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中文名称 英文名称 CAS号 化学式 结构式图片
—— 1-[3-(4-fluorophenyl)-1-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone —— C21H27FN4O
1-[3-(4-fluorophenyl)-1-[2-[(2S)-1-methylpyrrolidin-2-yl]ethyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone
—— N-[(3R,4R)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide —— C19H24N4O4S
N-[(3R,4R)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide
—— 1-benzyl-3-[5-(cyclopentylmethyl)-1,3,4-thiadiazol-2-yl]-1-[(2R)-1-morpholin-4-ylpropan-2-yl]urea —— C23H33N5O2S
1-benzyl-3-[5-(cyclopentylmethyl)-1,3,4-thiadiazol-2-yl]-1-[(2R)-1-morpholin-4-ylpropan-2-yl]urea
—— (3S)-3-acetyl-N-methyl-N-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C20H21N5O2S
(3S)-3-acetyl-N-methyl-N-[(6-methylimidazo[2,1-b][1,3]thiazol-5-yl)methyl]-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— (E)-2-phenyl-N-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]ethenesulfonamide —— C17H17N5O2S
(E)-2-phenyl-N-[(1R)-1-(1-phenyltetrazol-5-yl)ethyl]ethenesulfonamide
—— (E)-N-[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide —— C21H20FN3O2
(E)-N-[(1R)-1-(3-fluoro-4-methoxyphenyl)ethyl]-3-(1-phenylpyrazol-4-yl)prop-2-enamide
—— (1R)-N-methyl-N-(2-phenoxyethyl)-1-(1-phenyltetrazol-5-yl)ethanamine —— C18H21N5O
(1R)-N-methyl-N-(2-phenoxyethyl)-1-(1-phenyltetrazol-5-yl)ethanamine
—— (3S)-N-[2-(3-chlorophenyl)pyrazol-3-yl]-6-oxopiperidine-3-carboxamide —— C15H15ClN4O2
(3S)-N-[2-(3-chlorophenyl)pyrazol-3-yl]-6-oxopiperidine-3-carboxamide
—— (4R)-N-[(5-phenyl-1H-imidazol-2-yl)methyl]-3,4-dihydro-2H-chromene-4-carboxamide —— C20H19N3O2
(4R)-N-[(5-phenyl-1H-imidazol-2-yl)methyl]-3,4-dihydro-2H-chromene-4-carboxamide
—— (1S)-N-methyl-N-(2-phenoxyethyl)-1-(1-phenyltetrazol-5-yl)ethanamine —— C18H21N5O
(1S)-N-methyl-N-(2-phenoxyethyl)-1-(1-phenyltetrazol-5-yl)ethanamine
—— N'-[(3R)-1,1-dioxothiolane-3-carbonyl]-2-methyl-4-phenyl-1,3-thiazole-5-carbohydrazide —— C16H17N3O4S2
N'-[(3R)-1,1-dioxothiolane-3-carbonyl]-2-methyl-4-phenyl-1,3-thiazole-5-carbohydrazide
—— 5-[(1S)-1-[[butyl(methyl)sulfamoyl]amino]ethyl]-1-phenyltetrazole —— C14H22N6O2S
5-[(1S)-1-[[butyl(methyl)sulfamoyl]amino]ethyl]-1-phenyltetrazole
—— N'-[(3R)-1,1-dioxothiolane-3-carbonyl]-1-phenylpyrazole-4-carbohydrazide —— C15H16N4O4S
N'-[(3R)-1,1-dioxothiolane-3-carbonyl]-1-phenylpyrazole-4-carbohydrazide
—— (3R)-1,1-dioxo-N'-[(E)-3-(1-phenylpyrazol-4-yl)prop-2-enoyl]thiolane-3-carbohydrazide —— C17H18N4O4S
(3R)-1,1-dioxo-N'-[(E)-3-(1-phenylpyrazol-4-yl)prop-2-enoyl]thiolane-3-carbohydrazide
—— N'-[(3S)-1,1-dioxothiolane-3-carbonyl]-2-thiophen-3-yl-1,3-thiazole-4-carbohydrazide —— C13H13N3O4S3
N'-[(3S)-1,1-dioxothiolane-3-carbonyl]-2-thiophen-3-yl-1,3-thiazole-4-carbohydrazide
—— 1-benzyl-N'-[(3S)-1,1-dioxothiolane-3-carbonyl]pyrazole-4-carbohydrazide —— C16H18N4O4S
1-benzyl-N'-[(3S)-1,1-dioxothiolane-3-carbonyl]pyrazole-4-carbohydrazide
—— 2-[2-(3-bromophenyl)-1,3-thiazol-4-yl]-N-[(2-fluorophenyl)methyl]acetamide —— C18H14BrFN2OS
2-[2-(3-bromophenyl)-1,3-thiazol-4-yl]-N-[(2-fluorophenyl)methyl]acetamide
—— (4S)-N-[(5-phenyl-1H-imidazol-2-yl)methyl]-3,4-dihydro-2H-chromene-4-carboxamide —— C20H19N3O2
(4S)-N-[(5-phenyl-1H-imidazol-2-yl)methyl]-3,4-dihydro-2H-chromene-4-carboxamide
—— 3-ethyl-5-methyl-N-[4-(2,4,5-trimethylphenyl)-1,3-thiazol-2-yl]-1,2-oxazole-4-carboxamide —— C19H21N3O2S
3-ethyl-5-methyl-N-[4-(2,4,5-trimethylphenyl)-1,3-thiazol-2-yl]-1,2-oxazole-4-carboxamide
—— 1-benzyl-3-[5-(cyclopentylmethyl)-1,3,4-thiadiazol-2-yl]-1-[(2S)-1-morpholin-4-ylpropan-2-yl]urea —— C23H33N5O2S
1-benzyl-3-[5-(cyclopentylmethyl)-1,3,4-thiadiazol-2-yl]-1-[(2S)-1-morpholin-4-ylpropan-2-yl]urea
—— (1S,3R)-N-[4-(2H-tetrazol-5-yl)phenyl]-3-(trifluoromethyl)cyclohexane-1-carboxamide —— C15H16F3N5O
(1S,3R)-N-[4-(2H-tetrazol-5-yl)phenyl]-3-(trifluoromethyl)cyclohexane-1-carboxamide
—— 4-[[(2R)-oxolan-2-yl]methoxy]-N-[2-[(1-phenyltetrazol-5-yl)amino]ethyl]benzamide —— C21H24N6O3
4-[[(2R)-oxolan-2-yl]methoxy]-N-[2-[(1-phenyltetrazol-5-yl)amino]ethyl]benzamide
—— 1-[3-(4-fluorophenyl)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone —— C21H27FN4O
1-[3-(4-fluorophenyl)-1-[2-[(2R)-1-methylpyrrolidin-2-yl]ethyl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanone
—— N-[(3S,4R)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide —— C19H24N4O4S
N-[(3S,4R)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide
—— 3-ethyl-5-methyl-N-(tricyclo[3.3.1.1~3,7~]dec-1-ylmethyl)-1,2-oxazole-4-carboxamide —— C18H26N2O2
3-ethyl-5-methyl-N-(tricyclo[3.3.1.1~3,7~]dec-1-ylmethyl)-1,2-oxazole-4-carboxamide
—— 3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide —— C21H26FN5O2
3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide
—— 3-ethyl-5-methyl-N-[4-(2,4,6-trimethylphenyl)-1,3-thiazol-2-yl]-1,2-oxazole-4-carboxamide —— C19H21N3O2S
3-ethyl-5-methyl-N-[4-(2,4,6-trimethylphenyl)-1,3-thiazol-2-yl]-1,2-oxazole-4-carboxamide
—— N-[(2R)-4-(furan-2-yl)butan-2-yl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide —— C21H21N3O2S
N-[(2R)-4-(furan-2-yl)butan-2-yl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide
—— N-[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide —— C16H13F2N3O2S
N-[4-(3,4-difluorophenyl)-1,3-thiazol-2-yl]-3-ethyl-5-methyl-1,2-oxazole-4-carboxamide
—— N-(2,3-dihydro-1H-inden-5-yl)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide —— C23H25N3O
N-(2,3-dihydro-1H-inden-5-yl)-3-(3,5-dimethyl-1-phenylpyrazol-4-yl)propanamide
—— 3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(2-fluorophenyl)methyl]propanamide —— C21H22FN3O
3-(3,5-dimethyl-1-phenylpyrazol-4-yl)-N-[(2-fluorophenyl)methyl]propanamide
—— N-[(2S)-4-(furan-2-yl)butan-2-yl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide —— C21H21N3O2S
N-[(2S)-4-(furan-2-yl)butan-2-yl]-3-methyl-1-phenylthieno[2,3-c]pyrazole-5-carboxamide
—— N-[(3S,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide —— C19H24N4O4S
N-[(3S,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide
—— 3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide —— C21H24F2N4O2
3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-N-[(2S)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide
—— N-[(3R,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide —— C19H24N4O4S
N-[(3R,4S)-1,1-dioxo-4-pyrrolidin-1-ylthiolan-3-yl]-4-(4-methyl-2-oxo-1H-imidazol-3-yl)benzamide
—— 3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide —— C21H26FN5O2
3-[3-(3-fluoro-4-methylphenyl)-1,2,4-oxadiazol-5-yl]-N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide
—— 3-Cyclopropyl-5-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-1,2,4-triazol-4-amine —— C15H16N6OS
3-Cyclopropyl-5-[[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methylsulfanyl]-1,2,4-triazol-4-amine
—— 3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide —— C21H24F2N4O2
3-[5-(2,4-difluorophenyl)-1,3-oxazol-2-yl]-N-[(2R)-1-imidazol-1-yl-3,3-dimethylbutan-2-yl]propanamide
—— (2S)-N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenylbutanamide —— C19H18ClN3O2
(2S)-N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-phenylbutanamide
—— N-[(2S)-1-piperidin-1-ylpropan-2-yl]-3-(1,2,4-triazol-1-yl)benzamide —— C17H23N5O
N-[(2S)-1-piperidin-1-ylpropan-2-yl]-3-(1,2,4-triazol-1-yl)benzamide
—— N-[(2R)-3-methyl-2-(4-methylpiperidin-1-yl)butyl]-3-(1,2,4-triazol-1-yl)benzamide —— C20H29N5O
N-[(2R)-3-methyl-2-(4-methylpiperidin-1-yl)butyl]-3-(1,2,4-triazol-1-yl)benzamide
—— (2R)-5-(3-fluorophenyl)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxopentanenitrile —— C15H13FN2OS
(2R)-5-(3-fluorophenyl)-2-(4-methyl-1,3-thiazol-2-yl)-3-oxopentanenitrile
—— N-[(2R)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide —— C16H19F2N3O2S
N-[(2R)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide
—— N-[(1,3-diphenylpyrazol-4-yl)methyl]-2-(2-fluorophenoxy)-N-methylacetamide —— C25H22FN3O2
N-[(1,3-diphenylpyrazol-4-yl)methyl]-2-(2-fluorophenoxy)-N-methylacetamide
—— N-[(2S)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide —— C16H19F2N3O2S
N-[(2S)-2-(2,6-difluorophenyl)-2-(dimethylamino)ethyl]-2-(methoxymethyl)-1,3-thiazole-4-carboxamide
—— (2S)-N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-methylpentanamide —— C15H18ClN3O2
(2S)-N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-2-methylpentanamide
—— (2E,4E)-N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-methylhexa-2,4-dienamide —— C23H23N3O
(2E,4E)-N-[(1,3-diphenylpyrazol-4-yl)methyl]-N-methylhexa-2,4-dienamide
—— N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-[(2R)-oxolan-2-yl]propanamide —— C16H18ClN3O3
N-[[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl]-3-[(2R)-oxolan-2-yl]propanamide
—— N-[(1,3-diphenylpyrazol-4-yl)methyl]-2-(3-fluorophenyl)-N-methylacetamide —— C25H22FN3O
N-[(1,3-diphenylpyrazol-4-yl)methyl]-2-(3-fluorophenyl)-N-methylacetamide
—— N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-4-(2-oxo-1,3-benzoxazol-3-yl)butanamide —— C24H26N4O3
N-[(3,5-dimethyl-1-phenylpyrazol-4-yl)methyl]-N-methyl-4-(2-oxo-1,3-benzoxazol-3-yl)butanamide