5-(7-Chloro-4-oxo-4H-benzo[d][1,2,3]triazin-3-yl)-1-phenyl-1H-pyrazole-4-carboxylic acid ethyl ester | 454705-27-2

• 分子结构分类: 有机化合物 - 有机杂环化合物 - 唑类
• 英文名称: 5-(7-Chloro-4-oxo-4H-benzo[d][1,2,3]triazin-3-yl)-1-phenyl-1H-pyrazole-4-carboxylic acid ethyl ester
• CAS: 454705-27-2
• 化学式: C₁₉H₁₄ClN₅O₃
• 分子量: 395.805
• InChiKey: WWKSAIIAHNCPRY-UHFFFAOYSA-N

反应信息

• 作为反应物：
  描述：

  5-(7-Chloro-4-oxo-4H-benzo[d][1,2,3]triazin-3-yl)-1-phenyl-1H-pyrazole-4-carboxylic acid ethyl ester 在 溶剂黄146 、 potassium iodide 作用下， 反应 1.0h， 以75%的产率得到5-(4-Chloro-2-iodo-benzoylamino)-1-phenyl-1H-pyrazole-4-carboxylic acid ethyl ester
  参考文献：
  名称：

  Synthesis and antifungal activity of new N-(1-phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides

  摘要：

  N-(1-Phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides 6, with a Benodanil-like structure, were synthesized by refluxing in acetic acid the corresponding benzotriazin ones 5 with potassium iodide for 1 h in order to study the role on the antifungal activity of the N-substitution with an aromatic heterocyclic system on benzamide moiety. Among the tested iododerivatives, compounds 6d,f,g,h possess interesting activities toward some phytopathogenic fungal strains. (C) 2002 Editions scientifiques et medicales Elsevier SAS. All rights reserved.

  DOI：

  10.1016/s0014-827x(01)01190-9
• 作为产物：
  描述：

  5-(2-Amino-4-chloro-benzoylamino)-1-phenyl-1H-pyrazole-4-carboxylic acid ethyl ester 在 盐酸 、 sodium nitrite 作用下， 反应 1.0h， 以96%的产率得到5-(7-Chloro-4-oxo-4H-benzo[d][1,2,3]triazin-3-yl)-1-phenyl-1H-pyrazole-4-carboxylic acid ethyl ester
  参考文献：
  名称：

  Synthesis and antifungal activity of new N-(1-phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides

  摘要：

  N-(1-Phenyl-4-carbetoxypyrazol-5-yl)-, N-(indazol-3-yl)- and N-(indazol-5-yl)-2-iodobenzamides 6, with a Benodanil-like structure, were synthesized by refluxing in acetic acid the corresponding benzotriazin ones 5 with potassium iodide for 1 h in order to study the role on the antifungal activity of the N-substitution with an aromatic heterocyclic system on benzamide moiety. Among the tested iododerivatives, compounds 6d,f,g,h possess interesting activities toward some phytopathogenic fungal strains. (C) 2002 Editions scientifiques et medicales Elsevier SAS. All rights reserved.

  DOI：

  10.1016/s0014-827x(01)01190-9