O9S
2-[(1S,4R,6S,14R,18R)-18-(8-chloro-7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-4-(cyclopropylsulfonylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl]acetic acid
—— (1S,4R,6R,18R)-18-hydroxy-N-(1-methylcyclopropyl)sulfonyl-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C21H32N4O6S
(1S,4R,6R,18R)-18-hydroxy-N-(1-methylcyclopropyl)sulfonyl-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (6S,9S,12R)-12-benzyl-6-cyclohexyl-9-(hydroxymethyl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione —— C32H42N4O5
(6S,9S,12R)-12-benzyl-6-cyclohexyl-9-(hydroxymethyl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione
—— (3R,6S,9R,11S,12Z,19R)-N-cyclopropylsulfonyl-30,34-dimethoxy-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,29(37),30,32(36),33-hexaene-9-carboxamide —— C41H53N3O10S
(3R,6S,9R,11S,12Z,19R)-N-cyclopropylsulfonyl-30,34-dimethoxy-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,29(37),30,32(36),33-hexaene-9-carboxamide
—— (3R,6S,9R,11S,12Z,19R,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24,24-dimethyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide;(3R,6S,9R,11S,12Z,19R)-N-cyclopropylsulfonyl-30,34-dimethoxy-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,29(37),30,32(36),33-hexaene-9-carboxamide —— C84H108N6O20S2
(3R,6S,9R,11S,12Z,19R,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24,24-dimethyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide;(3R,6S,9R,11S,12Z,19R)-N-cyclopropylsulfonyl-30,34-dimethoxy-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,29(37),30,32(36),33-hexaene-9-carboxamide
—— N-[(4R,5S,8S)-5-benzyl-4-hydroxy-19-methoxy-7-oxo-2,6,14-triazatricyclo[13.6.1.016,21]docosa-1,17,19-trien-8-yl]-3,3,3-trifluoro-N-methylpropane-1-sulfonamide —— C31H43F3N4O5S
N-[(4R,5S,8S)-5-benzyl-4-hydroxy-19-methoxy-7-oxo-2,6,14-triazatricyclo[13.6.1.016,21]docosa-1,17,19-trien-8-yl]-3,3,3-trifluoro-N-methylpropane-1-sulfonamide
—— (3R,6S,9R,11S,12Z,19R,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24,24-dimethyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide —— C43H55N3O10S
(3R,6S,9R,11S,12Z,19R,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24,24-dimethyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide