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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(8S,9S,12S,13R,14S,16R)-19-[3-[3-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]propylamino]propylideneamino]-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C62H89N7O18
[(8S,9S,12S,13R,14S,16R)-19-[3-[3-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]propylamino]propylideneamino]-13,20,22-trihydroxy-10-(hydroxymethyl)-8,14-dimethoxy-4,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— 1-Azacyclododec-3-en-2-one —— C11H19NO
1-Azacyclododec-3-en-2-one
—— [(8S,9S,12S,13R,14S)-13,20,22-trihydroxy-19-[(4-hydroxybenzoyl)amino]-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C35H43N3O10
[(8S,9S,12S,13R,14S)-13,20,22-trihydroxy-19-[(4-hydroxybenzoyl)amino]-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— (2R)-4-[2-(1,3-benzoxazol-2-ylamino)-3-methylbutanoyl]-1-[(4-chlorophenyl)methyl]-N-[(5R)-3,4,13-trioxo-2,14-diazabicyclo[13.4.0]nonadeca-1(19),7,15,17-tetraen-5-yl]piperazine-2-carboxamide —— C41H46ClN7O6
(2R)-4-[2-(1,3-benzoxazol-2-ylamino)-3-methylbutanoyl]-1-[(4-chlorophenyl)methyl]-N-[(5R)-3,4,13-trioxo-2,14-diazabicyclo[13.4.0]nonadeca-1(19),7,15,17-tetraen-5-yl]piperazine-2-carboxamide
—— 2-Ethyl-3,4,10-trihydroxy-13-(5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl)oxy-3,5,6,8,10,12,14-heptamethyl-11-[(4-methyl-3,7-dioxabicyclo[4.1.0]heptan-2-yl)oxy]-1-oxa-6-azacyclopentadecan-7-one —— C36H65NO12
2-Ethyl-3,4,10-trihydroxy-13-(5-hydroxy-4-methoxy-4,6-dimethyloxan-2-yl)oxy-3,5,6,8,10,12,14-heptamethyl-11-[(4-methyl-3,7-dioxabicyclo[4.1.0]heptan-2-yl)oxy]-1-oxa-6-azacyclopentadecan-7-one
—— ethyl (1S,4R,6S,17R)-17-hydroxy-13-[(2-methylpropan-2-yl)oxycarbonylamino]-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C23H36N4O7
ethyl (1S,4R,6S,17R)-17-hydroxy-13-[(2-methylpropan-2-yl)oxycarbonylamino]-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— (3S,7S,10R,11R,12S)-10-but-3-enyl-7,11-dihydroxy-8,8,12,16-tetramethyl-3-[2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C29H44N2O5S
(3S,7S,10R,11R,12S)-10-but-3-enyl-7,11-dihydroxy-8,8,12,16-tetramethyl-3-[2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— (1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-14-[2-(3,3-difluorocyclohexyl)-2-oxoethyl]-18-[7-methoxy-8-methyl-2-[2-(propan-2-ylamino)-1,3-thiazol-4-yl]quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C46H58F2N6O8S2
(1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-14-[2-(3,3-difluorocyclohexyl)-2-oxoethyl]-18-[7-methoxy-8-methyl-2-[2-(propan-2-ylamino)-1,3-thiazol-4-yl]quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— 4-[[3-[3-[[1-[(11-Chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl)oxy]-1-oxopropan-2-yl]-methylamino]-3-oxopropyl]sulfanyl-2,5-dihydroxypyrrol-1-yl]methyl]cyclohexane-1-carboxylic acid —— C47H63ClN4O14S
4-[[3-[3-[[1-[(11-Chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl)oxy]-1-oxopropan-2-yl]-methylamino]-3-oxopropyl]sulfanyl-2,5-dihydroxypyrrol-1-yl]methyl]cyclohexane-1-carboxylic acid
—— [(9E,19E,21Z)-27-[2-[bis(2-methylpropyl)amino]-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate —— C47H66N2O13
[(9E,19E,21Z)-27-[2-[bis(2-methylpropyl)amino]-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate
—— [(1S,2S,17S)-7-(azetidin-1-yl)-8,20,24-trihydroxy-2,17-dimethoxy-4,13,22-trimethyl-12-oxo-21-oxa-11-azatricyclo[17.2.2.16,10]tetracosa-4,6(24),7,9,13,15,19(23)-heptaen-18-yl] carbamate —— C31H41N3O9
[(1S,2S,17S)-7-(azetidin-1-yl)-8,20,24-trihydroxy-2,17-dimethoxy-4,13,22-trimethyl-12-oxo-21-oxa-11-azatricyclo[17.2.2.16,10]tetracosa-4,6(24),7,9,13,15,19(23)-heptaen-18-yl] carbamate
—— (6Z,16Z,18Z)-11-chloro-21-hydroxy-12,15,20-trimethoxy-2,5,9,16-tetramethyl-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-6,10,12,14(26),16,18-hexaene-8,23-dione —— C29H37ClN2O8
(6Z,16Z,18Z)-11-chloro-21-hydroxy-12,15,20-trimethoxy-2,5,9,16-tetramethyl-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-6,10,12,14(26),16,18-hexaene-8,23-dione
—— 6-(4,4-Dimethylcyclohexyl)-13-methyl-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaene-5,7,12,14-tetrone;ethane —— C25H28N2O4
6-(4,4-Dimethylcyclohexyl)-13-methyl-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaene-5,7,12,14-tetrone;ethane
—— (1R,4R,6S,15R,17R)-17-[8-ethyl-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid —— C36H44N4O6S
(1R,4R,6S,15R,17R)-17-[8-ethyl-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylic acid
—— [(1S,4R,6S,14S)-4-[(3-bromophenyl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C29H39BrN4O7S
[(1S,4R,6S,14S)-4-[(3-bromophenyl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— Ethane;6-methylbenzimidazolo[1,2-a]quinazolin-5-one —— C19H23N3O
Ethane;6-methylbenzimidazolo[1,2-a]quinazolin-5-one
—— 1-[4-(6,13-Dibromo-4,15-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl)piperidin-1-yl]ethanone;ethane —— C28H45Br2N3O
1-[4-(6,13-Dibromo-4,15-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl)piperidin-1-yl]ethanone;ethane
—— [(9S)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(3-phosphonooxypropylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C31H46N3O12P
[(9S)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(3-phosphonooxypropylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— [(1S,4R,6S,14S)-2,15-dioxo-4-[[(1R)-1-phenylethyl]carbamoyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C31H44N4O5
[(1S,4R,6S,14S)-2,15-dioxo-4-[[(1R)-1-phenylethyl]carbamoyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— 8-Benzyl-24-cyclohexyl-9,10,11,12-tetramethyl-9-sulfanyl-15-oxa-1,8,10,12-tetrazapentacyclo[12.8.1.12,6.13,22.016,21]pentacosa-2,4,6(25),16,18,20,22(24)-heptaen-7-one —— C37H44N4O2S
8-Benzyl-24-cyclohexyl-9,10,11,12-tetramethyl-9-sulfanyl-15-oxa-1,8,10,12-tetrazapentacyclo[12.8.1.12,6.13,22.016,21]pentacosa-2,4,6(25),16,18,20,22(24)-heptaen-7-one
—— ethane;6-methyl-7H-quinazolino[3,2-a][1,4]benzodiazepine-5,13-dione —— C23H31N3O2
ethane;6-methyl-7H-quinazolino[3,2-a][1,4]benzodiazepine-5,13-dione
—— (1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[2-methoxy-6-(3-methoxyphenyl)pyrimidin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C33H41N5O8S
(1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[2-methoxy-6-(3-methoxyphenyl)pyrimidin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— (1S,4R,6S,14R,18R)-18-(5-chloro-6-methoxyisoquinolin-1-yl)oxy-N-cyclopropylsulfonyl-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C39H47ClF3N5O8S
(1S,4R,6S,14R,18R)-18-(5-chloro-6-methoxyisoquinolin-1-yl)oxy-N-cyclopropylsulfonyl-2,15-dioxo-14-[2-oxo-2-[4-(trifluoromethyl)piperidin-1-yl]ethyl]-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— 2-[(1R,4S,10R,13R,16R,19S,25R)-10-[4-[2-[2-[5-(2-amino-2-oxoethoxy)-4-oxopentoxy]ethoxy]ethoxy]butanoyl]-13-benzyl-25-[3-(diaminomethylideneamino)propyl]-4-[4-[[2-[2-[2-[2-[2-[2-[2-[(17E)-17-hydroxyimino-12-[2-[[(3E)-3-hydroxyimino-2-methylbutan-2-yl]amino]ethyl]-16,16-dimethyl-4,8-dioxooctadecoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethoxy]acetyl]amino]butyl]-3,6,12,15,18,21,24,27-octaoxo-8,29,30-trithia-2,5,11,17,23-pentazabicyclo[14.11.4]hentriacontan-19-yl]acetic acid —— C96H158N14O29S3
2-[(1R,4S,10R,13R,16R,19S,25R)-10-[4-[2-[2-[5-(2-amino-2-oxoethoxy)-4-oxopentoxy]ethoxy]ethoxy]butanoyl]-13-benzyl-25-[3-(diaminomethylideneamino)propyl]-4-[4-[[2-[2-[2-[2-[2-[2-[2-[(17E)-17-hydroxyimino-12-[2-[[(3E)-3-hydroxyimino-2-methylbutan-2-yl]amino]ethyl]-16,16-dimethyl-4,8-dioxooctadecoxy]ethoxy]ethoxy]ethoxy]ethoxy]ethylamino]-2-oxoethoxy]acetyl]amino]butyl]-3,6,12,15,18,21,24,27-octaoxo-8,29,30-trithia-2,5,11,17,23-pentazabicyclo[14.11.4]hentriacontan-19-yl]acetic acid
—— [13,20,22-Trihydroxy-4,8,10,12,16-pentamethyl-3-oxo-19-(2-pyrrolidin-1-ylethylamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C33H50N4O6
[13,20,22-Trihydroxy-4,8,10,12,16-pentamethyl-3-oxo-19-(2-pyrrolidin-1-ylethylamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— 5,6,7,8,14-Pentamethyl-10,12-dioxa-2,3-diazatetracyclo[11.8.0.04,9.016,21]henicosa-1(13),2,4,6,8,14,16,18,20-nonaene;propane —— C25H30N2O2
5,6,7,8,14-Pentamethyl-10,12-dioxa-2,3-diazatetracyclo[11.8.0.04,9.016,21]henicosa-1(13),2,4,6,8,14,16,18,20-nonaene;propane
—— 2-[(14R)-11-[3-(diaminomethylideneamino)propyl]-14-ethyl-12-methyl-4,7,10,13,16-pentaoxo-3,6,9,12,15-pentazabicyclo[15.3.1]henicosa-1(21),17,19-trien-5-yl]acetic acid —— C25H36N8O7
2-[(14R)-11-[3-(diaminomethylideneamino)propyl]-14-ethyl-12-methyl-4,7,10,13,16-pentaoxo-3,6,9,12,15-pentazabicyclo[15.3.1]henicosa-1(21),17,19-trien-5-yl]acetic acid
—— [(4E,8S,9S,10E,12S,13R,14S,16R)-13,20-dihydroxy-8,14-dimethoxy-10,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate;(8S,9S,10E,12S,13R,14S,16R)-5,13,20-trihydroxy-8,14-dimethoxy-9,10,12,16-tetramethyl-2-azabicyclo[16.3.1]docosa-1(21),10,18(22),19-tetraen-3-one —— C54H83N3O13
[(4E,8S,9S,10E,12S,13R,14S,16R)-13,20-dihydroxy-8,14-dimethoxy-10,12,16-trimethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate;(8S,9S,10E,12S,13R,14S,16R)-5,13,20-trihydroxy-8,14-dimethoxy-9,10,12,16-tetramethyl-2-azabicyclo[16.3.1]docosa-1(21),10,18(22),19-tetraen-3-one
—— [(1S,4R,6S,14S)-4-[(2,5-dichlorothiophen-3-yl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C27H36Cl2N4O7S2
[(1S,4R,6S,14S)-4-[(2,5-dichlorothiophen-3-yl)sulfonylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— 5-Chloro-22-methoxy-19-oxa-2,10,14,24,26-pentazatetracyclo[18.6.2.03,8.023,27]octacosa-1(26),3(8),4,6,20(28),21,23(27),24-octaene-11,15-dione —— C23H24ClN5O4
5-Chloro-22-methoxy-19-oxa-2,10,14,24,26-pentazatetracyclo[18.6.2.03,8.023,27]octacosa-1(26),3(8),4,6,20(28),21,23(27),24-octaene-11,15-dione
—— ethyl (1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-(4-nitrobenzoyl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylate —— C34H40N4O9
ethyl (1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-(4-nitrobenzoyl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylate
—— (1S,4R,6S,18R)-18-[8-chloro-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-14,14-dimethyl-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C39H48ClN5O7S2
(1S,4R,6S,18R)-18-[8-chloro-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-14,14-dimethyl-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— [(4Z,6Z,10Z)-13,14,17-trimethoxy-4,8,10,12,16-pentamethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl] carbamate —— C30H42N2O8
[(4Z,6Z,10Z)-13,14,17-trimethoxy-4,8,10,12,16-pentamethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl] carbamate
—— (4R)-4-[[(3S,7R)-3-[(2S)-2-amino-4-methylpentanoyl]-1-methyl-2,6,9-trioxo-1,4,8-triazacyclotetradec-12-en-7-yl]amino]-5-oxopentanoic acid —— C23H37N5O7
(4R)-4-[[(3S,7R)-3-[(2S)-2-amino-4-methylpentanoyl]-1-methyl-2,6,9-trioxo-1,4,8-triazacyclotetradec-12-en-7-yl]amino]-5-oxopentanoic acid
—— 3-[2-[[1-(3-Ethylphenyl)cyclopropyl]amino]-1-hydroxyethyl]-18-fluoro-10-propyl-7-prop-2-ynyl-2-oxa-4,10-diazatricyclo[14.3.1.06,8]icosa-1(19),16(20),17-triene-5,9-dione —— C36H46FN3O4
3-[2-[[1-(3-Ethylphenyl)cyclopropyl]amino]-1-hydroxyethyl]-18-fluoro-10-propyl-7-prop-2-ynyl-2-oxa-4,10-diazatricyclo[14.3.1.06,8]icosa-1(19),16(20),17-triene-5,9-dione
—— cyclopropanesulfonic acid {(1S,4R,6S,17R)-17-[2-(3-fluoro-phenyl)-7-methoxy-8-methyl-quinazolin-4-yloxy]-13-methyl-2,14-dioxo-3,13,15-triaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carbonyl}-amide —— C36H41FN6O7S
cyclopropanesulfonic acid {(1S,4R,6S,17R)-17-[2-(3-fluoro-phenyl)-7-methoxy-8-methyl-quinazolin-4-yloxy]-13-methyl-2,14-dioxo-3,13,15-triaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carbonyl}-amide
—— (2S)-N-[(7S,10S,11R)-10-benzyl-11-(hydroxymethoxy)-8-oxo-2-oxa-9,13-diazabicyclo[13.4.0]nonadeca-1(19),4,15,17-tetraen-7-yl]-N,2-dimethylhexanamide —— C32H45N3O5
(2S)-N-[(7S,10S,11R)-10-benzyl-11-(hydroxymethoxy)-8-oxo-2-oxa-9,13-diazabicyclo[13.4.0]nonadeca-1(19),4,15,17-tetraen-7-yl]-N,2-dimethylhexanamide
—— [(8S,9S,12S,14S)-19-benzamido-20,22-dihydroxy-8,14-dimethoxy-13-methoxyimino-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C36H44N4O9
[(8S,9S,12S,14S)-19-benzamido-20,22-dihydroxy-8,14-dimethoxy-13-methoxyimino-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— [(8S,9S,12S,13R,14S,16R)-13,20-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-9-yl] carbamate —— C29H44N2O8
[(8S,9S,12S,13R,14S,16R)-13,20-dihydroxy-8,14,19-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-9-yl] carbamate
—— 2-(dimethylamino)-N-[(13Z)-5,11-dioxo-3-phenyl-2-oxa-6,12-diazatricyclo[13.2.2.06,10]nonadeca-1(18),13,15(19),16-tetraen-4-yl]-3-phenylpropanamide —— C33H36N4O4
2-(dimethylamino)-N-[(13Z)-5,11-dioxo-3-phenyl-2-oxa-6,12-diazatricyclo[13.2.2.06,10]nonadeca-1(18),13,15(19),16-tetraen-4-yl]-3-phenylpropanamide
—— 18-[8-chloro-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-14-methyl-2,15-dioxo-13-oxa-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C37H44ClN5O8S2
18-[8-chloro-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-14-methyl-2,15-dioxo-13-oxa-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— ethyl (1R,6S,15R,17R)-17-[7-methoxy-8-methyl-2-(6-propan-2-ylpyridin-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C39H48N4O6
ethyl (1R,6S,15R,17R)-17-[7-methoxy-8-methyl-2-(6-propan-2-ylpyridin-2-yl)quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— (3R,6S,9R,12R)-6-cyclopropyl-12-(2-ethenylbut-2-enyl)-21-fluoro-3,8,9-trimethyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(18),19,21-triene-7,10,13-trione —— C29H41FN4O4
(3R,6S,9R,12R)-6-cyclopropyl-12-(2-ethenylbut-2-enyl)-21-fluoro-3,8,9-trimethyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(18),19,21-triene-7,10,13-trione
—— (6S,9R,12R)-6-butan-2-yl-12-[(4-fluorophenyl)methyl]-8,9-dimethyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10-dione —— C30H41FN4O3
(6S,9R,12R)-6-butan-2-yl-12-[(4-fluorophenyl)methyl]-8,9-dimethyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10-dione
—— (1R,4R,6S,15R,17R)-17-[8-chloro-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C37H44ClN5O7S2
(1R,4R,6S,15R,17R)-17-[8-chloro-7-methoxy-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— ethane;2-ethyl-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one —— C14H16N2OS
ethane;2-ethyl-3H-[1]benzothiolo[3,2-d]pyrimidin-4-one
—— [(6E,16E)-19-amino-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C28H39N3O8
[(6E,16E)-19-amino-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— [(16Z,18Z)-11-chloro-21-hydroxy-12,15,20-trimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] 2-(2-methylpropanoylamino)propanoate —— C36H50ClN3O11
[(16Z,18Z)-11-chloro-21-hydroxy-12,15,20-trimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] 2-(2-methylpropanoylamino)propanoate
—— (1S,4R,6S,14R,18R)-18-(5-chloro-6-methoxy-3-pyridin-2-ylisoquinolin-1-yl)oxy-N-cyclopropylsulfonyl-14-[2-(3,3-difluoropiperidin-1-yl)-2-oxoethyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C43H49ClF2N6O8S
(1S,4R,6S,14R,18R)-18-(5-chloro-6-methoxy-3-pyridin-2-ylisoquinolin-1-yl)oxy-N-cyclopropylsulfonyl-14-[2-(3,3-difluoropiperidin-1-yl)-2-oxoethyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— [(8S,9S,12S,13R,14S,16R)-19-[2-(dimethylamino)ethylideneamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C32H48N4O8
[(8S,9S,12S,13R,14S,16R)-19-[2-(dimethylamino)ethylideneamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate