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大环内酰胺类

中文名称 英文名称 CAS号 化学式 结构式图片
—— [(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-20-yl] N-methyl-N-[3-(methylamino)propyl]carbamate —— C34H54N4O8
[(8S,9S,12S,13R,14S,16R)-9-carbamoyloxy-13-hydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18(22),19-pentaen-20-yl] N-methyl-N-[3-(methylamino)propyl]carbamate
—— (1S,4R,6S,17R)-17-[7-methoxy-8-methyl-2-(6-methyl-pyridin-2-yl)-quinazolin-4-yloxy]-13-methyl-2,14-dioxo-3,13,15-triaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carboxylic acid —— C33H38N6O6
(1S,4R,6S,17R)-17-[7-methoxy-8-methyl-2-(6-methyl-pyridin-2-yl)-quinazolin-4-yloxy]-13-methyl-2,14-dioxo-3,13,15-triaza-tricyclo[13.3.0.0(4,6)]octadec-7-ene-4-carboxylic acid
—— (1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-(6-methoxy-2-phenylpyrimidin-4-yl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid —— C36H41N5O7
(1S,4R,6S,18R)-14-[(4-methoxyphenyl)methyl]-18-(6-methoxy-2-phenylpyrimidin-4-yl)oxy-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxylic acid
—— (20,22-Dihydroxy-8,13,14,17-tetramethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl) carbamate —— C30H42N2O9
(20,22-Dihydroxy-8,13,14,17-tetramethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl) carbamate
—— [(8R,9R,14R,16S)-19-[3-[3-[[(8S,9S,12S,14S)-9-carbamoyloxy-20,22-dihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,13-dioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-19-yl]amino]propylamino]propylideneamino]-20,22-dihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,13-dioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,11,18(22),19-hexaen-9-yl] carbamate —— C62H85N7O16
[(8R,9R,14R,16S)-19-[3-[3-[[(8S,9S,12S,14S)-9-carbamoyloxy-20,22-dihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,13-dioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-19-yl]amino]propylamino]propylideneamino]-20,22-dihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3,13-dioxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,11,18(22),19-hexaen-9-yl] carbamate
—— (6S,9S,12R)-12-[(4-chlorophenyl)methyl]-6-cyclopropyl-9-(hydroxymethyl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione —— C29H35ClN4O5
(6S,9S,12R)-12-[(4-chlorophenyl)methyl]-6-cyclopropyl-9-(hydroxymethyl)-8-methyl-2-oxa-5,8,11,14-tetrazabicyclo[16.4.0]docosa-1(22),16,18,20-tetraene-7,10,13-trione
—— (10S,14S,18S)-14-hydroxy-18-[(1S)-1-hydroxyprop-2-enyl]-10-methyl-12-methylidene-1-oxa-7-azacyclooctadec-15-ene-2,8-dione —— C21H33NO5
(10S,14S,18S)-14-hydroxy-18-[(1S)-1-hydroxyprop-2-enyl]-10-methyl-12-methylidene-1-oxa-7-azacyclooctadec-15-ene-2,8-dione
—— [(1S,7Z)-4-[2-(3-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate;[(1S,7Z)-4-[2-(4-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate —— C86H108F2N6O14
[(1S,7Z)-4-[2-(3-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate;[(1S,7Z)-4-[2-(4-methylphenyl)ethylcarbamoyl]-14-[2-[(2-methylpropan-2-yl)oxy]-2-oxoethyl]-2,15-dioxo-16-azatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] 4-fluoro-1,3-dihydroisoindole-2-carboxylate
—— (1S,3S,7S,10R,11S,12S,16S)-7,11-dihydroxy-8,8,10,12-tetramethyl-3-(2-methyl-1,3-benzothiazol-5-yl)-5,9-dioxo-17-oxa-4-azabicyclo[14.1.0]heptadecane-16-carbonitrile —— C28H37N3O5S
(1S,3S,7S,10R,11S,12S,16S)-7,11-dihydroxy-8,8,10,12-tetramethyl-3-(2-methyl-1,3-benzothiazol-5-yl)-5,9-dioxo-17-oxa-4-azabicyclo[14.1.0]heptadecane-16-carbonitrile
—— ethane;2,3,6-trimethyl-5H-pyrimido[1,2-a][1,4]benzodiazepine-1,7-dione —— C19H27N3O2
ethane;2,3,6-trimethyl-5H-pyrimido[1,2-a][1,4]benzodiazepine-1,7-dione
—— (1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-14-[2-(3,3-difluoropiperidin-1-yl)-2-oxoethyl]-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide —— C45H56F2N6O8S2
(1S,4R,6S,14R,18R)-N-cyclopropylsulfonyl-14-[2-(3,3-difluoropiperidin-1-yl)-2-oxoethyl]-18-[7-methoxy-8-methyl-2-(4-propan-2-yl-1,3-thiazol-2-yl)quinolin-4-yl]oxy-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-ene-4-carboxamide
—— [(8S,9S,12S,13R,14S)-19-[[4-(dimethylamino)benzoyl]amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C37H48N4O9
[(8S,9S,12S,13R,14S)-19-[[4-(dimethylamino)benzoyl]amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— tert-butyl N-[(6-butan-2-yl-8-methyl-5-oxo-10-oxa-1,6,14,15-tetrazabicyclo[10.3.0]pentadeca-12,14-dien-9-yl)methyl]-N-methylcarbamate —— C22H39N5O4
tert-butyl N-[(6-butan-2-yl-8-methyl-5-oxo-10-oxa-1,6,14,15-tetrazabicyclo[10.3.0]pentadeca-12,14-dien-9-yl)methyl]-N-methylcarbamate
—— tert-butyl (5S,8S)-8-[[(5R)-3,4,13-trioxo-2,14-diazabicyclo[13.4.0]nonadeca-1(19),7,15,17-tetraen-5-yl]carbamoyl]-2-oxa-7-azadispiro[3.0.45.14]decane-7-carboxylate —— C31H40N4O7
tert-butyl (5S,8S)-8-[[(5R)-3,4,13-trioxo-2,14-diazabicyclo[13.4.0]nonadeca-1(19),7,15,17-tetraen-5-yl]carbamoyl]-2-oxa-7-azadispiro[3.0.45.14]decane-7-carboxylate
—— acetic acid;12H-benzimidazolo[1,2-c]quinazolin-6-one;ethane —— C22H31N3O3
acetic acid;12H-benzimidazolo[1,2-c]quinazolin-6-one;ethane
—— [(1S,4R,6S,14S)-4-[[(R)-(4-methylphenyl)sulfinyl]carbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate —— C30H42N4O6S
[(1S,4R,6S,14S)-4-[[(R)-(4-methylphenyl)sulfinyl]carbamoyl]-2,15-dioxo-3,16-diazatricyclo[14.3.0.04,6]nonadec-7-en-14-yl] N-tert-butylcarbamate
—— [13,20,22-Trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C31H43N3O8
[13,20,22-Trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-19-(prop-2-enylideneamino)-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— ethyl (1S,4R,6S,17R)-13-methyl-17-(4-nitrobenzoyl)oxy-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C26H32N4O8
ethyl (1S,4R,6S,17R)-13-methyl-17-(4-nitrobenzoyl)oxy-2,14-dioxo-3,13,15-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— (5S,9S,14R)-20-methoxy-18-(methoxymethoxy)-7,7,14-trimethyl-6,8-dioxa-2-azatricyclo[15.4.0.05,9]henicosa-1(17),12,18,20-tetraene-3,10,16-trione —— C24H31NO8
(5S,9S,14R)-20-methoxy-18-(methoxymethoxy)-7,7,14-trimethyl-6,8-dioxa-2-azatricyclo[15.4.0.05,9]henicosa-1(17),12,18,20-tetraene-3,10,16-trione
—— (6S,7R,10S)-6-N-hydroxy-7-(2-methylpropyl)-8-oxo-10-N-[[4-[[[6-[[2-(trioxidanylsulfanyl)phenyl]methyldiazenyl]pyridine-3-carbonyl]amino]methyl]phenyl]methyl]-2-oxa-9-azabicyclo[10.2.2]hexadeca-1(14),12,15-triene-6,10-dicarboxamide —— C41H47N7O9S
(6S,7R,10S)-6-N-hydroxy-7-(2-methylpropyl)-8-oxo-10-N-[[4-[[[6-[[2-(trioxidanylsulfanyl)phenyl]methyldiazenyl]pyridine-3-carbonyl]amino]methyl]phenyl]methyl]-2-oxa-9-azabicyclo[10.2.2]hexadeca-1(14),12,15-triene-6,10-dicarboxamide
—— [(8S,9S,12S,13R,14S,16R)-19-[2-(dimethylamino)ethylideneamino]-20,22-dihydroxy-8,13,14-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate —— C33H50N4O8
[(8S,9S,12S,13R,14S,16R)-19-[2-(dimethylamino)ethylideneamino]-20,22-dihydroxy-8,13,14-trimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,18(22),19-hexaen-9-yl] carbamate
—— (1R,4R,6S,15R,17R)-17-(ethoxymethoxy)-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide —— C25H39N3O7S
(1R,4R,6S,15R,17R)-17-(ethoxymethoxy)-13-methyl-N-(1-methylcyclopropyl)sulfonyl-2,14-dioxo-3,13-diazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxamide
—— ethyl (4R,6S,15S,17S)-17-hydroxy-13-methyl-2,14-dioxo-1,3,13-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C19H29N3O5
ethyl (4R,6S,15S,17S)-17-hydroxy-13-methyl-2,14-dioxo-1,3,13-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— [2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-27-[2-[methyl(piperidin-1-yl)amino]-2-oxoethoxy]-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate —— C45H61N3O13
[2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-27-[2-[methyl(piperidin-1-yl)amino]-2-oxoethoxy]-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate
—— [27-[2-[ethyl(piperidin-1-yl)amino]-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate —— C46H63N3O13
[27-[2-[ethyl(piperidin-1-yl)amino]-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate
—— [(1S,4R,6S,18R)-4-[(1-methylcyclopropyl)sulfonylcarbamoyl]-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] N-[2-(4-ethyl-1,3-thiazol-2-yl)-5-methylphenyl]carbamate —— C34H44N6O7S2
[(1S,4R,6S,18R)-4-[(1-methylcyclopropyl)sulfonylcarbamoyl]-2,15-dioxo-3,14,16-triazatricyclo[14.3.0.04,6]nonadec-7-en-18-yl] N-[2-(4-ethyl-1,3-thiazol-2-yl)-5-methylphenyl]carbamate
—— ethyl (4R,6S,15S,17R)-17-[tert-butyl(dimethyl)silyl]oxy-13-methyl-2,14-dioxo-1,3,13-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate —— C25H43N3O5Si
ethyl (4R,6S,15S,17R)-17-[tert-butyl(dimethyl)silyl]oxy-13-methyl-2,14-dioxo-1,3,13-triazatricyclo[13.3.0.04,6]octadec-7-ene-4-carboxylate
—— [27-[2-(3,5-dimethylmorpholin-4-yl)-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate —— C45H60N2O14
[27-[2-(3,5-dimethylmorpholin-4-yl)-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate
—— [27-[2-[(dibutylamino)-propan-2-ylamino]-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate —— C50H73N3O13
[27-[2-[(dibutylamino)-propan-2-ylamino]-2-oxoethoxy]-2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate
—— [2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-27-[2-oxo-2-[piperidin-1-yl(propyl)amino]ethoxy]-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate —— C47H65N3O13
[2,15,17,29-tetrahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-27-[2-oxo-2-[piperidin-1-yl(propyl)amino]ethoxy]-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,25,27-octaen-13-yl] acetate
—— [(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] N-(3-phenylpropyl)carbamate —— C49H61N3O13
[(7S,11S,12R,13S,14R,15R,16R,17S,18S)-2,15,17-trihydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-26-morpholin-4-yl-6,23,27,29-tetraoxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(28),2,4,9,19,21,25-heptaen-13-yl] N-(3-phenylpropyl)carbamate
—— [(4S,7R,8S,9S)-4-hydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-2,6-dioxo-1-azacyclohexadeca-11,13-dien-8-yl] 2,2,2-trichloroethyl carbonate —— C30H41Cl3N2O6S
[(4S,7R,8S,9S)-4-hydroxy-5,5,7,9,13-pentamethyl-16-[1-(2-methyl-1,3-thiazol-4-yl)prop-1-en-2-yl]-2,6-dioxo-1-azacyclohexadeca-11,13-dien-8-yl] 2,2,2-trichloroethyl carbonate
—— [(8S,9S,12S,13R,14S)-19-[(4-fluorophenyl)methylcarbamoylamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C36H45FN4O9
[(8S,9S,12S,13R,14S)-19-[(4-fluorophenyl)methylcarbamoylamino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— N-[(1S,4R,5S,8S,14R)-5-[(3,5-difluorophenyl)methyl]-4-(hydroxymethoxy)-7-oxo-13-oxa-2,6-diazatricyclo[12.6.1.015,20]henicosa-10,15,17,19-tetraen-8-yl]-4,4,4-trifluoro-N,2-dimethylbutanamide —— C32H38F5N3O5
N-[(1S,4R,5S,8S,14R)-5-[(3,5-difluorophenyl)methyl]-4-(hydroxymethoxy)-7-oxo-13-oxa-2,6-diazatricyclo[12.6.1.015,20]henicosa-10,15,17,19-tetraen-8-yl]-4,4,4-trifluoro-N,2-dimethylbutanamide
—— (6S,7R,10S)-6-N-hydroxy-7-(2-methylpropyl)-8-oxo-10-N-[[4-[[[6-[[2-(trihydroxy-lambda4-sulfanyl)phenyl]methyldiazenyl]pyridine-3-carbonyl]amino]methyl]phenyl]methyl]-2-oxa-9-azabicyclo[10.2.2]hexadeca-1(14),12,15-triene-6,10-dicarboxamide —— C41H49N7O9S
(6S,7R,10S)-6-N-hydroxy-7-(2-methylpropyl)-8-oxo-10-N-[[4-[[[6-[[2-(trihydroxy-lambda4-sulfanyl)phenyl]methyldiazenyl]pyridine-3-carbonyl]amino]methyl]phenyl]methyl]-2-oxa-9-azabicyclo[10.2.2]hexadeca-1(14),12,15-triene-6,10-dicarboxamide
—— [(8S,9S,12S,13R,14S)-19-[(2-ethoxyacetyl)amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate —— C32H45N3O10
[(8S,9S,12S,13R,14S)-19-[(2-ethoxyacetyl)amino]-13,20,22-trihydroxy-8,14-dimethoxy-4,10,12,16-tetramethyl-3-oxo-2-azabicyclo[16.3.1]docosa-1(21),4,6,10,16,18(22),19-heptaen-9-yl] carbamate
—— [(5S,13R)-20-methoxy-18-(methoxymethoxy)-7,7,13-trimethyl-16-oxo-6,8-dioxa-15-azatricyclo[15.4.0.05,9]henicosa-1(17),2,11,18,20-pentaen-10-yl] benzoate —— C31H37NO8
[(5S,13R)-20-methoxy-18-(methoxymethoxy)-7,7,13-trimethyl-16-oxo-6,8-dioxa-15-azatricyclo[15.4.0.05,9]henicosa-1(17),2,11,18,20-pentaen-10-yl] benzoate
—— N-[1-(3,5-difluorophenyl)ethyl]-1-(fluoromethyl)-2-methyl-N-[3-(10-methyl-3-oxo-4,6,16-triazabicyclo[10.4.0]hexadeca-1(12),6,8,13,15-pentaen-14-yl)prop-2-enyl]cyclopropane-1-carboxamide —— C31H35F3N4O2
N-[1-(3,5-difluorophenyl)ethyl]-1-(fluoromethyl)-2-methyl-N-[3-(10-methyl-3-oxo-4,6,16-triazabicyclo[10.4.0]hexadeca-1(12),6,8,13,15-pentaen-14-yl)prop-2-enyl]cyclopropane-1-carboxamide
—— (3S,7S,10R,11R,12S)-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(3-methylbut-2-enyl)-3-[2-(2-methyl-1,3-oxazol-4-yl)ethenyl]-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C30H46N2O6
(3S,7S,10R,11R,12S)-7,11-dihydroxy-8,8,12,16-tetramethyl-10-(3-methylbut-2-enyl)-3-[2-(2-methyl-1,3-oxazol-4-yl)ethenyl]-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione
—— [(4E,8S,9R,10E,12S,14S,16S)-19-[2-(dimethylamino)ethylamino]-13-hydroxyimino-4,8,10,12,14,16-hexamethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18-tetraen-9-yl] carbamate —— C32H49N5O6
[(4E,8S,9R,10E,12S,14S,16S)-19-[2-(dimethylamino)ethylamino]-13-hydroxyimino-4,8,10,12,14,16-hexamethyl-3,20,22-trioxo-2-azabicyclo[16.3.1]docosa-1(21),4,10,18-tetraen-9-yl] carbamate
—— [2,15,17,27,29-pentahydroxy-11-methoxy-26-[(3-methoxybutoxyamino)methylidene]-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C43H58N2O14
[2,15,17,27,29-pentahydroxy-11-methoxy-26-[(3-methoxybutoxyamino)methylidene]-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— [2,15,17,27,29-pentahydroxy-26-[(6-hydroxyhexoxyamino)methylidene]-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C44H60N2O14
[2,15,17,27,29-pentahydroxy-26-[(6-hydroxyhexoxyamino)methylidene]-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— [26-[[2-(2-ethoxyethoxy)ethoxyamino]methylidene]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C44H60N2O15
[26-[[2-(2-ethoxyethoxy)ethoxyamino]methylidene]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— [26-[(5,6-dibromohexoxyamino)methylidene]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C44H58Br2N2O13
[26-[(5,6-dibromohexoxyamino)methylidene]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— [2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-26-[(10-phenoxydecoxyamino)methylidene]-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C54H72N2O14
[2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-26-[(10-phenoxydecoxyamino)methylidene]-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— [2,15,17,27,29-pentahydroxy-11-methoxy-26-[[2-(2-methoxyethoxy)ethoxyamino]methylidene]-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C43H58N2O15
[2,15,17,27,29-pentahydroxy-11-methoxy-26-[[2-(2-methoxyethoxy)ethoxyamino]methylidene]-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— [26-[[2-(2-butoxyethoxy)ethoxyamino]methylidene]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate —— C46H64N2O15
[26-[[2-(2-butoxyethoxy)ethoxyamino]methylidene]-2,15,17,27,29-pentahydroxy-11-methoxy-3,7,12,14,16,18,22-heptamethyl-6,23-dioxo-8,30-dioxa-24-azatetracyclo[23.3.1.14,7.05,28]triaconta-1(29),2,4,9,19,21,24,27-octaen-13-yl] acetate
—— (1S,4R,6S,18R)-18-[2-(4-fluoro-phenyl)-7-methoxy-8-methyl-quinazolin-4-yloxy]-14-(4-methoxy-benzyl)-2,15-dioxo-3,14,16-triaza-tricyclo[14.3.0.0(4,6)]nonadec-7-ene-4-carboxylic acid ethyl ester —— C43H48FN5O7
(1S,4R,6S,18R)-18-[2-(4-fluoro-phenyl)-7-methoxy-8-methyl-quinazolin-4-yloxy]-14-(4-methoxy-benzyl)-2,15-dioxo-3,14,16-triaza-tricyclo[14.3.0.0(4,6)]nonadec-7-ene-4-carboxylic acid ethyl ester
—— N-[(4R,5S,8S)-5-benzyl-4-hydroxy-7-oxo-19-phenoxy-14-oxa-2,6-diazatricyclo[13.6.1.016,21]docosa-1,17,19-trien-8-yl]-N-methylhexanamide —— C39H51N3O5
N-[(4R,5S,8S)-5-benzyl-4-hydroxy-7-oxo-19-phenoxy-14-oxa-2,6-diazatricyclo[13.6.1.016,21]docosa-1,17,19-trien-8-yl]-N-methylhexanamide
—— (3S,7S,11R,12S)-7,11-dihydroxy-8,8,12-trimethyl-16-(4-methylpent-3-enyl)-3-[2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione —— C30H46N2O5S
(3S,7S,11R,12S)-7,11-dihydroxy-8,8,12-trimethyl-16-(4-methylpent-3-enyl)-3-[2-(2-methyl-1,3-thiazol-4-yl)ethenyl]-17-oxa-4-azabicyclo[14.1.0]heptadecane-5,9-dione