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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-(cyclopropylamino)-N-[2-methyl-2-[[(1R)-1-phenylethyl]amino]propyl]-1,3-thiazole-4-carboxamide —— C19H26N4OS
2-(cyclopropylamino)-N-[2-methyl-2-[[(1R)-1-phenylethyl]amino]propyl]-1,3-thiazole-4-carboxamide
—— methyl 1-[2-[methyl-[(1R,2R)-2-methylcyclohexyl]amino]-2-oxoethyl]-1,2,4-triazole-3-carboxylate —— C14H22N4O3
methyl 1-[2-[methyl-[(1R,2R)-2-methylcyclohexyl]amino]-2-oxoethyl]-1,2,4-triazole-3-carboxylate
—— 1-(3-chlorophenyl)-N-[(2R)-3-(cyclopropylmethoxy)-2-hydroxypropyl]pyrazole-3-carboxamide —— C17H20ClN3O3
1-(3-chlorophenyl)-N-[(2R)-3-(cyclopropylmethoxy)-2-hydroxypropyl]pyrazole-3-carboxamide
—— 1-(3-chlorophenyl)-N-[(2S)-3-(cyclopropylmethoxy)-2-hydroxypropyl]pyrazole-3-carboxamide —— C17H20ClN3O3
1-(3-chlorophenyl)-N-[(2S)-3-(cyclopropylmethoxy)-2-hydroxypropyl]pyrazole-3-carboxamide
—— N-cyclopentyl-2-[2-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl]sulfanylacetamide —— C20H26N4O3S
N-cyclopentyl-2-[2-[(1,5-dimethyl-3-oxo-2-phenylpyrazol-4-yl)amino]-2-oxoethyl]sulfanylacetamide
—— 2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[2-propan-2-yl-4-[(2S)-1,1,1-trifluoro-2-hydroxypropan-2-yl]pyrazol-3-yl]acetamide —— C21H23F3N4O3
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[2-propan-2-yl-4-[(2S)-1,1,1-trifluoro-2-hydroxypropan-2-yl]pyrazol-3-yl]acetamide
—— 2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[2-propan-2-yl-4-[(2R)-1,1,1-trifluoro-2-hydroxypropan-2-yl]pyrazol-3-yl]acetamide —— C21H23F3N4O3
2-(5-methyl-2-phenyl-1,3-oxazol-4-yl)-N-[2-propan-2-yl-4-[(2R)-1,1,1-trifluoro-2-hydroxypropan-2-yl]pyrazol-3-yl]acetamide
—— 1-(2-fluorophenyl)-N-[(2R)-2-(hydroxymethyl)-3-[3-(trifluoromethoxy)phenyl]propyl]pyrazole-3-carboxamide —— C21H19F4N3O3
1-(2-fluorophenyl)-N-[(2R)-2-(hydroxymethyl)-3-[3-(trifluoromethoxy)phenyl]propyl]pyrazole-3-carboxamide
—— [1-(3,4-dichlorophenyl)pyrazol-3-yl]-[(3S)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C20H24Cl2N4O2
[1-(3,4-dichlorophenyl)pyrazol-3-yl]-[(3S)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1S,2R)-2-methylsulfonylcyclopentyl]butanamide —— C19H24ClN3O4S
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1S,2R)-2-methylsulfonylcyclopentyl]butanamide
—— 1-(4-fluorophenyl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C18H19FN4O3S2
1-(4-fluorophenyl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— [3-(2-chlorophenyl)-1-methylpyrazol-4-yl]-[(3S)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C21H27ClN4O2
[3-(2-chlorophenyl)-1-methylpyrazol-4-yl]-[(3S)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— [1-(3,4-dichlorophenyl)pyrazol-3-yl]-[(3R)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C20H24Cl2N4O2
[1-(3,4-dichlorophenyl)pyrazol-3-yl]-[(3R)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— N-[(1S,3R)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide —— C20H19N3O2S
N-[(1S,3R)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide
—— 2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]acetamide —— C16H19FN2O3S2
2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]acetamide
—— 1-(4-methylphenyl)-N-[(2S)-4-[(S)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide —— C22H25N3O2S
1-(4-methylphenyl)-N-[(2S)-4-[(S)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide
—— 3-[4-[(Z)-[(E)-(1-methyl-2-oxoindol-3-ylidene)hydrazinylidene]methyl]-3-phenylpyrazol-1-yl]propanenitrile —— C22H18N6O
3-[4-[(Z)-[(E)-(1-methyl-2-oxoindol-3-ylidene)hydrazinylidene]methyl]-3-phenylpyrazol-1-yl]propanenitrile
—— [3-(2-chlorophenyl)-1-methylpyrazol-4-yl]-[(3R)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone —— C21H27ClN4O2
[3-(2-chlorophenyl)-1-methylpyrazol-4-yl]-[(3R)-3-(morpholin-4-ylmethyl)piperidin-1-yl]methanone
—— 1-(4-methylphenyl)-N-[(2R)-4-[(R)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide —— C22H25N3O2S
1-(4-methylphenyl)-N-[(2R)-4-[(R)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide
—— N-[(1R,3R)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide —— C20H19N3O2S
N-[(1R,3R)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide
—— [(3S)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]-[4-(1,2,4-triazol-1-yl)phenyl]methanone —— C20H21N5O
[(3S)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]-[4-(1,2,4-triazol-1-yl)phenyl]methanone
—— N-[(1S,3S)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide —— C20H19N3O2S
N-[(1S,3S)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide
—— [2-(methoxymethyl)-1,3-thiazol-4-yl]-[(3R)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]methanone —— C17H21N3O2S
[2-(methoxymethyl)-1,3-thiazol-4-yl]-[(3R)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]methanone
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1S,2S)-2-methylsulfonylcyclopentyl]butanamide —— C19H24ClN3O4S
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1S,2S)-2-methylsulfonylcyclopentyl]butanamide
—— 1-(4-methylphenyl)-N-[(2S)-4-[(R)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide —— C22H25N3O2S
1-(4-methylphenyl)-N-[(2S)-4-[(R)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide
—— 1-(2-fluorophenyl)-N-[(2S)-2-(hydroxymethyl)-3-[3-(trifluoromethoxy)phenyl]propyl]pyrazole-3-carboxamide —— C21H19F4N3O3
1-(2-fluorophenyl)-N-[(2S)-2-(hydroxymethyl)-3-[3-(trifluoromethoxy)phenyl]propyl]pyrazole-3-carboxamide
—— 1-(4-methylphenyl)-N-[(2R)-4-[(S)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide —— C22H25N3O2S
1-(4-methylphenyl)-N-[(2R)-4-[(S)-methylsulfinyl]butan-2-yl]-3-phenylpyrazole-4-carboxamide
—— (E)-3-[1-[(3S)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-2-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)prop-2-enenitrile —— C18H17N5O3S2
(E)-3-[1-[(3S)-1,1-dioxothiolan-3-yl]-3,5-dimethylpyrazol-4-yl]-2-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)prop-2-enenitrile
—— (E)-3-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-2-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)prop-2-enenitrile —— C18H9ClN4OS2
(E)-3-[2-(4-chlorophenyl)-1,3-thiazol-4-yl]-2-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)prop-2-enenitrile
—— [(3R)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]-[4-(1,2,4-triazol-1-yl)phenyl]methanone —— C20H21N5O
[(3R)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]-[4-(1,2,4-triazol-1-yl)phenyl]methanone
—— 2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]acetamide —— C16H19FN2O3S2
2-[2-(3-fluorophenyl)-1,3-thiazol-4-yl]-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]acetamide
—— N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-3-(5-phenylpyrazol-1-yl)benzamide —— C21H23N3O3S
N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-3-(5-phenylpyrazol-1-yl)benzamide
—— 4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1R,2S)-2-methylsulfonylcyclopentyl]butanamide —— C19H24ClN3O4S
4-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1R,2S)-2-methylsulfonylcyclopentyl]butanamide
—— [2-(methoxymethyl)-1,3-thiazol-4-yl]-[(3S)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]methanone —— C17H21N3O2S
[2-(methoxymethyl)-1,3-thiazol-4-yl]-[(3S)-3-propan-2-yl-3,4-dihydro-2H-quinoxalin-1-yl]methanone
—— N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide —— C18H17N5O2
N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide
—— N-[(1R,3S)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide —— C20H19N3O2S
N-[(1R,3S)-1-oxothiolan-3-yl]-3-(5-phenylpyrazol-1-yl)benzamide
—— 1-[(1S,2R)-2-(hydroxymethyl)cyclohexyl]-3-(3-pyrazol-1-ylphenyl)urea —— C17H22N4O2
1-[(1S,2R)-2-(hydroxymethyl)cyclohexyl]-3-(3-pyrazol-1-ylphenyl)urea
—— 1-(4-fluorophenyl)-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C18H19FN4O3S2
1-(4-fluorophenyl)-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— methyl 5-[[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]carbamoyl]-1-phenylpyrazole-3-carboxylate —— C25H25N5O3
methyl 5-[[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]carbamoyl]-1-phenylpyrazole-3-carboxylate
—— N-[(2R)-2-(2,4-difluorophenyl)-2-hydroxypropyl]-1,5-dimethylpyrazole-4-carboxamide —— C15H17F2N3O2
N-[(2R)-2-(2,4-difluorophenyl)-2-hydroxypropyl]-1,5-dimethylpyrazole-4-carboxamide
—— N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide —— C18H17N5O2
N-[(1S,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-2-[4-(tetrazol-1-yl)phenyl]acetamide
—— N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C17H22N2O4S2
N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide
—— 1-(4-chlorophenyl)-5-(furan-2-yl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]pyrazole-3-carboxamide —— C19H20ClN3O4S
1-(4-chlorophenyl)-5-(furan-2-yl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]pyrazole-3-carboxamide
—— 2-(5-chlorothiophen-2-yl)-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-1,3-thiazole-4-carboxamide —— C13H15ClN2O3S3
2-(5-chlorothiophen-2-yl)-N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-1,3-thiazole-4-carboxamide
—— 1-[(1S,2R)-2-imidazol-1-ylcyclopentyl]-3-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]urea —— C19H19F3N6O
1-[(1S,2R)-2-imidazol-1-ylcyclopentyl]-3-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]urea
—— 2-(5-chlorothiophen-2-yl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-1,3-thiazole-4-carboxamide —— C13H15ClN2O3S3
2-(5-chlorothiophen-2-yl)-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-1,3-thiazole-4-carboxamide
—— 2-[(4-fluorophenyl)methyl]-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-1,3-thiazole-5-carboxamide —— C16H19FN2O3S2
2-[(4-fluorophenyl)methyl]-N-methyl-N-[(2R)-1-methylsulfonylpropan-2-yl]-1,3-thiazole-5-carboxamide
—— 1-[(1R,2R)-2-imidazol-1-ylcyclopentyl]-3-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]urea —— C19H19F3N6O
1-[(1R,2R)-2-imidazol-1-ylcyclopentyl]-3-[2-pyrazol-1-yl-5-(trifluoromethyl)phenyl]urea
—— 1-[(1S,2S)-2-(hydroxymethyl)cyclohexyl]-3-(3-pyrazol-1-ylphenyl)urea —— C17H22N4O2
1-[(1S,2S)-2-(hydroxymethyl)cyclohexyl]-3-(3-pyrazol-1-ylphenyl)urea
—— N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide —— C17H22N2O4S2
N-methyl-N-[(2S)-1-methylsulfonylpropan-2-yl]-2-[(2-phenyl-1,3-oxazol-4-yl)methylsulfanyl]acetamide