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中文名称 英文名称 CAS号 化学式 结构式图片
—— 3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(3-methylsulfanylphenyl)propanamide —— C18H16FN3O2S
3-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-(3-methylsulfanylphenyl)propanamide
—— (3S)-1-[5-pyrrol-1-yl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carbonyl]piperidine-3-carboxamide —— C21H20F3N5O2
(3S)-1-[5-pyrrol-1-yl-1-[3-(trifluoromethyl)phenyl]pyrazole-4-carbonyl]piperidine-3-carboxamide
—— 2-[(2S)-1-[[3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]ethanol —— C17H20F3N3O2
2-[(2S)-1-[[3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl]methyl]piperidin-2-yl]ethanol
—— 2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]benzamide —— C18H22N4O3
2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]benzamide
—— (2,4-dimethyl-1,3-thiazol-5-yl)methyl (3R)-3-cyclohexylbutanoate —— C16H25NO2S
(2,4-dimethyl-1,3-thiazol-5-yl)methyl (3R)-3-cyclohexylbutanoate
—— 2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2S)-2-(diethylamino)-2-(furan-2-yl)ethyl]benzamide —— C23H30N4O3
2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2S)-2-(diethylamino)-2-(furan-2-yl)ethyl]benzamide
—— 2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]benzamide —— C18H22N4O3
2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(3S)-1-methyl-5-oxopyrrolidin-3-yl]benzamide
—— (2,4-dimethyl-1,3-thiazol-5-yl)methyl (3S)-3-cyclohexylbutanoate —— C16H25NO2S
(2,4-dimethyl-1,3-thiazol-5-yl)methyl (3S)-3-cyclohexylbutanoate
—— (3S)-3-acetyl-N-(6-chloropyridin-3-yl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C17H15ClN4O2
(3S)-3-acetyl-N-(6-chloropyridin-3-yl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— 2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2R)-2-(diethylamino)-2-(furan-2-yl)ethyl]benzamide —— C23H30N4O3
2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2R)-2-(diethylamino)-2-(furan-2-yl)ethyl]benzamide
—— 2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2S)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]benzamide —— C24H30N4O2
2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2S)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]benzamide
—— ethyl (3S)-3-[2-cyanoethyl(methyl)carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C17H20N4O3
ethyl (3S)-3-[2-cyanoethyl(methyl)carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— (3R)-3-acetyl-N-(6-chloropyridin-3-yl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C17H15ClN4O2
(3R)-3-acetyl-N-(6-chloropyridin-3-yl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— 2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]benzamide —— C24H30N4O2
2-(3-tert-butyl-1,2,4-oxadiazol-5-yl)-N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]benzamide
—— ethyl (3R)-3-[2-cyanoethyl(methyl)carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate —— C17H20N4O3
ethyl (3R)-3-[2-cyanoethyl(methyl)carbamoyl]-2-phenyl-3,4-dihydropyrazole-5-carboxylate
—— (3S)-3-acetyl-N-(2-cyanoethyl)-N-(3-methylbutyl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C20H26N4O2
(3S)-3-acetyl-N-(2-cyanoethyl)-N-(3-methylbutyl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— 1-[[5-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropan-2-ol —— C18H25N3O3S
1-[[5-(4-methoxyphenyl)-4-[[(2R)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropan-2-ol
—— 2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[2-(thiophen-2-ylmethylsulfanyl)ethyl]acetamide —— C18H21N5OS3
2-[1-(3,5-dimethylphenyl)tetrazol-5-yl]sulfanyl-N-[2-(thiophen-2-ylmethylsulfanyl)ethyl]acetamide
—— (3R)-3-acetyl-N-(2-cyanoethyl)-N-(3-methylbutyl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C20H26N4O2
(3R)-3-acetyl-N-(2-cyanoethyl)-N-(3-methylbutyl)-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— 1-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropan-2-ol —— C18H25N3O3S
1-[[5-(4-methoxyphenyl)-4-[[(2S)-oxolan-2-yl]methyl]-1,2,4-triazol-3-yl]sulfanyl]-2-methylpropan-2-ol
—— (3R)-3-acetyl-N-[(2S)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C17H20N4O2
(3R)-3-acetyl-N-[(2S)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— (3R)-3-acetyl-N-[(2R)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C17H20N4O2
(3R)-3-acetyl-N-[(2R)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— 2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-thiophen-2-ylethyl)acetamide —— C18H21N5O2S2
2-[[4-amino-5-(4-ethoxyphenyl)-1,2,4-triazol-3-yl]sulfanyl]-N-(2-thiophen-2-ylethyl)acetamide
—— N-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1,3-thiazole-4-carboxamide —— C12H17N3O2S
N-[[(3R,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1,3-thiazole-4-carboxamide
—— [(3S)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 1-(2-fluorophenyl)cyclopentane-1-carboxylate —— C20H19FN2O3S
[(3S)-3-cyano-3-(4-methyl-1,3-thiazol-2-yl)-2-oxopropyl] 1-(2-fluorophenyl)cyclopentane-1-carboxylate
—— N-[(2S)-2-cyclopropyl-2-(1,3-thiazole-4-carbonylamino)ethyl]-1,3-thiazole-4-carboxamide —— C13H14N4O2S2
N-[(2S)-2-cyclopropyl-2-(1,3-thiazole-4-carbonylamino)ethyl]-1,3-thiazole-4-carboxamide
—— (3S)-3-acetyl-N-[(2S)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C17H20N4O2
(3S)-3-acetyl-N-[(2S)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide
—— N-[(2S)-2-(5-methylfuran-2-yl)-2-pyrrolidin-1-ylethyl]-1,3-thiazole-4-carboxamide —— C15H19N3O2S
N-[(2S)-2-(5-methylfuran-2-yl)-2-pyrrolidin-1-ylethyl]-1,3-thiazole-4-carboxamide
—— N-[(2R)-2-(4-methylphenyl)-2-pyrrolidin-1-ylethyl]-1,3-thiazole-4-carboxamide —— C17H21N3OS
N-[(2R)-2-(4-methylphenyl)-2-pyrrolidin-1-ylethyl]-1,3-thiazole-4-carboxamide
—— (2R)-4-[1-(3-chlorophenyl)tetrazol-5-yl]sulfanyl-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanenitrile —— C15H11ClN6OS2
(2R)-4-[1-(3-chlorophenyl)tetrazol-5-yl]sulfanyl-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanenitrile
—— (2S)-4-[1-(3-chlorophenyl)tetrazol-5-yl]sulfanyl-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanenitrile —— C15H11ClN6OS2
(2S)-4-[1-(3-chlorophenyl)tetrazol-5-yl]sulfanyl-2-(4-methyl-1,3-thiazol-2-yl)-3-oxobutanenitrile
—— [2-[[5-methyl-2-(4-methylphenyl)pyrazol-3-yl]amino]-2-oxoethyl] 2-[(1S)-cyclopent-2-en-1-yl]acetate —— C20H23N3O3
[2-[[5-methyl-2-(4-methylphenyl)pyrazol-3-yl]amino]-2-oxoethyl] 2-[(1S)-cyclopent-2-en-1-yl]acetate
—— N-[(3S)-6-oxopiperidin-3-yl]-1,3-thiazole-4-carboxamide —— C9H11N3O2S
N-[(3S)-6-oxopiperidin-3-yl]-1,3-thiazole-4-carboxamide
—— N-[(2R)-oxan-2-yl]oxy-1,3-thiazole-4-carboxamide —— C9H12N2O3S
N-[(2R)-oxan-2-yl]oxy-1,3-thiazole-4-carboxamide
—— [2-[[5-(4-chlorophenyl)-2-methylpyrazol-3-yl]amino]-2-oxoethyl] 2-[(1R)-cyclopent-2-en-1-yl]acetate —— C19H20ClN3O3
[2-[[5-(4-chlorophenyl)-2-methylpyrazol-3-yl]amino]-2-oxoethyl] 2-[(1R)-cyclopent-2-en-1-yl]acetate
—— [2-[[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 2-[(1R)-cyclopent-2-en-1-yl]acetate —— C21H25N3O3
[2-[[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 2-[(1R)-cyclopent-2-en-1-yl]acetate
—— [2-[[5-(4-chlorophenyl)-2-methylpyrazol-3-yl]amino]-2-oxoethyl] 2-[(1S)-cyclopent-2-en-1-yl]acetate —— C19H20ClN3O3
[2-[[5-(4-chlorophenyl)-2-methylpyrazol-3-yl]amino]-2-oxoethyl] 2-[(1S)-cyclopent-2-en-1-yl]acetate
—— N-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1,3-thiazole-4-carboxamide —— C12H17N3O2S
N-[[(3S,8aR)-3,4,6,7,8,8a-hexahydro-1H-pyrrolo[2,1-c][1,4]oxazin-3-yl]methyl]-1,3-thiazole-4-carboxamide
—— N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1,3-thiazole-4-carboxamide —— C15H19N3OS
N-[(2R)-2-(dimethylamino)-2-(4-methylphenyl)ethyl]-1,3-thiazole-4-carboxamide
—— tert-butyl N-[2-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2-methylpropyl]carbamate —— C17H30N4O3
tert-butyl N-[2-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2-methylpropyl]carbamate
—— N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1,3-thiazole-4-carboxamide —— C9H11N3O2S
N-[(3R)-1-methyl-5-oxopyrrolidin-3-yl]-1,3-thiazole-4-carboxamide
—— N-[(2R)-2-cyclopropyl-2-(1,3-thiazole-4-carbonylamino)ethyl]-1,3-thiazole-4-carboxamide —— C13H14N4O2S2
N-[(2R)-2-cyclopropyl-2-(1,3-thiazole-4-carbonylamino)ethyl]-1,3-thiazole-4-carboxamide
—— [2-[[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 2-[(1S)-cyclopent-2-en-1-yl]acetate —— C21H25N3O3
[2-[[3,5-dimethyl-1-(4-methylphenyl)pyrazol-4-yl]amino]-2-oxoethyl] 2-[(1S)-cyclopent-2-en-1-yl]acetate
—— [(2R)-2-(2,2-dimethylpropyl)pyrrolidin-1-yl]-(1,3-thiazol-4-yl)methanone —— C13H20N2OS
[(2R)-2-(2,2-dimethylpropyl)pyrrolidin-1-yl]-(1,3-thiazol-4-yl)methanone
—— N-[(2R)-2-(5-methylfuran-2-yl)-2-pyrrolidin-1-ylethyl]-1,3-thiazole-4-carboxamide —— C15H19N3O2S
N-[(2R)-2-(5-methylfuran-2-yl)-2-pyrrolidin-1-ylethyl]-1,3-thiazole-4-carboxamide
—— [(2S)-2-(2,2-dimethylpropyl)pyrrolidin-1-yl]-(1,3-thiazol-4-yl)methanone —— C13H20N2OS
[(2S)-2-(2,2-dimethylpropyl)pyrrolidin-1-yl]-(1,3-thiazol-4-yl)methanone
—— N-[(2R)-2-(diethylamino)-2-(furan-2-yl)ethyl]-1,3-thiazole-4-carboxamide —— C14H19N3O2S
N-[(2R)-2-(diethylamino)-2-(furan-2-yl)ethyl]-1,3-thiazole-4-carboxamide
—— N-[(2S)-2-(diethylamino)-2-(furan-2-yl)ethyl]-1,3-thiazole-4-carboxamide —— C14H19N3O2S
N-[(2S)-2-(diethylamino)-2-(furan-2-yl)ethyl]-1,3-thiazole-4-carboxamide
—— N-[(3R)-6-oxopiperidin-3-yl]-1,3-thiazole-4-carboxamide —— C9H11N3O2S
N-[(3R)-6-oxopiperidin-3-yl]-1,3-thiazole-4-carboxamide
—— (3S)-3-acetyl-N-[(2R)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide —— C17H20N4O2
(3S)-3-acetyl-N-[(2R)-1-cyanopropan-2-yl]-N-methyl-2-phenyl-3,4-dihydropyrazole-5-carboxamide