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—— (6S)-N-(2H-chromen-3-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C19H24N4O
(6S)-N-(2H-chromen-3-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(2S)-2-[(2S)-1-acetylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H26N4O3
6-[[(2S)-2-[(2S)-1-acetylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6R)-N-(2H-chromen-3-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C19H24N4O
(6R)-N-(2H-chromen-3-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-(1,3-benzodioxol-4-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H22N4O2
(6S)-N-(1,3-benzodioxol-4-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(N-[(1S)-1-cyclopropylethyl]-4-methoxyanilino)methyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H25N3O3
6-[(N-[(1S)-1-cyclopropylethyl]-4-methoxyanilino)methyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6R)-N-(1,3-benzodioxol-4-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H22N4O2
(6R)-N-(1,3-benzodioxol-4-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H21N5O
(6S)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(N-[(1R)-1-cyclopropylethyl]-4-methoxyanilino)methyl]-1,3-dimethylpyrimidine-2,4-dione —— C19H25N3O3
6-[(N-[(1R)-1-cyclopropylethyl]-4-methoxyanilino)methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-[[(2R)-2-[(2R)-1-acetylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H26N4O3
6-[[(2R)-2-[(2R)-1-acetylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-fluoro-N-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]quinazolin-4-amine —— C16H22FN5
6-fluoro-N-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]quinazolin-4-amine
—— 6-[(2R)-2-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]tetrazolo[1,5-b]pyridazine —— C14H19N9
6-[(2R)-2-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]tetrazolo[1,5-b]pyridazine
—— 6-[[(3S)-1-(2-methoxyethyl)piperidin-3-yl]amino]pyridine-3-carbonitrile —— C14H20N4O
6-[[(3S)-1-(2-methoxyethyl)piperidin-3-yl]amino]pyridine-3-carbonitrile
—— (6S)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H24N4O
(6S)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H24N4O
(6R)-N-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[(4-methylsulfonylphenyl)methyl]-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H24N4O2S
(6S)-N-[(4-methylsulfonylphenyl)methyl]-2-propan-2-yl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[2-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]-2-oxoethyl]-methylamino]pyridine-3-carbonitrile —— C17H25N5O2
6-[[2-[4-[(2S)-2-hydroxybutyl]piperazin-1-yl]-2-oxoethyl]-methylamino]pyridine-3-carbonitrile
—— 6-methyl-5-[(2R)-2-methylbutyl]-2-(2-methylpropylsulfanyl)-3H-thieno[2,3-d]pyrimidin-4-one —— C16H24N2OS2
6-methyl-5-[(2R)-2-methylbutyl]-2-(2-methylpropylsulfanyl)-3H-thieno[2,3-d]pyrimidin-4-one
—— 6-fluoro-N-[(2R)-1-(4-methylpiperazin-1-yl)propan-2-yl]quinazolin-4-amine —— C16H22FN5
6-fluoro-N-[(2R)-1-(4-methylpiperazin-1-yl)propan-2-yl]quinazolin-4-amine
—— 6-[[2-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]-2-oxoethyl]-methylamino]pyridine-3-carbonitrile —— C17H25N5O2
6-[[2-[4-[(2R)-2-hydroxybutyl]piperazin-1-yl]-2-oxoethyl]-methylamino]pyridine-3-carbonitrile
—— 6-[[(2S)-2-[(2R)-1-acetylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C17H26N4O3
6-[[(2S)-2-[(2R)-1-acetylpyrrolidin-2-yl]pyrrolidin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— 6-(3,5-dimethylpyrazol-1-yl)-N-[(3R)-1-ethylpyrrolidin-3-yl]-N-methylpyridine-3-carboxamide —— C18H25N5O
6-(3,5-dimethylpyrazol-1-yl)-N-[(3R)-1-ethylpyrrolidin-3-yl]-N-methylpyridine-3-carboxamide
—— 6-[(2S)-2-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]tetrazolo[1,5-b]pyridazine —— C14H19N9
6-[(2S)-2-[(3,5-dimethyl-1,2,4-triazol-1-yl)methyl]piperidin-1-yl]tetrazolo[1,5-b]pyridazine
—— 6-methyl-N-[(2R)-3-methyl-2-[(6-methylpyridine-3-carbonyl)amino]butyl]pyridine-3-carboxamide —— C19H24N4O2
6-methyl-N-[(2R)-3-methyl-2-[(6-methylpyridine-3-carbonyl)amino]butyl]pyridine-3-carboxamide
—— 6-(furan-2-yl)-3-[(3R)-3-pyrrolidin-1-ylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C19H23N3O3
6-(furan-2-yl)-3-[(3R)-3-pyrrolidin-1-ylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— 6-(furan-2-yl)-3-[(3S)-3-pyrrolidin-1-ylpiperidine-1-carbonyl]-1H-pyridin-2-one —— C19H23N3O3
6-(furan-2-yl)-3-[(3S)-3-pyrrolidin-1-ylpiperidine-1-carbonyl]-1H-pyridin-2-one
—— 6-[[(3R)-1-(2-methoxyethyl)piperidin-3-yl]amino]pyridine-3-carbonitrile —— C14H20N4O
6-[[(3R)-1-(2-methoxyethyl)piperidin-3-yl]amino]pyridine-3-carbonitrile
—— 6-butyl-2-[[(4R)-1,3-dioxan-4-yl]methylsulfanyl]-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine —— C16H24N4O2S
6-butyl-2-[[(4R)-1,3-dioxan-4-yl]methylsulfanyl]-5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine
—— 6-[[(R)-(3,5-dimethylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C18H20O3S
6-[[(R)-(3,5-dimethylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— 6-[[(S)-(3,5-dimethylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine —— C18H20O3S
6-[[(S)-(3,5-dimethylphenyl)methylsulfinyl]methyl]-2,3-dihydro-1,4-benzodioxine
—— (6S)-N,N-bis[[2-(2-fluorophenyl)-1,3-thiazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C26H22F2N6S2
(6S)-N,N-bis[[2-(2-fluorophenyl)-1,3-thiazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N,N-bis[[2-(2-fluorophenyl)-1,3-thiazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C26H22F2N6S2
(6R)-N,N-bis[[2-(2-fluorophenyl)-1,3-thiazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-methoxybenzoate —— C17H15ClO5
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-methoxybenzoate
—— (6R)-N-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H21N5O
(6R)-N-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H21N5O
(6S)-N-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-oxo-1H-quinoline-2-carboxylate —— C19H14ClNO5
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-oxo-1H-quinoline-2-carboxylate
—— 6-[5-[5-methyl-4-[(3R)-3-methylmorpholine-4-carbonyl]triazol-1-yl]-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile —— C24H25N7O2
6-[5-[5-methyl-4-[(3R)-3-methylmorpholine-4-carbonyl]triazol-1-yl]-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile
—— (6R)-2-ethyl-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H21N5O2
(6R)-2-ethyl-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-methyl-2-[3-[(6-methyl-1H-benzimidazol-2-yl)sulfanyl]propylsulfanyl]-1H-benzimidazole —— C19H20N4S2
6-methyl-2-[3-[(6-methyl-1H-benzimidazol-2-yl)sulfanyl]propylsulfanyl]-1H-benzimidazole
—— 6-[5-[5-methyl-4-[(3S)-3-methylmorpholine-4-carbonyl]triazol-1-yl]-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile —— C24H25N7O2
6-[5-[5-methyl-4-[(3S)-3-methylmorpholine-4-carbonyl]triazol-1-yl]-3,4-dihydro-1H-isoquinolin-2-yl]pyridine-3-carbonitrile
—— (6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-chloro-2-nitrobenzoate —— C16H11Cl2NO6
(6-chloro-4H-1,3-benzodioxin-8-yl)methyl 4-chloro-2-nitrobenzoate
—— (6S)-2-ethyl-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H21N5O2
(6S)-2-ethyl-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(3S)-4-(2-ethoxyethyl)-3-methylpiperazin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione —— C16H28N4O3
6-[[(3S)-4-(2-ethoxyethyl)-3-methylpiperazin-1-yl]methyl]-1,3-dimethylpyrimidine-2,4-dione
—— (6R)-5-benzyl-9,9-dimethyl-6-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H28N2O
(6R)-5-benzyl-9,9-dimethyl-6-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6S)-5-benzyl-9,9-dimethyl-6-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one —— C28H28N2O
(6S)-5-benzyl-9,9-dimethyl-6-phenyl-6,8,10,11-tetrahydrobenzo[b][1,4]benzodiazepin-7-one
—— (6R)-N-[[1-(2-fluoro-5-methylphenyl)tetrazol-5-yl]methyl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H19FN8
(6R)-N-[[1-(2-fluoro-5-methylphenyl)tetrazol-5-yl]methyl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[[1-(2-fluoro-5-methylphenyl)tetrazol-5-yl]methyl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H19FN8
(6S)-N-[[1-(2-fluoro-5-methylphenyl)tetrazol-5-yl]methyl]-2-methyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C17H18FNO3
6-[[[(1S)-1-(3-fluoro-4-methoxyphenyl)ethyl]amino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-[[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propylamino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one —— C19H26N4O2S
6-[[3-(4-cyclopentyl-5-methylsulfanyl-1,2,4-triazol-3-yl)propylamino]methylidene]-2-methoxycyclohexa-2,4-dien-1-one
—— 6-[[[(1R)-2-methyl-1-thiophen-2-ylpropyl]amino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one —— C15H16N2O3S
6-[[[(1R)-2-methyl-1-thiophen-2-ylpropyl]amino]methylidene]-4-nitrocyclohexa-2,4-dien-1-one
—— 6-[[[2-[(dimethylamino)methyl]phenyl]methylamino]methylidene]-4-methoxycyclohexa-2,4-dien-1-one —— C18H22N2O2
6-[[[2-[(dimethylamino)methyl]phenyl]methylamino]methylidene]-4-methoxycyclohexa-2,4-dien-1-one