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中文名称 英文名称 CAS号 化学式 结构式图片
—— N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-3-(2-chlorophenyl)-1-methylpyrazole-4-carboxamide —— C24H25Cl2FN4O2
N-[(2R)-2-(2-chloro-6-fluorophenyl)-2-[(2S)-2-methylmorpholin-4-yl]ethyl]-3-(2-chlorophenyl)-1-methylpyrazole-4-carboxamide
—— N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C22H32N4O3
N-[[(3S)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide —— C22H32N4O3
N-[[(3R)-1-(2-methoxyethyl)pyrrolidin-3-yl]methyl]-3-[3-(4-propan-2-ylphenyl)-1,2,4-oxadiazol-5-yl]propanamide
—— 1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(1R)-1-pyridin-4-ylethyl]urea —— C15H20N4OS
1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(1R)-1-pyridin-4-ylethyl]urea
—— (2R)-2-[4-[2-[5-(4-fluoro-3-methylphenyl)tetrazol-2-yl]acetyl]piperazin-1-yl]-2-phenylacetonitrile —— C22H22FN7O
(2R)-2-[4-[2-[5-(4-fluoro-3-methylphenyl)tetrazol-2-yl]acetyl]piperazin-1-yl]-2-phenylacetonitrile
—— 1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(1S)-1-pyridin-4-ylethyl]urea —— C15H20N4OS
1-[2-(2,4-dimethyl-1,3-thiazol-5-yl)ethyl]-3-[(1S)-1-pyridin-4-ylethyl]urea
—— (2S)-2-[4-[2-[5-(4-fluoro-3-methylphenyl)tetrazol-2-yl]acetyl]piperazin-1-yl]-2-phenylacetonitrile —— C22H22FN7O
(2S)-2-[4-[2-[5-(4-fluoro-3-methylphenyl)tetrazol-2-yl]acetyl]piperazin-1-yl]-2-phenylacetonitrile
—— 1-[4-(difluoromethoxy)phenyl]-N-[(1S)-6-(difluoromethoxy)-1,2,3,4-tetrahydronaphthalen-1-yl]-5-methyltriazole-4-carboxamide —— C22H20F4N4O3
1-[4-(difluoromethoxy)phenyl]-N-[(1S)-6-(difluoromethoxy)-1,2,3,4-tetrahydronaphthalen-1-yl]-5-methyltriazole-4-carboxamide
—— 1-(3-chloro-4-fluorophenyl)-N-[(2R)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]-5-methyltriazole-4-carboxamide —— C22H22ClF2N5O2
1-(3-chloro-4-fluorophenyl)-N-[(2R)-2-(3-fluorophenyl)-2-morpholin-4-ylethyl]-5-methyltriazole-4-carboxamide
—— 2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]acetamide —— C20H28N4OS
2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]acetamide
—— 5-ethyl-1-(4-fluorophenyl)-N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]pyrazole-4-carboxamide —— C20H28FN5O
5-ethyl-1-(4-fluorophenyl)-N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]pyrazole-4-carboxamide
—— 5-ethyl-1-(4-fluorophenyl)-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]pyrazole-4-carboxamide —— C20H28FN5O
5-ethyl-1-(4-fluorophenyl)-N-[(2S)-2-(4-methylpiperazin-1-yl)propyl]pyrazole-4-carboxamide
—— 2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]acetamide —— C20H28N4OS
2-(2-benzyl-1,3-thiazol-4-yl)-N-[(2R)-2-(4-methylpiperazin-1-yl)propyl]acetamide
—— N-[(3S)-1-(cyclopropylmethyl)pyrrolidin-3-yl]-2-(4-propan-2-yloxyphenyl)-1,3-thiazole-4-carboxamide —— C21H27N3O2S
N-[(3S)-1-(cyclopropylmethyl)pyrrolidin-3-yl]-2-(4-propan-2-yloxyphenyl)-1,3-thiazole-4-carboxamide
—— (1-ethylpyrazol-4-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C19H21N5O2
(1-ethylpyrazol-4-yl)-[(2S)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— (1-ethylpyrazol-4-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone —— C19H21N5O2
(1-ethylpyrazol-4-yl)-[(2R)-2-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methanone
—— 2,3,4,5-tetrafluoro-N-(1-phenylpyrazol-3-yl)benzamide —— C16H9F4N3O
2,3,4,5-tetrafluoro-N-(1-phenylpyrazol-3-yl)benzamide
—— tert-butyl N-[(2R)-2-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H34N4O3
tert-butyl N-[(2R)-2-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— tert-butyl N-[(2R)-2-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H34N4O3
tert-butyl N-[(2R)-2-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— N-[(3R)-1-(cyclopropylmethyl)pyrrolidin-3-yl]-2-(4-propan-2-yloxyphenyl)-1,3-thiazole-4-carboxamide —— C21H27N3O2S
N-[(3R)-1-(cyclopropylmethyl)pyrrolidin-3-yl]-2-(4-propan-2-yloxyphenyl)-1,3-thiazole-4-carboxamide
—— tert-butyl N-[(2S)-2-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H34N4O3
tert-butyl N-[(2S)-2-[[(2R)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— tert-butyl N-[(2S)-2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H33N3O4
tert-butyl N-[(2S)-2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— tert-butyl N-[(2R)-2-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H33N3O4
tert-butyl N-[(2R)-2-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— tert-butyl N-[(2S)-2-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H34N4O3
tert-butyl N-[(2S)-2-[[(2S)-2-(3,5-dimethylpyrazol-1-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— (2S)-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]oxolane-2-carboxamide —— C13H14N4O2
(2S)-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]oxolane-2-carboxamide
—— (3R,7aR)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide —— C16H17N5O2S
(3R,7aR)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide
—— (3R,7aS)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide —— C16H17N5O2S
(3R,7aS)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide
—— tert-butyl N-[(2R)-2,3-dimethyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]butyl]carbamate —— C16H27N3O3S
tert-butyl N-[(2R)-2,3-dimethyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]butyl]carbamate
—— 1-[2-[[(2S)-oxolane-2-carbonyl]amino]phenyl]pyrazole-3-carboxamide —— C15H16N4O3
1-[2-[[(2S)-oxolane-2-carbonyl]amino]phenyl]pyrazole-3-carboxamide
—— tert-butyl N-[(2R)-2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H33N3O4
tert-butyl N-[(2R)-2-[[(2R)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— tert-butyl N-[(2S)-2-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate —— C19H33N3O4
tert-butyl N-[(2S)-2-[[(2S)-2-(3,5-dimethyl-1,2-oxazol-4-yl)propanoyl]amino]-2,3-dimethylbutyl]carbamate
—— tert-butyl N-[(2S)-2,3-dimethyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]butyl]carbamate —— C16H27N3O3S
tert-butyl N-[(2S)-2,3-dimethyl-2-[(2-methyl-1,3-thiazole-4-carbonyl)amino]butyl]carbamate
—— 4-[(5S)-5-[(5-phenyltetrazol-2-yl)methyl]-4,5-dihydro-1,3-thiazol-2-yl]morpholine —— C15H18N6OS
4-[(5S)-5-[(5-phenyltetrazol-2-yl)methyl]-4,5-dihydro-1,3-thiazol-2-yl]morpholine
—— 1-[2-[[(2R)-oxolane-2-carbonyl]amino]phenyl]pyrazole-3-carboxamide —— C15H16N4O3
1-[2-[[(2R)-oxolane-2-carbonyl]amino]phenyl]pyrazole-3-carboxamide
—— (2R)-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]oxolane-2-carboxamide —— C13H14N4O2
(2R)-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]oxolane-2-carboxamide
—— [2-[[(3S)-3-methyl-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate —— C16H18N2O5S3
[2-[[(3S)-3-methyl-1,1-dioxothiolan-3-yl]amino]-2-oxoethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate
—— [2-oxo-2-[[(1S)-1-thiophen-2-ylethyl]amino]ethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate —— C17H16N2O3S3
[2-oxo-2-[[(1S)-1-thiophen-2-ylethyl]amino]ethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate
—— [5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate —— C17H12N2O4S2
[5-(Furan-2-yl)-1,2-oxazol-3-yl]methyl 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate
—— (5-Phenyl-1,2-oxazol-3-yl)methyl 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate —— C19H14N2O3S2
(5-Phenyl-1,2-oxazol-3-yl)methyl 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate
—— (3S,7aR)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide —— C16H17N5O2S
(3S,7aR)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide
—— 5-(4-Chlorophenyl)-2-[[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]methyl]-1,3-oxazole —— C22H24ClN3O2
5-(4-Chlorophenyl)-2-[[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]methyl]-1,3-oxazole
—— (2R)-2-phenyl-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]butanamide —— C18H18N4O
(2R)-2-phenyl-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]butanamide
—— [2-Oxo-2-(pentylamino)ethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate —— C16H20N2O3S2
[2-Oxo-2-(pentylamino)ethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate
—— (3S,7aS)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide —— C16H17N5O2S
(3S,7aS)-7a-methyl-5-oxo-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]-2,3,6,7-tetrahydropyrrolo[2,1-b][1,3]thiazole-3-carboxamide
—— (2S)-2-phenyl-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]butanamide —— C18H18N4O
(2S)-2-phenyl-N-[3-(1H-1,2,4-triazol-5-yl)phenyl]butanamide
—— N-[(R)-cyclopentyl(thiophen-2-yl)methyl]-1-phenylpyrazole-4-sulfonamide —— C19H21N3O2S2
N-[(R)-cyclopentyl(thiophen-2-yl)methyl]-1-phenylpyrazole-4-sulfonamide
—— 4-[(5R)-5-[(5-phenyltetrazol-2-yl)methyl]-4,5-dihydro-1,3-thiazol-2-yl]morpholine —— C15H18N6OS
4-[(5R)-5-[(5-phenyltetrazol-2-yl)methyl]-4,5-dihydro-1,3-thiazol-2-yl]morpholine
—— [2-[(2-Fluorophenyl)methyl-methylamino]-2-oxoethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate —— C19H17FN2O3S2
[2-[(2-Fluorophenyl)methyl-methylamino]-2-oxoethyl] 2-(2-thiophen-3-yl-1,3-thiazol-4-yl)acetate
—— (3S)-N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-(2-methylpropyl)morpholine-4-carboxamide —— C20H28N4O2
(3S)-N-(3,5-dimethyl-1-phenylpyrazol-4-yl)-3-(2-methylpropyl)morpholine-4-carboxamide
—— 5-(4-Fluorophenyl)-2-[[4-[(4-methoxyphenyl)methyl]piperazine-1,4-diium-1-yl]methyl]-1,3-oxazole —— C22H26FN3O2+2
5-(4-Fluorophenyl)-2-[[4-[(4-methoxyphenyl)methyl]piperazine-1,4-diium-1-yl]methyl]-1,3-oxazole