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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S,3S,7S,10R,11S,12S,16S)-16-chloro-7,11-dihydroxy-8,8,10,12-tetramethyl-3-(2-methyl-1,3-benzothiazol-5-yl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C27H37ClN2O5S
(1S,3S,7S,10R,11S,12S,16S)-16-chloro-7,11-dihydroxy-8,8,10,12-tetramethyl-3-(2-methyl-1,3-benzothiazol-5-yl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— [(1S,4R,6S,14S)-4-[(4-chlorophenyl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C29H39ClN4O7S
[(1S,4R,6S,14S)-4-[(4-chlorophenyl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— 2-[(4S,10S)-10-[3-(diaminomethylideneamino)propyl]-11-methyl-3,6,9,12,15-pentaoxo-13-[4-[[6-[(2-sulfophenyl)methyldiazenyl]pyridine-3-carbonyl]amino]butyl]-19-thia-2,5,8,11,14,20-hexazabicyclo[15.2.1]icosa-1(20),17-dien-4-yl]acetic acid —— C37H47N13O11S2
2-[(4S,10S)-10-[3-(diaminomethylideneamino)propyl]-11-methyl-3,6,9,12,15-pentaoxo-13-[4-[[6-[(2-sulfophenyl)methyldiazenyl]pyridine-3-carbonyl]amino]butyl]-19-thia-2,5,8,11,14,20-hexazabicyclo[15.2.1]icosa-1(20),17-dien-4-yl]acetic acid
—— [(1S,4R,6S,18R)-4-(cyclopropylsulfonylcarbamoyl)-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 5-methyl-2,3-dihydroindole-1-carboxylate —— C30H39N5O7S
[(1S,4R,6S,18R)-4-(cyclopropylsulfonylcarbamoyl)-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 5-methyl-2,3-dihydroindole-1-carboxylate
—— [(8S,9S,12S,13R,14S)-19-benzamido-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C35H43N3O10
[(8S,9S,12S,13R,14S)-19-benzamido-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— 3,10-Diazatricyclo[10.2.2.25,8]octadeca-1(15),12(16),13-triene-2,11-dione —— C16H20N2O2
3,10-Diazatricyclo[10.2.2.25,8]octadeca-1(15),12(16),13-triene-2,11-dione
—— Ethane;pyrrolo[2,1-c][1,4]benzothiazepine-6,11-dione —— C16H19NO2S
Ethane;pyrrolo[2,1-c][1,4]benzothiazepine-6,11-dione
—— (Cyclobutyloxycarbonylamino) 18-[2-(2,5-dimethylpyrazol-3-yl)thieno[3,2-d]pyrimidin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylate —— C34H41N7O7S
(Cyclobutyloxycarbonylamino) 18-[2-(2,5-dimethylpyrazol-3-yl)thieno[3,2-d]pyrimidin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylate
—— ethyl (1S,4R,6S,17R)-17-(3-chloro-6-methoxyisoquinolin-1-yl)oxy-13-methyl-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C29H35ClN4O6
ethyl (1S,4R,6S,17R)-17-(3-chloro-6-methoxyisoquinolin-1-yl)oxy-13-methyl-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— (6S,9S,12R)-6-butan-2-yl-9-(hydroxymethyl)-8-methyl-12-(1-phenylethyl)-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione —— C31H42N4O5
(6S,9S,12R)-6-butan-2-yl-9-(hydroxymethyl)-8-methyl-12-(1-phenylethyl)-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione
—— [(1S,2R,3R,5S,6S,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[acetyl(methyl)amino]propanoate —— C34H46ClN3O10
[(1S,2R,3R,5S,6S,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[acetyl(methyl)amino]propanoate
—— [(7S,11S,12R,13R,14R,15R,19S,20S,32R)-2-hydroxy-11-methoxy-3,7,12,14,17,17,20,24,32-nonamethyl-28-morpholin-4-yl-6,25,29,31-tetraoxo-8,16,18,33-tetraoxa-26-azapentacyclo[25.3.1.14,7.115,19.05,30]tritriaconta-1(30),2,4,9,21,23,27-heptaen-13-yl] 3-benzylimidazol-3-ium-1-carboxylate —— C53H63N4O13+
[(7S,11S,12R,13R,14R,15R,19S,20S,32R)-2-hydroxy-11-methoxy-3,7,12,14,17,17,20,24,32-nonamethyl-28-morpholin-4-yl-6,25,29,31-tetraoxo-8,16,18,33-tetraoxa-26-azapentacyclo[25.3.1.14,7.115,19.05,30]tritriaconta-1(30),2,4,9,21,23,27-heptaen-13-yl] 3-benzylimidazol-3-ium-1-carboxylate
—— 5-(1,3-Benzothiazol-2-yl)-10,10,16,16-tetramethyl-3-oxa-13-azatetracyclo[7.7.1.02,7.013,17]heptadeca-1,5,7,9(17)-tetraen-4-one;ethane —— C28H32N2O2S
5-(1,3-Benzothiazol-2-yl)-10,10,16,16-tetramethyl-3-oxa-13-azatetracyclo[7.7.1.02,7.013,17]heptadeca-1,5,7,9(17)-tetraen-4-one;ethane
—— 28-Cyclohexyl-22-methoxy-10,13,16-trimethyl-9-methylidene-9-oxo-9lambda6-thia-1,8,10,13,16-pentazapentacyclo[16.8.1.12,6.13,26.020,25]nonacosa-2,4,6(29),20(25),21,23,26(28)-heptaene-7,17-dione —— C34H45N5O4S
28-Cyclohexyl-22-methoxy-10,13,16-trimethyl-9-methylidene-9-oxo-9lambda6-thia-1,8,10,13,16-pentazapentacyclo[16.8.1.12,6.13,26.020,25]nonacosa-2,4,6(29),20(25),21,23,26(28)-heptaene-7,17-dione
—— N-[17-[[3-[2-[2-[2-(3-acetamido-6-ethyl-4-hydroxy-5-methyloxan-2-yl)oxyethoxy]ethoxy]ethylamino]-3-oxopropoxy]methyl]-33-(1-acetamido-2-hydroxypropyl)-41-ethyl-37-ethynyl-39-hydroxy-35,40-dimethyl-12,22-dioxo-2,5,8,15,19,26,29,32,34,42-decaoxa-11,23-diazabicyclo[36.4.0]dotetracontan-17-yl]-6-[[2,2-bis(octadeca-9,12-dienyl)-1,3-dioxolan-4-yl]methyl-(3-ethyl-3,4-dimethylhex-5-enyl)amino]hexanamide —— C117H209N7O26
N-[17-[[3-[2-[2-[2-(3-acetamido-6-ethyl-4-hydroxy-5-methyloxan-2-yl)oxyethoxy]ethoxy]ethylamino]-3-oxopropoxy]methyl]-33-(1-acetamido-2-hydroxypropyl)-41-ethyl-37-ethynyl-39-hydroxy-35,40-dimethyl-12,22-dioxo-2,5,8,15,19,26,29,32,34,42-decaoxa-11,23-diazabicyclo[36.4.0]dotetracontan-17-yl]-6-[[2,2-bis(octadeca-9,12-dienyl)-1,3-dioxolan-4-yl]methyl-(3-ethyl-3,4-dimethylhex-5-enyl)amino]hexanamide
—— [(9S,12S,13R,14S,16R)-20,22-dihydroxy-8,13,14-trimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(2-pyrrolidin-1-ylethylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C35H52N4O8
[(9S,12S,13R,14S,16R)-20,22-dihydroxy-8,13,14-trimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(2-pyrrolidin-1-ylethylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— (3R,6S,9R,11R,19R,24S)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide —— C42H57N3O10S
(3R,6S,9R,11R,19R,24S)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide
—— (3R,6S,9R,11S,12Z,19R,24S,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide —— C42H53N3O10S
(3R,6S,9R,11S,12Z,19R,24S,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide
—— (3R,6S,9R,11S,12Z,19R,24S,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide;(3R,6S,9R,11R,19R,24S)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide;(3R,6S,9R,11R,19R,24R)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide —— C126H167N9O30S3
(3R,6S,9R,11S,12Z,19R,24S,27E)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),12,27,29(37),30,32(36),33-heptaene-9-carboxamide;(3R,6S,9R,11R,19R,24S)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide;(3R,6S,9R,11R,19R,24R)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide
—— 25-Amino-13-fluoro-21-pentan-2-yl-5,8,28-triazapentacyclo[21.3.1.110,14.02,7.015,20]octacosa-2(7),3,5,10(28),11,13,15,17,19,21-decaen-9-one —— C30H33FN4O
25-Amino-13-fluoro-21-pentan-2-yl-5,8,28-triazapentacyclo[21.3.1.110,14.02,7.015,20]octacosa-2(7),3,5,10(28),11,13,15,17,19,21-decaen-9-one
—— (3R,6S,9R,11R,19R,24R)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide —— C42H57N3O10S
(3R,6S,9R,11R,19R,24R)-N-cyclopropylsulfonyl-30,34-dimethoxy-24-methyl-7,21,38-trioxo-2,22-dioxa-5,33-diazahexacyclo[27.6.2.13,6.15,19.09,11.032,36]nonatriaconta-1(35),29(37),30,32(36),33-pentaene-9-carboxamide
—— [(1S,7Z)-4-[2-(2-fluoro-6-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate;[(1S,7Z)-4-[2-(3-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate —— C86H107F3N6O14
[(1S,7Z)-4-[2-(2-fluoro-6-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate;[(1S,7Z)-4-[2-(3-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate
—— (1R,4R,6S,18S)-N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,14-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C38H47N5O7S2
(1R,4R,6S,18S)-N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,14-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— N-[[4-[(4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-2-ylamino)methyl]cyclohexyl]methyl]methanesulfonamide;ethane —— C22H33N3O3S2
N-[[4-[(4,5-dihydro-[1]benzoxepino[5,4-d][1,3]thiazol-2-ylamino)methyl]cyclohexyl]methyl]methanesulfonamide;ethane
—— (3R,6S,9R,11S,12Z,19R,26E)-N-cyclopropylsulfonyl-29,33-dimethoxy-7,21,37-trioxo-2,22-dioxa-5,32-diazahexacyclo[26.6.2.13,6.15,19.09,11.031,35]octatriaconta-1(34),12,26,28(36),29,31(35),32-heptaene-9-carboxamide —— C40H49N3O10S
(3R,6S,9R,11S,12Z,19R,26E)-N-cyclopropylsulfonyl-29,33-dimethoxy-7,21,37-trioxo-2,22-dioxa-5,32-diazahexacyclo[26.6.2.13,6.15,19.09,11.031,35]octatriaconta-1(34),12,26,28(36),29,31(35),32-heptaene-9-carboxamide
—— (1R,4R,6S,15R,17R)-17-(2-methoxy-6-phenylpyrimidin-4-yl)oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C29H34N4O6
(1R,4R,6S,15R,17R)-17-(2-methoxy-6-phenylpyrimidin-4-yl)oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— [(8S,9S,12S,13R,14S,16R)-13,20-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,6,10,18,20-hexaen-9-yl] carbamate —— C29H42N2O8
[(8S,9S,12S,13R,14S,16R)-13,20-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,6,10,18,20-hexaen-9-yl] carbamate
—— [(17S)-9-amino-15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaen-17-yl]methanol;ethane —— C17H22N4O2
[(17S)-9-amino-15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaen-17-yl]methanol;ethane
—— 5-Chloro-21-methoxy-18-oxa-2,10,15,23,25-pentazatetracyclo[17.6.2.03,8.022,26]heptacosa-1(25),3(8),4,6,19(27),20,22(26),23-octaene-11,16-dione —— C22H22ClN5O4
5-Chloro-21-methoxy-18-oxa-2,10,15,23,25-pentazatetracyclo[17.6.2.03,8.022,26]heptacosa-1(25),3(8),4,6,19(27),20,22(26),23-octaene-11,16-dione
—— ethane;3-methyl-3,3a-dihydro-1H-[1,3]thiazolo[4,3-c][1,4]benzothiazepine-4,10-dione —— C14H17NO2S2
ethane;3-methyl-3,3a-dihydro-1H-[1,3]thiazolo[4,3-c][1,4]benzothiazepine-4,10-dione
—— N-(12-cyano-17-methyl-14-oxa-3,10-diazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-1(21),2,5,7,12,15(20),16,18-octaen-11-ylidene)acetamide;ethane —— C26H28N4O2
N-(12-cyano-17-methyl-14-oxa-3,10-diazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-1(21),2,5,7,12,15(20),16,18-octaen-11-ylidene)acetamide;ethane
—— tert-butyl (1R,10R)-12-oxospiro[16-oxa-13-azatetracyclo[8.6.0.01,13.02,7]hexadeca-2,4,6-triene-8,3'-azetidine]-1'-carboxylate;ethane —— C23H32N2O4
tert-butyl (1R,10R)-12-oxospiro[16-oxa-13-azatetracyclo[8.6.0.01,13.02,7]hexadeca-2,4,6-triene-8,3'-azetidine]-1'-carboxylate;ethane
—— (1S,4R,6S,18S)-18-[2-(4-ethynyl-1,3-thiazol-2-yl)-7-methoxy-8-methylquinolin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13,15-triazatricyclo[13.4.0.04,6]nonadec-7-ene-4-carboxamide —— C38H44N6O7S2
(1S,4R,6S,18S)-18-[2-(4-ethynyl-1,3-thiazol-2-yl)-7-methoxy-8-methylquinolin-4-yl]oxy-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13,15-triazatricyclo[13.4.0.04,6]nonadec-7-ene-4-carboxamide
—— 5,7-dimethyl-7H-pyrrolo[1,2-a][1,5]benzodiazepin-6-one;ethane —— C16H20N2O
5,7-dimethyl-7H-pyrrolo[1,2-a][1,5]benzodiazepin-6-one;ethane
—— Ethane;12-methyl-21,28-dioxa-3,5,9,12-tetrazahexacyclo[27.3.1.116,20.03,7.09,14.022,27]tetratriaconta-1(32),4,6,16(34),17,19,22,24,26,29(33)-decaen-11-one —— C31H36N4O3
Ethane;12-methyl-21,28-dioxa-3,5,9,12-tetrazahexacyclo[27.3.1.116,20.03,7.09,14.022,27]tetratriaconta-1(32),4,6,16(34),17,19,22,24,26,29(33)-decaen-11-one
—— 29-Cyclohexyl-23-methoxy-10,17-dimethyl-9,9-dioxo-9lambda6-thia-1,8,10,17-tetrazapentacyclo[17.8.1.12,6.13,27.021,26]triaconta-2,4,6(30),19,22,24,27(29)-heptaen-18-one —— C34H46N4O4S
29-Cyclohexyl-23-methoxy-10,17-dimethyl-9,9-dioxo-9lambda6-thia-1,8,10,17-tetrazapentacyclo[17.8.1.12,6.13,27.021,26]triaconta-2,4,6(30),19,22,24,27(29)-heptaen-18-one
—— (22E)-23-fluoro-26-methyl-28-(2-methylpropanoyl)-2,10,17-triazapentacyclo[16.5.3.13,6.112,16.04,8]octacosa-1,12(27),13,15,17,22-hexaen-11-one —— C30H38FN3O2
(22E)-23-fluoro-26-methyl-28-(2-methylpropanoyl)-2,10,17-triazapentacyclo[16.5.3.13,6.112,16.04,8]octacosa-1,12(27),13,15,17,22-hexaen-11-one
—— [(8S,9S,12S,13R,14S,16R)-20,22-dihydroxy-19-[2-(1H-imidazol-5-yl)ethylideneamino]-8,13,14-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C34H47N5O8
[(8S,9S,12S,13R,14S,16R)-20,22-dihydroxy-19-[2-(1H-imidazol-5-yl)ethylideneamino]-8,13,14-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— N-[3-(3-aminopropanimidoyl)-12-(1-hydroxyethyl)-9-(2-hydroxyethyl)-6-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-10,20-dimethyl-2,5,8,11,14-pentaoxo-1,4,7,10,13,19-hexazabicyclo[19.3.0]tetracos-19-en-15-yl]acetamide —— C37H57N9O10
N-[3-(3-aminopropanimidoyl)-12-(1-hydroxyethyl)-9-(2-hydroxyethyl)-6-[2-hydroxy-2-(4-hydroxyphenyl)ethyl]-10,20-dimethyl-2,5,8,11,14-pentaoxo-1,4,7,10,13,19-hexazabicyclo[19.3.0]tetracos-19-en-15-yl]acetamide
—— (3R,14E,23R,29Z,31S,33R,36S)-33-(2-cyclopropylsulfonylacetyl)-18,18-dimethyl-4,20-dioxa-1,6-diazahexacyclo[21.13.1.13,36.16,9.08,13.031,33]nonatriaconta-8,10,12,14,29-pentaene-5,21,35,37-tetrone;(3R,6S,9R,11R,19R)-N-cyclopropylsulfonyl-33-ethoxy-29-methoxy-24,24-dimethyl-7,21,37-trioxo-2,22-dioxa-5,32-diazahexacyclo[26.6.2.13,6.15,19.09,11.031,35]octatriaconta-1(34),28(36),29,31(35),32-pentaene-9-carboxamide —— C85H113N5O19S2
(3R,14E,23R,29Z,31S,33R,36S)-33-(2-cyclopropylsulfonylacetyl)-18,18-dimethyl-4,20-dioxa-1,6-diazahexacyclo[21.13.1.13,36.16,9.08,13.031,33]nonatriaconta-8,10,12,14,29-pentaene-5,21,35,37-tetrone;(3R,6S,9R,11R,19R)-N-cyclopropylsulfonyl-33-ethoxy-29-methoxy-24,24-dimethyl-7,21,37-trioxo-2,22-dioxa-5,32-diazahexacyclo[26.6.2.13,6.15,19.09,11.031,35]octatriaconta-1(34),28(36),29,31(35),32-pentaene-9-carboxamide
—— (3R,14E,23R,29Z,31S,33R,36S)-33-(2-cyclopropylsulfonylacetyl)-18,18-dimethyl-4,20-dioxa-1,6-diazahexacyclo[21.13.1.13,36.16,9.08,13.031,33]nonatriaconta-8,10,12,14,29-pentaene-5,21,35,37-tetrone —— C42H54N2O9S
(3R,14E,23R,29Z,31S,33R,36S)-33-(2-cyclopropylsulfonylacetyl)-18,18-dimethyl-4,20-dioxa-1,6-diazahexacyclo[21.13.1.13,36.16,9.08,13.031,33]nonatriaconta-8,10,12,14,29-pentaene-5,21,35,37-tetrone
—— [(8S,9S,12S,13R,14S)-19-[[4-[(dipropylamino)methyl]benzoyl]amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C42H58N4O9
[(8S,9S,12S,13R,14S)-19-[[4-[(dipropylamino)methyl]benzoyl]amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— [(8S,9S,12S,13R,14S,16R)-2-(4-(18F)fluoranylbenzoyl)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C38H46FN3O9
[(8S,9S,12S,13R,14S,16R)-2-(4-(18F)fluoranylbenzoyl)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— Amino 19-[3-[3-[(9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl)imino]propylamino]propylideneamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaene-9-carboxylate —— C62H89N7O16
Amino 19-[3-[3-[(9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl)imino]propylamino]propylideneamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaene-9-carboxylate
—— [(4S,7R,8S,9S,16S)-4-hydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-2,6-dioxo-1-azacyclohexadeca-11,13-dien-8-yl] 2,2,2-trichloroethyl carbonate —— C30H41Cl3N2O6S
[(4S,7R,8S,9S,16S)-4-hydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-2,6-dioxo-1-azacyclohexadeca-11,13-dien-8-yl] 2,2,2-trichloroethyl carbonate
—— ethyl (1R,4R,6S,15R,17R)-17-[7-methoxy-8-methyl-2-(6-methylpyridin-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C37H44N4O6
ethyl (1R,4R,6S,15R,17R)-17-[7-methoxy-8-methyl-2-(6-methylpyridin-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— (4'R,6'R,8'R)-16'-chloro-17',19'-dihydroxy-4'-methylspiro[1,3-dithiane-2,13'-7-oxa-3-azatricyclo[13.4.0.06,8]nonadeca-1(15),9,11,16,18-pentaene]-2'-one —— C21H24ClNO4S2
(4'R,6'R,8'R)-16'-chloro-17',19'-dihydroxy-4'-methylspiro[1,3-dithiane-2,13'-7-oxa-3-azatricyclo[13.4.0.06,8]nonadeca-1(15),9,11,16,18-pentaene]-2'-one
—— (7S,9E,11R,12S,13S,14S,15S,16R,17S,18S,19E,21Z)-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,13,14,16,18,22-octamethyl-26-[[(3-methyl-1,3-diazetidin-1-yl)amino]methylidene]-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25(29)-heptaene-6,23,27-trione —— C40H54N4O10
(7S,9E,11R,12S,13S,14S,15S,16R,17S,18S,19E,21Z)-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,13,14,16,18,22-octamethyl-26-[[(3-methyl-1,3-diazetidin-1-yl)amino]methylidene]-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25(29)-heptaene-6,23,27-trione
—— (1S,4R,6S,17R)-17-(5-bromo-6-methoxyisoquinolin-1-yl)oxy-13-methyl-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C27H31BrN4O6
(1S,4R,6S,17R)-17-(5-bromo-6-methoxyisoquinolin-1-yl)oxy-13-methyl-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— 6H-[1]benzofuro[3,2-c]isoquinolin-5-one;ethane —— C32H24N2O4
6H-[1]benzofuro[3,2-c]isoquinolin-5-one;ethane