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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-1-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-1-methylurea —— C16H25N5OS
3-[(1R)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-1-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-1-methylurea
—— (2S,6R)-2,6-dimethyl-N-(4-methyl-1-phenylpyrazol-3-yl)morpholine-4-carboxamide —— C17H22N4O2
(2S,6R)-2,6-dimethyl-N-(4-methyl-1-phenylpyrazol-3-yl)morpholine-4-carboxamide
—— 1-(5-fluoro-2-pyrazol-1-ylphenyl)-3-[(3S)-2-oxoazepan-3-yl]urea —— C16H18FN5O2
1-(5-fluoro-2-pyrazol-1-ylphenyl)-3-[(3S)-2-oxoazepan-3-yl]urea
—— 1-(5-fluoro-2-pyrazol-1-ylphenyl)-3-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]urea —— C16H19FN4O2
1-(5-fluoro-2-pyrazol-1-ylphenyl)-3-[(1S)-1-[(2S)-oxolan-2-yl]ethyl]urea
—— [(3S)-oxolan-3-yl] 5-methyl-1-phenylpyrazole-3-carboxylate —— C15H16N2O3
[(3S)-oxolan-3-yl] 5-methyl-1-phenylpyrazole-3-carboxylate
—— 3-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-1-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-1-methylurea —— C16H25N5OS
3-[(1S)-1-(1,3-dimethylpyrazol-4-yl)ethyl]-1-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-1-methylurea
—— 1-[5-[(4-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]-3-[[(3R)-oxolan-3-yl]methyl]urea —— C15H17FN4O2S
1-[5-[(4-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]-3-[[(3R)-oxolan-3-yl]methyl]urea
—— N-[(1R,2S)-2-ethylcyclohexyl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C17H24N4O2
N-[(1R,2S)-2-ethylcyclohexyl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— N-[(1R,2R)-2-ethylcyclohexyl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C17H24N4O2
N-[(1R,2R)-2-ethylcyclohexyl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— (1-Phenyltetrazol-5-yl)methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate —— C20H18N4O3
(1-Phenyltetrazol-5-yl)methyl 2-(5,6-dimethyl-1-benzofuran-3-yl)acetate
—— N-[(1S,2R)-2-ethylcyclohexyl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C17H24N4O2
N-[(1S,2R)-2-ethylcyclohexyl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— tert-butyl N-[(3R)-1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]carbamate —— C17H29N3O3
tert-butyl N-[(3R)-1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]carbamate
—— [(2S)-oxan-2-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C15H19N3O4
[(2S)-oxan-2-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— N-cyclopropyl-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C16H20N4O4S
N-cyclopropyl-N-[(3S)-1,1-dioxothiolan-3-yl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— tert-butyl N-[(3S)-1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]carbamate —— C17H29N3O3
tert-butyl N-[(3S)-1-[(5-tert-butyl-1,3-oxazol-2-yl)methyl]pyrrolidin-3-yl]carbamate
—— [(1S,6S)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C17H21N3O3
[(1S,6S)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— [(1R)-cyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C16H19N3O3
[(1R)-cyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— 1-[(3R)-3-cyano-2-oxo-3-(4-phenyl-1,3-thiazol-2-yl)propyl]-1,2,4-triazole-3-carbonitrile —— C16H10N6OS
1-[(3R)-3-cyano-2-oxo-3-(4-phenyl-1,3-thiazol-2-yl)propyl]-1,2,4-triazole-3-carbonitrile
—— N-[(2R)-butan-2-yl]-N-butyl-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C17H26N4O2
N-[(2R)-butan-2-yl]-N-butyl-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— 1-[(3S)-3-cyano-2-oxo-3-(4-phenyl-1,3-thiazol-2-yl)propyl]-1,2,4-triazole-3-carbonitrile —— C16H10N6OS
1-[(3S)-3-cyano-2-oxo-3-(4-phenyl-1,3-thiazol-2-yl)propyl]-1,2,4-triazole-3-carbonitrile
—— N-cyclopropyl-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C16H20N4O4S
N-cyclopropyl-N-[(3R)-1,1-dioxothiolan-3-yl]-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— [(1S,6R)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C17H21N3O3
[(1S,6R)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— [(1R,6R)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C17H21N3O3
[(1R,6R)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— [(2R)-oxan-2-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C15H19N3O4
[(2R)-oxan-2-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— N-[(2S)-butan-2-yl]-N-butyl-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide —— C17H26N4O2
N-[(2S)-butan-2-yl]-N-butyl-3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanamide
—— [(1R,6S)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C17H21N3O3
[(1R,6S)-6-methylcyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— [(1S)-cyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate —— C16H19N3O3
[(1S)-cyclohex-3-en-1-yl]methyl 3-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)propanoate
—— (4R)-3-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]-N-methyl-N-propan-2-yl-1,3-thiazolidine-4-carboxamide —— C18H20Cl2N4O2S
(4R)-3-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]-N-methyl-N-propan-2-yl-1,3-thiazolidine-4-carboxamide
—— (2R)-4-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]morpholine-2-carboxamide —— C15H14Cl2N4O3
(2R)-4-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]morpholine-2-carboxamide
—— (4S)-3-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]-N-methyl-N-propan-2-yl-1,3-thiazolidine-4-carboxamide —— C18H20Cl2N4O2S
(4S)-3-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]-N-methyl-N-propan-2-yl-1,3-thiazolidine-4-carboxamide
—— 2-[(2R)-1-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]piperidin-2-yl]acetamide —— C17H18Cl2N4O2
2-[(2R)-1-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]piperidin-2-yl]acetamide
—— 1-(3,4-dichlorophenyl)-N-[(2S)-1-(dimethylamino)-4-methylpentan-2-yl]pyrazole-3-carboxamide —— C18H24Cl2N4O
1-(3,4-dichlorophenyl)-N-[(2S)-1-(dimethylamino)-4-methylpentan-2-yl]pyrazole-3-carboxamide
—— N-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1-(3,4-dichlorophenyl)pyrazole-3-carboxamide —— C18H20Cl2N4O2
N-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1-(3,4-dichlorophenyl)pyrazole-3-carboxamide
—— N-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1-(3,4-dichlorophenyl)pyrazole-3-carboxamide —— C18H20Cl2N4O2
N-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1-(3,4-dichlorophenyl)pyrazole-3-carboxamide
—— (2S)-4-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]morpholine-2-carboxamide —— C15H14Cl2N4O3
(2S)-4-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]morpholine-2-carboxamide
—— 2-[(2S)-1-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]piperidin-2-yl]acetamide —— C17H18Cl2N4O2
2-[(2S)-1-[1-(3,4-dichlorophenyl)pyrazole-3-carbonyl]piperidin-2-yl]acetamide
—— 1-(3,4-dichlorophenyl)-N-[(2R)-1-(dimethylamino)-4-methylpentan-2-yl]pyrazole-3-carboxamide —— C18H24Cl2N4O
1-(3,4-dichlorophenyl)-N-[(2R)-1-(dimethylamino)-4-methylpentan-2-yl]pyrazole-3-carboxamide
—— (2R)-3-(3-fluorophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-2-(5-methyltetrazol-1-yl)propanamide —— C21H20FN7O
(2R)-3-(3-fluorophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-2-(5-methyltetrazol-1-yl)propanamide
—— (4R)-3-(3,3-dimethylbutanoyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-1,3-thiazolidine-4-carboxamide —— C20H26N4O2S
(4R)-3-(3,3-dimethylbutanoyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-1,3-thiazolidine-4-carboxamide
—— 4-imidazol-1-yl-3-nitro-N-[5-[(1R)-1-phenylpropyl]-1,3,4-thiadiazol-2-yl]benzamide —— C21H18N6O3S
4-imidazol-1-yl-3-nitro-N-[5-[(1R)-1-phenylpropyl]-1,3,4-thiadiazol-2-yl]benzamide
—— (3R)-1-benzyl-N-(4-methyl-1-phenylpyrazol-3-yl)-3-(trifluoromethyl)pyrrolidine-3-carboxamide —— C23H23F3N4O
(3R)-1-benzyl-N-(4-methyl-1-phenylpyrazol-3-yl)-3-(trifluoromethyl)pyrrolidine-3-carboxamide
—— (3S)-1-benzyl-N-(4-methyl-1-phenylpyrazol-3-yl)-3-(trifluoromethyl)pyrrolidine-3-carboxamide —— C23H23F3N4O
(3S)-1-benzyl-N-(4-methyl-1-phenylpyrazol-3-yl)-3-(trifluoromethyl)pyrrolidine-3-carboxamide
—— (4S)-3-(3,3-dimethylbutanoyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-1,3-thiazolidine-4-carboxamide —— C20H26N4O2S
(4S)-3-(3,3-dimethylbutanoyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-1,3-thiazolidine-4-carboxamide
—— (2S)-3-(3-fluorophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-2-(5-methyltetrazol-1-yl)propanamide —— C21H20FN7O
(2S)-3-(3-fluorophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-2-(5-methyltetrazol-1-yl)propanamide
—— N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-N-methyl-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C21H21N5OS2
N-[(1S)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-N-methyl-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide
—— (3R)-1-(2-bromophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-5-oxopyrrolidine-3-carboxamide —— C21H19BrN4O2
(3R)-1-(2-bromophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-5-oxopyrrolidine-3-carboxamide
—— N-(4-methyl-1-phenylpyrazol-3-yl)-2-[(2S)-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]sulfanylpyridine-3-carboxamide —— C23H25N5O2S
N-(4-methyl-1-phenylpyrazol-3-yl)-2-[(2S)-1-oxo-1-pyrrolidin-1-ylpropan-2-yl]sulfanylpyridine-3-carboxamide
—— (3S)-1-(2-bromophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-5-oxopyrrolidine-3-carboxamide —— C21H19BrN4O2
(3S)-1-(2-bromophenyl)-N-(4-methyl-1-phenylpyrazol-3-yl)-5-oxopyrrolidine-3-carboxamide
—— (2S)-N-(4-methyl-1-phenylpyrazol-3-yl)-2-phenoxy-2-phenylacetamide —— C24H21N3O2
(2S)-N-(4-methyl-1-phenylpyrazol-3-yl)-2-phenoxy-2-phenylacetamide
—— N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-N-methyl-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide —— C21H21N5OS2
N-[(1R)-1-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-N-methyl-1-phenyl-5-thiophen-2-yl-1,2,4-triazole-3-carboxamide