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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)butanamide —— C22H23N5O2S
N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)butanamide
—— 2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R,2S)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C21H20ClFN4OS
2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R,2S)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]tetrazolo[1,5-b]pyridazin-6-amine —— C16H15FN8
N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]tetrazolo[1,5-b]pyridazin-6-amine
—— 2-(3-ethyl-2-oxobenzimidazol-1-yl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]acetamide —— C23H25N5O2
2-(3-ethyl-2-oxobenzimidazol-1-yl)-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]acetamide
—— N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-1-methylsulfonylpiperidine-4-carboxamide —— C19H26N4O3S
N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-1-methylsulfonylpiperidine-4-carboxamide
—— N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)butanamide —— C22H23N5O2S
N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(3-thiophen-2-yl-1,2,4-oxadiazol-5-yl)butanamide
—— 3-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]propanamide —— C24H33N5O
3-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]-N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]propanamide
—— 3-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]propanamide —— C24H33N5O
3-[3,5-dimethyl-1-(2-methylpropyl)pyrazol-4-yl]-N-[(1R)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]propanamide
—— (2S,3S)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine —— C19H21N5O2S2
(2S,3S)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine
—— (2R,3R)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine —— C19H21N5O2S2
(2R,3R)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine
—— 5-[[4-[(3R)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C18H21F3N4OS
5-[[4-[(3R)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one —— C20H24ClN3O2
1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
—— 1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one —— C20H25N3O2
1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
—— 1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one —— C20H24ClN3O2
1-[(4aR,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
—— 2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2R)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C21H20ClFN4OS
2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2R)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— 2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R,2R)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C21H20ClFN4OS
2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1R,2R)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— 1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one —— C20H24FN3O2
1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
—— 1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one —— C20H25N3O2
1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propan-1-one
—— 4-(5-methylpyrazol-1-yl)-N'-[2-(3-oxo-1,4-benzoxazin-4-yl)acetyl]benzohydrazide —— C21H19N5O4
4-(5-methylpyrazol-1-yl)-N'-[2-(3-oxo-1,4-benzoxazin-4-yl)acetyl]benzohydrazide
—— 1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propan-1-one —— C24H33N3O2
1-[(4aS,8aR)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propan-1-one
—— 1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one —— C20H24ClN3O2
1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
—— (2S,3R)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine —— C19H21N5O2S2
(2S,3R)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine
—— (2R,3S)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine —— C19H21N5O2S2
(2R,3S)-2,3-dimethyl-4-[[1-(4-methylsulfonylphenyl)tetrazol-5-yl]methyl]-2,3-dihydro-1,4-benzothiazine
—— N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-1-methylsulfonylpiperidine-4-carboxamide —— C19H26N4O3S
N-[(1S)-1-[4-(2-methylimidazol-1-yl)phenyl]ethyl]-1-methylsulfonylpiperidine-4-carboxamide
—— 5-[[4-[(3S)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole —— C18H21F3N4OS
5-[[4-[(3S)-thiolan-3-yl]piperazin-1-yl]methyl]-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole
—— 2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2S)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide —— C21H20ClFN4OS
2-[3-(4-chlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-4-yl]-N-[(1S,2S)-5-fluoro-2-methyl-1,2,3,4-tetrahydronaphthalen-1-yl]acetamide
—— 4,5-dichloro-N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-1H-pyrrole-2-carboxamide —— C17H15Cl2FN4O
4,5-dichloro-N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-1H-pyrrole-2-carboxamide
—— methyl 5-[(2S,3S)-2,3-dimethyl-2,3-dihydro-1,4-benzothiazine-4-carbonyl]-1-phenylpyrazole-3-carboxylate —— C22H21N3O3S
methyl 5-[(2S,3S)-2,3-dimethyl-2,3-dihydro-1,4-benzothiazine-4-carbonyl]-1-phenylpyrazole-3-carboxylate
—— 4,5-dichloro-N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-1H-pyrrole-2-carboxamide —— C17H15Cl2FN4O
4,5-dichloro-N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-1H-pyrrole-2-carboxamide
—— 1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propan-1-one —— C24H33N3O2
1-[(4aR,8aS)-3,4,4a,5,6,7,8,8a-octahydro-1H-isoquinolin-2-yl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propan-1-one
—— N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-oxochromene-2-carboxamide —— C22H18FN3O3
N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-oxochromene-2-carboxamide
—— N-[(1R)-1-(2,4-difluorophenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide —— C23H25F2N3O2
N-[(1R)-1-(2,4-difluorophenyl)ethyl]-3-[1-(3-methoxyphenyl)-3,5-dimethylpyrazol-4-yl]propanamide
—— (E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]prop-2-enamide —— C20H17ClFN5OS
(E)-3-(6-chloroimidazo[2,1-b][1,3]thiazol-5-yl)-N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]prop-2-enamide
—— N-[(1S)-1-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl]-2-naphthalen-1-ylacetamide —— C22H18ClN3O2
N-[(1S)-1-[5-(4-chlorophenyl)-1,2,4-oxadiazol-3-yl]ethyl]-2-naphthalen-1-ylacetamide
—— 2-(methylsulfanylmethyl)-5-[(S)-phenyl-(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl-1,3,4-oxadiazole —— C19H16N4O2S2
2-(methylsulfanylmethyl)-5-[(S)-phenyl-(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]sulfanyl-1,3,4-oxadiazole
—— [(3R)-3-(3-phenylpropoxy)pyrrolidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone —— C20H27N3O2
[(3R)-3-(3-phenylpropoxy)pyrrolidin-1-yl]-(1,3,5-trimethylpyrazol-4-yl)methanone
—— 5-[(R)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C22H17N5OS2
5-[(R)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(4-propylphenyl)propanamide —— C20H20FN3O2
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(4-propylphenyl)propanamide
—— 3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-(2,4-difluorophenyl)ethyl]propanamide —— C19H16ClF2N3O2
3-[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[(1S)-1-(2,4-difluorophenyl)ethyl]propanamide
—— 5-[(S)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C24H19N5O2S
5-[(S)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— (8aR)-7-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1,2,5,6,8,8a-hexahydroimidazo[1,5-a]pyrazin-3-one —— C16H16F3N5O2
(8aR)-7-[[3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]-1,2,5,6,8,8a-hexahydroimidazo[1,5-a]pyrazin-3-one
—— 5-[(R)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C24H19N5O2S
5-[(R)-[5-(furan-2-yl)-4-prop-2-enyl-1,2,4-triazol-3-yl]sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(4-oxo-3H-quinazolin-2-yl)butanamide —— C24H24FN5O2
N-[(1R)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(4-oxo-3H-quinazolin-2-yl)butanamide
—— N-[(1R)-1-(2,4-difluorophenyl)ethyl]-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C19H16F3N3O2
N-[(1R)-1-(2,4-difluorophenyl)ethyl]-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— methyl 5-[(2R,3S)-2,3-dimethyl-2,3-dihydro-1,4-benzothiazine-4-carbonyl]-1-phenylpyrazole-3-carboxylate —— C22H21N3O3S
methyl 5-[(2R,3S)-2,3-dimethyl-2,3-dihydro-1,4-benzothiazine-4-carbonyl]-1-phenylpyrazole-3-carboxylate
—— N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(4-oxo-3H-quinazolin-2-yl)butanamide —— C24H24FN5O2
N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]-4-(4-oxo-3H-quinazolin-2-yl)butanamide
—— N-[(1S)-1-(2,4-difluorophenyl)ethyl]-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C19H16F3N3O2
N-[(1S)-1-(2,4-difluorophenyl)ethyl]-3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— 5-[(S)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole —— C22H17N5OS2
5-[(S)-(4-methyl-5-thiophen-2-yl-1,2,4-triazol-3-yl)sulfanyl-phenylmethyl]-3-phenyl-1,2,4-oxadiazole
—— 3-(3-chlorophenyl)-N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]propanamide —— C21H21ClFN3O
3-(3-chlorophenyl)-N-[(1S)-1-[3-fluoro-4-(2-methylimidazol-1-yl)phenyl]ethyl]propanamide
—— methyl 5-[(2S,3R)-2,3-dimethyl-2,3-dihydro-1,4-benzothiazine-4-carbonyl]-1-phenylpyrazole-3-carboxylate —— C22H21N3O3S
methyl 5-[(2S,3R)-2,3-dimethyl-2,3-dihydro-1,4-benzothiazine-4-carbonyl]-1-phenylpyrazole-3-carboxylate