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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— (13,20,22-Trihydroxy-4,8,10,12,16-pentamethyl-3-oxo-19-pyrrolidin-1-yl-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl) carbamate —— C31H45N3O6
(13,20,22-Trihydroxy-4,8,10,12,16-pentamethyl-3-oxo-19-pyrrolidin-1-yl-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl) carbamate
—— 18-[8-chloro-7-methoxy-2-(3-propan-2-ylpyrazol-1-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-14-methyl-2,15-dioxo-13-oxa-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C37H45ClN6O8S
18-[8-chloro-7-methoxy-2-(3-propan-2-ylpyrazol-1-yl)quinolin-4-yl]oxy-N-cyclopropylsulfonyl-14-methyl-2,15-dioxo-13-oxa-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (1R,3S,12R,14R,16R)-14-(2-ethoxy-7-methoxy-8-methylquinolin-4-yl)oxy-10-methyl-18-oxa-10,20-diazatetracyclo[15.2.1.01,3.012,16]icosa-4,17(20)-diene-11,19-dione —— C31H37N3O6
(1R,3S,12R,14R,16R)-14-(2-ethoxy-7-methoxy-8-methylquinolin-4-yl)oxy-10-methyl-18-oxa-10,20-diazatetracyclo[15.2.1.01,3.012,16]icosa-4,17(20)-diene-11,19-dione
—— [(8S,9R,12S,13R,14S,16R)-19-fluoro-13-hydroxy-14-methoxy-4,8,10,12,16-pentamethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-9-yl] carbamate —— C28H41FN2O5
[(8S,9R,12S,13R,14S,16R)-19-fluoro-13-hydroxy-14-methoxy-4,8,10,12,16-pentamethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(22),4,10,18,20-pentaen-9-yl] carbamate
—— 6,9-Dithia-3-azatetracyclo[8.8.0.03,7.012,17]octadeca-1(18),10,12,14,16-pentaene-2,8-dione;ethane —— C17H17NO2S2
6,9-Dithia-3-azatetracyclo[8.8.0.03,7.012,17]octadeca-1(18),10,12,14,16-pentaene-2,8-dione;ethane
—— [(2R,6S,20R,21S)-11-chloro-21-hydroxy-12-(hydroxymethyl)-20-methoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10(26),11,13,16,18-pentaen-6-yl] 2-[methyl(3-methylsulfanylpropanoyl)amino]propanoate —— C36H50ClN3O10S
[(2R,6S,20R,21S)-11-chloro-21-hydroxy-12-(hydroxymethyl)-20-methoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10(26),11,13,16,18-pentaen-6-yl] 2-[methyl(3-methylsulfanylpropanoyl)amino]propanoate
—— (3S,7S,10R,11R,12S)-3-(1-fluoro-2-pyridin-2-ylethenyl)-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(oxiran-2-ylmethyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C29H41FN2O6
(3S,7S,10R,11R,12S)-3-(1-fluoro-2-pyridin-2-ylethenyl)-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(oxiran-2-ylmethyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— [(8S,9S,12S,13R,14S,16R)-7,13,20,22-tetrahydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate —— C31H45N3O9
[(8S,9S,12S,13R,14S,16R)-7,13,20,22-tetrahydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate
—— bis[2-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]ethyl] benzene-1,4-dicarboxylate —— C68H88N6O20
bis[2-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]ethyl] benzene-1,4-dicarboxylate
—— [(8S,9S,12S,13R,14S)-19-[[4-[(4-cyclohexylpiperazin-1-yl)methyl]benzoyl]amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C46H63N5O9
[(8S,9S,12S,13R,14S)-19-[[4-[(4-cyclohexylpiperazin-1-yl)methyl]benzoyl]amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— Ethane;3,10,17,24-tetrazaoctacyclo[13.13.2.02,10.04,9.012,29.016,24.018,23.026,30]triaconta-1(29),2,4,6,8,12,14,16,18,20,22,26(30),27-tridecaene-11,25-dione —— C30H24N4O2
Ethane;3,10,17,24-tetrazaoctacyclo[13.13.2.02,10.04,9.012,29.016,24.018,23.026,30]triaconta-1(29),2,4,6,8,12,14,16,18,20,22,26(30),27-tridecaene-11,25-dione
—— (17S)-17-(2-chloroethyl)-15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaen-9-amine;ethane —— C18H23ClN4O
(17S)-17-(2-chloroethyl)-15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaen-9-amine;ethane
—— [(8S,9S,12S,13R,14S,16R)-19-(2-(18F)fluoranylethylideneamino)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C30H42FN3O8
[(8S,9S,12S,13R,14S,16R)-19-(2-(18F)fluoranylethylideneamino)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— [(1S,4R,6S,14S)-4-(cyclobutylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C27H42N4O5
[(1S,4R,6S,14S)-4-(cyclobutylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— (3S,7S,10R,11R,12S)-10-but-3-enyl-7,11-dihydroxy-8,8,12,16-tetramethyl-3-(2-pyridin-2-ylethenyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C30H44N2O5
(3S,7S,10R,11R,12S)-10-but-3-enyl-7,11-dihydroxy-8,8,12,16-tetramethyl-3-(2-pyridin-2-ylethenyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— (11S)-7-hydroxy-17-methoxy-15-(methoxymethoxy)-11-methyl-12-oxa-2-azabicyclo[12.4.0]octadeca-1(14),15,17-triene-3,5,6,13-tetrone —— C20H25NO9
(11S)-7-hydroxy-17-methoxy-15-(methoxymethoxy)-11-methyl-12-oxa-2-azabicyclo[12.4.0]octadeca-1(14),15,17-triene-3,5,6,13-tetrone
—— [(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] N-(2-hydroxyethyl)carbamate —— C42H55N3O14
[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] N-(2-hydroxyethyl)carbamate
—— (4S,7R,8S,9S,16S)-4,8-dihydroxy-5,5,7,9,13-pentamethyl-16-quinolin-7-yl-1-azacyclohexadeca-11,13-diene-2,6-dione —— C29H38N2O4
(4S,7R,8S,9S,16S)-4,8-dihydroxy-5,5,7,9,13-pentamethyl-16-quinolin-7-yl-1-azacyclohexadeca-11,13-diene-2,6-dione
—— [(2R,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12-(hydroxymethyl)-20-methoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10(26),11,13,16,18-pentaen-6-yl] 2-[methyl(3-methylsulfanylpropanoyl)amino]propanoate —— C36H50ClN3O10S
[(2R,6S,16E,18E,20R,21S)-11-chloro-21-hydroxy-12-(hydroxymethyl)-20-methoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10(26),11,13,16,18-pentaen-6-yl] 2-[methyl(3-methylsulfanylpropanoyl)amino]propanoate
—— (13-Acetyloxy-15,17-dihydroxy-11-methoxy-3,7,12,22-tetramethyl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1,3,5(28),9,19,21,25-heptaen-2-yl) 4-methylbenzoate —— C42H45NO13
(13-Acetyloxy-15,17-dihydroxy-11-methoxy-3,7,12,22-tetramethyl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1,3,5(28),9,19,21,25-heptaen-2-yl) 4-methylbenzoate
—— [(8S,9R,12S,13R,14S,16R)-20,22-dihydroxy-13,14,19-trimethoxy-4,8,10,12,16-pentamethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C30H44N2O8
[(8S,9R,12S,13R,14S,16R)-20,22-dihydroxy-13,14,19-trimethoxy-4,8,10,12,16-pentamethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— (3S,7S,10R,11R,12S)-3-[1-fluoro-2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(oxiran-2-ylmethyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C28H41FN2O6S
(3S,7S,10R,11R,12S)-3-[1-fluoro-2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(oxiran-2-ylmethyl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— Ethane;10-phenyl-15-oxa-10,21,28-triazadecacyclo[17.14.1.14,8.02,17.03,14.05,33.021,29.022,27.030,34.012,35]pentatriaconta-1(33),2(17),3(14),4,6,8(35),12,18,22,24,26,28,30(34),31-tetradecaene-9,11,20-trione —— C43H35N3O4
Ethane;10-phenyl-15-oxa-10,21,28-triazadecacyclo[17.14.1.14,8.02,17.03,14.05,33.021,29.022,27.030,34.012,35]pentatriaconta-1(33),2(17),3(14),4,6,8(35),12,18,22,24,26,28,30(34),31-tetradecaene-9,11,20-trione
—— 2-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]ethylphosphonic acid —— C30H44N3O11P
2-[[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-19-yl]imino]ethylphosphonic acid
—— [(1S,4R,6S,14S)-4-(benzenesulfonylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C29H40N4O7S
[(1S,4R,6S,14S)-4-(benzenesulfonylcarbamoyl)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— (11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl) (2S)-2-[methyl-(4-methyl-4-sulfanylpentanoyl)amino]propanoate —— C38H54ClN3O10S
(11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl) (2S)-2-[methyl-(4-methyl-4-sulfanylpentanoyl)amino]propanoate
—— [(1S,2R,5R,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2R)-2-[methyl(3-sulfanylpropanoyl)amino]propanoate —— C35H48ClN3O10S
[(1S,2R,5R,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2R)-2-[methyl(3-sulfanylpropanoyl)amino]propanoate
—— ethane;1,2,5-trimethyl-4H-imidazo[1,2-a][1,4]benzodiazepin-6-one —— C18H27N3O
ethane;1,2,5-trimethyl-4H-imidazo[1,2-a][1,4]benzodiazepin-6-one
—— [(1S,4R,6S,14S)-4-[(4-fluorophenyl)sulfamoylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C29H40FN5O7S
[(1S,4R,6S,14S)-4-[(4-fluorophenyl)sulfamoylcarbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— (3S,7S,10R,11R,12S)-1-ethyl-7,11-dihydroxy-8,8,12,16-tetramethyl-3-[1-(2-methyl-1,3-oxazol-4-yl)prop-1-en-2-yl]-10-(oxiran-2-yl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C30H46N2O7
(3S,7S,10R,11R,12S)-1-ethyl-7,11-dihydroxy-8,8,12,16-tetramethyl-3-[1-(2-methyl-1,3-oxazol-4-yl)prop-1-en-2-yl]-10-(oxiran-2-yl)-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— Ethyl (2R,3aR,10Z,11aS,12aR,14aR)-2-{[2-(4-isopropyl-1,3-thiazol-2-yl)-7-methoxy-8-methyl-4-quinolinyl]oxy}-5-methyl-4,14-dioxo-2,3,3a,4,5,6,7,8,9,11a,12,13,14,14a-tetradecahydrocyclopenta[c]cycloprop a[g][1,6]diazacyclotetradecine-12a(1H)-carboxylate 923604-57-3 C37H46N4O6S
Ethyl (2R,3aR,10Z,11aS,12aR,14aR)-2-{[2-(4-isopropyl-1,3-thiazol-2-yl)-7-methoxy-8-methyl-4-quinolinyl]oxy}-5-methyl-4,14-dioxo-2,3,3a,4,5,6,7,8,9,11a,12,13,14,14a-tetradecahydrocyclopenta[c]cycloprop a[g][1,6]diazacyclotetradecine-12a(1H)-carboxylate
—— (1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-18-(7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-2,15-dioxo-14-(2-oxo-2-piperidin-1-ylethyl)-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C43H52N6O8S
(1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-18-(7-methoxy-2-pyridin-2-ylquinolin-4-yl)oxy-2,15-dioxo-14-(2-oxo-2-piperidin-1-ylethyl)-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (4R,6S,7E,16S)-18-[7,8-dimethyl-2-[4-(trifluoromethyl)-1,3-thiazol-2-yl]quinolin-4-yl]oxy-14-methyl-N-(1-methylcyclopropyl)sulfonyl-2,15-dioxo-1,14-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C38H44F3N5O6S2
(4R,6S,7E,16S)-18-[7,8-dimethyl-2-[4-(trifluoromethyl)-1,3-thiazol-2-yl]quinolin-4-yl]oxy-14-methyl-N-(1-methylcyclopropyl)sulfonyl-2,15-dioxo-1,14-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— (1R,4R,6S,14S,18S)-14-anilino-18-(5-fluoro-1-propan-2-ylbenzimidazol-2-yl)oxy-N-(1-methylcyclopropyl)sulfonyl-2,15-dioxo-3-azatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C39H48FN5O6S
(1R,4R,6S,14S,18S)-14-anilino-18-(5-fluoro-1-propan-2-ylbenzimidazol-2-yl)oxy-N-(1-methylcyclopropyl)sulfonyl-2,15-dioxo-3-azatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— Ethane;methyl 3-methyl-12-oxo-10,13,14-triazapentacyclo[12.6.1.02,10.04,9.017,21]henicosa-1(20),2,4(9),5,7,15,17(21),18-octaene-7-carboxylate —— C27H35N3O3
Ethane;methyl 3-methyl-12-oxo-10,13,14-triazapentacyclo[12.6.1.02,10.04,9.017,21]henicosa-1(20),2,4(9),5,7,15,17(21),18-octaene-7-carboxylate
—— (2R)-7-cyclopropylsulfonyl-2-fluoro-17-methoxy-4-methyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione —— C32H31FN4O7S
(2R)-7-cyclopropylsulfonyl-2-fluoro-17-methoxy-4-methyl-2-[(1-oxo-2H-isoquinolin-7-yl)amino]-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione
—— ethane;N-[(11R)-6-methyl-12-oxo-9-phenyl-1,10-diazatricyclo[6.4.1.04,13]trideca-4(13),5,7,9-tetraen-11-yl]pyridine-4-carboxamide —— C26H26N4O2
ethane;N-[(11R)-6-methyl-12-oxo-9-phenyl-1,10-diazatricyclo[6.4.1.04,13]trideca-4(13),5,7,9-tetraen-11-yl]pyridine-4-carboxamide
—— [(8S,9S,12S,13R,14S,16R)-20-chloro-13,19,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate —— C28H41ClN2O8
[(8S,9S,12S,13R,14S,16R)-20-chloro-13,19,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-9-yl] carbamate
—— Ethane;11-[2-(2-methoxyethoxy)phenyl]-5,17-dimethyl-8,14,24,27,32,35-hexaoxa-1,11,21-triazatetracyclo[19.8.8.02,7.015,20]heptatriaconta-2(7),3,5,15(20),16,18-hexaene —— C41H61N3O8
Ethane;11-[2-(2-methoxyethoxy)phenyl]-5,17-dimethyl-8,14,24,27,32,35-hexaoxa-1,11,21-triazatetracyclo[19.8.8.02,7.015,20]heptatriaconta-2(7),3,5,15(20),16,18-hexaene
—— (1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[7-methoxy-2-[2-(propan-2-ylamino)-1,3-thiazol-4-yl]quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C37H46N6O7S2
(1R,4R,6S,15R,17R)-N-cyclopropylsulfonyl-17-[7-methoxy-2-[2-(propan-2-ylamino)-1,3-thiazol-4-yl]quinolin-4-yl]oxy-13-methyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— [(1S,5S,6S,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[methyl-(4-methyl-4-sulfanylpentanoyl)amino]propanoate —— C38H54ClN3O10S
[(1S,5S,6S,20R,21S)-11-chloro-21-hydroxy-12,20-dimethoxy-2,5,9,16-tetramethyl-8,23-dioxo-4,24-dioxa-9,22-diazatetracyclo[19.3.1.110,14.03,5]hexacosa-10,12,14(26),16,18-pentaen-6-yl] (2S)-2-[methyl-(4-methyl-4-sulfanylpentanoyl)amino]propanoate
—— 2-[(18S,25R,35S)-35-[(S)-hydroxy(phenyl)methyl]-8-[4-(methanesulfonamido)-1,3-thiazol-2-yl]-28-(methoxymethyl)-21-methyl-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,7,10,12(42),14,19(41),21,26(40),28,36(39)-dodecaen-18-yl]-N-methylacetamide —— C48H49N13O9S7
2-[(18S,25R,35S)-35-[(S)-hydroxy(phenyl)methyl]-8-[4-(methanesulfonamido)-1,3-thiazol-2-yl]-28-(methoxymethyl)-21-methyl-16,23,30,33-tetraoxo-25-propan-2-yl-3,13,20,27,37-pentathia-7,17,24,31,34,39,40,41,42,43-decazaheptacyclo[34.2.1.12,5.112,15.119,22.126,29.06,11]tritetraconta-1(38),2(43),4,7,10,12(42),14,19(41),21,26(40),28,36(39)-dodecaen-18-yl]-N-methylacetamide
—— 6,11-Dihydropyridazino[4,3-c][1,5]benzodiazepin-5-one;ethane —— C13H14N4O
6,11-Dihydropyridazino[4,3-c][1,5]benzodiazepin-5-one;ethane
—— [(8S,9S,12S,13R,14S,16R)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(2-oxoethylamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C30H43N3O9
[(8S,9S,12S,13R,14S,16R)-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(2-oxoethylamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— Lopac-S-1316 —— C44H56N8O7
Lopac-S-1316
—— N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-14-propan-2-yl-13-oxa-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C40H51N5O8S2
N-cyclopropylsulfonyl-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-14-propan-2-yl-13-oxa-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— Ethane;methoxymethylbenzene;15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaen-17-ylmethanamine —— C25H32N4O2
Ethane;methoxymethylbenzene;15-oxa-8,11,18-triazatetracyclo[8.8.0.02,7.012,18]octadeca-1(10),2,4,6,8,11-hexaen-17-ylmethanamine
—— [(8S,9S,12S,13R,14S,16S)-9-carbamoyloxy-13-hydroxy-8,14,17-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-20-yl] N-ethyl-N-[2-(ethylamino)ethyl]carbamate —— C36H58N4O9
[(8S,9S,12S,13R,14S,16S)-9-carbamoyloxy-13-hydroxy-8,14,17-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-20-yl] N-ethyl-N-[2-(ethylamino)ethyl]carbamate
—— tert-butyl-[[(2R,8R)-2-[[(2R,8S)-8-ethyl-2,3,4,6,7,8-hexahydro-1H-pyrimido[1,2-a]pyrimidin-2-yl]methylsulfanylmethyl]-2,3,4,6,7,8-hexahydro-1H-pyrimido[1,2-a]pyrimidin-8-yl]methoxy]-diphenylsilane;[(4E,6Z,8S,9S,10E,12S,13R,14S,16R)-19-[3-[4-(2,5-dioxopyrrol-1-yl)butanoylamino]propylamino]-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl] carbamate —— C74H105N11O12SSi
tert-butyl-[[(2R,8R)-2-[[(2R,8S)-8-ethyl-2,3,4,6,7,8-hexahydro-1H-pyrimido[1,2-a]pyrimidin-2-yl]methylsulfanylmethyl]-2,3,4,6,7,8-hexahydro-1H-pyrimido[1,2-a]pyrimidin-8-yl]methoxy]-diphenylsilane;[(4E,6Z,8S,9S,10E,12S,13R,14S,16R)-19-[3-[4-(2,5-dioxopyrrol-1-yl)butanoylamino]propylamino]-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18-pentaen-9-yl] carbamate
—— 14-O-cyclopentyl 4-O-ethyl (1S,4R,6S,18R)-18-(3,4-dihydro-1H-isoquinoline-2-carbonyloxy)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4,14-dicarboxylate —— C36H47N3O8
14-O-cyclopentyl 4-O-ethyl (1S,4R,6S,18R)-18-(3,4-dihydro-1H-isoquinoline-2-carbonyloxy)-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4,14-dicarboxylate