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—— 6-[(E)-3-[4-(difluoromethoxy)phenyl]prop-2-enoyl]-4H-1,4-benzoxazin-3-one —— C18H13F2NO4
6-[(E)-3-[4-(difluoromethoxy)phenyl]prop-2-enoyl]-4H-1,4-benzoxazin-3-one
—— 6-[(E)-3-[3-methoxy-4-(3-methylbutoxy)phenyl]prop-2-enoyl]-4H-1,4-benzoxazin-3-one —— C23H25NO5
6-[(E)-3-[3-methoxy-4-(3-methylbutoxy)phenyl]prop-2-enoyl]-4H-1,4-benzoxazin-3-one
—— (6R)-N-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16FN5O
(6R)-N-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-2-ethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H19N5O
(6R)-2-ethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(E)-3-(2,3,4,5,6-pentafluorophenyl)prop-2-enoyl]-4H-1,4-benzoxazin-3-one —— C17H8F5NO3
6-[(E)-3-(2,3,4,5,6-pentafluorophenyl)prop-2-enoyl]-4H-1,4-benzoxazin-3-one
—— 6-[(E)-3-(2,4-dimethylphenyl)prop-2-enoyl]-4H-1,4-benzoxazin-3-one —— C19H17NO3
6-[(E)-3-(2,4-dimethylphenyl)prop-2-enoyl]-4H-1,4-benzoxazin-3-one
—— (6S)-6-[[[(2S)-1-(3-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6S)-6-[[[(2S)-1-(3-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C12H16N6O
(6R)-N-[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H19N5O
(6S)-N-[[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-Amino-3-methyl-5-[2-(4-methylpiperazin-1-yl)-1,3-thiazol-4-yl]-1-(2-methylpropyl)pyrimidine-2,4-dione —— C17H26N6O2S
6-Amino-3-methyl-5-[2-(4-methylpiperazin-1-yl)-1,3-thiazol-4-yl]-1-(2-methylpropyl)pyrimidine-2,4-dione
—— (6S)-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H17N5O2
(6S)-N-[[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(E)-3-[4-(trifluoromethyl)phenyl]prop-2-enoyl]-4H-1,4-benzoxazin-3-one —— C18H12F3NO3
6-[(E)-3-[4-(trifluoromethyl)phenyl]prop-2-enoyl]-4H-1,4-benzoxazin-3-one
—— (6S)-6-[[[(2R)-1-(3-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C18H25N5O2
(6S)-6-[[[(2R)-1-(3-methylphenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-N-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16FN5O
(6S)-N-[[2-(4-fluorophenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-2-ethyl-N-[[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H18N6O2
(6S)-2-ethyl-N-[[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[[2-(2,4-dimethylphenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H21N5O
(6S)-N-[[2-(2,4-dimethylphenyl)-1,3-oxazol-4-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-2-ethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H19N5O
(6S)-2-ethyl-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-Chloro-7-methyl-4-[(2-nitrophenoxy)methyl]chromen-2-one —— C17H12ClNO5
6-Chloro-7-methyl-4-[(2-nitrophenoxy)methyl]chromen-2-one
—— 6-[[(6S)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridine-3-carbonitrile —— C15H18N6
6-[[(6S)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridine-3-carbonitrile
—— (6R)-N-[(1-phenylpyrazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H18N6
(6R)-N-[(1-phenylpyrazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-2-ethyl-N-[(5-fluoroquinolin-8-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H20FN5
(6S)-2-ethyl-N-[(5-fluoroquinolin-8-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[[5-(3-methylfuran-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C14H16N6O2
(6R)-N-[[5-(3-methylfuran-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[[(6R)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridine-3-carbonitrile —— C15H18N6
6-[[(6R)-3-ethyl-5,6,7,8-tetrahydro-[1,2,4]triazolo[4,3-a]pyridin-6-yl]methylamino]pyridine-3-carbonitrile
—— (6R)-2-ethyl-N-[(5-fluoroquinolin-8-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C18H20FN5
(6R)-2-ethyl-N-[(5-fluoroquinolin-8-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6-methoxy-1H-indol-2-yl)-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C19H22N4O2
(6-methoxy-1H-indol-2-yl)-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— 6-methyl-2-[(3R)-3-methyl-4-(4-methyl-1,3-thiazol-2-yl)piperazin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole —— C14H18N6S2
6-methyl-2-[(3R)-3-methyl-4-(4-methyl-1,3-thiazol-2-yl)piperazin-1-yl]imidazo[2,1-b][1,3,4]thiadiazole
—— (6S)-N-[[3-(1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16N6O3
(6S)-N-[[3-(1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[4-[[(2R)-oxan-2-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine —— C15H22N6O
6-[4-[[(2R)-oxan-2-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine
—— (6-methoxy-1H-indol-2-yl)-[(3R)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C19H22N4O2
(6-methoxy-1H-indol-2-yl)-[(3R)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— 6-[4-[[(2S)-oxan-2-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine —— C15H22N6O
6-[4-[[(2S)-oxan-2-yl]methyl]piperazin-1-yl]-[1,2,4]triazolo[4,3-b]pyridazine
—— (6S)-N-[(1-phenylpyrazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H18N6
(6S)-N-[(1-phenylpyrazol-3-yl)methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6R)-N-[[3-(1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C16H16N6O3
(6R)-N-[[3-(1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— 6-[(1R)-1-cyano-2-cyclobutyl-2-oxoethyl]-N,N-diethylpyridine-3-sulfonamide —— C16H21N3O3S
6-[(1R)-1-cyano-2-cyclobutyl-2-oxoethyl]-N,N-diethylpyridine-3-sulfonamide
—— 6-chloro-2-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine —— C16H19ClN6
6-chloro-2-[[(3S)-3-(1,2,4-triazol-1-ylmethyl)piperidin-1-yl]methyl]imidazo[1,2-a]pyridine
—— 6-[(1S)-1-cyano-2-cyclobutyl-2-oxoethyl]-N,N-diethylpyridine-3-sulfonamide —— C16H21N3O3S
6-[(1S)-1-cyano-2-cyclobutyl-2-oxoethyl]-N,N-diethylpyridine-3-sulfonamide
—— [6-(dimethylamino)pyridazin-3-yl]-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C16H22N6O
[6-(dimethylamino)pyridazin-3-yl]-[(3S)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— (6R)-6-[[[(2S)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6R)-6-[[[(2S)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-N-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H20N6O
(6R)-N-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-N-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C17H20N6O
(6S)-N-[3-(3-phenyl-1,2,4-oxadiazol-5-yl)propyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— [6-(dimethylamino)pyridazin-3-yl]-[(3R)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone —— C16H22N6O
[6-(dimethylamino)pyridazin-3-yl]-[(3R)-3-(2-methylimidazol-1-yl)piperidin-1-yl]methanone
—— (6R)-5-acetyl-6-(3-nitrophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C21H19N3O4
(6R)-5-acetyl-6-(3-nitrophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one
—— (6S)-N-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H15FN6O
(6S)-N-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-6-[[[(2S)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6S)-6-[[[(2S)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6R)-N-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C15H15FN6O
(6R)-N-[[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 4-(hydroxymethyl)benzoate —— C19H15ClO5
(6-Chloro-7-methyl-2-oxochromen-4-yl)methyl 4-(hydroxymethyl)benzoate
—— (6R)-6-[[[(2R)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6R)-6-[[[(2R)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— (6S)-6-[[[(2R)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide —— C17H22FN5O2
(6S)-6-[[[(2R)-1-(3-fluorophenoxy)propan-2-yl]amino]methyl]-1,5,6,7-tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide
—— [6-(dimethylamino)pyridazin-3-yl]-[(3R)-3-(2-ethylimidazol-1-yl)piperidin-1-yl]methanone —— C17H24N6O
[6-(dimethylamino)pyridazin-3-yl]-[(3R)-3-(2-ethylimidazol-1-yl)piperidin-1-yl]methanone
—— (6R)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine —— C13H14N6O2
(6R)-N-[[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl]-5,6,7,8-tetrahydro-[1,2,4]triazolo[1,5-a]pyridin-6-amine
—— (6S)-5-acetyl-6-(3-nitrophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one —— C21H19N3O4
(6S)-5-acetyl-6-(3-nitrophenyl)-8,9,10,11-tetrahydro-6H-benzo[b][1,4]benzodiazepin-7-one