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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[(3S)-3-anilinopiperidin-1-yl]-3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one —— C23H26N4O3
1-[(3S)-3-anilinopiperidin-1-yl]-3-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
—— N-(2,3-dimethyl-5-sulfamoylphenyl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C19H19FN4O4S
N-(2,3-dimethyl-5-sulfamoylphenyl)-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— N-(2,3-dimethyl-5-sulfamoylphenyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide —— C19H20N4O4S
N-(2,3-dimethyl-5-sulfamoylphenyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
—— 3-[N-methyl-4-[(Z)-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]anilino]propanenitrile —— C20H20N6S
3-[N-methyl-4-[(Z)-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]anilino]propanenitrile
—— 3-[N-ethyl-3-methyl-4-[(Z)-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]anilino]propanenitrile —— C22H24N6S
3-[N-ethyl-3-methyl-4-[(Z)-[3-(4-methylphenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]iminomethyl]anilino]propanenitrile
—— 4-[(Z)-[4-[ethyl(2-hydroxyethyl)amino]-2-methylphenyl]methylideneamino]-3-(4-methylphenyl)-1H-1,2,4-triazole-5-thione —— C21H25N5OS
4-[(Z)-[4-[ethyl(2-hydroxyethyl)amino]-2-methylphenyl]methylideneamino]-3-(4-methylphenyl)-1H-1,2,4-triazole-5-thione
—— 2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-(4-methyl-3-sulfamoylphenyl)acetamide —— C20H22N4O3S
2-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-(4-methyl-3-sulfamoylphenyl)acetamide
—— 1-[(2R)-1-hydroxy-3,3-dimethylbutan-2-yl]-3-(2-pyrazol-1-ylphenyl)urea —— C16H22N4O2
1-[(2R)-1-hydroxy-3,3-dimethylbutan-2-yl]-3-(2-pyrazol-1-ylphenyl)urea
—— (3R,4R)-4-methyl-N-[3-(1,3-oxazol-5-yl)phenyl]-1-([1,2,4]triazolo[4,3-a]pyrazin-8-yl)pyrrolidine-3-carboxamide —— C20H19N7O2
(3R,4R)-4-methyl-N-[3-(1,3-oxazol-5-yl)phenyl]-1-([1,2,4]triazolo[4,3-a]pyrazin-8-yl)pyrrolidine-3-carboxamide
—— 1-[(2S)-2-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)ethane-1,2-dione —— C25H24N4O3
1-[(2S)-2-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)ethane-1,2-dione
—— (3R,4S)-4-methyl-N-[3-(1,3-oxazol-5-yl)phenyl]-1-([1,2,4]triazolo[4,3-a]pyrazin-8-yl)pyrrolidine-3-carboxamide —— C20H19N7O2
(3R,4S)-4-methyl-N-[3-(1,3-oxazol-5-yl)phenyl]-1-([1,2,4]triazolo[4,3-a]pyrazin-8-yl)pyrrolidine-3-carboxamide
—— (E)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2R)-2-cyano-1-methoxypropan-2-yl]prop-2-enamide —— C15H21N3O2S
(E)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2R)-2-cyano-1-methoxypropan-2-yl]prop-2-enamide
—— 1-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-3-(2-pyrazol-1-ylphenyl)urea —— C16H22N4O2
1-[(2S)-1-hydroxy-3,3-dimethylbutan-2-yl]-3-(2-pyrazol-1-ylphenyl)urea
—— 1-[(2R)-2-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)ethane-1,2-dione —— C25H24N4O3
1-[(2R)-2-(1,3-benzoxazol-2-yl)piperidin-1-yl]-2-(3,5-dimethyl-1-phenylpyrazol-4-yl)ethane-1,2-dione
—— N-(4-methyl-3-sulfamoylphenyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide —— C18H18N4O4S
N-(4-methyl-3-sulfamoylphenyl)-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
—— N-[(3S)-1-propanoylpyrrolidin-3-yl]-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C15H17N3O2S2
N-[(3S)-1-propanoylpyrrolidin-3-yl]-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— 2-[(2R)-1-[[3-(3-nitrophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]-1,3-benzoxazole —— C21H19N5O4
2-[(2R)-1-[[3-(3-nitrophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]-1,3-benzoxazole
—— (3-propyl-1,2,4-oxadiazol-5-yl)methyl (3R)-thiolane-3-carboxylate —— C11H16N2O3S
(3-propyl-1,2,4-oxadiazol-5-yl)methyl (3R)-thiolane-3-carboxylate
—— (E)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2S)-2-cyano-1-methoxypropan-2-yl]prop-2-enamide —— C15H21N3O2S
(E)-3-(2-tert-butyl-1,3-thiazol-5-yl)-N-[(2S)-2-cyano-1-methoxypropan-2-yl]prop-2-enamide
—— 2-[(2S)-1-[[3-(3-nitrophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]-1,3-benzoxazole —— C21H19N5O4
2-[(2S)-1-[[3-(3-nitrophenyl)-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]-1,3-benzoxazole
—— (3-propyl-1,2,4-oxadiazol-5-yl)methyl (3S)-thiolane-3-carboxylate —— C11H16N2O3S
(3-propyl-1,2,4-oxadiazol-5-yl)methyl (3S)-thiolane-3-carboxylate
—— N-[(3R)-1-propanoylpyrrolidin-3-yl]-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C15H17N3O2S2
N-[(3R)-1-propanoylpyrrolidin-3-yl]-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— 1-[(Z)-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]methylideneamino]-3-(3-methoxyphenyl)thiourea —— C21H20N6OS
1-[(Z)-[1-(2-cyanoethyl)-3-phenylpyrazol-4-yl]methylideneamino]-3-(3-methoxyphenyl)thiourea
—— (3R)-5-N-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide —— C20H27N5O3
(3R)-5-N-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide
—— (3S)-5-N-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide —— C20H27N5O3
(3S)-5-N-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide
—— N-[(2R)-2-methyl-3-pyrazol-1-ylpropyl]-2-(prop-2-enylamino)-1,3-thiazole-5-carboxamide —— C14H19N5OS
N-[(2R)-2-methyl-3-pyrazol-1-ylpropyl]-2-(prop-2-enylamino)-1,3-thiazole-5-carboxamide
—— (3S)-5-N-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide —— C20H27N5O3
(3S)-5-N-[1-[(3S)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide
—— 4-bromo-N'-[4-(5-methylpyrazol-1-yl)benzoyl]-1H-pyrrole-2-carbohydrazide —— C16H14BrN5O2
4-bromo-N'-[4-(5-methylpyrazol-1-yl)benzoyl]-1H-pyrrole-2-carbohydrazide
—— 4-bromo-N'-(4-pyrazol-1-ylbenzoyl)-1H-pyrrole-2-carbohydrazide —— C15H12BrN5O2
4-bromo-N'-(4-pyrazol-1-ylbenzoyl)-1H-pyrrole-2-carbohydrazide
—— (3R)-5-N-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide —— C20H27N5O3
(3R)-5-N-[1-[(3R)-oxolan-3-yl]piperidin-4-yl]-2-phenyl-3,4-dihydropyrazole-3,5-dicarboxamide
—— N-[(2S)-2-methyl-3-pyrazol-1-ylpropyl]-2-(prop-2-enylamino)-1,3-thiazole-5-carboxamide —— C14H19N5OS
N-[(2S)-2-methyl-3-pyrazol-1-ylpropyl]-2-(prop-2-enylamino)-1,3-thiazole-5-carboxamide
—— N-[[1-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]pyrazol-4-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)ethanamine —— C15H22N4O2S2
N-[[1-[(3S)-3-methyl-1,1-dioxothiolan-3-yl]pyrazol-4-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)ethanamine
—— 2-(4-methoxyphenyl)-N-[(4-methoxyphenyl)methyl]-1,3-thiazole-4-carboxamide —— C19H18N2O3S
2-(4-methoxyphenyl)-N-[(4-methoxyphenyl)methyl]-1,3-thiazole-4-carboxamide
—— 3-(3-fluoro-4-methylphenyl)-5-[3-[(3S)-3-(5-methyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl]propyl]-1,2,4-oxadiazole —— C20H25FN6O
3-(3-fluoro-4-methylphenyl)-5-[3-[(3S)-3-(5-methyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl]propyl]-1,2,4-oxadiazole
—— N-[[1-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]pyrazol-4-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)ethanamine —— C15H22N4O2S2
N-[[1-[(3R)-3-methyl-1,1-dioxothiolan-3-yl]pyrazol-4-yl]methyl]-2-(2-methyl-1,3-thiazol-4-yl)ethanamine
—— N-[(4R)-6-chloro-1,1-dioxo-3,4-dihydro-2H-thiochromen-4-yl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H16ClN5O2S
N-[(4R)-6-chloro-1,1-dioxo-3,4-dihydro-2H-thiochromen-4-yl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine
—— 3-(3-fluoro-4-methylphenyl)-5-[3-[(3R)-3-(5-methyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl]propyl]-1,2,4-oxadiazole —— C20H25FN6O
3-(3-fluoro-4-methylphenyl)-5-[3-[(3R)-3-(5-methyl-1H-1,2,4-triazol-3-yl)piperidin-1-yl]propyl]-1,2,4-oxadiazole
—— 2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]-N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]acetamide —— C20H19N5O3
2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]-N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]acetamide
—— 2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]-N-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]acetamide —— C20H19N5O3
2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]-N-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]acetamide
—— 5-bromo-N-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide —— C19H17BrN4O3
5-bromo-N-[(1R)-1-(1-phenyltriazol-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide
—— 5-bromo-N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide —— C19H17BrN4O3
5-bromo-N-[(1S)-1-(1-phenyltriazol-4-yl)ethyl]-2,3-dihydro-1,4-benzodioxine-7-carboxamide
—— N-[(4S)-6-chloro-1,1-dioxo-3,4-dihydro-2H-thiochromen-4-yl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine —— C20H16ClN5O2S
N-[(4S)-6-chloro-1,1-dioxo-3,4-dihydro-2H-thiochromen-4-yl]-1-phenylpyrazolo[3,4-d]pyrimidin-4-amine
—— 6-[[(2R)-oxolan-2-yl]methyl-(thiophen-2-ylmethyl)amino]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C21H21N5O2S
6-[[(2R)-oxolan-2-yl]methyl-(thiophen-2-ylmethyl)amino]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 6-[[(2S)-oxolan-2-yl]methyl-(thiophen-2-ylmethyl)amino]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one —— C21H21N5O2S
6-[[(2S)-oxolan-2-yl]methyl-(thiophen-2-ylmethyl)amino]-1-phenyl-2H-pyrazolo[3,4-d]pyrimidin-4-one
—— 1-[2-[(3R)-oxolan-3-yl]oxyphenyl]-3-[4-(1,2,4-triazol-1-yl)-3-(trifluoromethyl)phenyl]urea —— C20H18F3N5O3
1-[2-[(3R)-oxolan-3-yl]oxyphenyl]-3-[4-(1,2,4-triazol-1-yl)-3-(trifluoromethyl)phenyl]urea
—— 4-[[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]amino]-N-methyl-3-nitrobenzamide —— C21H23N5O3
4-[[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]amino]-N-methyl-3-nitrobenzamide
—— N-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-5-nitropyridin-2-amine —— C18H19N5O2
N-[(1S)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-5-nitropyridin-2-amine
—— N-[(2S)-4-(furan-2-yl)-4-oxobutan-2-yl]-4-(1,3-oxazol-5-yl)benzamide —— C18H16N2O4
N-[(2S)-4-(furan-2-yl)-4-oxobutan-2-yl]-4-(1,3-oxazol-5-yl)benzamide
—— N-[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-6,7-difluoroquinazolin-4-amine —— C21H19F2N5
N-[(1R)-1-[4-(3,5-dimethylpyrazol-1-yl)phenyl]ethyl]-6,7-difluoroquinazolin-4-amine
—— 4-[(3S)-5-(3-bromophenyl)-3-(3-methyl-1-phenylpyrazol-4-yl)-3,4-dihydropyrazol-2-yl]-4-oxobutanoic acid —— C23H21BrN4O3
4-[(3S)-5-(3-bromophenyl)-3-(3-methyl-1-phenylpyrazol-4-yl)-3,4-dihydropyrazol-2-yl]-4-oxobutanoic acid