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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-N-(5-bromo-2-pyrazol-1-ylphenyl)-5-oxo-1-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide —— C16H14BrF3N4O2
(3S)-N-(5-bromo-2-pyrazol-1-ylphenyl)-5-oxo-1-(2,2,2-trifluoroethyl)pyrrolidine-3-carboxamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-2-[2-[(4-fluorophenyl)methyl]-1,3-thiazol-4-yl]-N-(2-methoxyethyl)acetamide —— C19H23FN2O4S2
N-[(3S)-1,1-dioxothiolan-3-yl]-2-[2-[(4-fluorophenyl)methyl]-1,3-thiazol-4-yl]-N-(2-methoxyethyl)acetamide
—— N-[(S)-cyano-(2,3-dichlorophenyl)methyl]-1-(4-fluorophenyl)pyrazole-3-carboxamide —— C18H11Cl2FN4O
N-[(S)-cyano-(2,3-dichlorophenyl)methyl]-1-(4-fluorophenyl)pyrazole-3-carboxamide
—— ethyl (3S)-3-[[4-(1H-imidazol-2-yl)phenyl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C22H21N5O3
ethyl (3S)-3-[[4-(1H-imidazol-2-yl)phenyl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-2-(2-methylphenyl)-1,3-thiazole-4-carboxamide —— C18H22N2O4S2
N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-2-(2-methylphenyl)-1,3-thiazole-4-carboxamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-5-methyl-1-phenylpyrazole-3-carboxamide —— C18H23N3O4S
N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-5-methyl-1-phenylpyrazole-3-carboxamide
—— 2-(3,4-dichlorophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide —— C17H18Cl2N2O4S2
2-(3,4-dichlorophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide
—— 2-(3,4-dichlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide —— C17H18Cl2N2O4S2
2-(3,4-dichlorophenyl)-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide
—— 1-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-3-methoxyurea —— C11H20N4O2
1-[(2R)-3-(3,5-dimethylpyrazol-1-yl)-2-methylpropyl]-3-methoxyurea
—— 2-benzyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide —— C18H22N2O4S2
2-benzyl-N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide
—— 2-benzyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide —— C18H22N2O4S2
2-benzyl-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-1,3-thiazole-4-carboxamide
—— N-[(2S)-1-(2,4-dimethylphenyl)propan-2-yl]-2-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C23H28N4O2S
N-[(2S)-1-(2,4-dimethylphenyl)propan-2-yl]-2-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— ethyl (3S)-3-[[(2R)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C21H32N4O3
ethyl (3S)-3-[[(2R)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— N-[(3R)-1,1-dioxothiolan-3-yl]-2-[2-[(4-fluorophenyl)methyl]-1,3-thiazol-4-yl]-N-(2-methoxyethyl)acetamide —— C19H23FN2O4S2
N-[(3R)-1,1-dioxothiolan-3-yl]-2-[2-[(4-fluorophenyl)methyl]-1,3-thiazol-4-yl]-N-(2-methoxyethyl)acetamide
—— N-[(3R)-1,1-dioxothiolan-3-yl]-1-(2-fluorophenyl)-N-(2-methoxyethyl)pyrazole-3-carboxamide —— C17H20FN3O4S
N-[(3R)-1,1-dioxothiolan-3-yl]-1-(2-fluorophenyl)-N-(2-methoxyethyl)pyrazole-3-carboxamide
—— (3R)-1-[2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)benzoyl]pyrrolidine-3-carboxamide —— C18H22N4O3
(3R)-1-[2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)benzoyl]pyrrolidine-3-carboxamide
—— N-[(3S)-1,1-dioxothiolan-3-yl]-1-(4-fluorophenyl)-N-(2-methoxyethyl)pyrazole-3-carboxamide —— C17H20FN3O4S
N-[(3S)-1,1-dioxothiolan-3-yl]-1-(4-fluorophenyl)-N-(2-methoxyethyl)pyrazole-3-carboxamide
—— 3-(2-chlorophenyl)-1-methyl-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]pyrazole-4-carboxamide —— C16H17ClN4O2
3-(2-chlorophenyl)-1-methyl-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]pyrazole-4-carboxamide
—— 1-(4-bromophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)pyrazole-4-carboxamide —— C17H20BrN3O4S
1-(4-bromophenyl)-N-[(3S)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)pyrazole-4-carboxamide
—— ethyl (3R)-3-[[(2R)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C21H32N4O3
ethyl (3R)-3-[[(2R)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— ethyl (3R)-3-[[4-(1H-imidazol-2-yl)phenyl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C22H21N5O3
ethyl (3R)-3-[[4-(1H-imidazol-2-yl)phenyl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— 3-(2-chlorophenyl)-1-methyl-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]pyrazole-4-carboxamide —— C16H17ClN4O2
3-(2-chlorophenyl)-1-methyl-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]pyrazole-4-carboxamide
—— 1-[3-[3-(3-fluorophenyl)-1H-pyrazol-5-yl]propyl]-1-methyl-3-[[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]methyl]urea —— C25H32FN5OS
1-[3-[3-(3-fluorophenyl)-1H-pyrazol-5-yl]propyl]-1-methyl-3-[[(3R)-1-(thiophen-2-ylmethyl)piperidin-3-yl]methyl]urea
—— 1-[3-[3-(3-fluorophenyl)-1H-pyrazol-5-yl]propyl]-1-methyl-3-[[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]methyl]urea —— C25H32FN5OS
1-[3-[3-(3-fluorophenyl)-1H-pyrazol-5-yl]propyl]-1-methyl-3-[[(3S)-1-(thiophen-2-ylmethyl)piperidin-3-yl]methyl]urea
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-2-(2-methylphenyl)-1,3-thiazole-4-carboxamide —— C18H22N2O4S2
N-[(3R)-1,1-dioxothiolan-3-yl]-N-(2-methoxyethyl)-2-(2-methylphenyl)-1,3-thiazole-4-carboxamide
—— 4-(2-methoxyphenyl)-3-[(1R)-1-phenylpropyl]sulfanyl-1,2,4-triazole —— C18H19N3OS
4-(2-methoxyphenyl)-3-[(1R)-1-phenylpropyl]sulfanyl-1,2,4-triazole
—— 2-(2-chlorophenyl)-N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide —— C19H24ClN3O2S
2-(2-chlorophenyl)-N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide
—— 2-(2-chlorophenyl)-N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide —— C19H24ClN3O2S
2-(2-chlorophenyl)-N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide
—— ethyl (3R)-3-[[(2S)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C21H32N4O3
ethyl (3R)-3-[[(2S)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— 2-(2,4-dimethylphenyl)-4-methyl-N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide —— C22H31N3O2S
2-(2,4-dimethylphenyl)-4-methyl-N-[[(2S)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide
—— 1-(3-chloro-4-fluorophenyl)-N,5-dimethyl-N-[(1S)-1-pyridin-3-ylethyl]triazole-4-carboxamide —— C18H17ClFN5O
1-(3-chloro-4-fluorophenyl)-N,5-dimethyl-N-[(1S)-1-pyridin-3-ylethyl]triazole-4-carboxamide
—— ethyl (3S)-3-[[(2S)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C21H32N4O3
ethyl (3S)-3-[[(2S)-1-(dimethylamino)-4-methylpentan-2-yl]carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— N-[(3S)-1-[1-(3-chloro-4-fluorophenyl)-5-methyltriazole-4-carbonyl]piperidin-3-yl]butanamide —— C19H23ClFN5O2
N-[(3S)-1-[1-(3-chloro-4-fluorophenyl)-5-methyltriazole-4-carbonyl]piperidin-3-yl]butanamide
—— 3-(2-chlorophenyl)-1-methyl-N-[(2S)-2-morpholin-4-yl-2-[4-(trifluoromethyl)phenyl]ethyl]pyrazole-4-carboxamide —— C24H24ClF3N4O2
3-(2-chlorophenyl)-1-methyl-N-[(2S)-2-morpholin-4-yl-2-[4-(trifluoromethyl)phenyl]ethyl]pyrazole-4-carboxamide
—— tert-butyl (3R)-3-[[[1-(3-chloro-4-fluorophenyl)-5-methyltriazole-4-carbonyl]amino]methyl]piperidine-1-carboxylate —— C21H27ClFN5O3
tert-butyl (3R)-3-[[[1-(3-chloro-4-fluorophenyl)-5-methyltriazole-4-carbonyl]amino]methyl]piperidine-1-carboxylate
—— (3S)-1-[2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)benzoyl]pyrrolidine-3-carboxamide —— C18H22N4O3
(3S)-1-[2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)benzoyl]pyrrolidine-3-carboxamide
—— 3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-N-[(2S)-1-(2,4-dimethylphenyl)propan-2-yl]propanamide —— C23H24F2N2O2
3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-N-[(2S)-1-(2,4-dimethylphenyl)propan-2-yl]propanamide
—— 2-(2,4-dimethylphenyl)-4-methyl-N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide —— C22H31N3O2S
2-(2,4-dimethylphenyl)-4-methyl-N-[[(2R)-4-(2-methylpropyl)morpholin-2-yl]methyl]-1,3-thiazole-5-carboxamide
—— N-[(3S)-1-[1-[4-(difluoromethoxy)phenyl]-5-methyltriazole-4-carbonyl]piperidin-3-yl]butanamide —— C20H25F2N5O3
N-[(3S)-1-[1-[4-(difluoromethoxy)phenyl]-5-methyltriazole-4-carbonyl]piperidin-3-yl]butanamide
—— N-[(2R)-1-(2,4-dimethylphenyl)propan-2-yl]-2-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide —— C23H28N4O2S
N-[(2R)-1-(2,4-dimethylphenyl)propan-2-yl]-2-[[4-(4-methoxyphenyl)-5-methyl-1,2,4-triazol-3-yl]sulfanyl]acetamide
—— 3-(2-chlorophenyl)-1-methyl-N-[(2R)-2-morpholin-4-yl-2-[4-(trifluoromethyl)phenyl]ethyl]pyrazole-4-carboxamide —— C24H24ClF3N4O2
3-(2-chlorophenyl)-1-methyl-N-[(2R)-2-morpholin-4-yl-2-[4-(trifluoromethyl)phenyl]ethyl]pyrazole-4-carboxamide
—— [1-(3-chloro-4-fluorophenyl)-5-methyltriazol-4-yl]-[(2R)-2-(1-ethylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C23H22ClFN6O
[1-(3-chloro-4-fluorophenyl)-5-methyltriazol-4-yl]-[(2R)-2-(1-ethylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— 1-(3-chloro-4-fluorophenyl)-N-[(2S)-2-(3-chlorophenyl)-2-morpholin-4-ylethyl]-5-methyltriazole-4-carboxamide —— C22H22Cl2FN5O2
1-(3-chloro-4-fluorophenyl)-N-[(2S)-2-(3-chlorophenyl)-2-morpholin-4-ylethyl]-5-methyltriazole-4-carboxamide
—— 1-[4-(difluoromethoxy)phenyl]-N-[(3-fluorophenyl)methyl]-5-methyl-N-[[(2S)-oxolan-2-yl]methyl]triazole-4-carboxamide —— C23H23F3N4O3
1-[4-(difluoromethoxy)phenyl]-N-[(3-fluorophenyl)methyl]-5-methyl-N-[[(2S)-oxolan-2-yl]methyl]triazole-4-carboxamide
—— 1-(3-chloro-4-fluorophenyl)-5-methyl-N-[(1S)-2-methyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide —— C20H19ClFN7O
1-(3-chloro-4-fluorophenyl)-5-methyl-N-[(1S)-2-methyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide
—— 1-(3-chloro-4-fluorophenyl)-N-[(2S)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-5-methyltriazole-4-carboxamide —— C22H22Cl2FN5O2
1-(3-chloro-4-fluorophenyl)-N-[(2S)-2-(4-chlorophenyl)-2-morpholin-4-ylethyl]-5-methyltriazole-4-carboxamide
—— 1-[4-(difluoromethoxy)phenyl]-5-methyl-N-[(1R)-2-methyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide —— C21H21F2N7O2
1-[4-(difluoromethoxy)phenyl]-5-methyl-N-[(1R)-2-methyl-1-([1,2,4]triazolo[4,3-a]pyridin-3-yl)propyl]triazole-4-carboxamide
—— 3-(2-chlorophenyl)-N-[(1S)-6-(difluoromethoxy)-1,2,3,4-tetrahydronaphthalen-1-yl]-1-methylpyrazole-4-carboxamide —— C22H20ClF2N3O2
3-(2-chlorophenyl)-N-[(1S)-6-(difluoromethoxy)-1,2,3,4-tetrahydronaphthalen-1-yl]-1-methylpyrazole-4-carboxamide
—— [1-[4-(difluoromethoxy)phenyl]-5-methyltriazol-4-yl]-[(2S)-2-(1-ethylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone —— C24H24F2N6O2
[1-[4-(difluoromethoxy)phenyl]-5-methyltriazol-4-yl]-[(2S)-2-(1-ethylbenzimidazol-2-yl)pyrrolidin-1-yl]methanone
—— N-[(2R)-2-(3-chlorophenyl)-2-morpholin-4-ylethyl]-1-[4-(difluoromethoxy)phenyl]-5-methyltriazole-4-carboxamide —— C23H24ClF2N5O3
N-[(2R)-2-(3-chlorophenyl)-2-morpholin-4-ylethyl]-1-[4-(difluoromethoxy)phenyl]-5-methyltriazole-4-carboxamide