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中文名称 英文名称 CAS号 化学式 结构式图片
—— (3S)-3-ethyl-4-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperazin-2-one —— C16H17FN4O2
(3S)-3-ethyl-4-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperazin-2-one
—— (3R)-3-ethyl-4-(5-methyl-1-phenylpyrazole-4-carbonyl)piperazin-2-one —— C17H20N4O2
(3R)-3-ethyl-4-(5-methyl-1-phenylpyrazole-4-carbonyl)piperazin-2-one
—— (3R)-3-ethyl-4-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperazin-2-one —— C16H17FN4O2
(3R)-3-ethyl-4-[1-(2-fluorophenyl)pyrazole-3-carbonyl]piperazin-2-one
—— (3S)-3-ethyl-4-[3-(tetrazol-1-yl)benzoyl]piperazin-2-one —— C14H16N6O2
(3S)-3-ethyl-4-[3-(tetrazol-1-yl)benzoyl]piperazin-2-one
—— N-cyclopropyl-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C12H12N2OS2
N-cyclopropyl-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— (3R)-3-ethyl-4-[3-(tetrazol-1-yl)benzoyl]piperazin-2-one —— C14H16N6O2
(3R)-3-ethyl-4-[3-(tetrazol-1-yl)benzoyl]piperazin-2-one
—— (3R)-4-[(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoyl]-3-ethylpiperazin-2-one —— C20H24N4O2
(3R)-4-[(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoyl]-3-ethylpiperazin-2-one
—— N-[(1R)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-2-(2-methoxyethoxy)acetamide —— C14H24N2O3S
N-[(1R)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-2-(2-methoxyethoxy)acetamide
—— (3S)-4-[(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoyl]-3-ethylpiperazin-2-one —— C20H24N4O2
(3S)-4-[(E)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)prop-2-enoyl]-3-ethylpiperazin-2-one
—— (E)-N-cyclopropyl-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide —— C22H21N3O2
(E)-N-cyclopropyl-3-[3-(2-methoxyphenyl)-1-phenylpyrazol-4-yl]prop-2-enamide
—— 1-[(3R)-1,1-dioxothiolan-3-yl]-5-(4-methoxyphenyl)pyrazole-3-carboxylic acid —— C15H16N2O5S
1-[(3R)-1,1-dioxothiolan-3-yl]-5-(4-methoxyphenyl)pyrazole-3-carboxylic acid
—— (7S)-7-(3-hydroxy-4-methoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C20H16F3N3O3
(7S)-7-(3-hydroxy-4-methoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— N-[2-(4-chlorophenyl)-5-methylpyrazol-3-yl]pyridine-3-carboxamide —— C16H13ClN4O
N-[2-(4-chlorophenyl)-5-methylpyrazol-3-yl]pyridine-3-carboxamide
—— (7R)-7-(3-hydroxy-4-methoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C20H16F3N3O3
(7R)-7-(3-hydroxy-4-methoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— 3-(2-Ethylimidazo[2,1-B][1,3,4]thiadiazol-6-YL)phenyl morpholino sulfone —— C16H18N4O3S2
3-(2-Ethylimidazo[2,1-B][1,3,4]thiadiazol-6-YL)phenyl morpholino sulfone
—— 3-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-[(4-fluorophenyl)methyl]-1-methylurea —— C18H24FN3OS
3-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-[(4-fluorophenyl)methyl]-1-methylurea
—— [1-(3-bromophenyl)pyrazol-3-yl]-[(4R)-4-methylazepan-1-yl]methanone —— C17H20BrN3O
[1-(3-bromophenyl)pyrazol-3-yl]-[(4R)-4-methylazepan-1-yl]methanone
—— 1-benzyl-3-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-methylurea —— C18H25N3OS
1-benzyl-3-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-methylurea
—— 3-Imidazo[2,1-B][1,3]benzothiazol-2-ylphenyl morpholino sulfone —— C19H17N3O3S2
3-Imidazo[2,1-B][1,3]benzothiazol-2-ylphenyl morpholino sulfone
—— 1-(3,4-dichlorophenyl)-N-[(2S)-4-methoxybutan-2-yl]pyrazole-3-carboxamide —— C15H17Cl2N3O2
1-(3,4-dichlorophenyl)-N-[(2S)-4-methoxybutan-2-yl]pyrazole-3-carboxamide
—— 3-(2-Methylimidazo[2,1-B][1,3,4]thiadiazol-6-YL)phenyl morpholino sulfone —— C15H16N4O3S2
3-(2-Methylimidazo[2,1-B][1,3,4]thiadiazol-6-YL)phenyl morpholino sulfone
—— N-[(2-chlorophenyl)methyl]-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C19H18ClN3O2
N-[(2-chlorophenyl)methyl]-3-[3-(4-methylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— 2-[4-Methyl-3-(morpholin-4-ylsulfonyl)phenyl]imidazo[1,2-a]pyridine —— C18H19N3O3S
2-[4-Methyl-3-(morpholin-4-ylsulfonyl)phenyl]imidazo[1,2-a]pyridine
—— N-[(3-chlorophenyl)methyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C16H13ClN2OS2
N-[(3-chlorophenyl)methyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— N-[(2-chlorophenyl)methyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide —— C16H13ClN2OS2
N-[(2-chlorophenyl)methyl]-4-methyl-2-thiophen-3-yl-1,3-thiazole-5-carboxamide
—— 4-[4-(Piperidinosulfonyl)-2-thienyl]-1,3-thiazol-2-amine —— C12H15N3O2S3
4-[4-(Piperidinosulfonyl)-2-thienyl]-1,3-thiazol-2-amine
—— 3-Imidazo[2,1-B][1,3]thiazol-6-ylphenyl morpholino sulfone —— C15H15N3O3S2
3-Imidazo[2,1-B][1,3]thiazol-6-ylphenyl morpholino sulfone
—— (7R)-7-(3-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C20H16F3N3O2
(7R)-7-(3-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— 3-[(1R)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-[(4-fluorophenyl)methyl]-1-methylurea —— C18H24FN3OS
3-[(1R)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-[(4-fluorophenyl)methyl]-1-methylurea
—— (7R)-7-(3,4-dimethoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C21H18F3N3O3
(7R)-7-(3,4-dimethoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— N-(1-cyanocyclohexyl)-3-[3-(3-methylphenyl)-5-sulfanyl-4H-1,2,4-triazol-4-yl]propanamide —— C19H23N5OS
N-(1-cyanocyclohexyl)-3-[3-(3-methylphenyl)-5-sulfanyl-4H-1,2,4-triazol-4-yl]propanamide
—— (7S)-7-(3-hydroxy-4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C20H16F3N3O3
(7S)-7-(3-hydroxy-4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— (7R)-7-(3-hydroxy-4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C20H16F3N3O3
(7R)-7-(3-hydroxy-4-methoxyphenyl)-1-[3-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— (7S)-7-(4-hydroxyphenyl)-1-(3-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C19H17N3O3
(7S)-7-(4-hydroxyphenyl)-1-(3-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— (7R)-7-(4,7-dimethoxy-1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C22H21N3O6
(7R)-7-(4,7-dimethoxy-1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— 1-[(3R)-1,1-dioxothiolan-3-yl]-5-(4-methoxyphenyl)pyrazole-3-carboxylate —— C15H15N2O5S-
1-[(3R)-1,1-dioxothiolan-3-yl]-5-(4-methoxyphenyl)pyrazole-3-carboxylate
—— (7S)-7-(3,4-dimethoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C21H18F3N3O3
(7S)-7-(3,4-dimethoxyphenyl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— 1-(3-bromophenyl)-N-[(2S)-4-methoxybutan-2-yl]pyrazole-3-carboxamide —— C15H18BrN3O2
1-(3-bromophenyl)-N-[(2S)-4-methoxybutan-2-yl]pyrazole-3-carboxamide
—— (7R)-1-(3-methoxyphenyl)-7-(3,4,5-trimethoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C22H23N3O5
(7R)-1-(3-methoxyphenyl)-7-(3,4,5-trimethoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— (4R)-5-(4-hydroxyphenyl)-3-(4-methylphenyl)-4-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-6-one —— C24H19N3O2
(4R)-5-(4-hydroxyphenyl)-3-(4-methylphenyl)-4-phenyl-1,4-dihydropyrrolo[3,4-c]pyrazol-6-one
—— 1-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]-3-[2-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]urea —— C17H31N5OS
1-[(2S)-1-(4-methylpiperazin-1-yl)propan-2-yl]-3-[2-(2-propan-2-yl-1,3-thiazol-4-yl)ethyl]urea
—— 3-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-methyl-1-[(2-methylphenyl)methyl]urea —— C19H27N3OS
3-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-1-methyl-1-[(2-methylphenyl)methyl]urea
—— (7S)-7-(4,7-dimethoxy-1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C22H21N3O6
(7S)-7-(4,7-dimethoxy-1,3-benzodioxol-5-yl)-1-(4-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— [1-(3,4-dichlorophenyl)pyrazol-3-yl]-[(4R)-4-methylazepan-1-yl]methanone —— C17H19Cl2N3O
[1-(3,4-dichlorophenyl)pyrazol-3-yl]-[(4R)-4-methylazepan-1-yl]methanone
—— (7S)-7-(7-methoxy-1,3-benzodioxol-5-yl)-1-(3-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C21H19N3O5
(7S)-7-(7-methoxy-1,3-benzodioxol-5-yl)-1-(3-methoxyphenyl)-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— (7R)-7-(1,3-benzodioxol-5-yl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C20H14F3N3O3
(7R)-7-(1,3-benzodioxol-5-yl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— (7S)-7-(7-methoxy-1,3-benzodioxol-5-yl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one —— C21H16F3N3O4
(7S)-7-(7-methoxy-1,3-benzodioxol-5-yl)-1-[4-(trifluoromethyl)phenyl]-6,7-dihydro-4H-imidazo[4,5-b]pyridin-5-one
—— 1-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-3-phenylmethoxyurea —— C17H23N3O2S
1-[(1S)-1-(4-tert-butyl-1,3-thiazol-2-yl)ethyl]-3-phenylmethoxyurea
—— (3S)-1-cycloheptyl-5-oxo-N-(1-phenylpyrazol-4-yl)pyrrolidine-3-carboxamide —— C21H26N4O2
(3S)-1-cycloheptyl-5-oxo-N-(1-phenylpyrazol-4-yl)pyrrolidine-3-carboxamide
—— 3-[2-(Ethylsulfanyl)imidazo[2,1-B][1,3,4]thiadiazol-6-YL]phenyl morpholino sulfone —— C16H18N4O3S3
3-[2-(Ethylsulfanyl)imidazo[2,1-B][1,3,4]thiadiazol-6-YL]phenyl morpholino sulfone