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中文名称 英文名称 CAS号 化学式 结构式图片
—— 2-cyclopentyl-N-[2-[[(1S)-1-(1,3-thiazol-2-yl)ethyl]carbamoylamino]ethyl]acetamide —— C15H24N4O2S
2-cyclopentyl-N-[2-[[(1S)-1-(1,3-thiazol-2-yl)ethyl]carbamoylamino]ethyl]acetamide
—— 4-[[(S)-(1-cyclopropyltetrazol-5-yl)methylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole —— C13H13N5O2S2
4-[[(S)-(1-cyclopropyltetrazol-5-yl)methylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole
—— 4-[[(S)-cyclohexylmethylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole —— C15H19NO2S2
4-[[(S)-cyclohexylmethylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole
—— 2-cyclopentyl-N-[2-[[(1R)-1-(1,3-thiazol-2-yl)ethyl]carbamoylamino]ethyl]acetamide —— C15H24N4O2S
2-cyclopentyl-N-[2-[[(1R)-1-(1,3-thiazol-2-yl)ethyl]carbamoylamino]ethyl]acetamide
—— 4-[[(R)-(1-cyclopropyltetrazol-5-yl)methylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole —— C13H13N5O2S2
4-[[(R)-(1-cyclopropyltetrazol-5-yl)methylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole
—— 4-[[(R)-cyclohexylmethylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole —— C15H19NO2S2
4-[[(R)-cyclohexylmethylsulfinyl]methyl]-2-(furan-2-yl)-1,3-thiazole
—— 2-(furan-2-yl)-4-[[(S)-2-phenylethylsulfinyl]methyl]-1,3-thiazole —— C16H15NO2S2
2-(furan-2-yl)-4-[[(S)-2-phenylethylsulfinyl]methyl]-1,3-thiazole
—— [(3S)-thiolan-3-yl] 2-(2-thiophen-2-yl-1,3-oxazol-4-yl)acetate —— C13H13NO3S2
[(3S)-thiolan-3-yl] 2-(2-thiophen-2-yl-1,3-oxazol-4-yl)acetate
—— 2-(furan-2-yl)-4-[[(R)-2-phenylethylsulfinyl]methyl]-1,3-thiazole —— C16H15NO2S2
2-(furan-2-yl)-4-[[(R)-2-phenylethylsulfinyl]methyl]-1,3-thiazole
—— N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-phenyl-5-thiophen-2-ylpyrazole-3-carboxamide —— C20H21N3O3S2
N-[(3R)-1,1-dioxothiolan-3-yl]-N-ethyl-2-phenyl-5-thiophen-2-ylpyrazole-3-carboxamide
—— N-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]cyclopropanecarboxamide —— C14H13ClN2OS
N-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]cyclopropanecarboxamide
—— N-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-thiophen-2-ylacetamide —— C16H13ClN2OS2
N-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-thiophen-2-ylacetamide
—— N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide —— C21H16FN3OS2
N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
—— 2-[3-[(3R)-3-(dimethylamino)piperidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C16H23N5O2
2-[3-[(3R)-3-(dimethylamino)piperidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 2-[3-oxo-3-[(2R)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C18H25N5O2
2-[3-oxo-3-[(2R)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 2-[3-[(3S)-3-(dimethylamino)piperidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C16H23N5O2
2-[3-[(3S)-3-(dimethylamino)piperidin-1-yl]-3-oxopropyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 2-[3-oxo-3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one —— C18H25N5O2
2-[3-oxo-3-[(2S)-2-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]propyl]-[1,2,4]triazolo[4,3-a]pyridin-3-one
—— 3-N-[(2R)-2-(4-methylpiperidin-1-yl)propyl]-1-phenylpyrazole-3,5-dicarboxamide —— C20H27N5O2
3-N-[(2R)-2-(4-methylpiperidin-1-yl)propyl]-1-phenylpyrazole-3,5-dicarboxamide
—— tert-butyl N-[2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2-ethylbutyl]carbamate —— C19H33N3O4
tert-butyl N-[2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2-ethylbutyl]carbamate
—— tert-butyl N-[[1-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]cyclopentyl]methyl]carbamate —— C19H31N3O4
tert-butyl N-[[1-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]cyclopentyl]methyl]carbamate
—— 3-N-[(2S)-2-(4-methylpiperidin-1-yl)propyl]-1-phenylpyrazole-3,5-dicarboxamide —— C20H27N5O2
3-N-[(2S)-2-(4-methylpiperidin-1-yl)propyl]-1-phenylpyrazole-3,5-dicarboxamide
—— tert-butyl N-[2-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2-ethylbutyl]carbamate —— C19H33N3O4
tert-butyl N-[2-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2-ethylbutyl]carbamate
—— tert-butyl N-[[1-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]cyclopentyl]methyl]carbamate —— C19H31N3O4
tert-butyl N-[[1-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]cyclopentyl]methyl]carbamate
—— N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-2-phenyl-5-thiophen-2-ylpyrazole-3-carboxamide —— C20H21N3O3S2
N-[(3S)-1,1-dioxothiolan-3-yl]-N-ethyl-2-phenyl-5-thiophen-2-ylpyrazole-3-carboxamide
—— 2-(3-fluorophenoxy)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]acetamide —— C18H14F2N2O2S
2-(3-fluorophenoxy)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]acetamide
—— N-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-thiophen-3-ylacetamide —— C16H13ClN2OS2
N-[4-(4-chlorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-thiophen-3-ylacetamide
—— 2-(4-cyanophenoxy)-N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]acetamide —— C19H13F2N3O2S
2-(4-cyanophenoxy)-N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]acetamide
—— N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-(3-methylphenoxy)acetamide —— C19H16F2N2O2S
N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-(3-methylphenoxy)acetamide
—— N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide —— C21H16FN3O2S
N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-5-methyl-3-phenyl-1,2-oxazole-4-carboxamide
—— N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-3-(4-methoxyphenyl)propanamide —— C20H19FN2O2S
N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-3-(4-methoxyphenyl)propanamide
—— N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-phenoxyacetamide —— C18H14F2N2O2S
N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-phenoxyacetamide
—— 2-(4-fluorophenoxy)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]acetamide —— C18H14F2N2O2S
2-(4-fluorophenoxy)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]acetamide
—— (2S)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-phenoxypropanamide —— C19H17FN2O2S
(2S)-N-[4-(4-fluorophenyl)-5-methyl-1,3-thiazol-2-yl]-2-phenoxypropanamide
—— N-[(2R)-2-cyanopropyl]-4-methyl-2-(5-methylfuran-2-yl)-1,3-thiazole-5-carboxamide —— C14H15N3O2S
N-[(2R)-2-cyanopropyl]-4-methyl-2-(5-methylfuran-2-yl)-1,3-thiazole-5-carboxamide
—— N-[(2R)-2-cyanopropyl]-1-phenylpyrazole-3-carboxamide —— C14H14N4O
N-[(2R)-2-cyanopropyl]-1-phenylpyrazole-3-carboxamide
—— ethyl 1-[4-[[(2R)-2-cyanopropyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate —— C18H20N4O3
ethyl 1-[4-[[(2R)-2-cyanopropyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate
—— 1-(4-bromophenyl)-N-[(2S)-2-cyanopropyl]-5-methylpyrazole-4-carboxamide —— C15H15BrN4O
1-(4-bromophenyl)-N-[(2S)-2-cyanopropyl]-5-methylpyrazole-4-carboxamide
—— ethyl 1-[4-[[(2S)-2-cyanopropyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate —— C18H20N4O3
ethyl 1-[4-[[(2S)-2-cyanopropyl]carbamoyl]phenyl]-5-methylpyrazole-4-carboxylate
—— N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]-3-(4-methoxyphenyl)propanamide —— C20H18F2N2O2S
N-[4-(3,4-difluorophenyl)-5-methyl-1,3-thiazol-2-yl]-3-(4-methoxyphenyl)propanamide
—— N-[(2R)-2-cyanopropyl]-1,5-diphenyl-1,2,4-triazole-3-carboxamide —— C19H17N5O
N-[(2R)-2-cyanopropyl]-1,5-diphenyl-1,2,4-triazole-3-carboxamide
—— 2-methyl-N-[(2R)-4-methyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]pentyl]-1,3-thiazole-4-carboxamide —— C16H22N4O2S2
2-methyl-N-[(2R)-4-methyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]pentyl]-1,3-thiazole-4-carboxamide
—— 2-methyl-N-[(2S)-4-methyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]pentyl]-1,3-thiazole-4-carboxamide —— C16H22N4O2S2
2-methyl-N-[(2S)-4-methyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]pentyl]-1,3-thiazole-4-carboxamide
—— 1-(4-bromophenyl)-N-[(2R)-2-cyanopropyl]-5-methylpyrazole-4-carboxamide —— C15H15BrN4O
1-(4-bromophenyl)-N-[(2R)-2-cyanopropyl]-5-methylpyrazole-4-carboxamide
—— 2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2R)-2-cyanopropyl]acetamide —— C16H17N3OS
2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2R)-2-cyanopropyl]acetamide
—— tert-butyl N-[(2R)-2-cyclopropyl-2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]propyl]carbamate —— C19H31N3O4
tert-butyl N-[(2R)-2-cyclopropyl-2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]propyl]carbamate
—— 2-(5-chlorothiophen-2-yl)-N-[(2R)-2-cyanopropyl]-4-methyl-1,3-thiazole-5-carboxamide —— C13H12ClN3OS2
2-(5-chlorothiophen-2-yl)-N-[(2R)-2-cyanopropyl]-4-methyl-1,3-thiazole-5-carboxamide
—— N-[(2R)-2-cyanopropyl]-1-(4-methylphenyl)-3-phenylpyrazole-4-carboxamide —— C21H20N4O
N-[(2R)-2-cyanopropyl]-1-(4-methylphenyl)-3-phenylpyrazole-4-carboxamide
—— N-[(2R)-2-cyanopropyl]-3-[5-(2-fluorophenyl)-1,3-oxazol-2-yl]propanamide —— C16H16FN3O2
N-[(2R)-2-cyanopropyl]-3-[5-(2-fluorophenyl)-1,3-oxazol-2-yl]propanamide
—— 2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2S)-2-cyanopropyl]acetamide —— C16H17N3OS
2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2S)-2-cyanopropyl]acetamide
—— N-[(2R)-2-cyanopropyl]-2-(2-phenyl-1,3-oxazol-4-yl)acetamide —— C15H15N3O2
N-[(2R)-2-cyanopropyl]-2-(2-phenyl-1,3-oxazol-4-yl)acetamide