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中文名称 英文名称 CAS号 化学式 结构式图片
—— (1S)-N-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide —— C15H22N2O2S
(1S)-N-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide
—— (1R)-N-[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide —— C15H22N2O2S
(1R)-N-[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide
—— [(3aR,7aR)-1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl]-[1-(3-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone —— C21H21FN4OS
[(3aR,7aR)-1,3,3a,4,5,6,7,7a-octahydroisoindol-2-yl]-[1-(3-fluorophenyl)-5-thiophen-2-yl-1,2,4-triazol-3-yl]methanone
—— (1S)-N-[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide —— C15H22N2O2S
(1S)-N-[[2-[(1S)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide
—— (1R)-N-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide —— C15H22N2O2S
(1R)-N-[[2-[(1R)-1-methoxyethyl]-1,3-thiazol-4-yl]methyl]-N-methylcyclohex-3-ene-1-carboxamide
—— tert-butyl (3S)-3-[[(1R)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate —— C21H27FN4O4
tert-butyl (3S)-3-[[(1R)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate
—— [(3R)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]-(2-thiophen-2-yl-1,3-thiazol-4-yl)methanone —— C18H17N3O2S2
[(3R)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]-(2-thiophen-2-yl-1,3-thiazol-4-yl)methanone
—— tert-butyl (3R)-3-[[(1R)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate —— C21H27FN4O4
tert-butyl (3R)-3-[[(1R)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate
—— tert-butyl (3R)-3-[[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate —— C21H27FN4O4
tert-butyl (3R)-3-[[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate
—— tert-butyl (3S)-3-[[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate —— C21H27FN4O4
tert-butyl (3S)-3-[[(1S)-1-[3-(3-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl]carbamoyl]-3-methylpyrrolidine-1-carboxylate
—— (2R)-N-[4-fluoro-3-(5-methyltetrazol-1-yl)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C23H23FN8O
(2R)-N-[4-fluoro-3-(5-methyltetrazol-1-yl)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— 3-chloro-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-nitrobenzamide —— C19H16ClFN4O3
3-chloro-N-[(1R)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-nitrobenzamide
—— ethyl 2-[2-[[[(2R)-1-cyanopropan-2-yl]-methylcarbamoyl]amino]-1,3-thiazol-4-yl]acetate —— C13H18N4O3S
ethyl 2-[2-[[[(2R)-1-cyanopropan-2-yl]-methylcarbamoyl]amino]-1,3-thiazol-4-yl]acetate
—— [(3S)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]-(2-thiophen-2-yl-1,3-thiazol-4-yl)methanone —— C18H17N3O2S2
[(3S)-3-(pyridin-3-ylmethoxy)pyrrolidin-1-yl]-(2-thiophen-2-yl-1,3-thiazol-4-yl)methanone
—— (2S)-N-[4-fluoro-3-(5-methyltetrazol-1-yl)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C23H23FN8O
(2S)-N-[4-fluoro-3-(5-methyltetrazol-1-yl)phenyl]-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— (1S,3R)-3-[(R)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine —— C13H22N2OS2
(1S,3R)-3-[(R)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine
—— 5-(3-chloro-4-fluorophenyl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide —— C15H14ClFN4O2
5-(3-chloro-4-fluorophenyl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
—— (2S)-3-[5-(2-methylphenyl)tetrazol-2-yl]propane-1,2-diol —— C11H14N4O2
(2S)-3-[5-(2-methylphenyl)tetrazol-2-yl]propane-1,2-diol
—— 3-[(1R)-1-[ethyl-[(2-methyl-1,3-thiazol-4-yl)methyl]amino]ethyl]phenol —— C15H20N2OS
3-[(1R)-1-[ethyl-[(2-methyl-1,3-thiazol-4-yl)methyl]amino]ethyl]phenol
—— (1S,3S)-3-[(R)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine —— C13H22N2OS2
(1S,3S)-3-[(R)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine
—— 5-(3-chloro-4-fluorophenyl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide —— C15H14ClFN4O2
5-(3-chloro-4-fluorophenyl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1H-pyrazole-4-carboxamide
—— (2S)-3-(5-tert-butyltetrazol-1-yl)propane-1,2-diol —— C8H16N4O2
(2S)-3-(5-tert-butyltetrazol-1-yl)propane-1,2-diol
—— (1S,3S)-3-[(S)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine —— C13H22N2OS2
(1S,3S)-3-[(S)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine
—— (2S)-N-(4-chloro-2-fluorophenyl)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C21H20ClFN4O
(2S)-N-(4-chloro-2-fluorophenyl)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— (2R)-3-[5-(2-methylphenyl)tetrazol-2-yl]propane-1,2-diol —— C11H14N4O2
(2R)-3-[5-(2-methylphenyl)tetrazol-2-yl]propane-1,2-diol
—— (1S,3R)-3-[(S)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine —— C13H22N2OS2
(1S,3R)-3-[(S)-ethylsulfinyl]-N-[(2-methyl-1,3-thiazol-4-yl)methyl]cyclohexan-1-amine
—— 3-chloro-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-nitrobenzamide —— C19H16ClFN4O3
3-chloro-N-[(1S)-1-[1-(4-fluorophenyl)-5-methylpyrazol-4-yl]ethyl]-2-nitrobenzamide
—— (1R)-1-(5-ethyl-1,3-thiazol-2-yl)-N-(1H-pyrazol-5-ylmethyl)ethanamine —— C11H16N4S
(1R)-1-(5-ethyl-1,3-thiazol-2-yl)-N-(1H-pyrazol-5-ylmethyl)ethanamine
—— 3-[(1S)-1-[ethyl-[(2-methyl-1,3-thiazol-4-yl)methyl]amino]ethyl]phenol —— C15H20N2OS
3-[(1S)-1-[ethyl-[(2-methyl-1,3-thiazol-4-yl)methyl]amino]ethyl]phenol
—— (2R)-N-(4-chloro-2-fluorophenyl)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide —— C21H20ClFN4O
(2R)-N-(4-chloro-2-fluorophenyl)-2-(5-methyl-4-phenyl-1H-imidazol-2-yl)pyrrolidine-1-carboxamide
—— ethyl 2-[2-[[[(2S)-1-cyanopropan-2-yl]-methylcarbamoyl]amino]-1,3-thiazol-4-yl]acetate —— C13H18N4O3S
ethyl 2-[2-[[[(2S)-1-cyanopropan-2-yl]-methylcarbamoyl]amino]-1,3-thiazol-4-yl]acetate
—— (3R)-N-(3-chloro-2-fluorophenyl)-3-(5-phenyl-1H-imidazol-2-yl)piperidine-1-carboxamide —— C21H20ClFN4O
(3R)-N-(3-chloro-2-fluorophenyl)-3-(5-phenyl-1H-imidazol-2-yl)piperidine-1-carboxamide
—— (1S)-1-(5-ethyl-1,3-thiazol-2-yl)-N-(1H-pyrazol-5-ylmethyl)ethanamine —— C11H16N4S
(1S)-1-(5-ethyl-1,3-thiazol-2-yl)-N-(1H-pyrazol-5-ylmethyl)ethanamine
—— (3R)-3-(5-phenyl-1H-imidazol-2-yl)-N-[4-(pyrrolidine-1-carbonyl)phenyl]piperidine-1-carboxamide —— C26H29N5O2
(3R)-3-(5-phenyl-1H-imidazol-2-yl)-N-[4-(pyrrolidine-1-carbonyl)phenyl]piperidine-1-carboxamide
—— 1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1R,2R)-2-imidazol-1-ylcyclopentyl]urea —— C18H19ClN6O
1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1R,2R)-2-imidazol-1-ylcyclopentyl]urea
—— (2R)-7-chloro-2-methyl-5-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine —— C19H20ClN5O2S2
(2R)-7-chloro-2-methyl-5-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine
—— (2R)-N-[2-(difluoromethoxy)phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide —— C22H21F3N4O2
(2R)-N-[2-(difluoromethoxy)phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
—— 1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1S,2R)-2-imidazol-1-ylcyclopentyl]urea —— C18H19ClN6O
1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1S,2R)-2-imidazol-1-ylcyclopentyl]urea
—— (2R)-3-(5-tert-butyltetrazol-1-yl)propane-1,2-diol —— C8H16N4O2
(2R)-3-(5-tert-butyltetrazol-1-yl)propane-1,2-diol
—— (3S)-N-(3-chloro-2-fluorophenyl)-3-(5-phenyl-1H-imidazol-2-yl)piperidine-1-carboxamide —— C21H20ClFN4O
(3S)-N-(3-chloro-2-fluorophenyl)-3-(5-phenyl-1H-imidazol-2-yl)piperidine-1-carboxamide
—— (2S)-N-(3,5-dimethylphenyl)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide —— C23H25FN4O
(2S)-N-(3,5-dimethylphenyl)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
—— (2R)-N-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide —— C25H28FN5O2
(2R)-N-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
—— (2R)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]-N-(2-methylsulfanylphenyl)piperidine-1-carboxamide —— C22H23FN4OS
(2R)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]-N-(2-methylsulfanylphenyl)piperidine-1-carboxamide
—— tert-butyl (3R)-3-cyano-4-[1-(3-fluorophenyl)pyrazole-3-carbonyl]piperazine-1-carboxylate —— C20H22FN5O3
tert-butyl (3R)-3-cyano-4-[1-(3-fluorophenyl)pyrazole-3-carbonyl]piperazine-1-carboxylate
—— N-[2-[(1R)-1-(2,5-dichlorophenyl)ethyl]pyrazol-3-yl]-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)acetamide —— C19H16Cl2N6O2
N-[2-[(1R)-1-(2,5-dichlorophenyl)ethyl]pyrazol-3-yl]-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)acetamide
—— (2S)-7-chloro-2-methyl-5-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine —— C19H20ClN5O2S2
(2S)-7-chloro-2-methyl-5-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-3,4-dihydro-2H-1,5-benzothiazepine
—— (2S)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]-N-(2-methylsulfanylphenyl)piperidine-1-carboxamide —— C22H23FN4OS
(2S)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]-N-(2-methylsulfanylphenyl)piperidine-1-carboxamide
—— 1-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-3-[(2S)-1,1,1-trifluoro-3,3-dimethylbutan-2-yl]urea —— C17H21F3N4O2S
1-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-3-[(2S)-1,1,1-trifluoro-3,3-dimethylbutan-2-yl]urea
—— 1-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-3-[(2R)-1,1,1-trifluoro-3,3-dimethylbutan-2-yl]urea —— C17H21F3N4O2S
1-[5-[(3-methoxyphenyl)methyl]-1,3,4-thiadiazol-2-yl]-3-[(2R)-1,1,1-trifluoro-3,3-dimethylbutan-2-yl]urea
—— 1-(2-chlorophenyl)-5-methyl-N-[[(2S,3S)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide —— C19H25ClN4O2
1-(2-chlorophenyl)-5-methyl-N-[[(2S,3S)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide