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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[2-[(1S)-1-(2,5-dichlorophenyl)ethyl]pyrazol-3-yl]-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)acetamide —— C19H16Cl2N6O2
N-[2-[(1S)-1-(2,5-dichlorophenyl)ethyl]pyrazol-3-yl]-2-(3-oxo-[1,2,4]triazolo[4,3-a]pyridin-2-yl)acetamide
—— (2R)-N-(3,5-dimethylphenyl)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide —— C23H25FN4O
(2R)-N-(3,5-dimethylphenyl)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
—— (2S)-N-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide —— C25H28FN5O2
(2S)-N-[4-[2-(dimethylamino)-2-oxoethyl]phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
—— 1-(2-chlorophenyl)-5-methyl-N-[[(2R,3R)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide —— C19H25ClN4O2
1-(2-chlorophenyl)-5-methyl-N-[[(2R,3R)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide
—— tert-butyl (3S)-3-cyano-4-[1-(3-fluorophenyl)pyrazole-3-carbonyl]piperazine-1-carboxylate —— C20H22FN5O3
tert-butyl (3S)-3-cyano-4-[1-(3-fluorophenyl)pyrazole-3-carbonyl]piperazine-1-carboxylate
—— 2-[(1S)-1-methoxyethyl]-4-methyl-N-propan-2-yl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide —— C17H23N3O2S
2-[(1S)-1-methoxyethyl]-4-methyl-N-propan-2-yl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
—— (2S)-N-[2-(difluoromethoxy)phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide —— C22H21F3N4O2
(2S)-N-[2-(difluoromethoxy)phenyl]-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
—— 1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1S,2S)-2-imidazol-1-ylcyclopentyl]urea —— C18H19ClN6O
1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1S,2S)-2-imidazol-1-ylcyclopentyl]urea
—— (3S)-3-(5-phenyl-1H-imidazol-2-yl)-N-[4-(pyrrolidine-1-carbonyl)phenyl]piperidine-1-carboxamide —— C26H29N5O2
(3S)-3-(5-phenyl-1H-imidazol-2-yl)-N-[4-(pyrrolidine-1-carbonyl)phenyl]piperidine-1-carboxamide
—— 1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1R,2S)-2-imidazol-1-ylcyclopentyl]urea —— C18H19ClN6O
1-(3-chloro-4-pyrazol-1-ylphenyl)-3-[(1R,2S)-2-imidazol-1-ylcyclopentyl]urea
—— 1-(2-chlorophenyl)-5-methyl-N-[[(2R,3S)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide —— C19H25ClN4O2
1-(2-chlorophenyl)-5-methyl-N-[[(2R,3S)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide
—— 1-(2-chlorophenyl)-5-methyl-N-[[(2S,3R)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide —— C19H25ClN4O2
1-(2-chlorophenyl)-5-methyl-N-[[(2S,3R)-2-propan-2-yloxan-3-yl]methyl]triazole-4-carboxamide
—— 2-[(1S)-1-methoxyethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide —— C9H14N2O2S
2-[(1S)-1-methoxyethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
—— 2-[(1S)-1-methoxyethyl]-4-methyl-N-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-1,3-thiazole-5-carboxamide —— C13H19N5O2S
2-[(1S)-1-methoxyethyl]-4-methyl-N-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-1,3-thiazole-5-carboxamide
—— 2-[(1R)-1-methoxyethyl]-4-methyl-N-propan-2-yl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide —— C17H23N3O2S
2-[(1R)-1-methoxyethyl]-4-methyl-N-propan-2-yl-N-(pyridin-3-ylmethyl)-1,3-thiazole-5-carboxamide
—— (2S)-2-methyl-1-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)-3-(1,3,5-trimethylpyrazol-4-yl)propan-1-one —— C14H22N4OS
(2S)-2-methyl-1-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)-3-(1,3,5-trimethylpyrazol-4-yl)propan-1-one
—— ethyl 2-[2-[[(1R)-2-methyl-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]carbamoylamino]-1,3-thiazol-4-yl]acetate —— C15H22N6O3S
ethyl 2-[2-[[(1R)-2-methyl-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]carbamoylamino]-1,3-thiazol-4-yl]acetate
—— 2-[(1R)-1-methoxyethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide —— C9H14N2O2S
2-[(1R)-1-methoxyethyl]-N,4-dimethyl-1,3-thiazole-5-carboxamide
—— N-cyclopropyl-2-[(1S)-1-methoxyethyl]-4-methyl-N-[(1R)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide —— C18H23N3O2S
N-cyclopropyl-2-[(1S)-1-methoxyethyl]-4-methyl-N-[(1R)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide
—— 2-[(1S)-1-methoxyethyl]-4-methyl-N-(5-propyl-1H-pyrazol-3-yl)-1,3-thiazole-5-carboxamide —— C14H20N4O2S
2-[(1S)-1-methoxyethyl]-4-methyl-N-(5-propyl-1H-pyrazol-3-yl)-1,3-thiazole-5-carboxamide
—— (2R)-2-methyl-1-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)-3-(1,3,5-trimethylpyrazol-4-yl)propan-1-one —— C14H22N4OS
(2R)-2-methyl-1-(2-methylsulfanyl-4,5-dihydroimidazol-1-yl)-3-(1,3,5-trimethylpyrazol-4-yl)propan-1-one
—— 5-[(2S)-1-(5-nitroimidazo[2,1-b][1,3]thiazol-6-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C18H16N6O3S
5-[(2S)-1-(5-nitroimidazo[2,1-b][1,3]thiazol-6-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— N-cyclopropyl-2-[(1R)-1-methoxyethyl]-4-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide —— C18H23N3O2S
N-cyclopropyl-2-[(1R)-1-methoxyethyl]-4-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide
—— 2-[(1R)-1-methoxyethyl]-4-methyl-N-(5-propyl-1H-pyrazol-3-yl)-1,3-thiazole-5-carboxamide —— C14H20N4O2S
2-[(1R)-1-methoxyethyl]-4-methyl-N-(5-propyl-1H-pyrazol-3-yl)-1,3-thiazole-5-carboxamide
—— 1-cyclopropyl-1-[(3R)-1,1-dioxothiolan-3-yl]-3-(4-pyridin-3-yl-1,3-thiazol-2-yl)urea —— C16H18N4O3S2
1-cyclopropyl-1-[(3R)-1,1-dioxothiolan-3-yl]-3-(4-pyridin-3-yl-1,3-thiazol-2-yl)urea
—— N-cyclopropyl-2-[(1S)-1-methoxyethyl]-4-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide —— C18H23N3O2S
N-cyclopropyl-2-[(1S)-1-methoxyethyl]-4-methyl-N-[(1S)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide
—— [(1R)-1-(1-ethylimidazol-2-yl)-3-phenylpropyl] 2-(methoxymethyl)-1,3-thiazole-4-carboxylate —— C20H23N3O3S
[(1R)-1-(1-ethylimidazol-2-yl)-3-phenylpropyl] 2-(methoxymethyl)-1,3-thiazole-4-carboxylate
—— 2-[(1R)-1-methoxyethyl]-4-methyl-N-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-1,3-thiazole-5-carboxamide —— C13H19N5O2S
2-[(1R)-1-methoxyethyl]-4-methyl-N-(5-propan-2-yl-1H-1,2,4-triazol-3-yl)-1,3-thiazole-5-carboxamide
—— [(1S)-1-(1-ethylimidazol-2-yl)-3-phenylpropyl] 2-(methoxymethyl)-1,3-thiazole-4-carboxylate —— C20H23N3O3S
[(1S)-1-(1-ethylimidazol-2-yl)-3-phenylpropyl] 2-(methoxymethyl)-1,3-thiazole-4-carboxylate
—— N-cyclopropyl-2-[(1R)-1-methoxyethyl]-4-methyl-N-[(1R)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide —— C18H23N3O2S
N-cyclopropyl-2-[(1R)-1-methoxyethyl]-4-methyl-N-[(1R)-1-pyridin-2-ylethyl]-1,3-thiazole-5-carboxamide
—— ethyl 2-[2-[[(1S)-2-methyl-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]carbamoylamino]-1,3-thiazol-4-yl]acetate —— C15H22N6O3S
ethyl 2-[2-[[(1S)-2-methyl-1-(5-methyl-1H-1,2,4-triazol-3-yl)propyl]carbamoylamino]-1,3-thiazol-4-yl]acetate
—— 2-[(2S)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidin-1-yl]-4-pyrazol-1-ylpyrimidine —— C21H20FN7
2-[(2S)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidin-1-yl]-4-pyrazol-1-ylpyrimidine
—— 1-cyclopropyl-1-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-pyridin-3-yl-1,3-thiazol-2-yl)urea —— C16H18N4O3S2
1-cyclopropyl-1-[(3S)-1,1-dioxothiolan-3-yl]-3-(4-pyridin-3-yl-1,3-thiazol-2-yl)urea
—— 2-[(2R)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidin-1-yl]-4-pyrazol-1-ylpyrimidine —— C21H20FN7
2-[(2R)-2-[5-(3-fluorophenyl)-1H-imidazol-2-yl]piperidin-1-yl]-4-pyrazol-1-ylpyrimidine
—— 5-[(2S)-1-(5-bromopyrimidin-2-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C17H16BrN5O
5-[(2S)-1-(5-bromopyrimidin-2-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(2R)-1-(5-nitroimidazo[2,1-b][1,3]thiazol-6-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C18H16N6O3S
5-[(2R)-1-(5-nitroimidazo[2,1-b][1,3]thiazol-6-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— 5-[(2R)-1-(5-bromopyrimidin-2-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole —— C17H16BrN5O
5-[(2R)-1-(5-bromopyrimidin-2-yl)piperidin-2-yl]-3-phenyl-1,2,4-oxadiazole
—— N-(4-methoxyphenyl)-5-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-1,3,4-thiadiazol-2-amine —— C18H15N5O2S2
N-(4-methoxyphenyl)-5-[(3-phenyl-1,2,4-oxadiazol-5-yl)methylsulfanyl]-1,3,4-thiadiazol-2-amine
—— N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]-3-(4-nitrophenyl)-1,2,4-oxadiazol-5-amine —— C16H22N6O3
N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]-3-(4-nitrophenyl)-1,2,4-oxadiazol-5-amine
—— N-[(1S,2S)-2-carbamoylcyclohexyl]-3-pyrazol-1-ylbenzamide —— C17H20N4O2
N-[(1S,2S)-2-carbamoylcyclohexyl]-3-pyrazol-1-ylbenzamide
—— 2-[(2R)-oxolan-2-yl]ethyl 4-methyl-1,3-thiazole-5-carboxylate —— C11H15NO3S
2-[(2R)-oxolan-2-yl]ethyl 4-methyl-1,3-thiazole-5-carboxylate
—— 2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-(2-fluoro-5-methylphenyl)acetamide —— C19H19FN4OS
2-[(4-ethyl-5-phenyl-1,2,4-triazol-3-yl)sulfanyl]-N-(2-fluoro-5-methylphenyl)acetamide
—— [5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-[(3S)-3-(1H-1,2,4-triazol-5-yl)piperidin-1-yl]methanone —— C19H19F3N6O
[5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-[(3S)-3-(1H-1,2,4-triazol-5-yl)piperidin-1-yl]methanone
—— [5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-[(3R)-3-(1H-1,2,4-triazol-5-yl)piperidin-1-yl]methanone —— C19H19F3N6O
[5-methyl-1-[3-(trifluoromethyl)phenyl]pyrazol-4-yl]-[(3R)-3-(1H-1,2,4-triazol-5-yl)piperidin-1-yl]methanone
—— (2R)-2-(3,5-dimethylpyrazol-1-yl)-N-[3-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,2,4,4-tetramethylcyclobutyl]propanamide —— C24H38N6O2
(2R)-2-(3,5-dimethylpyrazol-1-yl)-N-[3-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,2,4,4-tetramethylcyclobutyl]propanamide
—— N-[5-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-3-yl]-2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]acetamide —— C19H16FN5O3
N-[5-[(4-fluorophenyl)methyl]-1H-1,2,4-triazol-3-yl]-2-[2-(furan-2-yl)-5-methyl-1,3-oxazol-4-yl]acetamide
—— (3S)-5-[3-[(3,5-dimethoxyphenyl)methyl]azetidine-1-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide —— C23H26N4O4
(3S)-5-[3-[(3,5-dimethoxyphenyl)methyl]azetidine-1-carbonyl]-2-phenyl-3,4-dihydropyrazole-3-carboxamide
—— tert-butyl (3R)-4-carbamoyl-3-[[4-(1,2,4-triazol-1-yl)phenyl]methylcarbamoyl]piperazine-1-carboxylate —— C20H27N7O4
tert-butyl (3R)-4-carbamoyl-3-[[4-(1,2,4-triazol-1-yl)phenyl]methylcarbamoyl]piperazine-1-carboxylate
—— N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]-3-(4-nitrophenyl)-1,2,4-oxadiazol-5-amine —— C16H22N6O3
N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]-3-(4-nitrophenyl)-1,2,4-oxadiazol-5-amine
—— (2R)-2-(3,5-dimethylpyrazol-1-yl)-N-[3-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,2,4,4-tetramethylcyclobutyl]propanamide —— C24H38N6O2
(2R)-2-(3,5-dimethylpyrazol-1-yl)-N-[3-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,2,4,4-tetramethylcyclobutyl]propanamide